4K0W
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![BU of 4k0w by Molmil](/molmil-images/mine/4k0w) | X-ray crystal structure of OXA-23 A220 duplication clinical variant | 分子名称: | 1,2-ETHANEDIOL, BICARBONATE ION, Beta-lactamase, ... | 著者 | Kaitany, K.J, Klinger, N.V, Leonard, D.A, Powers, R.A. | 登録日 | 2013-04-04 | 公開日 | 2013-08-07 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.2 Å) | 主引用文献 | Structures of the Class D Carbapenemases OXA-23 and OXA-146: Mechanistic Basis of Activity against Carbapenems, Extended-Spectrum Cephalosporins, and Aztreonam. Antimicrob.Agents Chemother., 57, 2013
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4JWI
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![BU of 4jwi by Molmil](/molmil-images/mine/4jwi) | |
4JWE
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![BU of 4jwe by Molmil](/molmil-images/mine/4jwe) | |
4JF6
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![BU of 4jf6 by Molmil](/molmil-images/mine/4jf6) | Structure of OXA-23 at pH 7.0 | 分子名称: | Beta-lactamase, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ... | 著者 | Smith, C.A, Vakulenko, S.B. | 登録日 | 2013-02-27 | 公開日 | 2013-09-25 | 最終更新日 | 2013-10-09 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structural Basis for Carbapenemase Activity of the OXA-23 beta-Lactamase from Acinetobacter baumannii. Chem.Biol., 20, 2013
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4JF5
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![BU of 4jf5 by Molmil](/molmil-images/mine/4jf5) | Structure of OXA-23 at pH 4.1 | 分子名称: | 1,2-ETHANEDIOL, Beta-lactamase, CITRATE ANION | 著者 | Smith, C.A, Vakulenko, S.B. | 登録日 | 2013-02-27 | 公開日 | 2013-09-25 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.15 Å) | 主引用文献 | Structural Basis for Carbapenemase Activity of the OXA-23 beta-Lactamase from Acinetobacter baumannii. Chem.Biol., 20, 2013
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4JF4
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![BU of 4jf4 by Molmil](/molmil-images/mine/4jf4) | OXA-23 meropenem complex | 分子名称: | (4R,5S)-3-{[(3S,5S)-5-(dimethylcarbamoyl)pyrrolidin-3-yl]sulfanyl}-5-[(2S,3R)-3-hydroxy-1-oxobutan-2-yl]-4-methyl-4,5-dihydro-1H-pyrrole-2-carboxylic acid, 1,2-ETHANEDIOL, Beta-lactamase | 著者 | Smith, C.A, Vakulenko, S.B, Toth, M. | 登録日 | 2013-02-27 | 公開日 | 2013-09-25 | 最終更新日 | 2013-10-09 | 実験手法 | X-RAY DIFFRACTION (2.14 Å) | 主引用文献 | Structural Basis for Carbapenemase Activity of the OXA-23 beta-Lactamase from Acinetobacter baumannii. Chem.Biol., 20, 2013
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4HNA
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![BU of 4hna by Molmil](/molmil-images/mine/4hna) | |
4GAB
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![BU of 4gab by Molmil](/molmil-images/mine/4gab) | Human AKR1B10 mutant V301L complexed with NADP+ and fidarestat | 分子名称: | (2S,4S)-2-AMINOFORMYL-6-FLUORO-SPIRO[CHROMAN-4,4'-IMIDAZOLIDINE]-2',5'-DIONE, Aldo-keto reductase family 1 member B10, CHLORIDE ION, ... | 著者 | Cousido-Siah, A, Ruiz Figueras, F.X, Mitschler, A, Podjarny, A. | 登録日 | 2012-07-25 | 公開日 | 2013-03-20 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.5971 Å) | 主引用文献 | X-ray structure of the V301L aldo-keto reductase 1B10 complexed with NADP(+) and the potent aldose reductase inhibitor fidarestat: Implications for inhibitor binding and selectivity. Chem.Biol.Interact, 202, 2013
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4F6R
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![BU of 4f6r by Molmil](/molmil-images/mine/4f6r) | Tubulin:Stathmin-like domain complex | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Designed ankyrin repeat protein (DARPIN) D2, GUANOSINE-5'-DIPHOSPHATE, ... | 著者 | Gigant, B, Mignot, I, Knossow, M. | 登録日 | 2012-05-15 | 公開日 | 2012-07-18 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.64 Å) | 主引用文献 | Design and characterization of modular scaffolds for tubulin assembly. J.Biol.Chem., 287, 2012
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4F61
