6HGM
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![BU of 6hgm by Molmil](/molmil-images/mine/6hgm) | |
5OM2
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![BU of 5om2 by Molmil](/molmil-images/mine/5om2) | Crystal structure of Alpha1-antichymotrypsin variant DBS-I1: a drug-binding serpin for doxycycline | Descriptor: | (4S,4AR,5S,5AR,6R,12AS)-4-(DIMETHYLAMINO)-3,5,10,12,12A-PENTAHYDROXY-6-METHYL-1,11-DIOXO-1,4,4A,5,5A,6,11,12A-OCTAHYDROTETRACENE-2-CARBOXAMIDE, 1,2-ETHANEDIOL, Alpha-1-antichymotrypsin | Authors: | Schmidt, K, Muller, Y.A. | Deposit date: | 2017-07-28 | Release date: | 2018-05-23 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (1.47 Å) | Cite: | Design of an allosterically modulated doxycycline and doxorubicin drug-binding protein. Proc. Natl. Acad. Sci. U.S.A., 115, 2018
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6HGN
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6HGI
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![BU of 6hgi by Molmil](/molmil-images/mine/6hgi) | |
5OM5
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![BU of 5om5 by Molmil](/molmil-images/mine/5om5) | |
6HGF
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![BU of 6hgf by Molmil](/molmil-images/mine/6hgf) | Crystal structure of Alpha1-antichymotrypsin variant NewBG-II: a new binding globulin in complex with cortisol | Descriptor: | (11alpha,14beta)-11,17,21-trihydroxypregn-4-ene-3,20-dione, 1,2-ETHANEDIOL, Alpha-1-antichymotrypsin | Authors: | Schmidt, K, Muller, Y.A. | Deposit date: | 2018-08-23 | Release date: | 2019-05-29 | Last modified: | 2024-01-17 | Method: | X-RAY DIFFRACTION (1.651 Å) | Cite: | NewBG: A surrogate corticosteroid-binding globulin with an unprecedentedly high ligand release efficacy. J.Struct.Biol., 207, 2019
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5OM7
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![BU of 5om7 by Molmil](/molmil-images/mine/5om7) | |
6HGG
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![BU of 6hgg by Molmil](/molmil-images/mine/6hgg) | Crystal structure of Alpha1-antichymotrypsin variant NewBG-III: a new binding globulin in complex with cortisol | Descriptor: | (11alpha,14beta)-11,17,21-trihydroxypregn-4-ene-3,20-dione, 1,2-ETHANEDIOL, Alpha-1-antichymotrypsin | Authors: | Schmidt, K, Muller, Y.A. | Deposit date: | 2018-08-23 | Release date: | 2019-05-29 | Last modified: | 2024-01-17 | Method: | X-RAY DIFFRACTION (1.787 Å) | Cite: | NewBG: A surrogate corticosteroid-binding globulin with an unprecedentedly high ligand release efficacy. J.Struct.Biol., 207, 2019
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6FTP
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![BU of 6ftp by Molmil](/molmil-images/mine/6ftp) | |
6HGJ
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![BU of 6hgj by Molmil](/molmil-images/mine/6hgj) | |
5OM6
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![BU of 5om6 by Molmil](/molmil-images/mine/5om6) | |
6HGK
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![BU of 6hgk by Molmil](/molmil-images/mine/6hgk) | |
6HGH
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![BU of 6hgh by Molmil](/molmil-images/mine/6hgh) | |
6HGD
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![BU of 6hgd by Molmil](/molmil-images/mine/6hgd) | |
6HGL
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![BU of 6hgl by Molmil](/molmil-images/mine/6hgl) | |
5OM3
