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7PXF
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BU of 7pxf by Molmil
Ca2+ free Drosophila Slo channel
分子名称: Isoform J of Calcium-activated potassium channel slowpoke, MAGNESIUM ION, POTASSIUM ION
著者Raisch, T, Brockmann, A, Ebbinghaus-Kintscher, U, Freigang, J, Gutbrod, O, Kubicek, J, Maertens, B, Hofnagel, O, Raunser, S.
登録日2021-10-08
公開日2021-12-15
最終更新日2024-07-17
実験手法ELECTRON MICROSCOPY (2.68 Å)
主引用文献Small molecule modulation of the Drosophila Slo channel elucidated by cryo-EM.
Nat Commun, 12, 2021
7PXE
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BU of 7pxe by Molmil
Ca2+ bound Drosophila Slo channel
分子名称: (4S,7R)-4-HYDROXY-N,N,N-TRIMETHYL-9-OXO-7-[(PALMITOYLOXY)METHYL]-3,5,8-TRIOXA-4-PHOSPHAHEXACOSAN-1-AMINIUM 4-OXIDE, CALCIUM ION, CHOLESTEROL, ...
著者Raisch, T, Brockmann, A, Ebbinghaus-Kintscher, U, Freigang, J, Gutbrod, O, Kubicek, J, Maertens, B, Hofnagel, O, Raunser, S.
登録日2021-10-08
公開日2021-12-15
最終更新日2024-07-17
実験手法ELECTRON MICROSCOPY (2.38 Å)
主引用文献Small molecule modulation of the Drosophila Slo channel elucidated by cryo-EM.
Nat Commun, 12, 2021
6EBL
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BU of 6ebl by Molmil
The voltage-activated Kv1.2-2.1 paddle chimera channel in lipid nanodiscs, cytosolic domain
分子名称: NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, Potassium voltage-gated channel subfamily A member 2,Potassium voltage-gated channel subfamily B member 2 chimera, Voltage-gated potassium channel subunit beta-2
著者Matthies, D, Bae, C, Fox, T, Bartesaghi, A, Subramaniam, S, Swartz, K.J.
登録日2018-08-06
公開日2018-08-22
最終更新日2024-03-13
実験手法ELECTRON MICROSCOPY (3 Å)
主引用文献Single-particle cryo-EM structure of a voltage-activated potassium channel in lipid nanodiscs.
Elife, 7, 2018
8TI1
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BU of 8ti1 by Molmil
Cryo-EM structure of a SUR1/Kir6.2-Q52R ATP-sensitive potassium channel in the presence of PIP2 in the open conformation
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, ATP-sensitive inward rectifier potassium channel 11, DI-PALMITOYL-3-SN-PHOSPHATIDYLETHANOLAMINE, ...
著者Driggers, C.M, Shyng, S.-L.
登録日2023-07-18
公開日2024-04-03
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献Structure of an open K ATP channel reveals tandem PIP 2 binding sites mediating the Kir6.2 and SUR1 regulatory interface.
Nat Commun, 15, 2024
8TI2
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BU of 8ti2 by Molmil
Cryo-EM structure of a SUR1/Kir6.2-Q52R ATP-sensitive potassium channel in the presence of PIP2 in the open conformation
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, ATP-sensitive inward rectifier potassium channel 11, DI-PALMITOYL-3-SN-PHOSPHATIDYLETHANOLAMINE, ...
著者Driggers, C.M, Shyng, S.-L.
登録日2023-07-18
公開日2024-04-03
実験手法ELECTRON MICROSCOPY (3.28 Å)
主引用文献Structure of an open K ATP channel reveals tandem PIP 2 binding sites mediating the Kir6.2 and SUR1 regulatory interface.
Nat Commun, 15, 2024
5YWD
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BU of 5ywd by Molmil
Structure of pancreatic ATP-sensitive potassium channel bound with Mg-ADP (focused refinement of SUR1 ABC transporter module at 4.22A)
分子名称: ADENOSINE-5'-DIPHOSPHATE, ATP-binding cassette sub-family C member 8 isoform X2, MAGNESIUM ION
著者Chen, L, Wu, J.X.
登録日2017-11-29
公開日2018-05-02
最終更新日2024-03-27
実験手法ELECTRON MICROSCOPY (4.2 Å)
主引用文献Ligand binding and conformational changes of SUR1 subunit in pancreatic ATP-sensitive potassium channels.
