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3C31	Crystal structure of GluR5 ligand-binding core in complex with lithium at 1.49 Angstrom resolution Descriptor: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, CHLORIDE ION, GLUTAMATE RECEPTOR, ... Authors: Mayer, M.L. Deposit date: 2008-01-27 Release date: 2008-06-17 Last modified: 2023-08-30 Method: X-RAY DIFFRACTION (1.49 Å) Cite: Molecular basis of kainate receptor modulation by sodium. Neuron, 58, 2008
1S9T	Crystal structure of the GLUR6 ligand binding core in complex with quisqualate at 1.8A resolution Descriptor: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, CHLORIDE ION, Glutamate receptor, ... Authors: Mayer, M.L. Deposit date: 2004-02-05 Release date: 2005-02-08 Last modified: 2023-10-25 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Crystal structures of the GluR5 and GluR6 ligand binding cores: molecular mechanisms underlying kainate receptor selectivity. Neuron, 45, 2005
1S7Y	Crystal structure of the GluR6 ligand binding core in complex with glutamate at 1.75 A resolution orthorhombic form Descriptor: GLUTAMIC ACID, Glutamate receptor, ionotropic kainate 2 precursor Authors: Mayer, M.L. Deposit date: 2004-01-30 Release date: 2005-02-08 Last modified: 2024-02-14 Method: X-RAY DIFFRACTION (1.75 Å) Cite: Crystal structures of the GluR5 and GluR6 ligand binding cores: Molecular mechanisms underlying kainate receptor selectivity Neuron, 45, 2005
2I0C	Crystal structure of the GluR6 ligand binding core dimer crosslinked by disulfide bonds between Y490C and L752C at 2.25 Angstroms Resolution Descriptor: GLUTAMIC ACID, Glutamate receptor, ionotropic kainate 2 Authors: Mayer, M.L. Deposit date: 2006-08-10 Release date: 2006-11-21 Last modified: 2024-04-03 Method: X-RAY DIFFRACTION (2.25 Å) Cite: Conformational restriction blocks glutamate receptor desensitization. Nat.Struct.Mol.Biol., 13, 2006
2I0B	Crystal structure of the GluR6 ligand binding core ELKQ mutant dimer at 1.96 Angstroms Resolution Descriptor: GLUTAMIC ACID, Glutamate receptor, ionotropic kainate 2, ... Authors: Mayer, M.L. Deposit date: 2006-08-10 Release date: 2006-11-21 Last modified: 2024-04-03 Method: X-RAY DIFFRACTION (1.96 Å) Cite: Conformational restriction blocks glutamate receptor desensitization. Nat.Struct.Mol.Biol., 13, 2006
2I3W	Measurement of conformational changes accompanying desensitization in an ionotropic glutamate receptor: Structure of S729C mutant Descriptor: GLUTAMATE RECEPTOR SUBUNIT 2, GLUTAMIC ACID Authors: Armstrong, N, Jasti, J, Beich-Frandsen, M, Gouaux, E. Deposit date: 2006-08-21 Release date: 2006-10-17 Last modified: 2023-08-30 Method: X-RAY DIFFRACTION (2.3 Å) Cite: Measurement of Conformational Changes accompanying Desensitization in an Ionotropic Glutamate Receptor. Cell(Cambridge,Mass.), 127, 2006
1SD3	Crystal structure of the GLUR6 ligand binding core in complex with 2S,4R-4-methylglutamate at 1.8 Angstrom resolution Descriptor: 2S,4R-4-METHYLGLUTAMATE, Glutamate receptor, ionotropic kainate 2 Authors: Mayer, M.L. Deposit date: 2004-02-12 Release date: 2005-02-15 Last modified: 2023-10-25 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Crystal structures of the GluR5 and GluR6 ligand binding cores: molecular mechanisms underlying kainate receptor selectivity. Neuron, 45, 2005
2I3V	Measurement of conformational changes accompanying desensitization in an ionotropic glutamate receptor: Structure of G725C mutant Descriptor: GLUTAMIC ACID, Glutamate receptor 2, ZINC ION Authors: Armstrong, N, Jasti, J, Beich-Frandsen, M, Gouaux, E. Deposit date: 2006-08-21 Release date: 2006-10-17 Last modified: 2023-08-30 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Measurement of Conformational Changes accompanying Desensitization in an Ionotropic Glutamate Receptor. Cell(Cambridge,Mass.), 127, 2006
3DP4	Crystal structure of the binding domain of the AMPA subunit GluR3 bound to AMPA Descriptor: (S)-ALPHA-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACID, Glutamate receptor 3, ZINC ION Authors: Ahmed, A.H, Wang, Q, Sondermann, H, Oswald, R.E. Deposit date: 2008-07-07 Release date: 2008-11-25 Last modified: 2023-08-30 Method: X-RAY DIFFRACTION (2.11 Å) Cite: Structure of the S1S2 glutamate binding domain of GLuR3. Proteins, 75, 2008
