1S6X
| Solution structure of VSTx | 分子名称: | KvAP CHANNEL | 著者 | Jung, H.J, Eu, Y.J, Kim, J.I. | 登録日 | 2004-01-28 | 公開日 | 2005-03-22 | 最終更新日 | 2022-03-02 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure and lipid membrane partitioning of VSTx1, an inhibitor of the KvAP potassium channel. Biochemistry, 44, 2005
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1SF4
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2HOG
| crystal structure of Chek1 in complex with inhibitor 20 | 分子名称: | (5-{3-[5-(PIPERIDIN-1-YLMETHYL)-1H-INDOL-2-YL]-1H-INDAZOL-6-YL}-2H-1,2,3-TRIAZOL-4-YL)METHANOL, Serine/threonine-protein kinase Chk1 | 著者 | Yan, Y, Ikuta, M. | 登録日 | 2006-07-14 | 公開日 | 2007-04-24 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | 3-(Indol-2-yl)indazoles as Chek1 kinase inhibitors: Optimization of potency and selectivity via substitution at C6. Bioorg.Med.Chem.Lett., 16, 2006
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2ZLT
| Horse methemoglobin high salt, pH 7.0 | 分子名称: | Hemoglobin subunit alpha, Hemoglobin subunit beta, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Kaushal, P.S, Sankaranarayanan, R, Vijayan, M. | 登録日 | 2008-04-10 | 公開日 | 2008-06-24 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Water-mediated variability in the structure of relaxed-state haemoglobin Acta Crystallogr.,Sect.F, 64, 2008
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1VSG
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2EVN
| NMR solution structures of At1g77540 | 分子名称: | Protein At1g77540 | 著者 | Tyler, R.C, Singh, S, Tonelli, M, Min, M.S, Markley, J.L, Center for Eukaryotic Structural Genomics (CESG) | 登録日 | 2005-10-31 | 公開日 | 2005-11-15 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Structure of Arabidopsis thaliana At1g77540 Protein, a Minimal Acetyltransferase from the COG2388 Family. Biochemistry, 45, 2006
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3TZE
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1K19
| NMR Solution Structure of the Chemosensory Protein CSP2 from Moth Mamestra brassicae | 分子名称: | Chemosensory Protein CSP2 | 著者 | Mosbah, A, Campanacci, V, Lartigue, A, Tegoni, M, Cambillau, C, Darbon, H. | 登録日 | 2001-09-24 | 公開日 | 2002-12-04 | 最終更新日 | 2022-02-23 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of a chemosensory protein from the moth Mamestra brassicae BIOCHEM.J., 369, 2003
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2W4C
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1BMM
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1KDU
| SEQUENTIAL 1H NMR ASSIGNMENTS AND SECONDARY STRUCTURE OF THE KRINGLE DOMAIN FROM UROKINASE | 分子名称: | PLASMINOGEN ACTIVATOR | 著者 | Li, X, Bokman, A.M, Llinas, M, Smith, R.A.G, Dobson, C.M. | 登録日 | 1993-07-15 | 公開日 | 1993-10-31 | 最終更新日 | 2024-06-05 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the kringle domain from urokinase-type plasminogen activator. J.Mol.Biol., 235, 1994
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1LRE
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2J5E
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1TLS
| THYMIDYLATE SYNTHASE TERNARY COMPLEX WITH FDUMP AND METHYLENETETRAHYDROFOLATE | 分子名称: | 5-FLUORO-2'-DEOXYURIDINE-5'-MONOPHOSPHATE, 5-METHYL-5,6,7,8-TETRAHYDROFOLIC ACID, THYMIDYLATE SYNTHASE | 著者 | Hyatt, D.C, Maley, F, Montfort, W.R. | 登録日 | 1996-12-03 | 公開日 | 1997-07-07 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Use of strain in a stereospecific catalytic mechanism: crystal structures of Escherichia coli thymidylate synthase bound to FdUMP and methylenetetrahydrofolate. Biochemistry, 36, 1997
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2J3W
| The crystal structure of the bet3-trs31-sedlin complex. | 分子名称: | PALMITIC ACID, TRAFFICKING PROTEIN PARTICLE COMPLEX PROTEIN 2, TRAFFICKING PROTEIN PARTICLE COMPLEX SUBUNIT 3, ... | 著者 | Kim, Y.-G, Oh, B.-H. | 登録日 | 2006-08-23 | 公開日 | 2006-11-27 | 最終更新日 | 2013-08-07 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | The Architecture of the Multisubunit Trapp I Complex Suggests a Model for Vesicle Tethering. Cell(Cambridge,Mass.), 127, 2006
