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8G2F
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BU of 8g2f by Molmil
Crystal Structure of PRMT3 with Compound II710
分子名称: 5'-S-[3-(N'-benzylcarbamimidamido)propyl]-5'-thioadenosine, Protein arginine N-methyltransferase 3
著者Song, X, Dong, A, Deng, Y, Huang, R, Arrowsmith, C.H, Edwards, A.M, Min, J, Structural Genomics Consortium (SGC)
登録日2023-02-03
公開日2023-05-10
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.06 Å)
主引用文献A unique binding pocket induced by a noncanonical SAH mimic to develop potent and selective PRMT inhibitors.
Acta Pharm Sin B, 13, 2023
1OWR
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BU of 1owr by Molmil
CRYSTAL STRUCTURE OF HUMAN NFAT1 BOUND MONOMERICALLY TO DNA
分子名称: NFAT1 Monomeric Binding Site, Minus Strand, Plus Strand, ...
著者Stroud, J.C, Chen, L.
登録日2003-03-29
公開日2004-02-10
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structure of NFAT Bound to DNA as a Monomer
J.Mol.Biol., 334, 2003
1VIB
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BU of 1vib by Molmil
NMR SOLUTION STRUCTURE OF THE NEUROTOXIN B-IV, 20 STRUCTURES
分子名称: NEUROTOXIN B-IV
著者Barnham, K.J, Dyke, T.R, Kem, W.R, Norton, R.S.
登録日1996-11-25
公開日1997-05-15
最終更新日2017-11-29
実験手法SOLUTION NMR
主引用文献Structure of neurotoxin B-IV from the marine worm Cerebratulus lacteus: a helical hairpin cross-linked by disulphide bonding.
J.Mol.Biol., 268, 1997
1VKJ
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BU of 1vkj by Molmil
Crystal structure of heparan sulfate 3-O-sulfotransferase isoform 1 in the presence of PAP
分子名称: ADENOSINE-3'-5'-DIPHOSPHATE, SULFATE ION, heparan sulfate (glucosamine) 3-O-sulfotransferase 1
著者Thorp, S, Lee, K.A, Negishi, M, Linhardt, R.J, Liu, J, Pedersen, L.C.
登録日2004-05-25
公開日2004-06-01
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure and mutational analysis of heparan sulfate 3-O-sulfotransferase isoform 1
J.Biol.Chem., 279, 2004
2NZ1
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BU of 2nz1 by Molmil
Viral Chemokine Binding Protein M3 From Murine Gammaherpesvirus68 In Complex With The CC-Chemokine CCL2/MCP-1
分子名称: Hypothetical protein GAMMAHV.M3, Small inducible cytokine A2
著者Alexander-Brett, J.M, Fremont, D.H.
登録日2006-11-22
公開日2007-12-25
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Dual GPCR and GAG mimicry by the M3 chemokine decoy receptor.
J.Exp.Med., 204, 2007
8UJW
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BU of 8ujw by Molmil
Crystal structure of the KETc7 antigen from Taenia solium
分子名称: GRAM domain-containing protein
著者Sotelo-Mundo, R.R, Gomez-Yanes, A.C, Lopez-Zavala, A.A, Ochoa-Leyva, A.
登録日2023-10-11
公開日2023-11-01
実験手法X-RAY DIFFRACTION (1.72 Å)
主引用文献Crystal structure of the KETc7 antigen from Taenia solium
To Be Published
1YEB
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BU of 1yeb by Molmil
STRUCTURE DETERMINATION AND ANALYSIS OF YEAST ISO-2-CYTOCHROME C AND A COMPOSITE MUTANT PROTEIN
分子名称: CYTOCHROME C, HEME C, SULFATE ION
著者Murphy, M.E.P, Brayer, G.D.
登録日1991-10-29
公開日1993-10-31
最終更新日2021-03-03
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Structure determination and analysis of yeast iso-2-cytochrome c and a composite mutant protein.
