Author results

1D4K
  • Download 1d4k
  • View 1d4k
Molmil generated image of 1d4k
HIV-1 PROTEASE COMPLEXED WITH A MACROCYCLIC PEPTIDOMIMETIC INHIBITOR
Descriptor:HIV-1 PROTEASE, SULFATE ION, N-13-[(10S,13S)-9,12-DIOXO-10-(2-BUTYL)-2-OXA-8,11-DIAZABICYCLO [13.2.2] NONADECA-15,17,18-TRIENE] (2R)-BENZYL-(4S)-HYDROXY-5-AMINOPENTANOIC (1R)-HYDROXY-(2S)-INDANEAMIDE
Authors:Tyndall, J.D., Reid, R.C., Tyssen, D.P., Jardine, D.K., Todd, B., Passmore, M., March, D.R., Pattenden, L.K., Alewood, D., Hu, S.H., Alewood, P.F., Birch, C.J., Martin, J.L., Fairlie, D.P.
Deposit date:1999-10-04
Release date:2000-10-11
Last modified:2017-10-04
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Synthesis, stability, antiviral activity, and protease-bound structures of substrate-mimicking constrained macrocyclic inhibitors of HIV-1 protease.
J.Med.Chem., 43, 2000
1D4L
  • Download 1d4l
  • View 1d4l
Molmil generated image of 1d4l
HIV-1 PROTEASE COMPLEXED WITH A MACROCYCLIC PEPTIDOMIMETIC INHIBITOR
Descriptor:HIV-1 PROTEASE, SULFATE ION, (10S,13S,1'R)-13-[1'-HYDROXY-2'-(N-P-AMINOBENZENESULFONYL-1''-AMINO-3''-METHYLBUTYL)ETHYL]-8,11-DIOXO-10-ISOPROPYL-2-OXA-9,12-DIAZABICYCLO [13.2.2]NONADECA-15,17,18-TRIENE
Authors:Tyndall, J.D., Reid, R.C., Tyssen, D.P., Jardine, D.K., Todd, B., Passmore, M., March, D.R., Pattenden, L.K., Alewood, D., Hu, S.H., Alewood, P.F., Birch, C.J., Martin, J.L., Fairlie, D.P.
Deposit date:1999-10-04
Release date:2000-10-11
Last modified:2017-10-04
Method:X-RAY DIFFRACTION (1.75 Å)
Cite:Synthesis, stability, antiviral activity, and protease-bound structures of substrate-mimicking constrained macrocyclic inhibitors of HIV-1 protease.
J.Med.Chem., 43, 2000
3BXR
  • Download 3bxr
  • View 3bxr
Molmil generated image of 3bxr
CRYSTAL STRUCTURES OF HIGHLY CONSTRAINED SUBSTRATE AND HYDROLYSIS PRODUCTS BOUND TO HIV-1 PROTEASE. IMPLICATIONS FOR CATALYTIC MECHANISM
Descriptor:Protease, SULFATE ION, (9S,12S)-9-(1-methylethyl)-N-[(8S,11S)-8-[(1S)-1-methylpropyl]-7,10-dioxo-2-oxa-6,9-diazabicyclo[11.2.2]heptadeca-1(15),13,16-trien-11-yl]-7,10-dioxo-2-oxa-8,11-diazabicyclo[12.2.2]octadeca-1(16),14,17-triene-12-carboxamide
Authors:Tyndall, J.D., Pattenden, L.K., Reid, R.C., Hu, S.H., Alewood, D., Alewood, P.F., Walsh, T., Fairlie, D.P., Martin, J.L.
Deposit date:2008-01-14
Release date:2008-03-25
Last modified:2017-10-25
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:Crystal Structures of Highly Constrained Substrate and Hydrolysis Products Bound to HIV-1 Protease. Implications for the Catalytic Mechanism
Biochemistry, 47, 2008
3BXS
  • Download 3bxs
  • View 3bxs
Molmil generated image of 3bxs
CRYSTAL STRUCTURES OF HIGHLY CONSTRAINED SUBSTRATE AND HYDROLYSIS PRODUCTS BOUND TO HIV-1 PROTEASE. IMPLICATIONS FOR CATALYTIC MECHANISM
Descriptor:Protease, SULFATE ION, (9S,12S)-9-(1-methylethyl)-7,10-dioxo-2-oxa-8,11-diazabicyclo[12.2.2]octadeca-1(16),14,17-triene-12-carboxylic acid
Authors:Tyndall, J.D., Pattenden, L.K., Reid, R.C., Hu, S.H., Alewood, D., Alewood, P.F., Walsh, T., Fairlie, D.P., Martin, J.L.
