6XXL
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![BU of 6xxl by Molmil](/molmil-images/mine/6xxl) | Crystal Structure of Human Deoxyhypusine Synthase in complex with spermine | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 1,2-ETHANEDIOL, ACETATE ION, ... | 著者 | Wator, E, Wilk, P, Grudnik, P. | 登録日 | 2020-01-27 | 公開日 | 2020-04-15 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.69 Å) | 主引用文献 | Half Way to Hypusine-Structural Basis for Substrate Recognition by Human Deoxyhypusine Synthase. Biomolecules, 10, 2020
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8QND
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![BU of 8qnd by Molmil](/molmil-images/mine/8qnd) | Crystal structure of the ribonucleoside hydrolase C from Lactobacillus reuteri | 分子名称: | CALCIUM ION, Inosine-uridine nucleoside N-ribohydrolase | 著者 | Matyuta, I.O, Minyaev, M.E, Shaposhnikov, L.A, Pometun, E.V, Tishkov, V.I, Popov, V.O, Boyko, K.M. | 登録日 | 2023-09-26 | 公開日 | 2023-12-20 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure-Functional Examination of Novel Ribonucleoside Hydrolase C (RihC) from Limosilactobacillus reuteri LR1. Int J Mol Sci, 25, 2023
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4MD8
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8FVB
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![BU of 8fvb by Molmil](/molmil-images/mine/8fvb) | E coli. CTP synthase in complex with CTP | 分子名称: | CTP synthase, CYTIDINE-5'-TRIPHOSPHATE, MALONIC ACID | 著者 | Holyoak, T, McLeod, M.J, Tran, N. | 登録日 | 2023-01-18 | 公開日 | 2023-05-24 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.03 Å) | 主引用文献 | A metal-dependent conformational change provides a structural basis for the inhibition of CTP synthase by gemcitabine-5'-triphosphate. Protein Sci., 32, 2023
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8FVE
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![BU of 8fve by Molmil](/molmil-images/mine/8fve) | E coli. CTP synthase in complex with CTP (potassium malonate + 100 mM MgCl2) | 分子名称: | CTP synthase, CYTIDINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ... | 著者 | Holyoak, T, McLeod, M.J, Tran, N. | 登録日 | 2023-01-18 | 公開日 | 2023-05-24 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | A metal-dependent conformational change provides a structural basis for the inhibition of CTP synthase by gemcitabine-5'-triphosphate. Protein Sci., 32, 2023
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8FVA
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![BU of 8fva by Molmil](/molmil-images/mine/8fva) | E coli. CTP synthase in complex with F-araCTP | 分子名称: | 4-amino-1-{2-deoxy-2-fluoro-5-O-[(R)-hydroxy{[(R)-hydroxy(phosphonooxy)phosphoryl]oxy}phosphoryl]-beta-D-arabinofuranosyl}pyrimidin-2(1H)-one, CTP synthase, MALONIC ACID, ... | 著者 | Holyoak, T, McLeod, M.J, Tran, N. | 登録日 | 2023-01-18 | 公開日 | 2023-05-24 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | A metal-dependent conformational change provides a structural basis for the inhibition of CTP synthase by gemcitabine-5'-triphosphate. Protein Sci., 32, 2023
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6EB9
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7SMG
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![BU of 7smg by Molmil](/molmil-images/mine/7smg) | Crystal structure of a (p)ppApp hydrolase from Bacteroides caccae | 分子名称: | (p)ppApp hydrolase, 1,2-ETHANEDIOL, CHLORIDE ION, ... | 著者 | Ahmad, S, Alexei, A.G, Tsang, K.K, Trilesky, S, Kim, Y, Whitney, J.C. | 登録日 | 2021-10-25 | 公開日 | 2022-11-09 | 最終更新日 | 2023-05-24 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Identification of a broadly conserved family of enzymes that hydrolyze (p)ppApp. Proc.Natl.Acad.Sci.USA, 120, 2023
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7ZQY
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4PQL
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7ZJE
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![BU of 7zje by Molmil](/molmil-images/mine/7zje) | C16-2 | 分子名称: | Transient receptor potential cation channel subfamily V member 2,Enhanced green fluorescent protein | 著者 | Zhang, L, Gourdon, P, Zygmunt, P.M. | 登録日 | 2022-04-10 | 公開日 | 2023-01-18 | 実験手法 | ELECTRON MICROSCOPY (3.12 Å) | 主引用文献 | Cannabinoid non-cannabidiol site modulation of TRPV2 structure and function. Nat Commun, 13, 2022
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7ZJG
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![BU of 7zjg by Molmil](/molmil-images/mine/7zjg) | Probenecid | 分子名称: | Transient receptor potential cation channel subfamily V member 2 | 著者 | Zhang, L, Gourdon, P, Zygmunt, P.M. | 登録日 | 2022-04-11 | 公開日 | 2023-01-18 | 実験手法 | ELECTRON MICROSCOPY (3.49 Å) | 主引用文献 | Cannabinoid non-cannabidiol site modulation of TRPV2 structure and function. Nat Commun, 13, 2022
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7ZJI
