8GHE
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![BU of 8ghe by Molmil](/molmil-images/mine/8ghe) | The structure of h12-LOX in tetrameric form bound to endogenous inhibitor oleoyl-CoA | 分子名称: | FE (II) ION, Polyunsaturated fatty acid lipoxygenase ALOX12, S-{(3R,5R,9R)-1-[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-hydroxy-3-(phosphonooxy)tetrahydrofuran-2-yl]-3,5,9-trihydroxy-8,8-dimethyl-3,5-dioxido-10,14-dioxo-2,4,6-trioxa-11,15-diaza-3lambda~5~,5lambda~5~-diphosphaheptadecan-17-yl} (9Z)-octadec-9-enethioate (non-preferred name) | 著者 | Black, K.A, Mobbs, J.I, Venugopal, H, Thal, D.M, Glukhova, A. | 登録日 | 2023-03-09 | 公開日 | 2023-08-09 | 最終更新日 | 2023-10-11 | 実験手法 | ELECTRON MICROSCOPY (2.05 Å) | 主引用文献 | Cryo-EM structures of human arachidonate 12S-lipoxygenase bound to endogenous and exogenous inhibitors. Blood, 142, 2023
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8GHB
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![BU of 8ghb by Molmil](/molmil-images/mine/8ghb) | The structure of h12-LOX in monomeric form | 分子名称: | FE (II) ION, Polyunsaturated fatty acid lipoxygenase ALOX12 | 著者 | Black, K.A, Mobbs, J.I, Venugopal, H, Thal, D.M, Glukhova, A. | 登録日 | 2023-03-09 | 公開日 | 2023-08-09 | 最終更新日 | 2024-05-01 | 実験手法 | ELECTRON MICROSCOPY (2.76 Å) | 主引用文献 | Cryo-EM structures of human arachidonate 12S-lipoxygenase bound to endogenous and exogenous inhibitors. Blood, 142, 2023
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1FAD
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![BU of 1fad by Molmil](/molmil-images/mine/1fad) | DEATH DOMAIN OF FAS-ASSOCIATED DEATH DOMAIN PROTEIN, RESIDUES 89-183 | 分子名称: | PROTEIN (FADD PROTEIN) | 著者 | Jeong, E.-J, Bang, S, Lee, T.H, Park, Y.-I, Sim, W.-S, Kim, K.-S. | 登録日 | 1999-03-23 | 公開日 | 1999-07-06 | 最終更新日 | 2023-12-27 | 実験手法 | SOLUTION NMR | 主引用文献 | The solution structure of FADD death domain. Structural basis of death domain interactions of Fas and FADD. J.Biol.Chem., 274, 1999
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8GRJ
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![BU of 8grj by Molmil](/molmil-images/mine/8grj) | Crystal structure of gamma-alpha subunit complex from Burkholderia cepacia FAD glucose dehydrogenase in complex with gluconolactone | 分子名称: | D-glucono-1,5-lactone, FE3-S4 CLUSTER, FLAVIN-ADENINE DINUCLEOTIDE, ... | 著者 | Yoshida, H, Kojima, K, Tsugawa, W, Okuda-Shimazaki, J, Kerrigan, J.A, Sode, K. | 登録日 | 2022-09-01 | 公開日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.95 Å) | 主引用文献 | Crystal structure of gamma-alpha subunit complex from Burkholderia cepacia FAD glucose dehydrogenase in complex with gluconolactone To Be Published
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6VCA
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![BU of 6vca by Molmil](/molmil-images/mine/6vca) | TB38 complex | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 5'-nucleotidase, ... | 著者 | Zhou, Y.F, Lord, D.M. | 登録日 | 2019-12-20 | 公開日 | 2020-11-11 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (3.73 Å) | 主引用文献 | A highly potent CD73 biparatopic antibody blocks organization of the enzyme active site through dual mechanisms. J.Biol.Chem., 295, 2020
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3AFF