J.Mol.Biol., 227, 1992
2OD1
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BU of 2od1 by Molmil
Solution structure of the MYND domain from human AML1-ETO
分子名称: Protein CBFA2T1, ZINC ION
著者Liu, Y.Z, Chen, W, Gaudet, J, Cheney, M.D, Roudaia, L, Cierpicki, T, Klet, R.C, Hartman, K, Laue, T.M, Speck, N.A, Bushweller, J.H.
登録日2006-12-21
公開日2007-06-19
最終更新日2023-12-27
実験手法SOLUTION NMR
主引用文献Structural basis for recognition of SMRT/N-CoR by the MYND domain and its contribution to AML1/ETO's activity.
Cancer Cell, 11, 2007
5XOG
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RNA Polymerase II elongation complex bound with Spt5 KOW5 and Elf1
分子名称: DIPHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER, DNA (30-MER), DNA (39-MER), ...
著者Ehara, H, Shirouzu, M, Sekine, S.
登録日2017-05-28
公開日2017-08-16
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structure of the complete elongation complex of RNA polymerase II with basal factors
Science, 357, 2017
8G58
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Tau (297-391) in vitro untwisted fibril
分子名称: Microtubule-associated protein tau
著者Duan, P, Dregni, A.J, Mammeri, N.E, Hong, M.
登録日2023-02-12
公開日2023-11-08
最終更新日2024-05-15
実験手法SOLID-STATE NMR
主引用文献Structure of the nonhelical filament of the Alzheimer's disease tau core.
Proc.Natl.Acad.Sci.USA, 120, 2023
8EHW
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BU of 8ehw by Molmil
cryo-EM structure of TMEM63A in nanodisc
分子名称: CSC1-like protein 1
著者Zheng, W, Fu, T.M, Holt, J.R.
登録日2022-09-14
公開日2023-08-23
最終更新日2023-11-01
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献TMEM63 proteins function as monomeric high-threshold mechanosensitive ion channels.
Neuron, 111, 2023
8Q3B
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BU of 8q3b by Molmil
The closed state of the ASFV apo-RNA polymerase
分子名称: DNA-directed RNA polymerase RPB1 homolog, DNA-directed RNA polymerase RPB10 homolog, DNA-directed RNA polymerase RPB2 homolog, ...
著者Pilotto, S, Sykora, M, Cackett, G, Werner, F.
登録日2023-08-03
公開日2024-02-14
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (2.69 Å)
主引用文献Structure of the recombinant RNA polymerase from African Swine Fever Virus.
Nat Commun, 15, 2024
2OAT
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BU of 2oat by Molmil
ORNITHINE AMINOTRANSFERASE COMPLEXED WITH 5-FLUOROMETHYLORNITHINE
分子名称: 1-AMINO-7-(2-METHYL-3-OXIDO-5-((PHOSPHONOXY)METHYL)-4-PYRIDOXAL-5-OXO-6-HEPTENATE, ORNITHINE AMINOTRANSFERASE
著者Storici, P, Schirmer, T.
登録日1998-05-07
公開日1998-12-09
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Crystal structure of human ornithine aminotransferase complexed with the highly specific and potent inhibitor 5-fluoromethylornithine.
J.Mol.Biol., 285, 1999
3ZU7
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BU of 3zu7 by Molmil
Crystal structure of a designed selected Ankyrin Repeat protein in complex with the MAP kinase ERK2
分子名称: DESIGNED ANKYRIN REPEAT PROTEIN, MITOGEN-ACTIVATED PROTEIN KINASE 1
著者Kummer, L, Mittl, P.R, Pluckthun, A.
登録日2011-07-16
公開日2012-06-27
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献Structural and Functional Analysis of Phosphorylation-Specific Binders of the Kinase Erk from Designed Ankyrin Repeat Protein Libraries.