Deposit date:2008-01-14
Release date:2008-03-25
Last modified:2017-10-25
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:Crystal Structures of Highly Constrained Substrate and Hydrolysis Products Bound to HIV-1 Protease. Implications for the Catalytic Mechanism
Biochemistry, 47, 2008
1RPV
  • Download 1rpv
  • View 1rpv
Molmil generated image of 1rpv
HIV-1 REV PROTEIN (RESIDUES 34-50)
Descriptor:HIV-1 REV PROTEIN
Authors:Scanlon, M.J., Fairlie, D.P., Craik, D.J., Englebretsen, D.R., West, M.L.
Deposit date:1995-05-04
Release date:1995-10-15
Last modified:2011-07-13
Method:SOLUTION NMR
Cite:NMR solution structure of the RNA-binding peptide from human immunodeficiency virus (type 1) Rev.
Biochemistry, 34, 1995
1B6J
  • Download 1b6j
  • View 1b6j
Molmil generated image of 1b6j
HIV-1 PROTEASE COMPLEXED WITH MACROCYCLIC PEPTIDOMIMETIC INHIBITOR 1
Descriptor:RETROPEPSIN, CYCLIC PEPTIDE INHIBITOR, SULFATE ION
Authors:Martin, J.L., Begun, J., Schindeler, A., Wickramasinghe, W.A., Alewood, D., Alewood, P.F., Bergman, D.A., Brinkworth, R.I., Abbenante, G., March, D.R., Reid, R.C., Fairlie, D.P.
Deposit date:1999-01-17
Release date:2000-01-07
Last modified:2013-03-13
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Molecular recognition of macrocyclic peptidomimetic inhibitors by HIV-1 protease.
Biochemistry, 38, 1999
1B6K
  • Download 1b6k
  • View 1b6k
Molmil generated image of 1b6k
HIV-1 PROTEASE COMPLEXED WITH MACROCYCLIC PEPTIDOMIMETIC INHIBITOR 5
Descriptor:RETROPEPSIN, SULFATE ION, N-[3-(8-SEC-BUTYL-7,10-DIOXO-2-OXA-6,9-DIAZA-BICYCLO[11.2.2]HEPTADECA-1(16),13(17),14- TRIEN-11-YLAMINO)-2-HYDROXY-1-(4-HYDROXY-BENZYL)-PROPYL]-3-METHYL-2- (2-OXO-PYRROLIDIN-1-YL)-BUTYRAMIDE
Authors:Martin, J.L., Begun, J., Schindeler, A., Wickramasinghe, W.A., Alewood, D., Alewood, P.F., Bergman, D.A., Brinkworth, R.I., Abbenante, G., March, D.R., Reid, R.C., Fairlie, D.P.
Deposit date:1999-01-17
Release date:2000-01-07
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Molecular recognition of macrocyclic peptidomimetic inhibitors by HIV-1 protease.
Biochemistry, 38, 1999
1B6L
  • Download 1b6l
  • View 1b6l
Molmil generated image of 1b6l
HIV-1 PROTEASE COMPLEXED WITH MACROCYCLIC PEPTIDOMIMETIC INHIBITOR 4
Descriptor:RETROPEPSIN, SULFATE ION, 1-[2-(8-CARBAMOYLMETHYL-6,9-DIOXO-2-OXA-7,10-DIAZA-BICYCLO[11.2.2]HEPTADECA- 1(16),13(17),14-TRIEN-11-YL)-2-HYDROXY-ETHYL]-PIPERIDINE-2-CARBOXYLIC ACID TERT-BUTYLAMIDE
Authors:Martin, J.L., Begun, J., Schindeler, A., Wickramasinghe, W.A., Alewood, D., Alewood, P.F., Bergman, D.A., Brinkworth, R.I., Abbenante, G., March, D.R., Reid, R.C., Fairlie, D.P.