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![BU of 3aff by Molmil](/molmil-images/mine/3aff) | Crystal structure of the HsaA monooxygenase from M. tuberculosis | 分子名称: | Hydroxylase, putative | 著者 | D'Angelo, I, Lin, L.Y, Dresen, C, Tocheva, E.I, Strynadka, N, Eltis, L.D. | 登録日 | 2010-02-28 | 公開日 | 2010-05-26 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | A flavin-dependent monooxygenase from Mycobacterium tuberculosis involved in cholesterol catabolism J.Biol.Chem., 285, 2010
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1FC7
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![BU of 1fc7 by Molmil](/molmil-images/mine/1fc7) | PHOTOSYSTEM II D1 C-TERMINAL PROCESSING PROTEASE | 分子名称: | PHOTOSYSTEM II D1 PROTEASE | 著者 | Liao, D.I, Qian, J, Chisholm, D.A, Jordan, D.B, Diner, B.A. | 登録日 | 2000-07-18 | 公開日 | 2001-01-18 | 最終更新日 | 2018-10-03 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal structures of the photosystem II D1 C-terminal processing protease. Nat.Struct.Biol., 7, 2000
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5C5U
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![BU of 5c5u by Molmil](/molmil-images/mine/5c5u) | The crystal structure of viral collagen prolyl hydroxylase vCPH from Paramecium Bursaria Chlorella virus-1 - Truncated Construct | 分子名称: | ACETATE ION, MANGANESE (II) ION, Prolyl 4-hydroxylase, ... | 著者 | Longbotham, J.E, Levy, C.W, Johannisen, L.O, Tarhonskaya, H, Jiang, S, Loenarz, C, Flashman, E, Hay, S, Schofiled, C.J, Scrutton, N.S. | 登録日 | 2015-06-22 | 公開日 | 2015-09-30 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structure and Mechanism of a Viral Collagen Prolyl Hydroxylase. Biochemistry, 54, 2015
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5C66
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![BU of 5c66 by Molmil](/molmil-images/mine/5c66) | |
8GO3
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![BU of 8go3 by Molmil](/molmil-images/mine/8go3) | |
5C7O
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![BU of 5c7o by Molmil](/molmil-images/mine/5c7o) | Structure of human testis-specific glyceraldehyde-3-phosphate dehydrogenase holo form with NAD+ | 分子名称: | Glyceraldehyde-3-phosphate dehydrogenase, testis-specific, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ... | 著者 | Betts, L, Machius, M, Danshina, P, O'Brien, D. | 登録日 | 2015-06-24 | 公開日 | 2016-03-09 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.729 Å) | 主引用文献 | Structural analyses to identify selective inhibitors of glyceraldehyde 3-phosphate dehydrogenase-S, a sperm-specific glycolytic enzyme. Mol. Hum. Reprod., 22, 2016
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1FG5
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![BU of 1fg5 by Molmil](/molmil-images/mine/1fg5) | CRYSTAL STRUCTURE OF BOVINE ALPHA-1,3-GALACTOSYLTRANSFERASE CATALYTIC DOMAIN. | 分子名称: | N-ACETYLLACTOSAMINIDE ALPHA-1,3-GALACTOSYLTRANSFERASE | 著者 | Gastinel, L.N, Bignon, C, Shaper, J.H, Joziasse, D.H. | 登録日 | 2000-07-28 | 公開日 | 2001-07-28 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Bovine alpha1,3-galactosyltransferase catalytic domain structure and its relationship with ABO histo-blood group and glycosphingolipid glycosyltransferases. EMBO J., 20, 2001
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6V18
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![BU of 6v18 by Molmil](/molmil-images/mine/6v18) | immune receptor complex | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Fibrinogen beta, GLYCEROL, ... | 著者 | Lim, J.J, Rossjohn, J. | 登録日 | 2019-11-20 | 公開日 | 2020-11-25 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | The shared susceptibility epitope of HLA-DR4 binds citrullinated self-antigens and the TCR. Sci Immunol, 6, 2021