Proc.Natl.Acad.Sci.USA, 109, 2012
3ZUV
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BU of 3zuv by Molmil
Crystal structure of a designed selected Ankyrin Repeat protein in complex with the phosphorylated MAP kinase ERK2
分子名称: DESIGNED ANKYRIN REPEAT PROTEIN, MITOGEN-ACTIVATED PROTEIN KINASE 1, SULFATE ION
著者Kummer, L, Mittl, P.R, Pluckthun, A.
登録日2011-07-20
公開日2012-06-27
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.72 Å)
主引用文献Structural and Functional Analysis of Phosphorylation-Specific Binders of the Kinase Erk from Designed Ankyrin Repeat Protein Libraries.
Proc.Natl.Acad.Sci.USA, 109, 2012
8Q3K
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BU of 8q3k by Molmil
The open state of the ASFV apo-RNA polymerase
分子名称: DNA-directed RNA polymerase RPB1 homolog, DNA-directed RNA polymerase RPB10 homolog, DNA-directed RNA polymerase RPB2 homolog, ...
著者Pilotto, S, Sykora, M, Cackett, G, Werner, F.
登録日2023-08-04
公開日2024-02-14
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (2.92 Å)
主引用文献Structure of the recombinant RNA polymerase from African Swine Fever Virus.
Nat Commun, 15, 2024
7QZR
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BU of 7qzr by Molmil
Structure of native leukocyte myeloperoxidase in complex with the Staphyloccal Peroxidase Inhibitor SPIN from Staphylococcus aureus
分子名称: 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Pfanzagl, V, Brito, J.A.
登録日2022-01-31
公開日2022-10-26
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献The staphylococcal inhibitory protein SPIN binds to human myeloperoxidase with picomolar affinity but only dampens halide oxidation.
J.Biol.Chem., 298, 2022
8G4S
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BU of 8g4s by Molmil
40S ribosomal subunit of the 80S Giardia intestinalis assemblage A ribosome with Emetine bound in V2 conformation with mRNA and three tRNAs.
分子名称: 18S rRNA, 40S ribosomal protein S21, 40S ribosomal protein S25, ...
著者Eiler, D.R, Wimberly, B.T, Bilodeau, D.Y, Rissland, O.S, Kieft, J.S.
登録日2023-02-10
公開日2024-01-31
最終更新日2024-04-17
実験手法ELECTRON MICROSCOPY (3.14 Å)
主引用文献The Giardia lamblia ribosome structure reveals divergence in several biological pathways and the mode of emetine function.
Structure, 32, 2024
2POO
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BU of 2poo by Molmil
THERMOSTABLE PHYTASE IN FULLY CALCIUM LOADED STATE
分子名称: CALCIUM ION, PROTEIN (PHYTASE)
著者Ha, N.-C, Oh, B.-H.
登録日1999-04-16
公開日2000-04-19
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Crystal structures of a novel, thermostable phytase in partially and fully calcium-loaded states.
Nat.Struct.Biol., 7, 2000
5W4U
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BU of 5w4u by Molmil
Pol II elongation complex with an N6-methyladenine-containing template
分子名称: 14mer non-template DNA, 29mer template DNA, 9mer RNA, ...
著者Wang, W, Wang, D.
登録日2017-06-13
公開日2018-06-20
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.6 Å)
主引用文献Epigenetic DNA Modification N6-Methyladenine Causes Site-Specific RNA Polymerase II Transcriptional Pausing.
J.Am.Chem.Soc., 139, 2017
8ICM
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BU of 8icm by Molmil
DNA POLYMERASE BETA (POL B) (E.C.2.7.7.7) COMPLEXED WITH SEVEN BASE PAIRS OF DNA; SOAKED IN THE PRESENCE OF DATP (1 MILLIMOLAR), MNCL2 (5 MILLIMOLAR), AND AMMONIUM SULFATE (75 MILLIMOLAR)
分子名称: DNA (5'-D(*CP*AP*TP*TP*AP*GP*AP*A)-3'), DNA (5'-D(*TP*CP*TP*AP*AP*TP*G)-3'), PROTEIN (DNA POLYMERASE BETA (E.C.2.7.7.7)), ...