Deposit date:1999-01-17
Release date:2000-01-07
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (1.75 Å)
Cite:Molecular recognition of macrocyclic peptidomimetic inhibitors by HIV-1 protease.
Biochemistry, 38, 1999
1B6M
  • Download 1b6m
  • View 1b6m
Molmil generated image of 1b6m
HIV-1 PROTEASE COMPLEXED WITH MACROCYCLIC PEPTIDOMIMETIC INHIBITOR 6
Descriptor:RETROPEPSIN, SULFATE ION, [1-BENZYL-3-(8-SEC-BUTYL-7,10-DIOXO-2-OXA-6,9-DIAZA-BICYCLO[11.2.2] HEPTADECA-1(16),13(17),14-TRIEN-11-YLAMINO)-2-HYDROXY-PROPYL]-CARBAMIC ACID TERT-BUTYL ESTER
Authors:Martin, J.L., Begun, J., Schindeler, A., Wickramasinghe, W.A., Alewood, D., Alewood, P.F., Bergman, D.A., Brinkworth, R.I., Abbenante, G., March, D.R., Reid, R.C., Fairlie, D.P.
Deposit date:1999-01-17
Release date:2000-01-07
Last modified:2013-02-27
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Molecular recognition of macrocyclic peptidomimetic inhibitors by HIV-1 protease.
Biochemistry, 38, 1999
1B6P
  • Download 1b6p
  • View 1b6p
Molmil generated image of 1b6p
HIV-1 PROTEASE COMPLEXED WITH MACROCYCLIC PEPTIDOMIMETIC INHIBITOR 7
Descriptor:RETROPEPSIN, SULFATE ION, N-[3-(8-SEC-BUTYL-7,10-DIOXO-2-OXA-6,9-DIAZA-BICYCLO[11.2.2] HEPTADECA-1(16),13(17),14-TRIEN-11-YAMINO)-2-HYDROXY-1-(4-HYDROXY-BENZYL) -PROPYL]-3-METHYL-2-PROPIONYLAMINO-BUTYRAMIDE
Authors:Martin, J.L., Begun, J., Schindeler, A., Wickramasinghe, W.A., Alewood, D., Alewood, P.F., Bergman, D.A., Brinkworth, R.I., Abbenante, G., March, D.R., Reid, R.C., Fairlie, D.P.
Deposit date:1999-01-17
Release date:2000-01-07
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (2 Å)
Cite:Molecular recognition of macrocyclic peptidomimetic inhibitors by HIV-1 protease.
Biochemistry, 38, 1999
1BA4
  • Download 1ba4
  • View 1ba4
Molmil generated image of 1ba4
THE SOLUTION STRUCTURE OF AMYLOID BETA-PEPTIDE (1-40) IN A WATER-MICELLE ENVIRONMENT. IS THE MEMBRANE-SPANNING DOMAIN WHERE WE THINK IT IS? NMR, 10 STRUCTURES
Descriptor:AMYLOID BETA-PEPTIDE
Authors:Coles, M., Bicknell, W., Watson, A.A., Fairlie, D.P., Craik, D.J.
Deposit date:1998-04-07
Release date:1998-06-17
Last modified:2011-07-13
Method:SOLUTION NMR
Cite:Solution structure of amyloid beta-peptide(1-40) in a water-micelle environment. Is the membrane-spanning domain where we think it is?
Biochemistry, 37, 1998
1BA6
  • Download 1ba6
  • View 1ba6
Molmil generated image of 1ba6
SOLUTION STRUCTURE OF THE METHIONINE-OXIDIZED AMYLOID BETA-PEPTIDE (1-40). DOES OXIDATION AFFECT CONFORMATIONAL SWITCHING? NMR, 10 STRUCTURES
Descriptor:AMYLOID BETA-PEPTIDE
Authors:Watson, A.A., Fairlie, D.P., Craik, D.J.
