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8ST0
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The 2alpha3beta stoichiometry of full-length human alpha4beta2 nicotinic acetylcholine receptor in complex with acetylcholine
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINE, IgG1 Heavy Chain, ...
著者Kang, G, Hibbs, R.E.
登録日2023-05-09
公開日2024-02-07
最終更新日2024-08-21
実験手法ELECTRON MICROSCOPY (2.4 Å)
主引用文献Structural bases for stoichiometry-selective calcium potentiation of a neuronal nicotinic receptor.
Br.J.Pharmacol., 181, 2024
8ST1
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The 3alpha2beta stoichiometry of human alpha4beta2 nicotinic acetylcholine receptor in complex with acetylcholine and calcium
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINE, CALCIUM ION, ...
著者Kang, G, Hibbs, R.E.
登録日2023-05-09
公開日2024-02-07
最終更新日2024-08-21
実験手法ELECTRON MICROSCOPY (3.41 Å)
主引用文献Structural bases for stoichiometry-selective calcium potentiation of a neuronal nicotinic receptor.
Br.J.Pharmacol., 181, 2024
8ST2
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The 3alpha2beta stoichiometry of human alpha4beta2 nicotinic acetylcholine receptor in complex with acetylcholine
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINE, IgG1 Heavy Chain, ...
著者Kang, G, Hibbs, R.E.
登録日2023-05-09
公開日2024-02-07
最終更新日2024-08-21
実験手法ELECTRON MICROSCOPY (2.94 Å)
主引用文献Structural bases for stoichiometry-selective calcium potentiation of a neuronal nicotinic receptor.
Br.J.Pharmacol., 181, 2024
6YBZ
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Crystal structure of the D116N mutant of the light-driven sodium pump KR2 in the pentameric form, pH 8.0
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, EICOSANE, RETINAL, ...
著者Kovalev, K, Gushchin, I, Gordeliy, V.
登録日2020-03-18
公開日2020-04-08
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Molecular mechanism of light-driven sodium pumping.
Nat Commun, 11, 2020
8ST4
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The 2alpha3beta stoichiometry of human alpha4beta2 nicotinic acetylcholine receptor in complex with acetylcholine
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, ACETYLCHOLINE, IgG1 Heavy Chain, ...
著者Kang, G, Hibbs, R.E.
登録日2023-05-09
公開日2024-02-07
最終更新日2024-08-21
実験手法ELECTRON MICROSCOPY (2.35 Å)
主引用文献Structural bases for stoichiometry-selective calcium potentiation of a neuronal nicotinic receptor.
Br.J.Pharmacol., 181, 2024
6YEN
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Crystal structure of AmpC from E. coli with Taniborbactam (VNRX-5133)
分子名称: (10aR)-2-(((1r,4R)-4-((2-aminoethyl)amino)cyclohexyl)methyl)-6-carboxy-4-hydroxy-4,10a-dihydro-10H-benzo[5,6][1,2]oxaborinino[2,3-b][1,4,2]oxazaborol-4-uide, (3~{R})-3-[2-[4-(2-azanylethylamino)cyclohexyl]ethanoylamino]-2-oxidanyl-3,4-dihydro-1,2-benzoxaborinine-8-carboxylic acid, 1,2-ETHANEDIOL, ...
著者Lang, P.A, Brem, J, Schofield, C.J.
登録日2020-03-25
公開日2020-06-24
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.418 Å)
主引用文献Bicyclic Boronates as Potent Inhibitors of AmpC, the Class C beta-Lactamase from Escherichia coli .
Biomolecules, 10, 2020
8F1Z
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EGFR kinase in complex with Bayer #33
分子名称: (2P)-3-(3-chloro-2-methoxyanilino)-2-[3-(2-methoxy-2-methylpropoxy)pyridin-4-yl]-1,5,6,7-tetrahydro-4H-pyrrolo[3,2-c]pyridin-4-one, CITRIC ACID, Epidermal growth factor receptor
著者Beyett, T.S, Eck, M.J.
登録日2022-11-06
公開日2023-11-08
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献EGFR kinase in complex with Bayer #33
To be published
5I79
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Crystal structure of a beta-1,4-endoglucanase mutant from Aspergillus niger in complex with sugar
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, Endo-beta-1, ...
著者Liu, W.D, Yan, J.J, Li, Y.J, Zheng, Y.Y, Chen, C.C, Guo, R.T.