1S50	X-ray structure of the GluR6 ligand binding core (S1S2A) in complex with glutamate at 1.65 A resolution Descriptor: GLUTAMIC ACID, Glutamate Receptor 6 Authors: Mayer, M.L. Deposit date: 2004-01-19 Release date: 2005-02-08 Last modified: 2023-08-23 Method: X-RAY DIFFRACTION (1.65 Å) Cite: Crystal structures of the GluR5 and GluR6 ligand binding cores: Molecular mechanisms underlying kainate receptor selectivity Neuron, 45, 2005
1VSO	Crystal Structure of the Ligand-Binding Core of iGluR5 in Complex With the Antagonist (S)-ATPO at 1.85 A resolution Descriptor: (S)-2-AMINO-3-(5-TERT-BUTYL-3-(PHOSPHONOMETHOXY)-4-ISOXAZOLYL)PROPIONIC ACID, GLYCEROL, Glutamate receptor, ... Authors: Hald, H, Naur, P, Gajhede, M, Kastrup, J.S. Deposit date: 2007-03-29 Release date: 2007-07-03 Last modified: 2023-08-23 Method: X-RAY DIFFRACTION (1.85 Å) Cite: Partial agonism and antagonism of the ionotropic glutamate receptor iGLuR5: structures of the ligand-binding core in complex with domoic acid and 2-amino-3-[5-tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl]propionic acid. J.Biol.Chem., 282, 2007
3DP6	Crystal structure of the binding domain of the AMPA subunit GluR2 bound to glutamate Descriptor: GLUTAMIC ACID, Glutamate receptor 2, ZINC ION Authors: Ahmed, A.H, Wang, Q, Sondermann, H, Oswald, R.E. Deposit date: 2008-07-07 Release date: 2008-11-25 Last modified: 2023-08-30 Method: X-RAY DIFFRACTION (1.55 Å) Cite: Structure of the S1S2 glutamate binding domain of GLuR3. Proteins, 75, 2008
3DLN	Crystal structure of the binding domain of the AMPA subunit GluR3 bound to glutamate Descriptor: GLUTAMIC ACID, Glutamate receptor 3, ZINC ION Authors: Ahmed, A.H, Wang, Q, Sondermann, H, Oswald, R.E. Deposit date: 2008-06-27 Release date: 2008-11-25 Last modified: 2023-08-30 Method: X-RAY DIFFRACTION (1.91 Å) Cite: Structure of the S1S2 glutamate binding domain of GLuR3. Proteins, 75, 2008
1TXF	CRYSTAL STRUCTURE OF THE GLUR5 LIGAND BINDING CORE IN COMPLEX WITH GLUTAMATE AT 2.1 ANGSTROM RESOLUTION Descriptor: GLUTAMIC ACID, Glutamate receptor, ionotropic kainate 1 Authors: Mayer, M.L. Deposit date: 2004-07-04 Release date: 2005-02-08 Last modified: 2023-08-23 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Crystal structures of the GluR5 and GluR6 ligand binding cores: Molecular mechanisms underlying kainate receptor selectivity Neuron, 45, 2005
1TT1	CRYSTAL STRUCTURE OF THE GLUR6 LIGAND BINDING CORE IN COMPLEX WITH KAINATE 1.93 A RESOLUTION Descriptor: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, Glutamate receptor, ionotropic kainate 2 Authors: Mayer, M.L. Deposit date: 2004-06-21 Release date: 2005-02-08 Last modified: 2023-08-23 Method: X-RAY DIFFRACTION (1.93 Å) Cite: Crystal structures of the GluR5 and GluR6 ligand binding cores: Molecular mechanisms underlying kainate receptor selectivity Neuron, 45, 2005
3EN3	Crystal Structure of the GluR4 Ligand-Binding domain in complex with kainate Descriptor: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, Glutamate receptor 4,Glutamate receptor Authors: Gill, A, Madden, D.R. Deposit date: 2008-09-25 Release date: 2009-05-19 Last modified: 2017-07-26 Method: X-RAY DIFFRACTION (2.43 Å) Cite: Correlating AMPA receptor activation and cleft closure across subunits: crystal structures of the GluR4 ligand-binding domain in complex with full and partial agonists Biochemistry, 47, 2008
3EPE	Crystal Structure of the GluR4 Ligand-Binding domain in complex with glutamate Descriptor: GLUTAMIC ACID, Glutamate receptor 4,Glutamate receptor Authors: Gill, A, Madden, D.R. Deposit date: 2008-09-29 Release date: 2009-05-19 Last modified: 2023-09-06 Method: X-RAY DIFFRACTION (1.85 Å) Cite: Correlating AMPA receptor activation and cleft closure across subunits: crystal structures of the GluR4 ligand-binding domain in complex with full and partial agonists Biochemistry, 47, 2008