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![BU of 4f61 by Molmil](/molmil-images/mine/4f61) | Tubulin:Stathmin-like domain complex | 分子名称: | GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ... | 著者 | Gigant, B, Mignot, I, Knossow, M. | 登録日 | 2012-05-14 | 公開日 | 2012-07-18 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (4.17 Å) | 主引用文献 | Design and characterization of modular scaffolds for tubulin assembly. J.Biol.Chem., 287, 2012
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4EB6
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![BU of 4eb6 by Molmil](/molmil-images/mine/4eb6) | Tubulin-Vinblastine: Stathmin-like complex | 分子名称: | (2ALPHA,2'BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLASTINE, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ... | 著者 | Ranaivoson, F.M, Gigant, B, Knossow, M. | 登録日 | 2012-03-23 | 公開日 | 2012-08-01 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (3.47 Å) | 主引用文献 | Structural plasticity of tubulin assembly probed by vinca-domain ligands. Acta Crystallogr.,Sect.D, 68, 2012
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4DRX
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![BU of 4drx by Molmil](/molmil-images/mine/4drx) | GTP-Tubulin in complex with a DARPIN | 分子名称: | Designed ankyrin repeat protein (DARPIN) D1, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ... | 著者 | Pecqueur, L, Gigant, B, Knossow, M. | 登録日 | 2012-02-17 | 公開日 | 2012-07-11 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.22 Å) | 主引用文献 | A designed ankyrin repeat protein selected to bind to tubulin caps the microtubule plus end. Proc.Natl.Acad.Sci.USA, 109, 2012
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4CK4
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![BU of 4ck4 by Molmil](/molmil-images/mine/4ck4) | Ovine beta-Lactoglobulin at Atomic Resolution | 分子名称: | ACETATE ION, AMMONIUM ION, BETA_LACTOGLOBULIN-1/B, ... | 著者 | Kontopidis, G, Nordle, A, Sawyer, L. | 登録日 | 2013-12-27 | 公開日 | 2014-10-08 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.12 Å) | 主引用文献 | Ovine Beta-Lactoglobulin at Atomic Resolution Acta Crystallogr.,Sect.F, 70, 2014
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3UT5
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![BU of 3ut5 by Molmil](/molmil-images/mine/3ut5) | Tubulin-Colchicine-Ustiloxin: Stathmin-like domain complex | 分子名称: | GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ... | 著者 | Ranaivoson, F.M, Gigant, B, Knossow, M. | 登録日 | 2011-11-25 | 公開日 | 2012-08-01 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.73 Å) | 主引用文献 | Structural plasticity of tubulin assembly probed by vinca-domain ligands. Acta Crystallogr.,Sect.D, 68, 2012
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3RYI
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![BU of 3ryi by Molmil](/molmil-images/mine/3ryi) | GDP-Tubulin: rb3 stathmin-like domain complex | 分子名称: | GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ... | 著者 | Nawrotek, A, Knossow, M, Gigant, B. | 登録日 | 2011-05-11 | 公開日 | 2011-10-05 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | The Determinants That Govern Microtubule Assembly from the Atomic Structure of GTP-Tubulin. J.Mol.Biol., 412, 2011
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3RYH
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![BU of 3ryh by Molmil](/molmil-images/mine/3ryh) | GMPCPP-Tubulin: RB3 Stathmin-like domain complex | 分子名称: | GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID GUANYLATE ESTER, ... | 著者 | Nawrotek, A, Knossow, M, Gigant, B. | 登録日 | 2011-05-11 | 公開日 | 2011-10-05 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | The Determinants That Govern Microtubule Assembly from the Atomic Structure of GTP-Tubulin. J.Mol.Biol., 412, 2011
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3RYF
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![BU of 3ryf by Molmil](/molmil-images/mine/3ryf) | GTP-Tubulin: RB3 Stathmin-like domain complex | 分子名称: | GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, SULFATE ION, ... | 著者 | Nawrotek, A, Knossow, M, Gigant, B. | 登録日 | 2011-05-11 | 公開日 | 2011-10-05 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.52 Å) | 主引用文献 | The Determinants That Govern Microtubule Assembly from the Atomic Structure of GTP-Tubulin. J.Mol.Biol., 412, 2011
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3RYC
