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1SC7
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Human DNA Topoisomerase I (70 Kda) In Complex With The Indenoisoquinoline MJ-II-38 and Covalent Complex With A 22 Base Pair DNA Duplex
分子名称: 4-(5,11-DIOXO-5H-INDENO[1,2-C]ISOQUINOLIN-6(11H)-YL)BUTANOATE, 5'-D(*(TGP)P*GP*AP*AP*AP*AP*AP*TP*TP*TP*TP*T)-3', 5'-D(*AP*AP*AP*AP*AP*GP*AP*CP*TP*T)-3', ...
著者Staker, B.L, Feese, M.D, Cushman, M, Pommier, Y, Zembower, D, Stewart, L, Burgin, A.B.
登録日2004-02-11
公開日2005-04-19
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structures of three classes of anticancer agents bound to the human topoisomerase I-DNA covalent complex
J.Med.Chem., 48, 2005
1SC8
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Urokinase Plasminogen Activator B-Chain-J435 Complex
分子名称: N-(BENZYLSULFONYL)SERYL-N~1~-{4-[AMINO(IMINO)METHYL]BENZYL}GLYCINAMIDE, SULFATE ION, plasminogen activator, ...
著者Schweinitz, A, Steinmetzer, T, Banke, I.J, Arlt, M.J.E, Stuerzebecher, A, Schuster, O, Geissler, A, Giersiefen, H, Zeslawska, E, Jacob, U, Kruger, A, Stuerzebecher, J.
登録日2004-02-12
公開日2004-06-22
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Design of novel and selective inhibitors of urokinase-type plasminogen activator with improved pharmacokinetic properties for use as antimetastatic agents
J.Biol.Chem., 279, 2004
1SC9
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Hydroxynitrile Lyase from Hevea brasiliensis in complex with the natural substrate acetone cyanohydrin
分子名称: (S)-acetone-cyanohydrin lyase, 2-HYDROXY-2-METHYLPROPANENITRILE, SULFATE ION
著者Gruber, K, Gartler, G, Krammer, B, Schwab, H, Kratky, C.
登録日2004-02-12
公開日2004-06-29
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Reaction mechanism of hydroxynitrile lyases of the alpha/beta-hydrolase superfamily: the three-dimensional structure of the transient enzyme-substrate complex certifies the crucial role of LYS236
J.Biol.Chem., 279, 2004
1SCA
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ENZYME CRYSTAL STRUCTURE IN A NEAT ORGANIC SOLVENT
分子名称: CALCIUM ION, SODIUM ION, SUBTILISIN CARLSBERG
著者Fitzpatrick, P.A, Steinmetz, A.C.U, Ringe, D, Klibanov, A.M.
登録日1993-07-19
公開日1994-01-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Enzyme crystal structure in a neat organic solvent.
Proc.Natl.Acad.Sci.USA, 90, 1993
1SCB
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ENZYME CRYSTAL STRUCTURE IN A NEAT ORGANIC SOLVENT
分子名称: ACETONITRILE, CALCIUM ION, SUBTILISIN CARLSBERG
著者Fitzpatrick, P.A, Steinmetz, A.C.U, Ringe, D, Klibanov, A.M.
登録日1993-07-13
公開日1994-01-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Enzyme crystal structure in a neat organic solvent.
Proc.Natl.Acad.Sci.USA, 90, 1993
1SCD
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X-RAY CRYSTAL STRUCTURE OF CROSS-LINKED SUBTILISM CARLSBERG IN WATER VS. ACETONITRILE
分子名称: CALCIUM ION, SUBTILISIN CARLSBERG
著者Fitzpatrick, P.A, Ringe, D, Klibanov, A.M.
登録日1993-08-23
公開日1994-01-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献X-ray crystal structure of cross-linked subtilisin Carlsberg in water vs. acetonitrile.
Biochem.Biophys.Res.Commun., 198, 1994
1SCE
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CRYSTAL STRUCTURE OF THE CELL CYCLE REGULATORY PROTEIN SUC1 REVEALS A NOVEL BETA-HINGE CONFORMATIONAL SWITCH
分子名称: CHLORIDE ION, SUC1
著者Bourne, Y, Tainer, J.A.