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![BU of 5om3 by Molmil](/molmil-images/mine/5om3) | Crystal structure of Alpha1-antichymotrypsin variant DBS-I5: a MMP14-cleavable drug-binding serpin for doxycycline | Descriptor: | (4S,4AR,5S,5AR,6R,12AS)-4-(DIMETHYLAMINO)-3,5,10,12,12A-PENTAHYDROXY-6-METHYL-1,11-DIOXO-1,4,4A,5,5A,6,11,12A-OCTAHYDROTETRACENE-2-CARBOXAMIDE, Alpha-1-antichymotrypsin, DI(HYDROXYETHYL)ETHER | Authors: | Schmidt, K, Muller, Y.A. | Deposit date: | 2017-07-28 | Release date: | 2018-05-23 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Design of an allosterically modulated doxycycline and doxorubicin drug-binding protein. Proc. Natl. Acad. Sci. U.S.A., 115, 2018
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1AS4
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![BU of 1as4 by Molmil](/molmil-images/mine/1as4) | CLEAVED ANTICHYMOTRYPSIN A349R | Descriptor: | ACETATE ION, ANTICHYMOTRYPSIN | Authors: | Lukacs, C.M, Christianson, D.W. | Deposit date: | 1997-08-12 | Release date: | 1998-02-25 | Last modified: | 2024-02-07 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | Engineering an anion-binding cavity in antichymotrypsin modulates the "spring-loaded" serpin-protease interaction. Biochemistry, 37, 1998
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5OM8
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![BU of 5om8 by Molmil](/molmil-images/mine/5om8) | |
1QMN
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![BU of 1qmn by Molmil](/molmil-images/mine/1qmn) | |
3CAA
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![BU of 3caa by Molmil](/molmil-images/mine/3caa) | CLEAVED ANTICHYMOTRYPSIN A347R | Descriptor: | ANTICHYMOTRYPSIN | Authors: | Lukacs, C.M, Christianson, D.W. | Deposit date: | 1997-08-18 | Release date: | 1998-02-25 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (2.4 Å) | Cite: | Engineering an anion-binding cavity in antichymotrypsin modulates the "spring-loaded" serpin-protease interaction. Biochemistry, 37, 1998
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3DLW
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![BU of 3dlw by Molmil](/molmil-images/mine/3dlw) | Antichymotrypsin | Descriptor: | Alpha-1-antichymotrypsin | Authors: | Feil, S.C. | Deposit date: | 2008-06-29 | Release date: | 2009-07-07 | Last modified: | 2023-11-01 | Method: | X-RAY DIFFRACTION (2.7 Å) | Cite: | Identification and characterization of a misfolded monomeric serpin formed at physiological temperature J.Mol.Biol., 403, 2010
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2ACH
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![BU of 2ach by Molmil](/molmil-images/mine/2ach) | CRYSTAL STRUCTURE OF CLEAVED HUMAN ALPHA1-ANTICHYMOTRYPSIN AT 2.7 ANGSTROMS RESOLUTION AND ITS COMPARISON WITH OTHER SERPINS | Descriptor: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ALPHA 1-ANTICHYMOTRYPSIN, PHOSPHATE ION, ... | Authors: | Baumann, U, Huber, R, Bode, W, Grosse, D, Lesjak, M, Laurell, C.B. | Deposit date: | 1993-04-26 | Release date: | 1993-07-15 | Last modified: | 2020-07-29 | Method: | X-RAY DIFFRACTION (2.7 Å) | Cite: | Crystal structure of cleaved human alpha 1-antichymotrypsin at 2.7 A resolution and its comparison with other serpins. J.Mol.Biol., 218, 1991
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6HGE
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![BU of 6hge by Molmil](/molmil-images/mine/6hge) | |
4CAA
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![BU of 4caa by Molmil](/molmil-images/mine/4caa) | CLEAVED ANTICHYMOTRYPSIN T345R | Descriptor: | ANTICHYMOTRYPSIN | Authors: | Lukacs, C.M, Christianson, D.W. | Deposit date: | 1997-08-14 | Release date: | 1998-02-25 | Last modified: | 2024-05-22 | Method: | X-RAY DIFFRACTION (2.9 Å) | Cite: | Engineering an anion-binding cavity in antichymotrypsin modulates the "spring-loaded" serpin-protease interaction. Biochemistry, 37, 1998
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