1SYI	X-RAY STRUCTURE OF THE Y702F MUTANT OF THE GLUR2 LIGAND-BINDING CORE (S1S2J) IN COMPLEX WITH (S)-CPW399 AT 2.1 A RESOLUTION. Descriptor: (S)-2-AMINO-3-(1,3,5,7-PENTAHYDRO-2,4-DIOXO-CYCLOPENTA[E]PYRIMIDIN-1-YL) PROIONIC ACID, Glutamate receptor 2 Authors: Frandsen, A, Pickering, D.S, Vestergaard, B, Kasper, C, Nielsen, B.B, Greenwood, J.R, Campiani, G, Gajhede, M, Schousboe, A, Kastrup, J.S. Deposit date: 2004-04-01 Release date: 2005-03-22 Last modified: 2023-08-23 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Tyr702 Is an Important Determinant of Agonist Binding and Domain Closure of the Ligand-Binding Core of GluR2. Mol.Pharmacol., 67, 2005
1XHY	X-ray structure of the Y702F mutant of the GluR2 ligand-binding core (S1S2J) in complex with kainate at 1.85 A resolution Descriptor: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, Glutamate receptor, SULFATE ION Authors: Frandsen, A, Pickering, D.S, Vestergaard, B, Kasper, C, Nielsen, B.B, Greenwood, J.R, Campiani, G, Gajhede, M, Schousboe, A, Kastrup, J.S. Deposit date: 2004-09-21 Release date: 2005-03-22 Last modified: 2023-08-23 Method: X-RAY DIFFRACTION (1.85 Å) Cite: Tyr702 Is an Important Determinant of Agonist Binding and Domain Closure of the Ligand-Binding Core of GluR2. Mol.Pharmacol., 67, 2005
1Y20	Crystal structure of the NR1 ligand-binding core in complex with ACPC Descriptor: 1-AMINOCYCLOPROPANECARBOXYLIC ACID, Glutamate [NMDA] receptor subunit zeta 1 Authors: Inanobe, A, Gouaux, E. Deposit date: 2004-11-19 Release date: 2005-07-12 Last modified: 2017-07-26 Method: X-RAY DIFFRACTION (1.4 Å) Cite: Mechanism of Partial Agonist Action at the NR1 Subunit of NMDA Receptors. Neuron, 47, 2005
1Y1M	Crystal structure of the NR1 ligand binding core in complex with cycloleucine Descriptor: 1-AMINOCYCLOPENTANECARBOXYLIC ACID, Glutamate [NMDA] receptor subunit zeta 1 Authors: Inanobe, A, Gouaux, E. Deposit date: 2004-11-18 Release date: 2005-07-12 Last modified: 2017-07-26 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Mechanism of Partial Agonist Action at the NR1 Subunit of NMDA Receptors. Neuron, 47, 2005
1Y1Z	Crystal structure of the NR1 ligand binding core in complex with ACBC Descriptor: 1-AMINOCYCLOBUTANECARBOXLIC ACID, Glutamate [NMDA] receptor subunit zeta 1 Authors: Inanobe, A, Gouaux, E. Deposit date: 2004-11-19 Release date: 2005-07-12 Last modified: 2017-07-26 Method: X-RAY DIFFRACTION (1.5 Å) Cite: Mechanism of Partial Agonist Action at the NR1 Subunit of NMDA Receptors. Neuron, 47, 2005
1YCJ	Crystal structure of the kainate receptor GluR5 ligand-binding core in complex with (S)-glutamate Descriptor: GLUTAMIC ACID, Ionotropic glutamate receptor 5, SULFATE ION Authors: Naur, P, Vestergaard, B, Skov, L.K, Egebjerg, J, Gajhede, M, Kastrup, J.S. Deposit date: 2004-12-22 Release date: 2005-02-01 Last modified: 2023-10-25 Method: X-RAY DIFFRACTION (1.95 Å) Cite: Crystal structure of the kainate receptor GluR5 ligand-binding core in complex with (S)-glutamate Febs Lett., 579, 2005
2F36	Crystal Structure of the GluR5 Ligand Binding Core Dimer with Glutamate At 2.1 Angstroms Resolution Descriptor: GLUTAMATE RECEPTOR, IONOTROPIC KAINATE 1, GLUTAMIC ACID, ... Authors: Mayer, M.L. Deposit date: 2005-11-18 Release date: 2006-04-04 Last modified: 2023-08-23 Method: X-RAY DIFFRACTION (2.11 Å) Cite: Crystal structures of the kainate receptor GluR5 ligand binding core dimer with novel GluR5-selective antagonists. J.Neurosci., 26, 2006
1YAE	Structure of the Kainate Receptor Subunit GluR6 Agonist Binding Domain Complexed with Domoic Acid Descriptor: (2S,3S,4S)-2-CARBOXY-4-[(1Z,3E,5R)-5-CARBOXY-1-METHYL-1,3-HEXADIENYL]-3-PYRROLIDINEACETIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor, ... Authors: Nanao, M.H, Green, T, Stern-Bach, Y, Heinemann, S.F, Choe, S. Deposit date: 2004-12-17 Release date: 2005-02-01 Last modified: 2023-08-23 Method: X-RAY DIFFRACTION (3.11 Å) Cite: Structure of the kainate receptor subunit GluR6 agonist-binding domain complexed with domoic acid. Proc.Natl.Acad.Sci.USA, 102, 2005

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