登録日1995-05-11
公開日1996-01-29
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal structure of the cell cycle-regulatory protein suc1 reveals a beta-hinge conformational switch.
Proc.Natl.Acad.Sci.USA, 92, 1995
1SCF
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BU of 1scf by Molmil
HUMAN RECOMBINANT STEM CELL FACTOR
分子名称: CALCIUM ION, PENTAETHYLENE GLYCOL, STEM CELL FACTOR
著者Jiang, X, Gurel, O, Langley, K.E, Hendrickson, W.A.
登録日1998-06-04
公開日2000-07-07
最終更新日2022-12-21
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure of the active core of human stem cell factor and analysis of binding to its receptor kit.
EMBO J., 19, 2000
1SCH
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BU of 1sch by Molmil
PEANUT PEROXIDASE
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, PEANUT PEROXIDASE, ...
著者Schuller, D.J, Poulos, T.L.
登録日1996-01-23
公開日1996-07-11
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.56 Å)
主引用文献The crystal structure of peanut peroxidase.
Structure, 4, 1996
1SCI
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BU of 1sci by Molmil
K236L mutant of hydroxynitrile lyase from Hevea brasiliensis
分子名称: (S)-acetone-cyanohydrin lyase, SULFATE ION
著者Gruber, K, Gartler, G, Krammer, B, Schwab, H, Kratky, C.
登録日2004-02-12
公開日2004-06-29
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献Reaction mechanism of hydroxynitrile lyases of the alpha/beta-hydrolase superfamily: the three-dimensional structure of the transient enzyme-substrate complex certifies the crucial role of LYS236
J.Biol.Chem., 279, 2004
1SCJ
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CRYSTAL STRUCTURE OF SUBTILISIN-PROPEPTIDE COMPLEX
分子名称: CALCIUM ION, SUBTILISIN E
著者Berman, H.M, Jain, S.C.
登録日1998-04-29
公開日1998-12-09
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The crystal structure of an autoprocessed Ser221Cys-subtilisin E-propeptide complex at 2.0 A resolution.
J.Mol.Biol., 284, 1998
1SCK
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BU of 1sck by Molmil
K236L mutant of hydroxynitrile lyase from Hevea brasiliensis in complex with acetone
分子名称: (S)-acetone-cyanohydrin lyase, ACETONE, SULFATE ION
著者Gruber, K, Gartler, G, Krammer, B, Schwab, H, Kratky, C.
登録日2004-02-12
公開日2004-06-29
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Reaction mechanism of hydroxynitrile lyases of the alpha/beta-hydrolase superfamily: the three-dimensional structure of the transient enzyme-substrate complex certifies the crucial role of LYS236
J.Biol.Chem., 279, 2004
1SCL
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BU of 1scl by Molmil
THE SARCIN-RICIN LOOP, A MODULAR RNA
分子名称: RNA SARCIN-RICIN LOOP
著者Szewczak, A.A, Moore, P.B.
登録日1994-11-11
公開日1995-01-26
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献The conformation of the sarcin/ricin loop from 28S ribosomal RNA.
Proc.Natl.Acad.Sci.USA, 90, 1993
1SCM
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BU of 1scm by Molmil
STRUCTURE OF THE REGULATORY DOMAIN OF SCALLOP MYOSIN AT 2.8 ANGSTROMS RESOLUTION
分子名称: CALCIUM ION, MYOSIN ESSENTIAL LIGHT CHAIN, MYOSIN HEAVY CHAIN, ...
著者Cohen, C, Xie, X.
登録日1994-01-06
公開日1994-04-30
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure of the regulatory domain of scallop myosin at 2.8 A resolution.
