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4K0W
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BU of 4k0w by Molmil
X-ray crystal structure of OXA-23 A220 duplication clinical variant
分子名称: 1,2-ETHANEDIOL, BICARBONATE ION, Beta-lactamase, ...
著者Kaitany, K.J, Klinger, N.V, Leonard, D.A, Powers, R.A.
登録日2013-04-04
公開日2013-08-07
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Structures of the Class D Carbapenemases OXA-23 and OXA-146: Mechanistic Basis of Activity against Carbapenems, Extended-Spectrum Cephalosporins, and Aztreonam.
Antimicrob.Agents Chemother., 57, 2013
4JWI
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BU of 4jwi by Molmil
Crystal structure of the substrate binding domain of E.coli DnaK in complex with sheep Bac7(35-43)
分子名称: Cathelicidin-3, Chaperone protein DnaK, SULFATE ION
著者Zahn, M, Straeter, N.
登録日2013-03-27
公開日2013-11-13
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural Identification of DnaK Binding Sites within Bovine and Sheep Bactenecin Bac7.
Protein Pept.Lett., 21, 2014
4JWE
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BU of 4jwe by Molmil
Crystal structure of the substrate binding domain of E.coli DnaK in complex with sheep Bac7(1-21)
分子名称: Cathelicidin-3, Chaperone protein DnaK, SULFATE ION
著者Zahn, M, Straeter, N.
登録日2013-03-27
公開日2013-11-13
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Structural Identification of DnaK Binding Sites within Bovine and Sheep Bactenecin Bac7.
Protein Pept.Lett., 21, 2014
4JF6
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BU of 4jf6 by Molmil
Structure of OXA-23 at pH 7.0
分子名称: Beta-lactamase, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ...
著者Smith, C.A, Vakulenko, S.B.
登録日2013-02-27
公開日2013-09-25
最終更新日2013-10-09
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural Basis for Carbapenemase Activity of the OXA-23 beta-Lactamase from Acinetobacter baumannii.
Chem.Biol., 20, 2013
4JF5
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BU of 4jf5 by Molmil
Structure of OXA-23 at pH 4.1
分子名称: 1,2-ETHANEDIOL, Beta-lactamase, CITRATE ANION
著者Smith, C.A, Vakulenko, S.B.
登録日2013-02-27
公開日2013-09-25
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献Structural Basis for Carbapenemase Activity of the OXA-23 beta-Lactamase from Acinetobacter baumannii.
Chem.Biol., 20, 2013
4JF4
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BU of 4jf4 by Molmil
OXA-23 meropenem complex
分子名称: (4R,5S)-3-{[(3S,5S)-5-(dimethylcarbamoyl)pyrrolidin-3-yl]sulfanyl}-5-[(2S,3R)-3-hydroxy-1-oxobutan-2-yl]-4-methyl-4,5-dihydro-1H-pyrrole-2-carboxylic acid, 1,2-ETHANEDIOL, Beta-lactamase
著者Smith, C.A, Vakulenko, S.B, Toth, M.
登録日2013-02-27
公開日2013-09-25
最終更新日2013-10-09
実験手法X-RAY DIFFRACTION (2.14 Å)
主引用文献Structural Basis for Carbapenemase Activity of the OXA-23 beta-Lactamase from Acinetobacter baumannii.
Chem.Biol., 20, 2013
4HNA
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BU of 4hna by Molmil
Kinesin motor domain in the ADP-MG-ALFX state in complex with tubulin and a DARPIN
分子名称: ADENOSINE-5'-DIPHOSPHATE, DESIGNED ANKYRIN REPEAT PROTEIN (DARPIN) D2, GUANOSINE-5'-DIPHOSPHATE, ...
著者Gigant, B, Knossow, M.
登録日2012-10-19
公開日2013-06-12
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (3.19 Å)
主引用文献Structure of a kinesin-tubulin complex and implications for kinesin motility.
Nat.Struct.Mol.Biol., 20, 2013
4GAB
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BU of 4gab by Molmil
Human AKR1B10 mutant V301L complexed with NADP+ and fidarestat
分子名称: (2S,4S)-2-AMINOFORMYL-6-FLUORO-SPIRO[CHROMAN-4,4'-IMIDAZOLIDINE]-2',5'-DIONE, Aldo-keto reductase family 1 member B10, CHLORIDE ION, ...
