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4Z71
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Crystal structure of inorganic pyrophosphatase from Mycobacterium tuberculosis in complex with Mg ions
分子名称: Inorganic pyrophosphatase, MAGNESIUM ION
著者Pratt, A.C, Biswas, T, Tsodikov, O.V.
登録日2015-04-06
公開日2015-08-26
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Structural and computational dissection of the catalytic mechanism of the inorganic pyrophosphatase from Mycobacterium tuberculosis.
J.Struct.Biol., 192, 2015
1MP5
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Y177F VARIANT OF S. ENTERICA RmlA
分子名称: URIDINE-5'-DIPHOSPHATE-GLUCOSE, Y177F VARIANT OF S. ENTERICA RmlA BOUND TO UDP-GLUCOSE
著者Barton, W.A, Biggins, J.B, Jiang, J, Thorson, J.S, Nikolov, D.B.
登録日2002-09-11
公開日2002-10-09
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Expanding pyrimidine diphosphosugar libraries via structure-based nucleotidylyltransferase engineering
Proc.Natl.Acad.Sci.USA, 99, 2002
4Z7C
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Diphosphomevalonate decarboxylase from the Sulfolobus solfataricus, space group h32
分子名称: Diphosphomevalonate decarboxylase, GLYCEROL, PHOSPHATE ION, ...
著者Unno, H, Hattori, A, Hemmi, H.
登録日2015-04-07
公開日2015-09-16
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献In Vivo Formation of the Protein Disulfide Bond That Enhances the Thermostability of Diphosphomevalonate Decarboxylase, an Intracellular Enzyme from the Hyperthermophilic Archaeon Sulfolobus solfataricus
J.Bacteriol., 197, 2015
1MQ5
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Crystal Structure of 3-chloro-N-[4-chloro-2-[[(4-chlorophenyl)amino]carbonyl]phenyl]-4-[(4-methyl-1-piperazinyl)methyl]-2-thiophenecarboxamide Complexed with Human Factor Xa
分子名称: 3-CHLORO-N-[4-CHLORO-2-[[(4-CHLOROPHENYL)AMINO]CARBONYL]PHENYL]-4-[(4-METHYL-1-PIPERAZINYL)METHYL]-2-THIOPHENECARBOXAMIDE, CALCIUM ION, COAGULATION FACTOR X HEAVY CHAIN, ...
著者Adler, M, Whitlow, M.
登録日2002-09-13
公開日2003-01-28
最終更新日2017-10-11
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystal Structures of Two Potent Nonamidine Inhibitors Bound to Factor Xa
Biochemistry, 41, 2002
4Z7J
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Structure of Acetobacter aceti PurE-S57A
分子名称: 1,2-ETHANEDIOL, 2-(2-METHOXYETHOXY)ETHANOL, 5-O-phosphono-beta-D-ribofuranose, ...
著者Kappock, T.J, Sullivan, K.L.
登録日2015-04-07
公開日2016-04-13
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.502 Å)
主引用文献Mutation of the conserved serine in two PurE classes
To Be Published
1MPQ
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MALTOPORIN TREHALOSE COMPLEX
分子名称: MALTOPORIN, alpha-D-glucopyranose-(1-1)-alpha-D-glucopyranose
著者Dutzler, R, Schirmer, T.
登録日1997-03-24
公開日1998-03-25
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Channel specificity: structural basis for sugar discrimination and differential flux rates in maltoporin.
J.Mol.Biol., 272, 1997
4Z7P
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BU of 4z7p by Molmil
X-ray structure of racemic ShK Q16K toxin
分子名称: Potassium channel toxin kappa-stichotoxin-She1a, SULFATE ION
著者Sickmier, E.A.
登録日2015-04-07
公開日2015-09-09
最終更新日2015-09-23
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Pharmaceutical Optimization of Peptide Toxins for Ion Channel Targets: Potent, Selective, and Long-Lived Antagonists of Kv1.3.
J.Med.Chem., 58, 2015
1MQJ
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Crystal structure of the GluR2 ligand binding core (S1S2J) in complex with willardiine at 1.65 angstroms resolution
分子名称: 2-AMINO-3-(2,4-DIOXO-3,4-DIHYDRO-2H-PYRIMIDIN-1-YL)-PROPIONIC ACID, ZINC ION, glutamate receptor 2
著者Jin, R, Banke, T.G, Mayer, M.L, Traynelis, S.F, Gouaux, E.
登録日2002-09-16
公開日2003-08-05
最終更新日2017-08-02
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Structural basis for partial agonist action at ionotropic glutamate receptors
Nat.Neurosci., 6, 2003
4Z7Q
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Integrin alphaIIbbeta3 in complex with AGDV-NH2 peptide
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Lin, F.-Y, Zhu, J, Springer, T.A.