Nature, 368, 1994
1SCN
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BU of 1scn by Molmil
INACTIVATION OF SUBTILISIN CARLSBERG BY N-(TERT-BUTOXYCARBONYL-ALANYL-PROLYL-PHENYLALANYL)-O-BENZOL HYDROXYLAMINE: FORMATION OF COVALENT ENZYME-INHIBITOR LINKAGE IN THE FORM OF A CARBAMATE DERIVATIVE
分子名称: CALCIUM ION, N-(tert-butoxycarbonyl)-L-alanyl-N-[(1R)-1-(carboxyamino)-2-phenylethyl]-L-prolinamide, SODIUM ION, ...
著者Steinmetz, A.C.U, Demuth, H.-U, Ringe, D.
登録日1994-03-02
公開日1994-08-31
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Inactivation of subtilisin Carlsberg by N-((tert-butoxycarbonyl)alanylprolylphenylalanyl)-O-benzolhydroxyl- amine: formation of a covalent enzyme-inhibitor linkage in the form of a carbamate derivative.
Biochemistry, 33, 1994
1SCO
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BU of 1sco by Molmil
SCORPION TOXIN (OSK1 TOXIN) WITH HIGH AFFINITY FOR SMALL CONDUCTANCE CA(2+)-ACTIVATED K+ CHANNEL IN NEUROBLASTOMA-X-GLUOMA NG 108-15 HYBRID CELLS, NMR, 30 STRUCTURES
分子名称: SCORPION TOXIN OSK1
著者Jaravine, V.A, Nolde, D.E, Pluzhnikov, K.A, Grishin, E.V, Arseniev, A.S.
登録日1996-04-01
公開日1997-01-27
最終更新日2017-11-29
実験手法SOLUTION NMR
主引用文献Three-dimensional structure of toxin OSK1 from Orthochirus scrobiculosus scorpion venom.
Biochemistry, 36, 1997
1SCQ
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BU of 1scq by Molmil
K236L mutant of hydroxynitrile lyase from Hevea brasiliensis in complex with acetonecyanohydrin
分子名称: (S)-acetone-cyanohydrin lyase, 2-HYDROXY-2-METHYLPROPANENITRILE, SULFATE ION
著者Gruber, K, Gartler, G, Krammer, B, Schwab, H, Kratky, C.
登録日2004-02-12
公開日2004-06-29
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Reaction mechanism of hydroxynitrile lyases of the alpha/beta-hydrolase superfamily: the three-dimensional structure of the transient enzyme-substrate complex certifies the crucial role of LYS236
J.Biol.Chem., 279, 2004
1SCR
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BU of 1scr by Molmil
HIGH-RESOLUTION STRUCTURES OF SINGLE-METAL-SUBSTITUTED CONCANAVALIN A: THE CO,CA-PROTEIN AT 1.6 ANGSTROMS AND THE NI,CA-PROTEIN AT 2.0 ANGSTROMS
分子名称: CALCIUM ION, CONCANAVALIN A, NICKEL (II) ION
著者Emmerich, C, Helliwell, J.R, Redshaw, M, Naismith, J.H, Harrop, S.J, Raftery, J, Kalb, A.J, Yariv, J, Dauter, Z, Wilson, K.S.
登録日1993-12-06
公開日1994-05-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献High-resolution structures of single-metal-substituted concanavalin A: the Co,Ca-protein at 1.6 A and the Ni,Ca-protein at 2.0 A.
Acta Crystallogr.,Sect.D, 50, 1994
1SCS
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BU of 1scs by Molmil
HIGH-RESOLUTION STRUCTURES OF SINGLE-METAL-SUBSTITUTED CONCANAVALIN A: THE CO,CA-PROTEIN AT 1.6 ANGSTROMS AND THE NI,CA-PROTEIN AT 2.0 ANGSTROMS
分子名称: CALCIUM ION, COBALT (II) ION, CONCANAVALIN A
著者Emmerich, C, Helliwell, J.R, Redshaw, M, Naismith, J.H, Harrop, S.J, Raftery, J, Kalb, A.J, Yariv, J, Dauter, Z, Wilson, K.S.
登録日1993-12-06
公開日1994-05-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献High-resolution structures of single-metal-substituted concanavalin A: the Co,Ca-protein at 1.6 A and the Ni,Ca-protein at 2.0 A.
