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PDB: 3 results

7LCI
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BU of 7lci by Molmil
PF 06882961 bound to the glucagon-like peptide-1 receptor (GLP-1R):Gs complex
Descriptor: 2-[(4-{6-[(4-cyano-2-fluorophenyl)methoxy]pyridin-2-yl}piperidin-1-yl)methyl]-1-{[(2S)-oxetan-2-yl]methyl}-1H-benzimidazole-6-carboxylic acid, Glucagon-like peptide 1 receptor, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ...
Authors:Belousoff, M.J, Johnson, R.M, Drulyte, I, Yu, L, Kotecha, A, Danev, R, Wootten, D, Zhang, X, Sexton, P.M.
Deposit date:2021-01-11
Release date:2021-01-20
Last modified:2021-09-15
Method:ELECTRON MICROSCOPY (2.9 Å)
Cite:Evolving cryo-EM structural approaches for GPCR drug discovery.
Structure, 29, 2021
7LCJ
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BU of 7lcj by Molmil
PF 06882961 bound to the glucagon-like peptide-1 receptor (GLP-1R):Gs complex
Descriptor: 2-[(4-{6-[(4-cyano-2-fluorophenyl)methoxy]pyridin-2-yl}piperidin-1-yl)methyl]-1-{[(2S)-oxetan-2-yl]methyl}-1H-benzimidazole-6-carboxylic acid, Glucagon-like peptide 1 receptor
Authors:Belousoff, M.J, Johnson, R.M, Drulyte, I, Yu, L, Kotecha, A, Danev, R, Wootten, D, Zhang, X, Sexton, P.M.
Deposit date:2021-01-11
Release date:2021-01-20
Last modified:2021-09-15
Method:ELECTRON MICROSCOPY (2.82 Å)
Cite:Evolving cryo-EM structural approaches for GPCR drug discovery.
Structure, 29, 2021
7LCK
DownloadVisualize
BU of 7lck by Molmil
PF 06882961 bound to the glucagon-like peptide-1 receptor (GLP-1R)
Descriptor: 2-[(4-{6-[(4-cyano-2-fluorophenyl)methoxy]pyridin-2-yl}piperidin-1-yl)methyl]-1-{[(2S)-oxetan-2-yl]methyl}-1H-benzimidazole-6-carboxylic acid, Glucagon-like peptide 1 receptor
Authors:Belousoff, M.J, Johnson, R.M, Drulyte, I, Yu, L, Kotecha, A, Danev, R, Wootten, D, Zhang, X, Sexton, P.M.
Deposit date:2021-01-11
Release date:2021-01-20
Last modified:2021-09-15
Method:ELECTRON MICROSCOPY (3.24 Å)
Cite:Evolving cryo-EM structural approaches for GPCR drug discovery.
Structure, 29, 2021

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