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5ES3
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Co-crystal structure of LDH liganded with oxamate
分子名称: L-lactate dehydrogenase A chain, OXAMIC ACID
著者Nowicki, M.W, Wear, M.A, McNae, I.W, Blackburn, E.A.
登録日2015-11-16
公開日2016-01-13
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.29 Å)
主引用文献A Streamlined, Automated Protocol for the Production of Milligram Quantities of Untagged Recombinant Rat Lactate Dehydrogenase A Using AKTAxpressTM.
Plos One, 10, 2015
2X0J
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2.8 A RESOLUTION STRUCTURE OF MALATE DEHYDROGENASE FROM ARCHAEOGLOBUS FULGIDUS IN COMPLEX WITH ETHENO-NAD
分子名称: ETHENO-NAD, MALATE DEHYDROGENASE, SULFATE ION
著者Irimia, A, Madern, D, Zaccai, G, Vellieux, F.M, Karshikoff, A, Tibbelin, G, Ladenstein, R, Lien, T, Birkeland, N.K.
登録日2009-12-14
公開日2009-12-22
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.786 Å)
主引用文献The 2.9A Resolution Crystal Structure of Malate Dehydrogenase from Archaeoglobus Fulgidus: Mechanisms of Oligomerisation and Thermal Stabilisation.
J.Mol.Biol., 335, 2004
3P7M
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Structure of putative lactate dehydrogenase from Francisella tularensis subsp. tularensis SCHU S4
分子名称: Malate dehydrogenase, PHOSPHATE ION
著者Osinski, T, Cymborowski, M, Zimmerman, M.D, Gordon, E, Grimshaw, S, Skarina, T, Chruszcz, M, Savchenko, A, Anderson, W, Minor, W, Center for Structural Genomics of Infectious Diseases (CSGID)
登録日2010-10-12
公開日2010-10-20
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure of putative lactate dehydrogenase from Francisella tularensis subsp. tularensis SCHU S4
To be Published
3OM9
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T. Gondii bradyzoite-specific LDH (LDH1) in complex with NAD and OXQ
分子名称: 4-HYDROXY-1,2,5-OXADIAZOLE-3-CARBOXYLIC ACID, Lactate dehydrogenase, NICOTINAMIDE-ADENINE-DINUCLEOTIDE
著者Susko, M.S, Wilson, D.K.
登録日2010-08-26
公開日2010-10-27
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献T.Gondii bradyzoite-specific LDH (LDH1) in complex with NAD and OXQ
To be Published
2XXB
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Penta-mutant of Thermus thermophilus lactate dehydrogenase, complex with AMP
分子名称: ADENOSINE MONOPHOSPHATE, L-LACTATE DEHYDROGENASE
著者Diop, F, Coquelle, N, Vellieux, F.M.D.
登録日2010-11-09
公開日2010-11-17
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Lactate Dehydrogenase from T. Thermophilus, Penta-Mutant (Complex with AMP)
To be Published
5KKC
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l-lactate dehydrogenase from rabbit muscle with the inhibitor 6DHNAD
分子名称: L-lactate dehydrogenase A chain, SULFATE ION, [[(2~{R},3~{S},4~{R},5~{R})-5-(5-aminocarbonyl-2~{H}-pyridin-1-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methoxy-oxidanyl-phosphoryl] [(2~{R},3~{S},4~{R},5~{R})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl hydrogen phosphate
著者Meneely, K.M, Moran, G.R, Lamb, A.L.
登録日2016-06-21
公開日2016-11-02
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.859 Å)
主引用文献Ligand binding phenomena that pertain to the metabolic function of renalase.
Arch.Biochem.Biophys., 612, 2016
2XXJ
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Penta mutant of lactate dehydrogenase from Thermus thermophilus, ternary complex
分子名称: L-LACTATE DEHYDROGENASE, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, OXAMIC ACID, ...
著者Tickle, J, de Mendoza Barbera, E, Vellieux, F.M.D.
登録日2010-11-10
公開日2010-11-24
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.964 Å)
主引用文献Lactate Dehydrogenase from T. Thermophilus, Penta- Mutant (Ternary Complex)
To be Published
5KVV
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Structure of Malate Dehydrogenase in complex with NADH from Mycobacterium tuberculosis
分子名称: 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, GLYCEROL, ...
著者Cheng, Y.S, Sacchettini, J.C, TB Structural Genomics Consortium (TBSGC)
登録日2016-07-15
公開日2016-09-14
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.01 Å)
主引用文献Structure of Malate Dehydrogenase in complex with NADH from Mycobacterium tuberculosis
To Be Published
5KKA
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E. coli malate dehydrogenase with the inhibitor 6DHNAD
分子名称: Malate dehydrogenase, [[(2~{R},3~{S},4~{R},5~{R})-5-(5-aminocarbonyl-2~{H}-pyridin-1-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methoxy-oxidanyl-phosphoryl] [(2~{R},3~{S},4~{R},5~{R})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl hydrogen phosphate
著者Meneely, K.M, Lamb, A.L, Moran, G.R.
