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1P48
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REVERSE PROTONATION IS THE KEY TO GENERAL ACID-BASE CATALYSIS IN ENOLASE
分子名称: Enolase 1, MAGNESIUM ION, PHOSPHOENOLPYRUVATE
著者Sims, P.A, Larsen, T.M, Poyner, R.R, Cleland, W.W, Reed, G.H.
登録日2003-04-21
公開日2003-11-18
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Reverse protonation is the key to general acid-base catalysis in enolase
Biochemistry, 42, 2003
1P49
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Structure of Human Placental Estrone/DHEA Sulfatase
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, PHOSPHATE ION, ...
著者Hernandez-Guzman, F.G, Higashiyama, T, Pangborn, W, Osawa, Y, Ghosh, D.
登録日2003-04-21
公開日2003-08-12
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structure of Human Estrone Sulfatase Suggests Functional Roles of Membrane Association
J.Biol.Chem., 278, 2003
1P4A
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Crystal Structure of the PurR complexed with cPRPP
分子名称: 1-ALPHA-PYROPHOSPHORYL-2-ALPHA,3-ALPHA-DIHYDROXY-4-BETA-CYCLOPENTANE-METHANOL-5-PHOSPHATE, Pur operon repressor
著者Bera, A.K, Zhu, J, Zalkin, H, Smith, J.L.
登録日2003-04-22
公開日2003-12-09
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.22 Å)
主引用文献Functional dissection of the Bacillus subtilis pur operator site.
J.Bacteriol., 185, 2003
1P4B
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Three-Dimensional Structure Of a Single Chain Fv Fragment Complexed With The peptide GCN4(7P-14P).
分子名称: Antibody Variable heavy chain, Antibody Variable light chain, GCN4(7P-14P) peptide
著者Zahnd, C, Spinelli, S, Luginbuhl, B, Jermutus, L, Amstutz, P, Cambillau, C, Pluckthun, A.
登録日2003-04-22
公開日2004-05-04
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Directed in Vitro Evolution and Crystallographic Analysis of a Peptide-binding Single Chain Antibody Fragment (scFv) with Low Picomolar Affinity.
J.Biol.Chem., 279, 2004
1P4C
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High Resolution Structure of Oxidized Active Mutant of (S)-Mandelate Dehydrogenase
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, FLAVIN MONONUCLEOTIDE, L(+)-Mandelate Dehydrogenase, ...
著者Sukumar, N, Mitra, B, Mathews, F.S.
登録日2003-04-22
公開日2003-10-28
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.35 Å)
主引用文献High Resolution Structures of an Oxidized and Reduced Flavoprotein: THE WATER SWITCH IN A SOLUBLE FORM OF (S)-MANDELATE DEHYDROGENASE
J.Biol.Chem., 279, 2004
1P4D
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F factor TraI Relaxase Domain
分子名称: 1,2-ETHANEDIOL, MAGNESIUM ION, TraI protein
著者Datta, S, Larkin, C, Schildbach, J.F.
登録日2003-04-22
公開日2003-10-14
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structural insights into single-stranded DNA binding and cleavage by F factor TraI.
Structure, 11, 2003
1P4E
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Flpe W330F mutant-DNA Holliday Junction Complex
分子名称: 33-MER, 5'-D(*TP*AP*AP*GP*TP*TP*CP*CP*TP*AP*TP*TP*C)-3', 5'-D(*TP*TP*TP*AP*AP*AP*AP*GP*AP*AP*TP*AP*GP*GP*AP*AP*CP*TP*TP*C)-3', ...
著者Rice, P.A, Chen, Y.
登録日2003-04-23
公開日2003-05-20
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献The role of the conserved Trp330 in Flp-mediated recombination. Functional and structural analysis
J.Biol.Chem., 278, 2003
1P4F
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DEATH ASSOCIATED PROTEIN KINASE CATALYTIC DOMAIN WITH BOUND INHIBITOR FRAGMENT
分子名称: 5,6-Dihydro-benzo[H]cinnolin-3-ylamine, Death-associated protein kinase 1
著者Velentza, A.V, Wainwright, M.S, Zasadzki, M, Mirzoeva, S, Haiech, J, Focia, P.J, Egli, M, Watterson, D.M.
登録日2003-04-23
公開日2004-09-28
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献An aminopyridazine-based inhibitor of a pro-apoptotic protein kinase attenuates hypoxia-ischemia induced acute brain injury.
Bioorg.Med.Chem.Lett., 13, 2003
1P4G
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Crystal structure of glycogen phosphorylase b in complex with C-(1-azido-alpha-D-glucopyranosyl)formamide
分子名称: C-(1-AZIDO-ALPHA-D-GLUCOPYRANOSYL) FORMAMIDE, Glycogen phosphorylase, muscle form, ...
著者Chrysina, E.D, Oikonomakos, N.G, Zographos, S.E, Kosmopoulou, M.N, Bischler, N, Leonidas, D.D, Nagy, V, Somsak, L, Gergely, P, Praly, J.-P.