著者Cousido-Siah, A, Ruiz Figueras, F.X, Mitschler, A, Podjarny, A.
登録日2012-07-25
公開日2013-03-20
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.5971 Å)
主引用文献X-ray structure of the V301L aldo-keto reductase 1B10 complexed with NADP(+) and the potent aldose reductase inhibitor fidarestat: Implications for inhibitor binding and selectivity.
Chem.Biol.Interact, 202, 2013
4F6R
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BU of 4f6r by Molmil
Tubulin:Stathmin-like domain complex
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Designed ankyrin repeat protein (DARPIN) D2, GUANOSINE-5'-DIPHOSPHATE, ...
著者Gigant, B, Mignot, I, Knossow, M.
登録日2012-05-15
公開日2012-07-18
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.64 Å)
主引用文献Design and characterization of modular scaffolds for tubulin assembly.
J.Biol.Chem., 287, 2012
4F61
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BU of 4f61 by Molmil
Tubulin:Stathmin-like domain complex
分子名称: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
著者Gigant, B, Mignot, I, Knossow, M.
登録日2012-05-14
公開日2012-07-18
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (4.17 Å)
主引用文献Design and characterization of modular scaffolds for tubulin assembly.
J.Biol.Chem., 287, 2012
4EB6
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BU of 4eb6 by Molmil
Tubulin-Vinblastine: Stathmin-like complex
分子名称: (2ALPHA,2'BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLASTINE, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ...
著者Ranaivoson, F.M, Gigant, B, Knossow, M.
登録日2012-03-23
公開日2012-08-01
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.47 Å)
主引用文献Structural plasticity of tubulin assembly probed by vinca-domain ligands.
Acta Crystallogr.,Sect.D, 68, 2012
4DRX
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BU of 4drx by Molmil
GTP-Tubulin in complex with a DARPIN
分子名称: Designed ankyrin repeat protein (DARPIN) D1, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
著者Pecqueur, L, Gigant, B, Knossow, M.
登録日2012-02-17
公開日2012-07-11
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.22 Å)
主引用文献A designed ankyrin repeat protein selected to bind to tubulin caps the microtubule plus end.
Proc.Natl.Acad.Sci.USA, 109, 2012
4CK4
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BU of 4ck4 by Molmil
Ovine beta-Lactoglobulin at Atomic Resolution
分子名称: ACETATE ION, AMMONIUM ION, BETA_LACTOGLOBULIN-1/B, ...
著者Kontopidis, G, Nordle, A, Sawyer, L.
登録日2013-12-27
公開日2014-10-08
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.12 Å)
主引用文献Ovine Beta-Lactoglobulin at Atomic Resolution
Acta Crystallogr.,Sect.F, 70, 2014
3UT5
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BU of 3ut5 by Molmil
Tubulin-Colchicine-Ustiloxin: Stathmin-like domain complex
分子名称: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
著者Ranaivoson, F.M, Gigant, B, Knossow, M.
登録日2011-11-25
公開日2012-08-01
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.73 Å)
主引用文献Structural plasticity of tubulin assembly probed by vinca-domain ligands.
Acta Crystallogr.,Sect.D, 68, 2012
3RYI
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BU of 3ryi by Molmil
GDP-Tubulin: rb3 stathmin-like domain complex
分子名称: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
著者Nawrotek, A, Knossow, M, Gigant, B.
登録日2011-05-11
公開日2011-10-05
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The Determinants That Govern Microtubule Assembly from the Atomic Structure of GTP-Tubulin.
J.Mol.Biol., 412, 2011
3RYH
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BU of 3ryh by Molmil
GMPCPP-Tubulin: RB3 Stathmin-like domain complex
分子名称: GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID GUANYLATE ESTER, ...
著者Nawrotek, A, Knossow, M, Gigant, B.
登録日2011-05-11
公開日2011-10-05
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The Determinants That Govern Microtubule Assembly from the Atomic Structure of GTP-Tubulin.
J.Mol.Biol., 412, 2011
3RYF
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BU of 3ryf by Molmil
GTP-Tubulin: RB3 Stathmin-like domain complex
分子名称: GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, SULFATE ION, ...
著者Nawrotek, A, Knossow, M, Gigant, B.