登録日2015-04-07
公開日2015-12-16
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献beta-Subunit Binding Is Sufficient for Ligands to Open the Integrin alpha IIb beta 3 Headpiece.
J.Biol.Chem., 291, 2016
1MQ4
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Crystal Structure of Aurora-A Protein Kinase
分子名称: ADENOSINE-5'-DIPHOSPHATE, AURORA-RELATED KINASE 1, MAGNESIUM ION, ...
著者Nowakowski, J, Cronin, C.N, McRee, D.E, Knuth, M.W, Nelson, C, Pavletich, N.P, Rodgers, J, Sang, B.-C, Scheibe, D.N, Swanson, R.V, Thompson, D.A.
登録日2002-09-13
公開日2003-09-16
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structures of the Cancer-Related Aurora-A, FAK and EphA2 Protein Kinases from Nanovolume Crystallography
Structure, 10, 2002
4Z9N
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BU of 4z9n by Molmil
ABC transporter / periplasmic binding protein from Brucella ovis with glutathione bound
分子名称: 1,2-ETHANEDIOL, Amino acid ABC transporter, periplasmic amino acid-binding protein, ...
著者Seattle Structural Genomics Center for Infectious Disease (SSGCID)
登録日2015-04-10
公開日2015-06-17
実験手法X-RAY DIFFRACTION (1.745 Å)
主引用文献ABC transporter / periplasmic binding protein from Brucella ovis with glutathione bound
To Be Published
1M51
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BU of 1m51 by Molmil
PEPCK complex with a GTP-competitive inhibitor
分子名称: 1,2-ETHANEDIOL, ACETATE ION, MANGANESE (II) ION, ...
著者Foley, L.H, Wang, P, Dunten, P, Wertheimer, S.J.
登録日2002-07-06
公開日2003-09-30
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献X-ray Structures of two xanthine inhibitors bound to PEPCK and N-3 modifications of substituted 1,8-Dibenzylxanthines
Bioorg.Med.Chem.Lett., 13, 2003
4ZB3
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BU of 4zb3 by Molmil
Crystal structure of the apo AtNUDT7
分子名称: Nudix hydrolase 7, SULFATE ION
著者Tang, Q, Liu, C, Zhong, C, Ding, J.
登録日2015-04-14
公開日2015-09-09
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal Structures of Arabidopsis thaliana Nudix Hydrolase NUDT7 Reveal a Previously Unobserved Conformation.
Mol Plant, 8, 2015
1MQD
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X-ray structure of the GluR2 ligand-binding core (S1S2J) in complex with (S)-Des-Me-AMPA at 1.46 A resolution. Crystallization in the presence of lithium sulfate.
分子名称: (S)-2-AMINO-3-(3-HYDROXY-ISOXAZOL-4-YL)PROPIONIC ACID, GLYCEROL, Glutamate receptor subunit 2, ...
著者Kasper, C, Lunn, M.-L, Liljefors, T, Gouaux, E, Egebjerg, J, Kastrup, J.S.
登録日2002-09-16
公開日2003-07-01
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.46 Å)
主引用文献GluR2 ligand-binding core complexes: Importance of the isoxazolol moiety and 5-substituent for the binding mode of AMPA-type agonists.
FEBS Lett., 531, 2002
4ZBC
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BU of 4zbc by Molmil
A dehydrated form of glucose isomerase collected at 100K.
分子名称: MANGANESE (II) ION, Xylose isomerase, alpha-D-glucopyranose, ...
著者Sandy, J.
登録日2015-04-14
公開日2016-03-23
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A generic protocol for protein crystal dehydration using the HC1b humidity controller.
Acta Crystallogr D Struct Biol, 72, 2016
1M5D
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X-RAY STRUCTURE OF THE GLUR2 LIGAND BINDING CORE (S1S2J-Y702F) IN COMPLEX WITH Br-HIBO AT 1.73 A RESOLUTION
分子名称: (S)-2-AMINO-3-(4-BROMO-3-HYDROXY-ISOXAZOL-5-YL)PROPIONIC ACID, Glutamate receptor 2, SULFATE ION
著者Hogner, A, Kastrup, J.S, Jin, R, Liljefors, T, Mayer, M.L, Egebjerg, J, Larsen, I.K, Gouaux, E.