登録日2003-04-23
公開日2004-05-18
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crsytallographic Studies on alpha- and beta-D-glucopyranosyl Formamide Analogues, Inhibitors of Glycogen Phosphorylase
Biocatal.Biotransfor., 21, 2003
1P4H
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Crystal structure of glycogen phosphorylase b in complex with C-(1-acetamido-alpha-D-glucopyranosyl) formamide
分子名称: 1-DEOXY-1-ACETYLAMINO-BETA-D-GLUCO-2-HEPTULOPYRANOSONAMIDE, Glycogen phosphorylase, muscle form, ...
著者Chrysina, E.D, Oikonomakos, N.G, Zographos, S.E, Kosmopoulou, M.N, Bischler, N, Leonidas, D.D, Nagy, V, Somsak, L, Gergely, P, Praly, J.-P.
登録日2003-04-23
公開日2004-05-18
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.06 Å)
主引用文献Crsytallographic Studies on alpha- and beta-D-glucopyranosyl Formamide Analogues, Inhibitors of Glycogen Phosphorylase
Biocatal.Biotransfor., 21, 2003
1P4I
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Crystal Structure of scFv against peptide GCN4
分子名称: ANTIBODY VARIABLE LIGHT CHAIN, antibody variable heavy chain
著者Zahnd, C, Spinelli, S, Luginbuhl, B, Jermutus, L, Amstutz, P, Cambillau, C, Pluckthun, A.
登録日2003-04-23
公開日2004-05-04
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Directed in Vitro Evolution and Crystallographic Analysis of a Peptide-binding Single Chain Antibody Fragment (scFv) with Low Picomolar Affinity.
J.Biol.Chem., 279, 2004
1P4J
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Crystal structure of glycogen phosphorylase b in complex with C-(1-hydroxy-beta-D-glucopyranosyl)formamide
分子名称: (2R,3R,4S,5S,6R)-2,3,4,5-tetrahydroxy-6-(hydroxymethyl)oxane-2-carboxamide, Glycogen phosphorylase, muscle form, ...
著者Chrysina, E.D, Oikonomakos, N.G, Zographos, S.E, Kosmopoulou, M.N, Bischler, N, Leonidas, D.D, Nagy, V, Somsak, L, Gergely, P, Praly, J.-P.
登録日2003-04-23
公開日2004-05-18
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crsytallographic Studies on alpha- and beta-D-glucopyranosyl Formamide Analogues, Inhibitors of Glycogen Phosphorylase
Biocatal.Biotransfor., 21, 2003
1P4K
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CRYSTAL STRUCTURE OF THE GLYCOSYLASPARAGINASE PRECURSOR D151N MUTANT
分子名称: GLYCEROL, N(4)-(Beta-N-acetylglucosaminyl)-L-asparaginase
著者Qian, X, Guan, C, Guo, H.C.
登録日2003-04-23
公開日2003-05-06
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献A dual role for an aspartic acid in glycosylasparaginase autoproteolysis.
Structure, 11, 2003
1P4L
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Crystal structure of NK receptor Ly49C mutant with its MHC class I ligand H-2Kb
分子名称: Beta-2-microglobulin, LY49-C, MHC CLASS I H-2KB HEAVY CHAIN, ...
著者Dam, J, Guan, R, Natarajan, K, Dimasi, N, Mariuzza, R.A.
登録日2003-04-23
公開日2003-11-11
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Variable MHC class I engagement by Ly49 natural killer cell receptors demonstrated by the crystal structure of Ly49C bound to H-2K(b).
Nat.Immunol., 4, 2003
1P4M
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CRYSTAL STRUCTURE OF RIBOFLAVIN KINASE
分子名称: ADENOSINE-5'-DIPHOSPHATE, FLAVIN MONONUCLEOTIDE, MAGNESIUM ION, ...
著者Karthikeyan, S, Zhou, Q, Mseeh, F, Grishin, N.V, Osterman, A.L, Zhang, H.
登録日2003-04-23
公開日2003-05-13
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal Structure of Human Riboflavin Kinase Reveals a Beta Barrel Fold and a Novel Active Site Arch
Structure, 11, 2003
1P4N
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Crystal Structure of Weissella viridescens FemX:UDP-MurNAc-pentapeptide complex
分子名称: FemX, GLYCEROL, MAGNESIUM ION, ...
著者Biarrotte-Sorin, S, Maillard, A, Delettre, J, Sougakoff, W, Arthur, M, Mayer, C.
登録日2003-04-23
公開日2004-02-10
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structures of Weissella viridescens FemX and its complex with UDP-MurNAc-pentapeptide: insights into FemABX family substrates recognition.
Structure, 12, 2004
1P4O
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Structure of Apo unactivated IGF-1R KInase domain at 1.5A resolution.
