8DYV
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![BU of 8dyv by Molmil](/molmil-images/mine/8dyv) | Structure of human cytoplasmic dynein-1 bound to one Lis1 | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, Cytoplasmic dynein 1 heavy chain 1, ... | 著者 | Reimer, J.M, DeSantis, M, Reck-Peterson, S.L, Leschziner, A.E. | 登録日 | 2022-08-05 | 公開日 | 2023-02-01 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.97 Å) | 主引用文献 | Structures of human dynein in complex with the lissencephaly 1 protein, LIS1. Elife, 12, 2023
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4RDK
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![BU of 4rdk by Molmil](/molmil-images/mine/4rdk) | Crystal structure of Norovirus Boxer P domain in complex with Lewis b tetrasaccharide | 分子名称: | Capsid, alpha-L-fucopyranose-(1-2)-beta-D-galactopyranose-(1-3)-[alpha-L-fucopyranose-(1-4)]2-acetamido-2-deoxy-alpha-D-glucopyranose | 著者 | Hao, N, Chen, Y, Xia, M, Liu, W, Tan, M, Jiang, X, Li, X. | 登録日 | 2014-09-19 | 公開日 | 2015-01-14 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.629 Å) | 主引用文献 | Crystal structures of GI.8 Boxer virus P dimers in complex with HBGAs, a novel evolutionary path selected by the Lewis epitope. Protein Cell, 6, 2015
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3NJ4
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![BU of 3nj4 by Molmil](/molmil-images/mine/3nj4) | Fluoro-neplanocin A in Human S-Adenosylhomocysteine Hydrolase | 分子名称: | (4S,5S)-4-(6-amino-9H-purin-9-yl)-3-fluoro-5-hydroxy-2-(hydroxymethyl)cyclopent-2-en-1-one, Adenosylhomocysteinase, NICOTINAMIDE-ADENINE-DINUCLEOTIDE | 著者 | Jeong, L.S, Lee, K.M, Hwang, K.Y, Choi, S, Heo, Y.S. | 登録日 | 2010-06-17 | 公開日 | 2011-05-04 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | X-ray crystal structure and binding mode analysis of human S-adenosylhomocysteine hydrolase complexed with novel mechanism-based inhibitors, haloneplanocin A analogues. J.Med.Chem., 54, 2011
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6PQZ
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8DYU
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![BU of 8dyu by Molmil](/molmil-images/mine/8dyu) | Structure of human cytoplasmic dynein-1 bound to two Lis1 proteins | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, Cytoplasmic dynein 1 heavy chain 1, ... | 著者 | Reimer, J.M, DeSantis, M, Reck-Peterson, S.L, Leschziner, A.E. | 登録日 | 2022-08-05 | 公開日 | 2023-02-01 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (4 Å) | 主引用文献 | Structures of human dynein in complex with the lissencephaly 1 protein, LIS1. Elife, 12, 2023
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8AY2
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6P5Z
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5NBJ
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![BU of 5nbj by Molmil](/molmil-images/mine/5nbj) | DLS Tetragonal - ReHEWL | 分子名称: | CHLORIDE ION, Lysozyme C, RHENIUM, ... | 著者 | Brink, A, Helliwell, J.R. | 登録日 | 2017-03-02 | 公開日 | 2017-05-10 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.266 Å) | 主引用文献 | New leads for fragment-based design of rhenium/technetium radiopharmaceutical agents. IUCrJ, 4, 2017
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3NAG
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![BU of 3nag by Molmil](/molmil-images/mine/3nag) | Crystal structure of the phosphoribosylpyrophosphate (PRPP) synthetase from Thermoplasma Volcanium in complex with ADP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Ribose-phosphate pyrophosphokinase, ... | 著者 | Cherney, M.M, Cherney, L.T, Garen, C.R, James, M.N.G. | 登録日 | 2010-06-02 | 公開日 | 2011-06-08 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | The structures of Thermoplasma volcanium phosphoribosyl pyrophosphate synthetase bound to ribose-5-phosphate and ATP analogs. J.Mol.Biol., 413, 2011
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8AFY
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![BU of 8afy by Molmil](/molmil-images/mine/8afy) | Subtomogram average of membrane-bound Atg18 oligomers | 分子名称: | Autophagy-related protein 18 | 著者 | Mann, D, Fromm, S, Martinez-Sanchez, A, Gopaldass, N, Mayer, A, Sachse, C. | 登録日 | 2022-07-18 | 公開日 | 2023-11-01 | 最終更新日 | 2024-05-15 | 実験手法 | ELECTRON MICROSCOPY (26 Å) | 主引用文献 | Atg18 oligomer organization in assembled tubes and on lipid membrane scaffolds. Nat Commun, 14, 2023
