Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
PDB: 9 results

5U1X
DownloadVisualize
BU of 5u1x by Molmil
Crystal structure of the ATP-gated P2X7 ion channel bound to allosteric antagonist JNJ47965567
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, N-{[4-(4-phenylpiperazin-1-yl)oxan-4-yl]methyl}-2-(phenylsulfanyl)pyridine-3-carboxamide, ...
Authors:Karasawa, A, Kawate, T.
Deposit date:2016-11-29
Release date:2017-01-04
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (3.201 Å)
Cite:Structural basis for subtype-specific inhibition of the P2X7 receptor.
Elife, 5, 2016
5U1Y
DownloadVisualize
BU of 5u1y by Molmil
Crystal structure of the ATP-gated P2X7 ion channel bound to allosteric antagonist GW791343
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, N~2~-(3,4-difluorophenyl)-N-{2-methyl-5-[(piperazin-1-yl)methyl]phenyl}glycinamide, P2X purinoceptor
Authors:Karasawa, A, Kawate, T.
Deposit date:2016-11-29
Release date:2017-01-04
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (3.3 Å)
Cite:Structural basis for subtype-specific inhibition of the P2X7 receptor.
Elife, 5, 2016
8JV8
DownloadVisualize
BU of 8jv8 by Molmil
Cryo-EM structure of the panda P2X7 receptor in complex with PPNDS
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 3-[(E)-{4-formyl-5-hydroxy-6-methyl-3-[(phosphonooxy)methyl]pyridin-2-yl}diazenyl]-7-nitronaphthalene-1,5-disulfonic acid, P2X purinoceptor
Authors:Sheng, D, Hattori, M.
Deposit date:2023-06-27
Release date:2023-11-29
Last modified:2024-05-15
Method:ELECTRON MICROSCOPY (3.34 Å)
Cite:Structural insights into the orthosteric inhibition of P2X receptors by non-ATP analog antagonists.
Elife, 12, 2024
5U1V
DownloadVisualize
BU of 5u1v by Molmil
Crystal structure of the ATP-gated P2X7 ion channel bound to allosteric antagonist A804598
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, N-cyano-N'-[(1R)-1-phenylethyl]-N''-quinolin-5-ylguanidine, ...
Authors:Karasawa, A, Kawate, T.
Deposit date:2016-11-29
Release date:2017-01-11
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (3.4 Å)
Cite:Structural basis for subtype-specific inhibition of the P2X7 receptor.
Elife, 5, 2016
5U1L
DownloadVisualize
BU of 5u1l by Molmil
Crystal structure of the ATP-gated P2X7 ion channel in the closed, apo state
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, P2X purinoceptor
Authors:Karasawa, A, Kawate, T.
Deposit date:2016-11-28
Release date:2017-01-04
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (3.4 Å)
Cite:Structural basis for subtype-specific inhibition of the P2X7 receptor.
Elife, 5, 2016
5U1W
DownloadVisualize
BU of 5u1w by Molmil
Crystal structure of the ATP-gated P2X7 ion channel bound to allosteric antagonist AZ10606120
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, N-[2-({2-[(2-hydroxyethyl)amino]ethyl}amino)quinolin-5-yl]-2-[(3s,5s,7s)-tricyclo[3.3.1.1~3,7~]decan-1-yl]acetamide, ...
Authors:Karasawa, A, Kawate, T.
Deposit date:2016-11-29
Release date:2017-01-04
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (3.501 Å)
Cite:Structural basis for subtype-specific inhibition of the P2X7 receptor.
Elife, 5, 2016
8JV7
DownloadVisualize
BU of 8jv7 by Molmil
Cryo-EM structure of the panda P2X7 receptor in complex with PPADS
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-[(E)-[4-methanoyl-6-methyl-5-oxidanyl-3-(phosphonooxymethyl)pyridin-2-yl]diazenyl]benzene-1,3-disulfonic acid, P2X purinoceptor
Authors:Sheng, D, Hattori, M.
Deposit date:2023-06-27
Release date:2023-11-29
Last modified:2024-05-15
Method:ELECTRON MICROSCOPY (3.6 Å)
Cite:Structural insights into the orthosteric inhibition of P2X receptors by non-ATP analog antagonists.
Elife, 12, 2024
5U1U
DownloadVisualize
BU of 5u1u by Molmil
Crystal structure of the ATP-gated P2X7 ion channel bound to allosteric antagonist A740003
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, N-{(1R)-1-[N''-cyano-N'-(quinolin-5-yl)carbamimidamido]-2,2-dimethylpropyl}-2-(3,4-dimethoxyphenyl)acetamide, P2X purinoceptor
Authors:Karasawa, A, Kawate, T.
Deposit date:2016-11-29
Release date:2017-01-11
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (3.604 Å)
Cite:Structural basis for subtype-specific inhibition of the P2X7 receptor.
Elife, 5, 2016
5U2H
DownloadVisualize
BU of 5u2h by Molmil
Crystal structure of the ATP-gated P2X7 ion channel bound to ATP and allosteric antagonist A804598
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ADENOSINE-5'-TRIPHOSPHATE, ...
Authors:Karasawa, A, Kawate, T.
Deposit date:2016-11-30
Release date:2017-01-04
Last modified:2024-04-03
Method:X-RAY DIFFRACTION (3.903 Å)
Cite:Structural basis for subtype-specific inhibition of the P2X7 receptor.
Elife, 5, 2016

223166

PDB entries from 2024-07-31

PDB statisticsPDBj update infoContact PDBjnumon