登録日2016-06-21
公開日2016-11-02
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Ligand binding phenomena that pertain to the metabolic function of renalase.
Arch.Biochem.Biophys., 612, 2016
3PQE
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Crystal structure of L-lactate dehydrogenase from Bacillus subtilis with H171C mutation
分子名称: L-lactate dehydrogenase
著者Zhang, Y, Garavito, R.M.
登録日2010-11-26
公開日2011-12-14
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal structure of L-lactate dehydrogenase from Bacillus subtilis with H171C mutation
To be Published
3PQF
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Crystal structure of L-lactate dehydrogenase from Bacillus subtilis mutation H171C complexed with NAD+
分子名称: L-lactate dehydrogenase, NICOTINAMIDE-ADENINE-DINUCLEOTIDE
著者Zhang, Y, Garavito, R.M.
登録日2010-11-26
公開日2012-01-11
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.49 Å)
主引用文献Crystal structure of L-lactate dehydrogenase from Bacillus subtilis mutation H171C complexed with NAD+
To be Published
3PQD
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Crystal structure of L-lactate dehydrogenase from Bacillus subtilis complexed with FBP and NAD+
分子名称: 1,6-di-O-phosphono-beta-D-fructofuranose, L-lactate dehydrogenase, NICOTINAMIDE-ADENINE-DINUCLEOTIDE
著者Zhang, Y, Garavito, R.M.
登録日2010-11-26
公開日2012-01-18
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.376 Å)
主引用文献Crystal structure of L-lactate dehydrogenase from Bacillus subtilis complexed with FBP and NAD+
To be Published
2ZQY
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T-state structure of allosteric L-lactate dehydrogenase from Lactobacillus casei
分子名称: L-lactate dehydrogenase, NITRATE ION
著者Arai, K, Ishimitsu, T, Fushinobu, S, Uchikoba, H, Matsuzawa, H, Taguchi, H.
登録日2008-08-22
公開日2009-09-08
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Active and inactive state structures of unliganded Lactobacillus casei allosteric L-lactate dehydrogenase.
Proteins, 78, 2010
5LDH
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STRUCTURE OF THE ACTIVE TERNARY COMPLEX OF PIG HEART LACTATE DEHYDROGENASE WITH S-LAC-NAD AT 2.7 ANGSTROMS RESOLUTION
分子名称: (3S)-5-(3-CARBOXY-3-HYDROXYPROPYL) NICOTINAMIDE-ADENINE-DINUCLEOTIDE, CITRIC ACID, LACTATE DEHYDROGENASE
著者Grau, U.M, Rossmann, M.G.
登録日1980-10-29
公開日1981-03-04
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structure of the active ternary complex of pig heart lactate dehydrogenase with S-lac-NAD at 2.7 A resolution.
J.Mol.Biol., 151, 1981
2ZQZ
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R-state structure of allosteric L-lactate dehydrogenase from Lactobacillus casei
分子名称: L-lactate dehydrogenase, SULFATE ION
著者Arai, K, Ishimitsu, T, Fushinobu, S, Uchikoba, H, Matsuzawa, H, Taguchi, H.
登録日2008-08-22
公開日2009-09-08
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Active and inactive state structures of unliganded Lactobacillus casei allosteric L-lactate dehydrogenase.
Proteins, 78, 2010
5MDH
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CRYSTAL STRUCTURE OF TERNARY COMPLEX OF PORCINE CYTOPLASMIC MALATE DEHYDROGENASE ALPHA-KETOMALONATE AND TNAD AT 2.4 ANGSTROMS RESOLUTION
分子名称: ALPHA-KETOMALONIC ACID, MALATE DEHYDROGENASE, NICOTINAMIDE-ADENINE-DINUCLEOTIDE
著者Chapman, A.D.M, Cortes, A, Dafforn, T.R, Clarke, A.R, Brady, R.L.
登録日1998-10-08
公開日1999-05-18
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural basis of substrate specificity in malate dehydrogenases: crystal structure of a ternary complex of porcine cytoplasmic malate dehydrogenase, alpha-ketomalonate and tetrahydoNAD.
J.Mol.Biol., 285, 1999
5HTO
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BU of 5hto by Molmil
Crystal structure of Plasmodium Vivax LDH in complex with a DNA aptamer called pL1 (tetrameric LDH in an asymmetric unit)
分子名称: DNA (30-MER), DNA (34-MER), L-lactate dehydrogenase, ...
著者Choi, S.J, Ban, C.
登録日2016-01-27
公開日2016-10-19
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structure of a DNA aptamer bound to PvLDH elucidates novel single-stranded DNA structural elements for folding and recognition
Sci Rep, 6, 2016
5HS4
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Plasmdoium Vivax Lactate dehydrogenase
分子名称: L-lactate dehydrogenase
著者Choi, S.J, Ban, C.