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7ZJH
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![BU of 7zjh by Molmil](/molmil-images/mine/7zjh) | TRPV2-C16+Pro-2 | 分子名称: | Transient receptor potential cation channel subfamily V member 2 | 著者 | Zhang, L, Gourdon, P, Zygmunt, P.M. | 登録日 | 2022-04-11 | 公開日 | 2023-01-18 | 実験手法 | ELECTRON MICROSCOPY (3.39 Å) | 主引用文献 | Cannabinoid non-cannabidiol site modulation of TRPV2 structure and function. Nat Commun, 13, 2022
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7ZJD
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4PNC
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![BU of 4pnc by Molmil](/molmil-images/mine/4pnc) | E. COLI METHIONINE AMINOPEPTIDASE IN COMPLEX WITH INHIBITOR 7-METHOXY-2-METHYLEN-3,4-DIHYDRONAPHTHALEN-1(2H)-ONE | 分子名称: | (2S)-7-methoxy-2-methyl-3,4-dihydronaphthalen-1(2H)-one, COBALT (II) ION, Methionine aminopeptidase, ... | 著者 | Scheidig, A.J, Altmeyer, M, Klein, C.D. | 登録日 | 2014-05-23 | 公開日 | 2014-07-23 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.54 Å) | 主引用文献 | Beta-aminoketones as prodrugs for selective irreversible inhibitors of type-1 methionine aminopeptidases. Bioorg.Med.Chem.Lett., 24, 2014
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4MD7
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4P9O
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4PFN
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![BU of 4pfn by Molmil](/molmil-images/mine/4pfn) | Crystal structure of Plasmodium vivax SHMT with L-serine Schiff base | 分子名称: | CHLORIDE ION, PYRIDOXAL-5'-PHOSPHATE, SERINE, ... | 著者 | Chitnumsub, P, Jaruwat, A, Leartsakulpanich, U. | 登録日 | 2014-04-30 | 公開日 | 2014-12-17 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structures of Plasmodium vivax serine hydroxymethyltransferase: implications for ligand-binding specificity and functional control. Acta Crystallogr.,Sect.D, 70, 2014
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4HRH
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![BU of 4hrh by Molmil](/molmil-images/mine/4hrh) | Crystal Structure of p11-Annexin A2(N-terminal) Fusion Protein in Complex with SMARCA3 Peptide | 分子名称: | Helicase-like transcription factor, Protein S100-A10, Annexin A2, ... | 著者 | Gao, P, Patel, D.J. | 登録日 | 2012-10-27 | 公開日 | 2013-03-06 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (3.001 Å) | 主引用文献 | SMARCA3, a Chromatin-Remodeling Factor, Is Required for p11-Dependent Antidepressant Action. Cell(Cambridge,Mass.), 152, 2013
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4HRG
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8JJ5
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![BU of 8jj5 by Molmil](/molmil-images/mine/8jj5) | Porcine uroplakin complex | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Tetraspanin, ... | 著者 | Oda, T, Yanagisawa, H, Kikkawa, M. | 登録日 | 2023-05-29 | 公開日 | 2023-06-14 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Cryo-EM elucidates the uroplakin complex structure within liquid-crystalline lipids in the porcine urothelial membrane. Commun Biol, 6, 2023
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4PTA
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![BU of 4pta by Molmil](/molmil-images/mine/4pta) | Structure of MDR initiator | 分子名称: | Replication initiator protein | 著者 | Schumacher, M.A. | 登録日 | 2014-03-10 | 公開日 | 2014-06-25 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.6003 Å) | 主引用文献 | Mechanism of staphylococcal multiresistance plasmid replication origin assembly by the RepA protein. Proc.Natl.Acad.Sci.USA, 111, 2014
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4PFF
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![BU of 4pff by Molmil](/molmil-images/mine/4pff) | Crystal structure of Plasmodium vivax SHMT with PLP Schiff base | 分子名称: | PYRIDOXAL-5'-PHOSPHATE, Serine hydroxymethyltransferase, putative | 著者 | Chitnumsub, P, Jaruwat, A, Leartsakulpanich, U. | 登録日 | 2014-04-29 | 公開日 | 2014-12-17 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structures of Plasmodium vivax serine hydroxymethyltransferase: implications for ligand-binding specificity and functional control. Acta Crystallogr.,Sect.D, 70, 2014
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4PA7
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![BU of 4pa7 by Molmil](/molmil-images/mine/4pa7) | Structure of NavMS pore and C-terminal domain crystallised in presence of channel blocking compound | 分子名称: | DODECAETHYLENE GLYCOL, HEGA-10, Ion transport protein, ... | 著者 | Naylor, C.E, Bagneris, C, Wallace, B.A. | 登録日 | 2014-04-07 | 公開日 | 2014-06-04 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (3.02 Å) | 主引用文献 | Prokaryotic NavMs channel as a structural and functional model for eukaryotic sodium channel antagonism. Proc.Natl.Acad.Sci.USA, 111, 2014
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