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6E3S

Crystal Structure of the Heterodimeric HIF-2 Complex with Antagonist PT2385

Experimental procedure
Experimental methodSINGLE WAVELENGTH
Source typeSYNCHROTRON
Source detailsAPS BEAMLINE 19-ID
Synchrotron siteAPS
Beamline19-ID
Temperature [K]100
Detector technologyCCD
Collection date2015-11-25
DetectorADSC QUANTUM 315r
Wavelength(s)0.97929
Spacegroup nameP 1 21 1
Unit cell lengths49.009, 97.895, 77.965
Unit cell angles90.00, 107.43, 90.00
Refinement procedure
Resolution48.948 - 3.000
R-factor0.2139
Rwork0.212
R-free0.24910
Structure solution methodMOLECULAR REPLACEMENT
Starting model (for MR)4zp4
RMSD bond length0.010
RMSD bond angle1.257
Data scaling softwareHKL-3000
Phasing softwarePHASER
Refinement softwarePHENIX ((1.10.1_2155: ???))
Data quality characteristics
 OverallOuter shell
Low resolution limit [Å]50.0002.950
High resolution limit [Å]2.9002.900
Rmerge0.0990.765
Number of reflections14037
<I/σ(I)>11.4
Completeness [%]99.0
Redundancy2.6
Crystallization Conditions
crystal IDmethodpHtemperaturedetails
1VAPOR DIFFUSION, SITTING DROP72892% TACSIMATE, PH 7.0, 6% PEG3350

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