Deposit date:1998-04-22
Release date:1998-06-17
Last modified:2011-07-13
Method:SOLUTION NMR
Cite:Solution structure of methionine-oxidized amyloid beta-peptide (1-40). Does oxidation affect conformational switching?
Biochemistry, 37, 1998
1J1A
  • Download 1j1a
  • View 1j1a
Molmil generated image of 1j1a
PANCREATIC SECRETORY PHOSPHOLIPASE A2 (IIA) WITH ANTI-INFLAMMATORY ACTIVITY
Descriptor:Phospholipase A2, CALCIUM ION, (S)-5-(4-BENZYLOXY-PHENYL)-4-(7-PHENYL-HEPTANOYLAMINO)-PENTANOIC ACID
Authors:Hansford, K.A., Reid, R.C., Clark, C.I., Tyndall, J.D.A., Whitehouse, M.W., Guthrie, T., McGeary, R.P., Schafer, K., Martin, J.L., Fairlie, D.P.
Deposit date:2002-12-03
Release date:2003-03-18
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:D-Tyrosine as a Chiral Precusor to Potent Inhibitors of Human Nonpancreatic Secretory Phospholipase A2 (IIa) with Antiinflammatory Activity
Chembiochem, 4, 2003
1Z1H
  • Download 1z1h
  • View 1z1h
Molmil generated image of 1z1h
HIV-1 PROTEASE COMPLEXED WITH MACROCYCLIC PEPTIDOMIMETIC INHIBITOR 3
Descriptor:Pol polyprotein, SULFATE ION, N-{(2R)-2-HYDROXY-2-[(8S,11S)-8-ISOPROPYL-6,9-DIOXO-2-OXA-7,10-DIAZABICYCLO[11.2.2]HEPTADECA-1(15),13,16-TRIEN-11-YL]ETHYL}-N-ISOPENTYLBENZENESULFONAMIDE
Authors:Martin, J.L., Begun, J., Schindeler, A., Wickramasinghe, W.A., Alewood, D., Alewood, P.F., Bergman, D.A., Brinkworth, R.I., Abbenante, G., March, D.R., Reid, R.C., Fairlie, D.P.
Deposit date:2005-03-04
Release date:2005-03-22
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Molecular recognition of macrocyclic peptidomimetic inhibitors by HIV-1 protease
Biochemistry, 38, 1999
1Z1R
  • Download 1z1r
  • View 1z1r
Molmil generated image of 1z1r
HIV-1 PROTEASE COMPLEXED WITH MACROCYCLIC PEPTIDOMIMETIC INHIBITOR 2
Descriptor:Pol polyprotein, SULFATE ION, 2-[(8S,11S)-11-{(1R)-1-HYDROXY-2-[ISOPENTYL(PHENYLSULFONYL)AMINO]ETHYL}-6,9-DIOXO-2-OXA-7,10-DIAZABICYCLO[11.2.2]HEPTADECA-1(15),13,16-TRIEN-8-YL]ACETAMIDE
Authors:Martin, J.L., Begun, J., Schindeler, A., Wickramasinghe, W.A., Alewood, D., Alewood, P.F., Bergman, D.A., Brinkworth, R.I., Abbenante, G., March, D.R., Reid, R.C., Fairlie, D.P.
Deposit date:2005-03-06
Release date:2005-03-22
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Molecular recognition of macrocyclic peptidomimetic inhibitors by HIV-1 protease
Biochemistry, 38, 1999
2MBS
  • Download 2mbs
  • View 2mbs
Molmil generated image of 2mbs
NMR SOLUTION STRUCTURE OF OXIDIZED KPDSBA
Descriptor:Thiol:disulfide interchange protein
Authors:Kurth, F., Rimmer, K., Premkumar, L., Mohanty, B., Duprez, W., Halili, M.A., Shouldice, S.R., Heras, B., Fairlie, D.P., Scanlon, M.J., Martin, J.L.
Deposit date:2013-08-03
Release date:2013-12-11
Method:SOLUTION NMR
Cite:Comparative Sequence, Structure and Redox Analyses of Klebsiella pneumoniae DsbA Show That Anti-Virulence Target DsbA Enzymes Fall into Distinct Classes.