分子名称: Insulin-like growth factor I receptor protein
著者Munshi, S, Kornienko, M, Hall, D.L, Darke, P.L, Waxman, L, Kuo, L.C.
登録日2003-04-23
公開日2003-04-29
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Structure of apo, unactivated insulin-like growth factor-1 receptor kinase at 1.5 A resolution.
Acta Crystallogr.,Sect.D, 59, 2003
1P4P
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Outer Surface Protein B of B. burgdorferi: crystal structure of the C-terminal fragment
分子名称: Outer surface protein B
著者Becker, M, Bunikis, J, Lade, B.D, Dunn, J.J, Barbour, A.G, Lawson, C.L.
登録日2003-04-23
公開日2004-05-04
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural Investigation of Borrelia burgdorferi OspB, a BactericidalFab Target.
J.Biol.Chem., 280, 2005
1P4Q
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Solution structure of the CITED2 transactivation domain in complex with the p300 CH1 domain
分子名称: Cbp/p300-interacting transactivator 2, E1A-associated protein p300, ZINC ION
著者Freedman, S.J, Sun, Z.-Y.J, Kung, A.L, France, D.S, Wagner, G, Eck, M.J.
登録日2003-04-23
公開日2003-07-01
最終更新日2017-02-01
実験手法SOLUTION NMR
主引用文献Structural basis for negative regulation of hypoxia-inducible factor-1alpha by CITED2.
Nat.Struct.Biol., 10, 2003
1P4R
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Crystal Structure of Human ATIC in complex with folate-based inhibitor BW1540U88UD
分子名称: AMINOIMIDAZOLE 4-CARBOXAMIDE RIBONUCLEOTIDE, Bifunctional purine biosynthesis protein PURH, N-[(S)-(4-{[(2-AMINO-4-HYDROXYQUINAZOLIN-6-YL)(DIHYDROXY)-LAMBDA~4~-SULFANYL]AMINO}PHENYL)(HYDROXY)METHYL]-L-GLUTAMIC ACID, ...
著者Cheong, C.-G, Greasley, S.E, Horton, P.A, Beardsley, G.P, Wilson, I.A.
登録日2003-04-23
公開日2004-03-30
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献Crystal structures of human bifunctional enzyme aminoimidazole-4-carboxamide ribonucleotide transformylase/IMP cyclohydrolase in complex with potent sulfonyl-containing antifolates
J.Biol.Chem., 279, 2004
1P4S
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Solution structure of Mycobacterium tuberculosis adenylate kinase
分子名称: Adenylate kinase
著者Miron, S, Munier-Lehmann, H, Craescu, C.T.
登録日2003-04-24
公開日2004-01-20
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Structural and Dynamic Studies on Ligand-Free Adenylate Kinase from Mycobacterium tuberculosis Revealed a Closed Conformation that Can Be Related to the Reduced Catalytic Activity.
Biochemistry, 43, 2004
1P4T
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Crystal structure of Neisserial surface protein A (NspA)
分子名称: ETHANOLAMINE, PENTAETHYLENE GLYCOL MONODECYL ETHER, SULFATE ION, ...
著者Vandeputte-Rutten, L, Bos, M.P, Tommassen, J, Gros, P.
登録日2003-04-24
公開日2003-07-22
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献Crystal structure of Neisserial Surface Protein A (NspA), a conserved outer membrane protein with vaccine potential
J.Biol.Chem., 278, 2003
1P4U
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CRYSTAL STRUCTURE OF GGA3 GAE DOMAIN IN COMPLEX WITH RABAPTIN-5 PEPTIDE
分子名称: ADP-ribosylation factor binding protein GGA3, Rabaptin-5
著者Miller, G.J, Mattera, R, Bonifacino, J.S, Hurley, J.H.
登録日2003-04-24
公開日2003-07-29
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献RECOGNITION OF ACCESSORY PROTEIN MOTIFS BY THE GAMMA-ADAPTIN EAR DOMAIN OF GGA3
Nat.Struct.Biol., 10, 2003
1P4V
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CRYSTAL STRUCTURE OF THE GLYCOSYLASPARAGINASE PRECURSOR D151N MUTANT WITH GLYCINE
分子名称: GLYCINE, N(4)-(Beta-N-acetylglucosaminyl)-L-asparaginase precursor
著者Qian, X, Guan, C, Guo, H.C.
登録日2003-04-24
公開日2003-05-06
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献A dual role for an aspartic acid in glycosylasparaginase autoproteolysis.
Structure, 11, 2003
1P4W
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Solution structure of the DNA-binding domain of the Erwinia amylovora RcsB protein
分子名称: rcsB
著者Pristovsek, P, Sengupta, K, Loehr, F, Schaefer, B, Wehland von Trebra, M, Rueterjans, H, Bernhard, F.
登録日2003-04-24
公開日2003-06-17
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Structural analysis of the DNA-binding domain of the Erwinia amylovora RcsB protein and its interaction with the RcsAB box.
J.Biol.Chem., 278, 2003

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