Protein Cell, 9, 2018
5YW7
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Structure of pancreatic ATP-sensitive potassium channel bound with glibenclamide and ATPgammaS (focused refinement on SUR1 ABC transporter module at 4.4A)
分子名称: 5-chloro-N-(2-{4-[(cyclohexylcarbamoyl)sulfamoyl]phenyl}ethyl)-2-methoxybenzamide, ATP-binding cassette sub-family C member 8 isoform X2, PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER
著者Chen, L, Wu, J.X.
登録日2017-11-29
公開日2018-05-02
最終更新日2024-03-27
実験手法ELECTRON MICROSCOPY (4.4 Å)
主引用文献Ligand binding and conformational changes of SUR1 subunit in pancreatic ATP-sensitive potassium channels.
Protein Cell, 9, 2018
2A79
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BU of 2a79 by Molmil
Mammalian Shaker Kv1.2 potassium channel- beta subunit complex
分子名称: NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, POTASSIUM ION, Potassium voltage-gated channel subfamily A member 2, ...
著者Long, S.B, Campbell, E.B, MacKinnon, R.
登録日2005-07-05
公開日2005-07-12
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal structure of a mammalian voltage-dependent Shaker family K+ channel.
Science, 309, 2005
1AGT
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BU of 1agt by Molmil
SOLUTION STRUCTURE OF THE POTASSIUM CHANNEL INHIBITOR AGITOXIN 2: CALIPER FOR PROBING CHANNEL GEOMETRY
分子名称: AGITOXIN 2
著者Krezel, A.M, Kasibhatla, C, Hidalgo, P, Mackinnon, R, Wagner, G.
登録日1995-04-14
公開日1995-07-10
最終更新日2017-11-29
実験手法SOLUTION NMR
主引用文献Solution structure of the potassium channel inhibitor agitoxin 2: caliper for probing channel geometry.
Protein Sci., 4, 1995
8F1D
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BU of 8f1d by Molmil
Voltage-gated potassium channel Kv3.1 apo
分子名称: CHOLESTEROL, POTASSIUM ION, Potassium voltage-gated channel subfamily C member 1, ...
著者Chen, Y, Ishchenko, A.
登録日2022-11-04
公開日2023-10-25
実験手法ELECTRON MICROSCOPY (2.94 Å)
主引用文献Identification and structural and biophysical characterization of a positive modulator of human Kv3.1 channels.
Proc.Natl.Acad.Sci.USA, 120, 2023
8F1C
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BU of 8f1c by Molmil
Voltage-gated potassium channel Kv3.1 with novel positive modulator (9M)-9-{5-chloro-6-[(3,3-dimethyl-2,3-dihydro-1-benzofuran-4-yl)oxy]-4-methylpyridin-3-yl}-2-methyl-7,9-dihydro-8H-purin-8-one (compound 4)
分子名称: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, (9M)-9-{5-chloro-6-[(3,3-dimethyl-2,3-dihydro-1-benzofuran-4-yl)oxy]-4-methylpyridin-3-yl}-2-methyl-7,9-dihydro-8H-purin-8-one, POTASSIUM ION, ...
著者Chen, Y, Ishchenko, A.
登録日2022-11-04
公開日2023-10-25
実験手法ELECTRON MICROSCOPY (2.92 Å)
主引用文献Identification and structural and biophysical characterization of a positive modulator of human Kv3.1 channels.
Proc.Natl.Acad.Sci.USA, 120, 2023
2JK5
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BU of 2jk5 by Molmil
Potassium Channel KcsA in complex with Tetrabutylammonium in high K
分子名称: (2S)-3-HYDROXY-2-(NONANOYLOXY)PROPYL LAURATE, ANTIBODY FAB FRAGMENT HEAVY CHAIN, ANTIBODY FAB FRAGMENT LIGHT CHAIN, ...
著者Lenaeus, M.J, Focia, P.J, Wagner, T, Gross, A.
登録日2008-08-15
公開日2009-11-17
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structures of Kcsa in Complex with Symmetrical Quaternary Ammonium Compounds Reveal a Hydrophobic Binding Site.
Biochemistry, 53, 2014
6U5R
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BU of 6u5r by Molmil
Calcium-bound MthK closed state
分子名称: CALCIUM ION, Calcium-gated potassium channel MthK
著者Fan, C, Nimigean, C.M.