著者Pelletier, H, Sawaya, M.R.
登録日1996-01-04
公開日1996-11-15
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献A structural basis for metal ion mutagenicity and nucleotide selectivity in human DNA polymerase beta.
Biochemistry, 35, 1996
8ICJ
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BU of 8icj by Molmil
DNA POLYMERASE BETA (E.C.2.7.7.7)/DNA COMPLEX + THYMIDINE-5'-TRIPHOSPHATE, SOAKED IN THE PRESENCE OF DTTP AND MGCL2
分子名称: DNA (5'-D(*CP*AP*TP*TP*AP*GP*AP*A)-3'), DNA (5'-D(*TP*CP*TP*AP*AP*TP*G)-3'), PROTEIN (DNA POLYMERASE BETA (E.C.2.7.7.7)), ...
著者Pelletier, H, Sawaya, M.R.
登録日1996-04-19
公開日1996-11-15
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献A structural basis for metal ion mutagenicity and nucleotide selectivity in human DNA polymerase beta
Biochemistry, 35, 1996
8ICH
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DNA POLYMERASE BETA (POL B) (E.C.2.7.7.7) COMPLEXED WITH SEVEN BASE PAIRS OF DNA; SOAKED IN THE PRESENCE OF DCTP (1 MILLIMOLAR) AND MGCL2 (5 MILLIMOLAR)
分子名称: DNA (5'-D(*CP*AP*TP*TP*AP*GP*AP*A)-3'), DNA (5'-D(*TP*CP*TP*AP*AP*TP*G)-3'), PROTEIN (DNA POLYMERASE BETA (E.C.2.7.7.7)), ...
著者Pelletier, H, Sawaya, M.R.
登録日1996-04-19
公開日1996-11-15
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Characterization of the metal ion binding helix-hairpin-helix motifs in human DNA polymerase beta by X-ray structural analysis.
Biochemistry, 35, 1996
8ICU
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BU of 8icu by Molmil
DNA POLYMERASE BETA (POL B) (E.C.2.7.7.7) COMPLEXED WITH SEVEN BASE PAIRS OF DNA; SOAKED IN THE PRESENCE OF DDATP (1 MILLIMOLAR) AND MNCL2 (5 MILLIMOLAR)
分子名称: 2',3'-DIDEOXYADENOSINE-5'-TRIPHOSPHATE, DNA (5'-D(*CP*AP*TP*TP*AP*GP*AP*A)-3'), DNA (5'-D(*TP*CP*TP*AP*AP*TP*GP*A)-3'), ...
著者Pelletier, H, Sawaya, M.R.
登録日1995-12-15
公開日1996-11-15
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献A structural basis for metal ion mutagenicity and nucleotide selectivity in human DNA polymerase beta
Biochemistry, 35, 1996
8ICV
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BU of 8icv by Molmil
DNA POLYMERASE BETA (POL B) (E.C.2.7.7.7) COMPLEXED WITH SEVEN BASE PAIRS OF DNA; SOAKED IN THE PRESENCE OF DGTP (1 MILLIMOLAR) AND MNCL2 (5 MILLIMOLAR)
分子名称: 2'-DEOXYGUANOSINE-5'-TRIPHOSPHATE, DNA (5'-D(*CP*AP*TP*TP*AP*GP*AP*A)-3'), DNA (5'-D(*TP*CP*TP*AP*AP*TP*GP*G)-3'), ...
著者Pelletier, H, Sawaya, M.R.
登録日1996-01-04
公開日1996-11-15
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献A structural basis for metal ion mutagenicity and nucleotide selectivity in human DNA polymerase beta
Biochemistry, 35, 1996

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