登録日2016-01-25
公開日2016-10-19
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.339 Å)
主引用文献Crystal structure of a DNA aptamer bound to PvLDH elucidates novel single-stranded DNA structural elements for folding and recognition
Sci Rep, 6, 2016
5HRU
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Crystal structure of Plasmodium vivax LDH in complex with a DNA aptamer called pL1
分子名称: DNA (32-MER), L-lactate dehydrogenase, MAGNESIUM ION
著者Choi, S.J, Ban, C.
登録日2016-01-24
公開日2016-10-19
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.71 Å)
主引用文献Crystal structure of a DNA aptamer bound to PvLDH elucidates novel single-stranded DNA structural elements for folding and recognition
Sci Rep, 6, 2016
5IXY
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Lactate Dehydrogenase in complex with hydroxylactam inhibitor compound 31: (2~{S})-5-(2-chlorophenyl)sulfanyl-2-(4-morpholin-4-ylphenyl)-4-oxidanyl-2-thiophen-3-yl-1,3-dihydropyridin-6-one
分子名称: (2~{S})-5-(2-chlorophenyl)sulfanyl-2-(4-morpholin-4-ylphenyl)-4-oxidanyl-2-thiophen-3-yl-1,3-dihydropyridin-6-one, L-lactate dehydrogenase A chain, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ...
著者Chen, Z, Eigenbrot, C.
登録日2016-03-23
公開日2016-09-14
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Cell Active Hydroxylactam Inhibitors of Human Lactate Dehydrogenase with Oral Bioavailability in Mice.
Acs Med.Chem.Lett., 7, 2016
5IXS
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Lactate Dehydrogenase in complex with hydroxylactam inhibitor compound 9: (6R)-3-[(2-chlorophenyl)sulfanyl]-4-hydroxy-6-(3-hydroxyphenyl)-6-(thiophen-3-yl)-5,6-dihydropyridin-2(1H)-one
分子名称: (6R)-3-[(2-chlorophenyl)sulfanyl]-4-hydroxy-6-(3-hydroxyphenyl)-6-(thiophen-3-yl)-5,6-dihydropyridin-2(1H)-one, 1,4,5,6-TETRAHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, ...
著者Ultsch, M, Eigenbrot, C.
登録日2016-03-23
公開日2016-09-14
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Cell Active Hydroxylactam Inhibitors of Human Lactate Dehydrogenase with Oral Bioavailability in Mice.
Acs Med.Chem.Lett., 7, 2016
3TL2
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Crystal structure of Bacillus anthracis str. Ames malate dehydrogenase in closed conformation.
分子名称: 1,2-ETHANEDIOL, Malate dehydrogenase, THIOCYANATE ION
著者Blus, B.J, Chruszcz, M, Tkaczuk, K.L, Osinski, T, Cymborowski, M, Kudritska, M, Grimshaw, S, Savchenko, A, Anderson, W.F, Minor, W, Center for Structural Genomics of Infectious Diseases (CSGID)
登録日2011-08-29
公開日2011-09-21
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structure of Bacillus anthracis str. Ames malate dehydrogenase in closed conformation.
TO BE PUBLISHED
2HLP
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CRYSTAL STRUCTURE OF THE E267R MUTANT OF A HALOPHILIC MALATE DEHYDROGENASE IN THE APO FORM
分子名称: CHLORIDE ION, MALATE DEHYDROGENASE, SODIUM ION
著者Richard, S.B, Madern, D, Garcin, E, Zaccai, G.
登録日1999-04-23
公開日2000-02-04
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.59 Å)
主引用文献Halophilic adaptation: novel solvent protein interactions observed in the 2.9 and 2.6 A resolution structures of the wild type and a mutant of malate dehydrogenase from Haloarcula marismortui.
Biochemistry, 39, 2000
2I6T
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Orthorhombic Structure of the LDH domain of Human Ubiquitin-conjugating Enzyme E2-like Isoform A
分子名称: GLYCEROL, SULFATE ION, UBIQUITIN-CONJUGATING ENZYME E2-LIKE ISOFORM A
著者Walker, J.R, Avvakumov, G.V, Xue, S, Newman, E.M, Finerty Jr, P.J, Butler-Cole, C, Tempel, W, Weigelt, J, Sundstrom, M, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Dhe-Paganon, S.
登録日2006-08-29
公開日2006-10-24
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structural Investigation into the L-lactate Dehydrogenase Domain of Human Ubiquitin-conjugating Enzyme E2-like Isoform A
To be Published
6ZZR
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The Crystal Structure of human LDHA from Biortus.
分子名称: 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, L-lactate dehydrogenase A chain
著者Wang, F, Lin, D, Cheng, W, Bao, X, Zhu, B, Shang, H.
登録日2020-08-05
公開日2020-08-19
最終更新日2024-04-24
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献The Crystal Structure of human LDHA from Biortus
To Be Published

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