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3BEZ
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8AMS
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![BU of 8ams by Molmil](/molmil-images/mine/8ams) | Complex of human TRIM2 RING domain, UBCH5C, and Ubiquitin | 分子名称: | 3,6,9,12,15,18,21-HEPTAOXATRICOSANE-1,23-DIOL, GLYCEROL, Polyubiquitin-C, ... | 著者 | Perez-Borrajero, C, Kotova, I, Murciano, B, Hennig, J. | 登録日 | 2022-08-04 | 公開日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structural and biophysical studies of TRIM2 and TRIM3 To Be Published
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3DVO
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![BU of 3dvo by Molmil](/molmil-images/mine/3dvo) | SgrAI with cognate DNA and calcium bound | 分子名称: | CALCIUM ION, DNA (5'-D(*DGP*DAP*DGP*DTP*DCP*DCP*DAP*DCP*DCP*DGP*DGP*DTP*DGP*DGP*DAP*DCP*DTP*DC)-3'), SgraIR restriction enzyme | 著者 | Dunten, P.W, Horton, N.C, Little, E.J. | 登録日 | 2008-07-18 | 公開日 | 2008-08-19 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.892 Å) | 主引用文献 | The structure of SgrAI bound to DNA; recognition of an 8 base pair target. Nucleic Acids Res., 36, 2008
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5NJX
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![BU of 5njx by Molmil](/molmil-images/mine/5njx) | Human FKBP51 protein in complex with C-terminal peptide of Human HSP 90-alpha | 分子名称: | HSP90AA1 protein, Peptidyl-prolyl cis-trans isomerase FKBP5, SULFATE ION | 著者 | Kumar, R, Moche, M, Winblad, B, Pavlov, P. | 登録日 | 2017-03-30 | 公開日 | 2017-11-08 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.49 Å) | 主引用文献 | Combined x-ray crystallography and computational modeling approach to investigate the Hsp90 C-terminal peptide binding to FKBP51. Sci Rep, 7, 2017
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8SY5
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![BU of 8sy5 by Molmil](/molmil-images/mine/8sy5) | E. coli DNA-directed RNA polymerase transcription elongation complex bound the unnatural dS-BTP base pair in the active site | 分子名称: | 2-oxo-2-hydroadenosine 5'-(tetrahydrogen triphosphate), DNA-directed RNA polymerase subunit alpha, DNA-directed RNA polymerase subunit beta, ... | 著者 | Shan, Z, Lyumkis, D, Oh, J, Wang, D. | 登録日 | 2023-05-24 | 公開日 | 2023-12-27 | 実験手法 | ELECTRON MICROSCOPY (2.7 Å) | 主引用文献 | A unified Watson-Crick geometry drives transcription of six-letter expanded DNA alphabets by E. coli RNA polymerase. Nat Commun, 14, 2023
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2ZEB
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![BU of 2zeb by Molmil](/molmil-images/mine/2zeb) | Potent, Nonpeptide Inhibitors of Human Mast Cell Tryptase | 分子名称: | 1-(1'-{[3-(methylsulfanyl)-2-benzothiophen-1-yl]carbonyl}spiro[1-benzofuran-3,4'-piperidin]-5-yl)methanamine, Tryptase beta 2 | 著者 | Spurlino, J.C, Lewandowski, F, Milligan, C. | 登録日 | 2007-12-08 | 公開日 | 2008-12-09 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Potent, nonpeptide inhibitors of human mast cell tryptase. Synthesis and biological evaluation of novel spirocyclic piperidine amide derivatives Bioorg.Med.Chem.Lett., 18, 2008
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3P5Q
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![BU of 3p5q by Molmil](/molmil-images/mine/3p5q) | Ferric R-state human aquomethemoglobin | 分子名称: | Hemoglobin subunit alpha, Hemoglobin subunit beta, PROTOPORPHYRIN IX CONTAINING FE, ... | 著者 | Yi, J, Thomas, L.M, Richter-Addo, G.B. | 登録日 | 2010-10-10 | 公開日 | 2011-06-08 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure of human R-state aquomethemoglobin at 2.0 A resolution Acta Crystallogr.,Sect.F, 67, 2011
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6WMF
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![BU of 6wmf by Molmil](/molmil-images/mine/6wmf) | Human Sun2-KASH5 complex | 分子名称: | POTASSIUM ION, Protein KASH5, SUN domain-containing protein 2 | 著者 | Cruz, V.E, Schwartz, T.U. | 登録日 | 2020-04-21 | 公開日 | 2020-12-02 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structural Analysis of Different LINC Complexes Reveals Distinct Binding Modes. J.Mol.Biol., 432, 2020
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6PU3