登録日2016-02-17
公開日2016-12-21
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Functional and structural analysis of Pichia pastoris-expressed Aspergillus niger 1,4-beta-endoglucanase
Biochem. Biophys. Res. Commun., 475, 2016
8SDF
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BU of 8sdf by Molmil
Crystal structure of SARS-CoV-2 receptor binding domain in complex with neutralizing antibody CC25.4
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Yuan, M, Wilson, I.A.
登録日2023-04-06
公開日2024-03-13
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (1.79 Å)
主引用文献Broadly neutralizing antibodies targeting a conserved silent face of spike RBD resist extreme SARS-CoV-2 antigenic drift.
Biorxiv, 2023
8F1Y
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BU of 8f1y by Molmil
EGFR kinase in complex with poziotinib
分子名称: 1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-one, CITRIC ACID, Epidermal growth factor receptor
著者Beyett, T.S, Eck, M.J.
登録日2022-11-06
公開日2023-11-08
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献EGFR kinase in complex with poziotinib
To be published
8SJK
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BU of 8sjk by Molmil
Pembrolizumab Caffeine crystal
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ANTIBODY HEAVY CHAIN, ANTIBODY LIGHT CHAIN, ...
著者Larpent, P, Codan, L, Bothe, J.R, Stueber, D, Reichert, P, Fischmann, T, Su, Y, Pabit, S, Gupta, S, Iuzzolino, L, Cote, A.
登録日2023-04-18
公開日2024-04-24
最終更新日2024-08-21
実験手法X-RAY DIFFRACTION (2.22 Å)
主引用文献Small-Angle X-ray Scattering as a Powerful Tool for Phase and Crystallinity Assessment of Monoclonal Antibody Crystallites in Support of Batch Crystallization.
Mol Pharm., 21, 2024
8SGM
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BU of 8sgm by Molmil
Crystal Structure of CD1d-lipid complexed with Beta-2-Microglobulin, TCR Alpha-Chain and TCR Beta-Chain
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Antigen-presenting glycoprotein CD1d, ...
著者Chan Yew Poa, K.T.O, Le Nours, J, Rossjohn, J.
登録日2023-04-12
公開日2024-04-24
実験手法X-RAY DIFFRACTION (2.50000215 Å)
主引用文献Semi-invariant human type II Natural Killer T cells recognise CD1d independently of bound lipids.
To Be Published
5BO8
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BU of 5bo8 by Molmil
Structure of human sialyltransferase ST8SiaIII
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CITRIC ACID, ...
著者Volkers, G, Worrall, L, Strynadka, N.C.J.
登録日2015-05-27
公開日2015-07-15
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structure of human ST8SiaIII sialyltransferase provides insight into cell-surface polysialylation.
Nat.Struct.Mol.Biol., 22, 2015
8SGB
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BU of 8sgb by Molmil
Crystal Structure of CD1d-lipid complexed with Beta-2-Microglobulin, TCR Alpha-Chain and TCR Beta-Chain
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Antigen-presenting glycoprotein CD1d, Beta-2-microglobulin, ...
著者Chan Yew Poa, K.T.O, Le Nours, J, Rossjohn, J.
登録日2023-04-12
公開日2024-04-24
実験手法X-RAY DIFFRACTION (2.80001545 Å)
主引用文献Semi-invariant human type II Natural Killer T cells recognise CD1d independently of bound lipids.
To Be Published
1BDG
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BU of 1bdg by Molmil
HEXOKINASE FROM SCHISTOSOMA MANSONI COMPLEXED WITH GLUCOSE
分子名称: HEXOKINASE, SULFATE ION, alpha-D-glucopyranose
著者Mulichak, A.M, Garavito, R.M.
登録日1998-05-08
公開日1999-05-11
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献The structure of mammalian hexokinase-1.
Nat.Struct.Biol., 5, 1998
7KQH
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BU of 7kqh by Molmil
Antibodies that engage the hemagglutinin receptor-binding site of influenza B viruses
分子名称: 2365 Fab heavy chain, 2365 Fab light chain, Hemagglutinin, ...
著者Bajic, G, Harrison, S.C.
登録日2020-11-16
公開日2020-12-16
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (3.5 Å)
主引用文献Antibodies That Engage the Hemagglutinin Receptor-Binding Site of Influenza B Viruses.
Acs Infect Dis., 7, 2021
8CWH
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BU of 8cwh by Molmil
200us Temperature-Jump (Dark2) XFEL structure of Lysozyme Bound to N,N'-diacetylchitobiose
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-alpha-D-glucopyranose, CHLORIDE ION, Lysozyme C, ...
著者Wolff, A.M, Thompson, M.C, Fraser, J.S, Nango, E.
