6R11
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![BU of 6r11 by Molmil](/molmil-images/mine/6r11) | Cereblon isoform 4 from Magnetospirillum gryphiswaldense in complex with compound 5b | Descriptor: | 5-azanyl-2-[(3~{S})-2,5-bis(oxidanylidene)pyrrolidin-3-yl]isoindole-1,3-dione, CHLORIDE ION, Cereblon isoform 4, ... | Authors: | Heim, C, Hartmann, M.D. | Deposit date: | 2019-03-13 | Release date: | 2019-08-07 | Last modified: | 2024-01-24 | Method: | X-RAY DIFFRACTION (1.75 Å) | Cite: | De-Novo Design of Cereblon (CRBN) Effectors Guided by Natural Hydrolysis Products of Thalidomide Derivatives. J.Med.Chem., 62, 2019
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6R13
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6R12
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6R18
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6R19
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6R1A
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6R1D
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6R1K
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6R1W
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6R1X
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6R1C
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1C3T
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5SWK
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1VL3
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![BU of 1vl3 by Molmil](/molmil-images/mine/1vl3) | DESIGN OF NEW MIMOCHROMES WITH UNIQUE TOPOLOGY | Descriptor: | CO(III)-(DEUTEROPORPHYRIN IX), GLU-SER-GLN-LEU-HIS-SER-ASN-LYS-ARG | Authors: | Lombardi, A, Nastri, F, Marasco, D, Maglio, O, De Sanctis, G, Sinibaldi, F, Santucci, R, Coletta, M, Pavone, V. | Deposit date: | 2004-07-05 | Release date: | 2004-07-20 | Last modified: | 2023-12-27 | Method: | SOLUTION NMR | Cite: | Design of a New Mimochrome with Unique Topology. Chemistry, 9, 2003
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7PWY
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![BU of 7pwy by Molmil](/molmil-images/mine/7pwy) | Structure of human dimeric ACMSD in complex with the inhibitor TES-1025 | Descriptor: | 2-[3-[(5-cyano-6-oxidanylidene-4-thiophen-2-yl-1H-pyrimidin-2-yl)sulfanylmethyl]phenyl]ethanoic acid, 2-amino-3-carboxymuconate-6-semialdehyde decarboxylase, POTASSIUM ION, ... | Authors: | Cianci, M, Giacche, N, Carotti, A, Liscio, P, Amici, A, Cialabrini, L, De Franco, F, Pellicciari, R, Raffaelli, N. | Deposit date: | 2021-10-07 | Release date: | 2022-04-20 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Structural Basis of Human Dimeric alpha-Amino-beta-Carboxymuconate-epsilon-Semialdehyde Decarboxylase Inhibition With TES-1025. Front Mol Biosci, 9, 2022
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1KVF
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1KVG
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![BU of 1kvg by Molmil](/molmil-images/mine/1kvg) | EPO-3 beta Hairpin Peptide | Descriptor: | Protein: EPO-3 Receptor Agonist | Authors: | Skelton, N.J, Russell, S, de Sauvage, F, Cochran, A.G. | Deposit date: | 2002-01-25 | Release date: | 2002-03-06 | Last modified: | 2022-02-23 | Method: | SOLUTION NMR | Cite: | Amino Acid Determinants of beta-Hairpin Conformation in Erythropoeitin
Receptor Agonist Peptides Derived from a Phage Display Library J.Mol.Biol., 316, 2002
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1AO0
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1GX5
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1GX6
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6F0Q
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6F0S
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6F0T
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![BU of 6f0t by Molmil](/molmil-images/mine/6f0t) | Crystal structure of Pizza6-SFW | Descriptor: | GLYCEROL, Pizza6-SFW | Authors: | Noguchi, H, De Zitter, E, Van Meervelt, L, Voet, A.R.D. | Deposit date: | 2017-11-20 | Release date: | 2018-03-21 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (1.74 Å) | Cite: | Design of tryptophan-containing mutants of the symmetrical Pizza protein for biophysical studies. Biochem. Biophys. Res. Commun., 497, 2018
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6NBR
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6OP5
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