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![BU of 6pu3 by Molmil](/molmil-images/mine/6pu3) | ABC transporter-associated periplasmic binding protein DppA from Helicobacter pylori | 分子名称: | Heme-binding protein A, SER-THR-SER-ALA | 著者 | Rahman, M.M, Machuca, M.A, Khan, M.F, Barlow, C.K, Schittenhelm, R.B, Roujeinikova, A. | 登録日 | 2019-07-16 | 公開日 | 2019-08-21 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Molecular Basis of Unexpected Specificity of ABC Transporter-Associated Substrate-Binding Protein DppA from Helicobacter pylori. J.Bacteriol., 201, 2019
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6NNW
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![BU of 6nnw by Molmil](/molmil-images/mine/6nnw) | Tsn15 in complex with substrate intermediate | 分子名称: | (3E)-3-{(1S,4S,4aS,5R,8aS)-1-[(2E,4R,7S,8E,10S)-1,7-dihydroxy-10-{(2R,3S,5R)-5-[(1S)-1-methoxyethyl]-3-methyloxolan-2-yl}-4-methylundeca-2,8-dien-2-yl]-4,5-dimethyloctahydro-3H-2-benzopyran-3-ylidene}oxolane-2,4-dione, PHOSPHATE ION, PROPANOIC ACID, ... | 著者 | Paiva, F.C.R, Little, R, Leadlay, P, Dias, M.V.B. | 登録日 | 2019-01-15 | 公開日 | 2019-10-23 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Unexpected enzyme-catalysed [4+2] cycloaddition and rearrangement in polyether antibiotic biosynthesis Nat Catal, 2019
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3FUB
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![BU of 3fub by Molmil](/molmil-images/mine/3fub) | Crystal structure of GDNF-GFRalpha1 complex | 分子名称: | 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Parkash, V, Goldman, A. | 登録日 | 2009-01-14 | 公開日 | 2009-06-02 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Comparison of GFL-GFRalpha complexes: further evidence relating GFL bend angle to RET signalling Acta Crystallogr.,Sect.F, 65, 2009
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6VOE
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![BU of 6voe by Molmil](/molmil-images/mine/6voe) | HIV-1 wild type protease with GRL-019-17A, a tricyclic cyclohexane fused tetrahydrofuranofuran (CHf-THF) derivative as the P2 ligand and a aminobenzothiazole(Abt)-based P2'-ligand | 分子名称: | (1S,3aR,5S,6R,7aS)-octahydro-1,6-epoxy-2-benzofuran-5-yl {(2S,3R)-3-hydroxy-4-[(2-methylpropyl)({2-[(propan-2-yl)amino]-1,3-benzoxazol-6-yl}sulfonyl)amino]-1-phenylbutan-2-yl}carbamate, ACETATE ION, CHLORIDE ION, ... | 著者 | Wang, Y.-F, Agniswamy, J, Weber, I.T. | 登録日 | 2020-01-30 | 公開日 | 2020-05-13 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Structure-Based Design of Highly Potent HIV-1 Protease Inhibitors Containing New Tricyclic Ring P2-Ligands: Design, Synthesis, Biological, and X-ray Structural Studies. J.Med.Chem., 63, 2020
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6WAG
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![BU of 6wag by Molmil](/molmil-images/mine/6wag) | Crystal Structure of SmcR S76A from Vibrio Vulnificus | 分子名称: | 1,2-ETHANEDIOL, LuxR family transcriptional regulator, SULFATE ION | 著者 | Newman, J.D, Russell, M.M, Gonzalez-Gutierrez, G, van Kessel, J.C. | 登録日 | 2020-03-25 | 公開日 | 2020-06-17 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.575 Å) | 主引用文献 | The DNA binding domain of the Vibrio vulnificus SmcR transcription factor is flexible and binds diverse DNA sequences. Nucleic Acids Res., 49, 2021
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2CJX
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![BU of 2cjx by Molmil](/molmil-images/mine/2cjx) | Extended substrate recognition in caspase-3 revealed by high resolution X-ray structure analysis | 分子名称: | CASPASE-3, PHQ-ASP-GLU-VAL-ASP-CHLOROMETHYLKETONE | 著者 | Ganesan, R, Mittl, P.R.E, Jelakovic, S, Grutter, M.G. | 登録日 | 2006-04-09 | 公開日 | 2006-06-27 | 最終更新日 | 2017-06-28 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Extended Substrate Recognition in Caspase-3 Revealed by High Resolution X-Ray Structure Analysis J.Mol.Biol., 359, 2006
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8E08
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![BU of 8e08 by Molmil](/molmil-images/mine/8e08) | Crystal structure of HPSE P6 in complex with tetraose pentosan inhibitor | 分子名称: | 2,3,4-tri-O-sulfo-beta-D-xylopyranose-(1-4)-2,3-di-O-sulfo-beta-D-xylopyranose-(1-4)-2,3-di-O-sulfo-beta-D-xylopyranose-(1-4)-2,3-di-O-sulfo-beta-D-xylopyranose, ACETATE ION, Heparanase 50 kDa subunit, ... | 著者 | Whitefield, C, Jackson, C.J. | 登録日 | 2022-08-08 | 公開日 | 2023-07-12 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.93 Å) | 主引用文献 | Complex Inhibitory Mechanism of Glycomimetics with Heparanase. Biochemistry, 62, 2023
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