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3BGR
| Crystal structure of K103N/Y181C mutant HIV-1 reverse transcriptase (RT) in complex with TMC278 (Rilpivirine), a non-nucleoside RT inhibitor | 分子名称: | 1,2-ETHANEDIOL, 4-{[4-({4-[(E)-2-cyanoethenyl]-2,6-dimethylphenyl}amino)pyrimidin-2-yl]amino}benzonitrile, Reverse transcriptase/ribonuclease H, ... | 著者 | Das, K, Bauman, J.D, Clark Jr, A.D, Shatkin, A.J, Arnold, E. | 登録日 | 2007-11-27 | 公開日 | 2008-02-12 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | High-resolution structures of HIV-1 reverse transcriptase/TMC278 complexes: Strategic flexibility explains potency against resistance mutations. Proc.Natl.Acad.Sci.Usa, 105, 2008
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3DN5
| Aldose Reductase in complex with novel biarylic inhibitor | 分子名称: | 3-[5-(3-nitrophenyl)thiophen-2-yl]propanoic acid, Aldose reductase, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE | 著者 | Steuber, H, Klebe, G. | 登録日 | 2008-07-01 | 公開日 | 2009-04-07 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Structure-Based Optimization of Aldose Reductase Inhibitors Originating from Virtual Screening Chemmedchem, 4, 2009
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1W9H
| The Structure of a Piwi protein from Archaeoglobus fulgidus. | 分子名称: | CADMIUM ION, CHLORIDE ION, HYPOTHETICAL PROTEIN AF1318, ... | 著者 | Parker, J.S, Roe, S.M, Barford, D. | 登録日 | 2004-10-13 | 公開日 | 2005-01-13 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Crystal Structure of a Piwi Protein Suggests Mechanisms for Sirna Recognition and Slicer Activity Embo J., 23, 2004
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1FI6
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1A9N
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1TUS
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3CBP
| Set7/9-ER-Sinefungin complex | 分子名称: | BETA-MERCAPTOETHANOL, Estrogen receptor, GLYCEROL, ... | 著者 | Cheng, X, Jia, D. | 登録日 | 2008-02-22 | 公開日 | 2008-05-13 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.42 Å) | 主引用文献 | Regulation of estrogen receptor alpha by the SET7 lysine methyltransferase. Mol.Cell, 30, 2008
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2ETT
| Solution Structure of Human Sorting Nexin 22 PX Domain | 分子名称: | Sorting nexin-22 | 著者 | Song, J, Zhao, Q, Tyler, R.C, Lee, M.S, Newman, C.L, Markley, J.L, Center for Eukaryotic Structural Genomics (CESG) | 登録日 | 2005-10-27 | 公開日 | 2005-11-15 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of human sorting nexin 22. Protein Sci., 16, 2007
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2V3O
| Thrombin with 3-cycle with F | 分子名称: | (2R)-[(4-CARBAMIMIDOYLPHENYL)AMINO]{3-[3-(DIMETHYLAMINO)-2,2-DIMETHYLPROPOXY]-5-ETHYL-2-FLUOROPHENYL}ETHANOIC ACID, CALCIUM ION, HIRUDIN IIA, ... | 著者 | Banner, D.W, Wessel, H.P. | 登録日 | 2007-06-19 | 公開日 | 2008-06-24 | 最終更新日 | 2013-10-23 | 実験手法 | X-RAY DIFFRACTION (1.79 Å) | 主引用文献 | Fluorine in Pharmaceuticals: Looking Beyond Intuition. Science, 317, 2007
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1LUH
| SOLUTION NMR STRUCTURE OF SELF-COMPLIMENTARY DUPLEX 5'-D(TCCG*CGGA)2 CONTAINING A TRIMETHYLENE CROSSLINK AT THE N2 POSITION OF G* | 分子名称: | 5'-D(*TP*CP*CP*(TME)GP*CP*GP*GP*A)-3', PROPANE | 著者 | Dooley, P.D, Zhang, M, Korbel, G.A, Nechev, L.V, Harris, C.M, Stone, M.P, Harris, T.M. | 登録日 | 2002-05-22 | 公開日 | 2003-02-11 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | NMR Determination of the Conformation of a Trimethylene Interstrand Cross-Link in an Oligodeoxynucleotide Duplex Containing a 5'-d(GpC) Motif J.AM.CHEM.SOC., 125, 2003
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