登録日2011-05-11
公開日2011-10-05
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.52 Å)
主引用文献The Determinants That Govern Microtubule Assembly from the Atomic Structure of GTP-Tubulin.
J.Mol.Biol., 412, 2011
3RYC
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BU of 3ryc by Molmil
Tubulin: RB3 stathmin-like domain complex
分子名称: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
著者Nawrotek, A, Knossow, M, Gigant, B.
登録日2011-05-11
公開日2011-10-05
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The Determinants That Govern Microtubule Assembly from the Atomic Structure of GTP-Tubulin.
J.Mol.Biol., 412, 2011
3QE3
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BU of 3qe3 by Molmil
Sheep liver sorbitol dehydrogenase
分子名称: ACETIC ACID, GLYCEROL, Sorbitol dehydrogenase, ...
著者Yennawar, N.H, Yennawar, H.P.
登録日2011-01-19
公開日2011-04-27
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献X-ray crystal structure and small-angle X-ray scattering of sheep liver sorbitol dehydrogenase.
Acta Crystallogr.,Sect.D, 67, 2011
3PTL
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BU of 3ptl by Molmil
Crystal structure of proteinase K inhibited by a lactoferrin nonapeptide, Lys-Gly-Glu-Ala-Asp-Ala-Leu-Ser-Leu-Asp at 1.3 A resolution.
分子名称: 10-mer peptide from Lactoferrin, Proteinase K
著者Shukla, P.K, Sinha, M, Kaur, P, Sharma, S, Singh, T.P.
登録日2010-12-03
公開日2010-12-22
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Crystal structure of proteinase K inhibited by a lactoferrin nonapeptide, Lys-Gly-Glu-Ala-Asp-Ala-Leu-Ser-Leu-Asp at 1.3 A resolution.
TO BE PUBLISHED
3N8Z
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BU of 3n8z by Molmil
Crystal Structure of Cyclooxygenase-1 in Complex with Flurbiprofen
分子名称: 2-acetamido-2-deoxy-alpha-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, FLURBIPROFEN, ...
著者Sidhu, R.S.
登録日2010-05-28
公開日2010-07-28
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Comparison of Cyclooxygenase-1 Crystal Structures: Cross-Talk between Monomers Comprising Cyclooxygenase-1 Homodimers
Biochemistry, 49, 2010
3N8Y
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BU of 3n8y by Molmil
Structure of Aspirin Acetylated Cyclooxygenase-1 in Complex with Diclofenac
分子名称: 2-HYDROXYBENZOIC ACID, 2-[2,6-DICHLOROPHENYL)AMINO]BENZENEACETIC ACID, 2-acetamido-2-deoxy-alpha-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Sidhu, R.S.
登録日2010-05-28
公開日2010-07-28
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Comparison of Cyclooxygenase-1 Crystal Structures: Cross-Talk between Monomers Comprising Cyclooxygenase-1 Homodimers
Biochemistry, 49, 2010
3N8X
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Crystal Structure of Cyclooxygenase-1 in Complex with Nimesulide
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 4-NITRO-2-PHENOXYMETHANESULFONANILIDE, ...
著者Lee, J.Y.
登録日2010-05-28
公開日2010-07-28
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Comparison of Cyclooxygenase-1 Crystal Structures: Cross-Talk between Monomers Comprising Cyclooxygenase-1 Homodimers
Biochemistry, 49, 2010
3N8W
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Crystal Structure of R120Q/Native Cyclooxygenase-1 Heterodimer mutant in complex with Flurbiprofen
分子名称: 2-acetamido-2-deoxy-alpha-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, FLURBIPROFEN, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Sidhu, R.S.
登録日2010-05-28
公開日2010-07-28
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Comparison of Cyclooxygenase-1 Crystal Structures: Cross-Talk between Monomers Comprising Cyclooxygenase-1 Homodimers
Biochemistry, 49, 2010
3N8V
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BU of 3n8v by Molmil
Crystal Structure of Unoccupied Cyclooxygenase-1
分子名称: 2-acetamido-2-deoxy-alpha-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, GLYCEROL, ...
著者Sidhu, R.S.
登録日2010-05-28
公開日2010-07-28
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (3.05 Å)
主引用文献Comparison of Cyclooxygenase-1 Crystal Structures: Cross-Talk between Monomers Comprising Cyclooxygenase-1 Homodimers
Biochemistry, 49, 2010

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