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![BU of 3ryc by Molmil](/molmil-images/mine/3ryc) | Tubulin: RB3 stathmin-like domain complex | 分子名称: | GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ... | 著者 | Nawrotek, A, Knossow, M, Gigant, B. | 登録日 | 2011-05-11 | 公開日 | 2011-10-05 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | The Determinants That Govern Microtubule Assembly from the Atomic Structure of GTP-Tubulin. J.Mol.Biol., 412, 2011
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3QE3
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![BU of 3qe3 by Molmil](/molmil-images/mine/3qe3) | Sheep liver sorbitol dehydrogenase | 分子名称: | ACETIC ACID, GLYCEROL, Sorbitol dehydrogenase, ... | 著者 | Yennawar, N.H, Yennawar, H.P. | 登録日 | 2011-01-19 | 公開日 | 2011-04-27 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | X-ray crystal structure and small-angle X-ray scattering of sheep liver sorbitol dehydrogenase. Acta Crystallogr.,Sect.D, 67, 2011
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3PTL
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![BU of 3ptl by Molmil](/molmil-images/mine/3ptl) | Crystal structure of proteinase K inhibited by a lactoferrin nonapeptide, Lys-Gly-Glu-Ala-Asp-Ala-Leu-Ser-Leu-Asp at 1.3 A resolution. | 分子名称: | 10-mer peptide from Lactoferrin, Proteinase K | 著者 | Shukla, P.K, Sinha, M, Kaur, P, Sharma, S, Singh, T.P. | 登録日 | 2010-12-03 | 公開日 | 2010-12-22 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Crystal structure of proteinase K inhibited by a lactoferrin nonapeptide, Lys-Gly-Glu-Ala-Asp-Ala-Leu-Ser-Leu-Asp at 1.3 A resolution. TO BE PUBLISHED
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3N8Z
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![BU of 3n8z by Molmil](/molmil-images/mine/3n8z) | Crystal Structure of Cyclooxygenase-1 in Complex with Flurbiprofen | 分子名称: | 2-acetamido-2-deoxy-alpha-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, FLURBIPROFEN, ... | 著者 | Sidhu, R.S. | 登録日 | 2010-05-28 | 公開日 | 2010-07-28 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Comparison of Cyclooxygenase-1 Crystal Structures: Cross-Talk between Monomers Comprising Cyclooxygenase-1 Homodimers Biochemistry, 49, 2010
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3N8Y
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![BU of 3n8y by Molmil](/molmil-images/mine/3n8y) | Structure of Aspirin Acetylated Cyclooxygenase-1 in Complex with Diclofenac | 分子名称: | 2-HYDROXYBENZOIC ACID, 2-[2,6-DICHLOROPHENYL)AMINO]BENZENEACETIC ACID, 2-acetamido-2-deoxy-alpha-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Sidhu, R.S. | 登録日 | 2010-05-28 | 公開日 | 2010-07-28 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Comparison of Cyclooxygenase-1 Crystal Structures: Cross-Talk between Monomers Comprising Cyclooxygenase-1 Homodimers Biochemistry, 49, 2010
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3N8X
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![BU of 3n8x by Molmil](/molmil-images/mine/3n8x) | Crystal Structure of Cyclooxygenase-1 in Complex with Nimesulide | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 4-NITRO-2-PHENOXYMETHANESULFONANILIDE, ... | 著者 | Lee, J.Y. | 登録日 | 2010-05-28 | 公開日 | 2010-07-28 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.75 Å) | 主引用文献 | Comparison of Cyclooxygenase-1 Crystal Structures: Cross-Talk between Monomers Comprising Cyclooxygenase-1 Homodimers Biochemistry, 49, 2010
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3N8W
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![BU of 3n8w by Molmil](/molmil-images/mine/3n8w) | |
3N8V
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![BU of 3n8v by Molmil](/molmil-images/mine/3n8v) | Crystal Structure of Unoccupied Cyclooxygenase-1 | 分子名称: | 2-acetamido-2-deoxy-alpha-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, GLYCEROL, ... | 著者 | Sidhu, R.S. | 登録日 | 2010-05-28 | 公開日 | 2010-07-28 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (3.05 Å) | 主引用文献 | Comparison of Cyclooxygenase-1 Crystal Structures: Cross-Talk between Monomers Comprising Cyclooxygenase-1 Homodimers Biochemistry, 49, 2010
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