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8GQ1
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![BU of 8gq1 by Molmil](/molmil-images/mine/8gq1) | HyHEL10 Fab complexed with hen egg lysozyme carrying arginine cluster in framework region of light chain. | 分子名称: | Heavy Chain of HyHel10 Antibody Fragment (Fab), Light Chain of HyHel10 Antibody Fragment (Fab), Lysozyme C, ... | 著者 | Matsuura, H, Hirata, K, Sakai, N, Nakakido, M, Tsumoto, K. | 登録日 | 2022-08-28 | 公開日 | 2023-08-30 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (3.13 Å) | 主引用文献 | Arginine cluster introduction on framework region in anti-lysozyme antibody improved association rate constant by changing conformational diversity of CDR loops. Protein Sci., 32, 2023
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6V38
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![BU of 6v38 by Molmil](/molmil-images/mine/6v38) | Cryo-EM structure of Ca2+-bound hsSlo1 channel | 分子名称: | (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, CALCIUM ION, CHOLESTEROL, ... | 著者 | Tao, X, MacKinnon, R. | 登録日 | 2019-11-25 | 公開日 | 2019-12-25 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | Molecular structures of the human Slo1 K + channel in complex with beta 4. Elife, 8, 2019
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4QNQ
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5CB3
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![BU of 5cb3 by Molmil](/molmil-images/mine/5cb3) | Structural Insights into the Mechanism of Escherichia coli Ymdb | 分子名称: | ADENOSINE-5-DIPHOSPHORIBOSE, O-acetyl-ADP-ribose deacetylase | 著者 | Zhang, W, Wang, C, Song, Y, Shao, C, Zhang, X, Zang, J. | 登録日 | 2015-06-30 | 公開日 | 2015-11-04 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structural insights into the mechanism of Escherichia coli YmdB: A 2'-O-acetyl-ADP-ribose deacetylase J.Struct.Biol., 192, 2015
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8GYK
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![BU of 8gyk by Molmil](/molmil-images/mine/8gyk) | CryoEM structure of the RAD51_ADP filament | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, DNA repair protein RAD51 homolog 1, MAGNESIUM ION | 著者 | Miki, Y, Luo, S.C, Ho, M.C. | 登録日 | 2022-09-22 | 公開日 | 2023-08-30 | 実験手法 | ELECTRON MICROSCOPY (3.14 Å) | 主引用文献 | A RAD51-ADP double filament structure unveils the mechanism of filament dynamics in homologous recombination. Nat Commun, 14, 2023
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1FJD
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![BU of 1fjd by Molmil](/molmil-images/mine/1fjd) | HUMAN PARVULIN-LIKE PEPTIDYL PROLYL CIS/TRANS ISOMERASE, HPAR14 | 分子名称: | PEPTIDYL PROLYL CIS/TRANS ISOMERASE (PPIASE) | 著者 | Terada, T, Shirouzu, M, Fukumori, Y, Fujimori, F, Ito, Y, Kigawa, T, Yokoyama, S, Uchida, T, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2000-08-08 | 公開日 | 2001-08-08 | 最終更新日 | 2024-05-22 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the human parvulin-like peptidyl prolyl cis/trans isomerase, hPar14. J.Mol.Biol., 305, 2001
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6V7D
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![BU of 6v7d by Molmil](/molmil-images/mine/6v7d) | Human Arginase1 Complexed with Bicyclic Inhibitor Compound 10 | 分子名称: | Arginase-1, MANGANESE (II) ION, {3-[(3aR,4R,5S,6aR)-4-azaniumyl-4-carboxyoctahydrocyclopenta[b]pyrrol-1-ium-5-yl]propyl}(trihydroxy)borate(1-) | 著者 | Palte, R.L, Lesburg, C.A. | 登録日 | 2019-12-08 | 公開日 | 2020-05-06 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.82 Å) | 主引用文献 | Discovery and Optimization of Rationally Designed Bicyclic Inhibitors of Human Arginase to Enhance Cancer Immunotherapy. Acs Med.Chem.Lett., 11, 2020
