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3EQY

Crystal structure of human MDMX in complex with a 12-mer peptide inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
A0043066biological_processnegative regulation of apoptotic process
A0051726biological_processregulation of cell cycle
B0005634cellular_componentnucleus
B0043066biological_processnegative regulation of apoptotic process
B0051726biological_processregulation of cell cycle
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE GAI A 302
ChainResidue
AHIS38
AGLY44
AGLU45
AHOH391

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE PO4 A 303
ChainResidue
BGLN88
AGLN26
ATHR48
AGLU51
AHOH400
BARG87

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE PO4 A 306
ChainResidue
ATYR59
ALYS63
AASP79
ALEU80
AHOH381

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE GAI B 301
ChainResidue
BHIS38
BGLY44
BGLU45
BHOH460

site_idAC5
Number of Residues8
DetailsBINDING SITE FOR RESIDUE PO4 B 304
ChainResidue
AARG87
AGLN88
BGLN26
BTHR48
BGLU51
BHOH439
BHOH449
BHOH472

site_idAC6
Number of Residues6
DetailsBINDING SITE FOR RESIDUE PO4 B 305
ChainResidue
BTYR59
BLYS63
BASP79
BLEU80
BHOH432
BHOH443

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PDB entries from 2024-07-17

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