Plos One, 8, 2013
2N08
  • Download 2n08
  • View 2n08
Molmil generated image of 2n08
NMR STRUCTURE OF A SHORT HYDROPHOBIC 11MER PEPTIDE IN 25 MM SDS SOLUTION
Descriptor:Short hydrophobic peptide with cyclic constraints
Authors:Hoang, H.N., Song, K., Hill, T.A., Derksen, D.R., Edmonds, D.J., Kok, W.M., Limberakis, C., Liras, S., Loria, P.M., Mascitti, V., Mathiowetz, A.M., Mitchell, J.M., Piotrowski, D.W., Price, D.A., Stanton, R.V., Suen, J.Y., Withka, J.M., Griffith, D.A., Fairlie, D.P.
Deposit date:2015-03-04
Release date:2015-04-15
Last modified:2015-05-27
Method:SOLUTION NMR
Cite:Short Hydrophobic Peptides with Cyclic Constraints Are Potent Glucagon-like Peptide-1 Receptor (GLP-1R) Agonists.
J.Med.Chem., 58, 2015
2N09
  • Download 2n09
  • View 2n09
Molmil generated image of 2n09
NMR STRUCTURE OF A SHORT HYDROPHOBIC 11MER PEPTIDE IN DMSO-D6/H2O (1:3) SOLUTION
Descriptor:Short hydrophobic peptide with cyclic constraints
Authors:Hoang, H.N., Song, K., Hill, T.A., Derksen, D.R., Edmonds, D.J., Kok, W.M., Limberakis, C., Liras, S., Loria, P.M., Mascitti, V., Mathiowetz, A.M., Mitchell, J.M., Piotrowski, D.W., Price, D.A., Stanton, R.V., Suen, J.Y., Withka, J.M., Griffith, D.A., Fairlie, D.P.
Deposit date:2015-03-04
Release date:2015-04-15
Last modified:2015-05-27
Method:SOLUTION NMR
Cite:Short Hydrophobic Peptides with Cyclic Constraints Are Potent Glucagon-like Peptide-1 Receptor (GLP-1R) Agonists.
J.Med.Chem., 58, 2015
2N0I
  • Download 2n0i
  • View 2n0i
Molmil generated image of 2n0i
NMR SOLUTION STRUCTURE FOR DI-SULFIDE 11MER PEPTIDE
Descriptor:di-sulfide 11mer peptide
Authors:Hoang, H.N., Song, K., Hill, T.A., Derksen, D.R., Edmonds, D.J., Kok, W.M., Limberakis, C., Liras, S., Loria, P.M., Mascitti, V., Mathiowetz, A.M., Mitchell, J.M., Piotrowski, D.W., Price, D.A., Stanton, R.V., Suen, J.Y., Withka, J.M., Griffith, D.A., Fairlie, D.P.
Deposit date:2015-03-09
Release date:2015-04-15
Last modified:2015-05-27
Method:SOLUTION NMR
Cite:Short Hydrophobic Peptides with Cyclic Constraints Are Potent Glucagon-like Peptide-1 Receptor (GLP-1R) Agonists.
J.Med.Chem., 58, 2015
2N0N
  • Download 2n0n
  • View 2n0n
Molmil generated image of 2n0n
NMR SOLUTION STRUCTURE FOR LACTAM (5,9) 11MER
Descriptor:lactam (5,9) 11mer peptide
Authors:Hoang, H.N., Song, K., Hill, T.A., Derksen, D.R., Edmonds, D.J., Kok, W.M., Limberakis, C., Liras, S., Loria, P.M., Mascitti, V., Mathiowetz, A.M., Mitchell, J.M., Piotrowski, D.W., Price, D.A., Stanton, R.V., Suen, J.Y., Withka, J.M., Griffith, D.A., Fairlie, D.P.
Deposit date:2015-03-10
Release date:2015-04-15
Last modified:2015-05-27
Method:SOLUTION NMR
Cite:Short Hydrophobic Peptides with Cyclic Constraints Are Potent Glucagon-like Peptide-1 Receptor (GLP-1R) Agonists.