Acta Crystallogr.,Sect.D, 50, 1994
1SCU
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BU of 1scu by Molmil
THE CRYSTAL STRUCTURE OF SUCCINYL-COA SYNTHETASE FROM ESCHERICHIA COLI AT 2.5 ANGSTROMS RESOLUTION
分子名称: COENZYME A, SUCCINYL-COA SYNTHETASE, ALPHA SUBUNIT, ...
著者Wolodko, W.T, Fraser, M.E, James, M.N.G, Bridger, W.A.
登録日1993-11-18
公開日1995-04-20
最終更新日2019-08-14
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The crystal structure of succinyl-CoA synthetase from Escherichia coli at 2.5-A resolution.
J.Biol.Chem., 269, 1994
1SCV
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BU of 1scv by Molmil
NMR STRUCTURE OF THE C TERMINAL DOMAIN OF CARDIAC TROPONIN C BOUND TO THE N TERMINAL DOMAIN OF CARDIAC TROPONIN I
分子名称: CALCIUM ION, Troponin C, slow skeletal and cardiac muscles
著者Finley, N.L, Howarth, J.W, Rosevear, P.R.
登録日2004-02-12
公開日2004-11-23
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Structure of the Mg2+-loaded C-lobe of cardiac troponin C bound to the N-domain of cardiac troponin I: comparison with the Ca2+-loaded structure.
Biochemistry, 43, 2004
1SCW
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BU of 1scw by Molmil
TOWARD BETTER ANTIBIOTICS: CRYSTAL STRUCTURE OF R61 DD-PEPTIDASE INHIBITED BY A NOVEL MONOCYCLIC PHOSPHATE INHIBITOR
分子名称: (2Z)-3-{[OXIDO(OXO)PHOSPHINO]OXY}-2-PHENYLACRYLATE, D-alanyl-D-alanine carboxypeptidase, GLYCEROL
著者Silvaggi, N.R, Kaur, K, Adediran, S.A, Pratt, R.F, Kelly, J.A.
登録日2004-02-12
公開日2004-06-22
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.13 Å)
主引用文献Toward Better Antibiotics: Crystallographic Studies of a Novel Class of DD-Peptidase/beta-Lactamase Inhibitors.
Biochemistry, 43, 2004
1SCY
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DETERMINATION OF THE THREE-DIMENSIONAL STRUCTURE OF SCYLLATOXIN BY 1H NUCLEAR MAGNETIC RESONANCE
分子名称: SCYLLATOXIN
著者Martins, J.C, Van De Ven, F.J.M, Borremans, F.A.M.
登録日1994-06-02
公開日1995-01-26
最終更新日2017-11-29
実験手法SOLUTION NMR
主引用文献Determination of the three-dimensional solution structure of scyllatoxin by 1H nuclear magnetic resonance.
J.Mol.Biol., 253, 1995
1SCZ
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Improved structural model for the catalytic domain of E.coli dihydrolipoamide succinyltransferase
分子名称: Dihydrolipoamide Succinyltransferase
著者Schormann, N, Symersky, J, Carson, M, Luo, M, Tsao, J, Johnson, D, Huang, W.-Y, Pruett, P, Lin, G, Li, S, Qiu, S, Arabashi, A, Bunzel, B, Luo, D, Nagy, L, Gray, R, Luan, C.-H, Zhang, Z, Lu, S, DeLucas, L.
登録日2004-02-12
公開日2004-03-02
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Improved structural model for the catalytic domain of E.coli dihydrolipoamide succinyltransferase
To be Published
1SD0
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Structure of arginine kinase C271A mutant
分子名称: ADENOSINE-5'-DIPHOSPHATE, ARGININE, Arginine kinase, ...
著者Gattis, J.L, Ruben, E, Fenley, M.O, Ellington, W.R, Chapman, M.S.
登録日2004-02-12
公開日2004-07-27
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献The active site cysteine of arginine kinase: structural and functional analysis of partially active mutants
Biochemistry, 43, 2004

224004

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