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6V51
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![BU of 6v51 by Molmil](/molmil-images/mine/6v51) | Spin-labeled T4 Lysozyme (9/131FnbY)-(4-Amino-TEMPO) | 分子名称: | 4-amino-2,2,6,6-tetramethylpiperidin-1-ol, Endolysin | 著者 | Liu, J, Morizumi, T, Ou, W.L, Wang, L, Ernst, O.P. | 登録日 | 2019-12-02 | 公開日 | 2020-10-07 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Genetically Encoded Quinone Methides Enabling Rapid, Site-Specific, and Photocontrolled Protein Modification with Amine Reagents. J.Am.Chem.Soc., 142, 2020
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6V6L
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![BU of 6v6l by Molmil](/molmil-images/mine/6v6l) | Co-structure of human glycogen synthase kinase beta with 1-(6-((2-((6-amino-5-nitropyridin-2-yl)amino)ethyl)amino)-2-(2,4-dichlorophenyl)pyridin-3-yl)-4-methylpiperazin-2-one | 分子名称: | 1-(6-((2-((6-amino-5-nitropyridin-2-yl)amino)ethyl)amino)-2-(2,4-dichlorophenyl)pyridin-3-yl)-4-methylpiperazin-2-one, Glycogen synthase kinase-3 beta, PHOSPHATE ION | 著者 | Bussiere, D.E, Fang, E, Shu, W. | 登録日 | 2019-12-05 | 公開日 | 2020-01-15 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.19 Å) | 主引用文献 | Discovery and optimization of novel pyridines as highly potent and selective glycogen synthase kinase 3 inhibitors. Bioorg.Med.Chem.Lett., 30, 2020
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6VAX
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![BU of 6vax by Molmil](/molmil-images/mine/6vax) | Crystal structure of human SDHA-SDHAF2 assembly intermediate | 分子名称: | 1,2-ETHANEDIOL, FLAVIN-ADENINE DINUCLEOTIDE, GLYCEROL, ... | 著者 | Sharma, P, Maklashina, E, Cecchini, G, Iverson, T.M. | 登録日 | 2019-12-18 | 公開日 | 2020-08-26 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.59 Å) | 主引用文献 | The roles of SDHAF2 and dicarboxylate in covalent flavinylation of SDHA, the human complex II flavoprotein. Proc.Natl.Acad.Sci.USA, 117, 2020
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1FGX
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![BU of 1fgx by Molmil](/molmil-images/mine/1fgx) | CRYSTAL STRUCTURE OF THE BOVINE BETA 1,4 GALACTOSYLTRANSFERASE (B4GALT1) CATALYTIC DOMAIN COMPLEXED WITH UMP | 分子名称: | BETA 1,4 GALACTOSYLTRANSFERASE, URIDINE-5'-MONOPHOSPHATE | 著者 | Gastinel, L.N, Cambillau, C, Bourne, Y. | 登録日 | 2000-07-29 | 公開日 | 2000-08-16 | 最終更新日 | 2021-07-21 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Crystal structures of the bovine beta4galactosyltransferase catalytic domain and its complex with uridine diphosphogalactose. EMBO J., 18, 1999
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6VCM
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![BU of 6vcm by Molmil](/molmil-images/mine/6vcm) | Crystal structure of E.coli RppH-DapF in complex with GTP, Mg2+ and F- | 分子名称: | CHLORIDE ION, Diaminopimelate epimerase, FLUORIDE ION, ... | 著者 | Gao, A, Vasilyev, N, Kaushik, A, Duan, W, Serganov, A. | 登録日 | 2019-12-21 | 公開日 | 2020-02-05 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Principles of RNA and nucleotide discrimination by the RNA processing enzyme RppH. Nucleic Acids Res., 48, 2020
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