J.Med.Chem., 58, 2015
4L4T
  • Download 4l4t
  • View 4l4t
Molmil generated image of 4l4t
STRUCTURE OF HUMAN MAIT TCR IN COMPLEX WITH HUMAN MR1-6-FP
Descriptor:Major histocompatibility complex class I-related gene protein, Beta-2-microglobulin, MAIT T-cell receptor alpha chain, ...
Authors:Patel, O., Kjer-Nielsen, L., Le Nours, J., Eckle, S.B.G., Birkinshaw, R.W., Beddoe, T., Corbett, A.J., Liu, L., Miles, J.J., Meehan, B., Reantragoon, R., Sandoval-Romero, M.L., Sullivan, L.C., Brooks, A.G., Chen, Z., Fairlie, D.P., McCluskey, J., Rossjohn, J.
Deposit date:2013-06-09
Release date:2013-07-17
Last modified:2013-09-11
Method:X-RAY DIFFRACTION (2 Å)
Cite:Recognition of vitamin B metabolites by mucosal-associated invariant T cells.
Nat Commun, 4, 2013
4L4V
  • Download 4l4v
  • View 4l4v
Molmil generated image of 4l4v
STRUCTURE OF HUMAN MAIT TCR IN COMPLEX WITH HUMAN MR1-RL-6-ME-7-OH
Descriptor:Major histocompatibility complex class I-related gene protein, Beta-2-microglobulin, MAIT T-cell receptor alpha chain, ...
Authors:Patel, O., Kjer-Nielsen, L., Le Nours, J., Eckle, S.B.G., Birkinshaw, R.W., Beddoe, T., Corbett, A.J., Liu, L., Miles, J.J., Meehan, B., Reantragoon, R., Sandoval-Romero, M.L., Sullivan, L.C., Brooks, A.G., Chen, Z., Fairlie, D.P., McCluskey, J., Rossjohn, J.
Deposit date:2013-06-09
Release date:2013-07-17
Last modified:2013-09-11
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Recognition of vitamin B metabolites by mucosal-associated invariant T cells.
Nat Commun, 4, 2013
5TWI
  • Download 5twi
  • View 5twi
Molmil generated image of 5twi
ALPHA HELIX NUCLEATION BY A SIMPLE CYCLIC TETRAPEPTIDE
Descriptor:Cyclic tetrapeptide ALA-ARG-ALA-UN1
Authors:Hoang, H.N., Fairlie, D.P.
Deposit date:2016-11-13
Release date:2016-12-14
Method:SOLUTION NMR
Cite:Alpha Helix Nucleation by a Simple Cyclic Tetrapeptide
To Be Published
1KQU
  • Download 1kqu
  • View 1kqu
Molmil generated image of 1kqu
HUMAN PHOSPHOLIPASE A2 COMPLEXED WITH A SUBSTRATE ANOLOGUE
Descriptor:Phospholipase A2, membrane associated, CALCIUM ION, ...
Authors:Tyndall, J.D., Martin, J.L.
Deposit date:2002-01-07
Release date:2003-11-11
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:D-Tyrosine as a chiral precusor to potent inhibitors of human nonpancreatic secretory phospholipase A2 (IIa) with antiinflammatory activity.
Chembiochem, 4, 2003
1CPI
  • Download 1cpi
  • View 1cpi
Molmil generated image of 1cpi
REGIOSELECTIVE STRUCTURAL AND FUNCTIONAL MIMICRY OF PEPTIDES. DESIGN OF HYDROLYTICALLY STABLE CYCLIC PEPTIDOMIMETIC INHIBITORS OF HIV-1 PROTEASE
Descriptor:HIV-1 PROTEASE, CYCLIC PEPTIDE INHIBITOR, SULFATE ION
Authors:Martin, J.L.
Deposit date:1995-10-16
Release date:1996-03-08
Last modified:2012-12-12
Method:X-RAY DIFFRACTION (2.05 Å)
Cite:REGIOSELECTIVE STRUCTURAL AND FUNCTIONAL MIMICRY OF PEPTIDES - DESIGN OF HYDROLYTICALLY-STABLE CYCLIC PEPTIDOMIMETIC INHIBITORS OF HIV-1 PROTEASE.
J.Am.Chem.Soc., 117, 1995
<123>