登録日2002-07-09
公開日2002-09-18
最終更新日2021-10-27
実験手法X-RAY DIFFRACTION (1.73 Å)
主引用文献Structural Basis for AMPA Receptor Activation and Ligand Selectivity: Crystal Structures of Five Agonist Complexes with the GluR2 Ligand-binding Core
J.Mol.Biol., 322, 2002
4ZBM
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BU of 4zbm by Molmil
Crystal structure of Drosophila cyclic nucleotide gated channel pore mimicking NaK mutant
分子名称: BARIUM ION, POTASSIUM ION, Potassium channel protein
著者Lam, Y, Zeng, W, Derebe, M.G, Jiang, Y.
登録日2015-04-14
公開日2015-07-29
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural implications of weak Ca2+ block in Drosophila cyclic nucleotide-gated channels.
J.Gen.Physiol., 146, 2015
1M5N
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Crystal structure of HEAT repeats (1-11) of importin b bound to the non-classical NLS(67-94) of PTHrP
分子名称: Importin beta-1 subunit, Parathyroid hormone-related protein
著者Cingolani, G, Bednenko, J, Gillespie, M.T, Gerace, L.
登録日2002-07-09
公開日2003-01-21
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Molecular basis for the recognition of a nonclassical nuclear localization signal by importin beta
Mol.Cell, 10, 2002
4ZBR
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Crystal Structure of Equine Serum Albumin in complex with Diclofenac and Naproxen
分子名称: (2S)-2-(6-methoxynaphthalen-2-yl)propanoic acid, (2S)-2-hydroxybutanedioic acid, 2-[2,6-DICHLOROPHENYL)AMINO]BENZENEACETIC ACID, ...
著者Sekula, B, Bujacz, A, Bujacz, G.
登録日2015-04-15
公開日2015-12-23
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.19 Å)
主引用文献Structural Insights into the Competitive Binding of Diclofenac and Naproxen by Equine Serum Albumin.
J.Med.Chem., 59, 2016
1LZJ
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Glycosyltransferase B + UDP + H antigen acceptor
分子名称: Glycosyltransferase B, MANGANESE (II) ION, MERCURY (II) ION, ...
著者Patenaude, S.I, Seto, N.O.L, Borisova, S.N, Szpacenko, A, Marcus, S.L, Palcic, M.M, Evans, S.V.
登録日2002-06-10
公開日2002-08-28
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.32 Å)
主引用文献The structural basis for specificity in human ABO(H) blood group biosynthesis.
Nat.Struct.Biol., 9, 2002
4ZCA
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Eg5 motor domain mutant Y231F
分子名称: ADENOSINE-5'-DIPHOSPHATE, Kinesin-like protein KIF11, MAGNESIUM ION
著者Luo, M, Parke, C, Worthylake, D.
登録日2015-04-15
公開日2016-06-22
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Eg5
To Be Published
1M5R
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Ternary complex of T4 phage BGT with UDP and a 13 mer DNA duplex
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 5'-D(*CP*TP*AP*TP*CP*TP*GP*AP*GP*TP*AP*TP*C)-3', ...
著者Lariviere, L, Morera, S.
登録日2002-07-10
公開日2002-12-11
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献A Base-flipping mechanism for the T4 phage beta-glucosyltransferase and identification of a transition state analog
J.Mol.Biol., 324, 2002
4ZCL
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Crystal Structure of Escherichia coli GTPase BipA/TypA Complexed with GDP
分子名称: COBALT HEXAMMINE(III), GTP-binding protein TypA/BipA, GUANOSINE-5'-DIPHOSPHATE, ...
著者Fan, H.T, Hahm, J, Diggs, S, Blaha, G.
登録日2015-04-16
公開日2015-07-29
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3.06 Å)
主引用文献Structural and Functional Analysis of BipA, a Regulator of Virulence in Enteropathogenic Escherichia coli.
J.Biol.Chem., 290, 2015
1M6A
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NMR structure of the i-Motif Tetramer Formed by XC2
分子名称: 5'-D(*CP*C)-3'
著者Malliavin, T.E, Snoussi, K, Leroy, J.-L.
登録日2002-07-15
公開日2002-08-07
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献The NMR structure of [Xd(C2)]4 investigated by molecular dynamics simulations
MAGN.RESON.CHEM., 41, 2003
4ZD6
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Halohydrin hydrogen-halide-lyase, HheB
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CHLORIDE ION, Halohydrin epoxidase B, ...
著者Watanabe, F, Yu, F, Ohtaki, A, Yamanaka, Y, Noguchi, K, Yohda, M, Odaka, M.
登録日2015-04-17
公開日2015-11-04
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Crystal structures of halohydrin hydrogen-halide-lyases from Corynebacterium sp. N-1074
Proteins, 83, 2015

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