登録日2019-08-28
公開日2020-03-25
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6U5P
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BU of 6u5p by Molmil
Calcium-bound MthK gating ring state 1
分子名称: CALCIUM ION, Calcium-gated potassium channel MthK
著者Fan, C, Nimigean, C.M.
登録日2019-08-28
公開日2020-03-25
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6U68
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BU of 6u68 by Molmil
Calcium-bound MthK open-inactivated state 1
分子名称: Calcium-gated potassium channel MthK
著者Fan, C, Nimigean, C.M.
登録日2019-08-29
公開日2020-03-25
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (4.5 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6U5N
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BU of 6u5n by Molmil
Calcium-bound MthK gating ring state 2
分子名称: CALCIUM ION, Calcium-gated potassium channel MthK
著者Fan, C, Nimigean, C.M.
登録日2019-08-28
公開日2020-03-25
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6U6H
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BU of 6u6h by Molmil
Calcium-bound MthK open-inactivated state 3
分子名称: Calcium-gated potassium channel MthK
著者Chen, F, Crina, N.
登録日2019-08-29
公開日2020-04-22
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (5 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6U6E
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BU of 6u6e by Molmil
Calcium-bound MthK open-inactivated state 2
分子名称: Calcium-gated potassium channel MthK
著者Fan, C, Nimigean, C.M.
登録日2019-08-29
公開日2020-03-25
最終更新日2024-03-20
実験手法ELECTRON MICROSCOPY (6.3 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6UWN
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BU of 6uwn by Molmil
MthK N-terminal truncation RCK domain state 1 bound with calcium
分子名称: CALCIUM ION, Calcium-gated potassium channel MthK
著者Chen, F, Crina, N.
登録日2019-11-05
公開日2020-03-18
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6UX4
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BU of 6ux4 by Molmil
MthK N-terminal truncation RCK domain state 2 bound with calcium
分子名称: CALCIUM ION, Calcium-gated potassium channel MthK
著者Chen, F, Crina, N.
登録日2019-11-06
公開日2020-03-18
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6UXB
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BU of 6uxb by Molmil
MthK N-terminal truncation state 3 bound with calcium
分子名称: Calcium-gated potassium channel MthK
著者Chen, F, Crina, N.
登録日2019-11-07
公開日2020-03-18
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (4.9 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6UXA
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BU of 6uxa by Molmil
MthK N-terminal truncation state 2 bound with calcium
分子名称: Calcium-gated potassium channel MthK
著者Chen, F, Crina, N.
登録日2019-11-07
公開日2020-03-18
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (4.5 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
6UX7
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BU of 6ux7 by Molmil
MthK N-terminal truncation state 1 bound with calcium
分子名称: Calcium-gated potassium channel MthK
著者Chen, F, Crina, N.
登録日2019-11-06
公開日2020-03-18
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (6.7 Å)
主引用文献Ball-and-chain inactivation in a calcium-gated potassium channel.
Nature, 580, 2020
7SQW
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BU of 7sqw by Molmil
Structure of the KcsA-W67F mutant with the activation gate in the closed conformation
分子名称: (1S)-2-HYDROXY-1-[(NONANOYLOXY)METHYL]ETHYL MYRISTATE, Antibody Fragment, KcsA potassium channel, ...
著者Cuello, L.G, Labro, A.J.
登録日2021-11-07
公開日2022-10-12
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (3.21 Å)
主引用文献The nonconducting W434F mutant adopts upon membrane depolarization an inactivated-like state that differs from wild-type Shaker-IR potassium channels.
Sci Adv, 8, 2022
2R9R
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BU of 2r9r by Molmil
Shaker family voltage dependent potassium channel (kv1.2-kv2.1 paddle chimera channel) in association with beta subunit
分子名称: (1R)-2-{[(S)-{[(2S)-2,3-dihydroxypropyl]oxy}(hydroxy)phosphoryl]oxy}-1-[(hexadecanoyloxy)methyl]ethyl (9Z)-octadec-9-enoate, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, POTASSIUM ION, ...
著者Long, S.B, Tao, X, Campbell, E.B, Mackinnon, R.
登録日2007-09-13
公開日2007-11-20
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Atomic structure of a voltage-dependent K+ channel in a lipid membrane-like environment.
Nature, 450, 2007

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