登録日2022-05-19
公開日2022-06-22
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Mapping protein dynamics at high spatial resolution with temperature-jump X-ray crystallography.
Nat.Chem., 15, 2023
7KZB
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Potent SARS-CoV-2 binding and neutralization through maturation of iconic SARS-CoV-1antibodies
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, Fab heavy chain of CR3014-C8 antibody, ...
著者Langley, D.B, Christ, D.
登録日2020-12-10
公開日2021-02-03
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.83 Å)
主引用文献Potent SARS-CoV-2 binding and neutralization through maturation of iconic SARS-CoV-1 antibodies.
Mabs, 13
8CWG
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BU of 8cwg by Molmil
200us Temperature-Jump (Dark1) XFEL structure of Lysozyme Bound to N,N'-diacetylchitobiose
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-alpha-D-glucopyranose, CHLORIDE ION, Lysozyme C, ...
著者Wolff, A.M, Thompson, M.C, Fraser, J.S, Nango, E.
登録日2022-05-19
公開日2022-06-22
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Mapping protein dynamics at high spatial resolution with temperature-jump X-ray crystallography.
Nat.Chem., 15, 2023
8CWB
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BU of 8cwb by Molmil
Laser Off Temperature-Jump XFEL structure of Lysozyme Bound to N,N'-diacetylchitobiose
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-alpha-D-glucopyranose, CHLORIDE ION, Lysozyme C, ...
著者Wolff, A.M, Thompson, M.C, Fraser, J.S, Nango, E.
登録日2022-05-19
公開日2022-06-22
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.51 Å)
主引用文献Mapping protein dynamics at high spatial resolution with temperature-jump X-ray crystallography.
Nat.Chem., 15, 2023
8SIQ
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BU of 8siq by Molmil
Crystal structure of SARS-CoV-2 spike receptor-binding domain in complex with broadly neutralizing antibodies CC25.36 and CV38-142 Fab
分子名称: CC25.36 Fab heavy chain, CC25.36 Fab light chain, CV38-142 Fab heavy chain, ...
著者Liu, H, Wilson, I.A.
登録日2023-04-16
公開日2024-03-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Broadly neutralizing antibodies targeting a conserved silent face of spike RBD resist extreme SARS-CoV-2 antigenic drift
Biorxiv, 2023
1ARP
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BU of 1arp by Molmil
Crystal structure of the fungal peroxidase from Arthromyces ramosus at 1.9 angstroms resolution: structural comparisons with the lignin and cytochrome C peroxidases
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, PEROXIDASE, ...
著者Kunishima, N, Fukuyama, K.
登録日1993-06-18
公開日1994-01-31
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structure of the fungal peroxidase from Arthromyces ramosus at 1.9 A resolution. Structural comparisons with the lignin and cytochrome c peroxidases.
J.Mol.Biol., 235, 1994
8CWE
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BU of 8cwe by Molmil
20ns Temperature-Jump (Dark2) XFEL structure of Lysozyme Bound to N,N'-diacetylchitobiose
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-alpha-D-glucopyranose, CHLORIDE ION, Lysozyme C, ...
著者Wolff, A.M, Thompson, M.C, Fraser, J.S, Nango, E.
登録日2022-05-19
公開日2022-06-22
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.48 Å)
主引用文献Mapping protein dynamics at high spatial resolution with temperature-jump X-ray crystallography.
Nat.Chem., 15, 2023
8CWD
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BU of 8cwd by Molmil
20ns Temperature-Jump (Dark1) XFEL structure of Lysozyme Bound to N,N'-diacetylchitobiose
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-alpha-D-glucopyranose, CHLORIDE ION, Lysozyme C, ...
著者Wolff, A.M, Thompson, M.C, Fraser, J.S, Nango, E.
登録日2022-05-19
公開日2022-06-22
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.48 Å)
主引用文献Mapping protein dynamics at high spatial resolution with temperature-jump X-ray crystallography.
Nat.Chem., 15, 2023
8SGN
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BU of 8sgn by Molmil
Crystal structure of Epstein-Barr virus glycoprotein 350 (gp350) in complex with Cy651H02, a monoclonal antibody isolated from macaques immunized with a gp350 nanoparticle vaccine
分子名称: 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Joyce, M.G, Jensen, J.L, Chen, W.H, Kanekiyo, M.
登録日2023-04-12
公開日2024-04-17
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal structure of Epstein-Barr virus glycoprotein 350 (gp350) in complex with Cy651H02, a monoclonal antibody isolated from macaques immunized with a gp350 nanoparticle vaccine
To Be Published

224004

件を2024-08-21に公開中

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