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8E96
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Glycine and glutamate bound Human GluN1a-GluN2D NMDA receptor
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, GLUTAMIC ACID, GLYCINE, ...
著者Kang, H, Furukawa, H.
登録日2022-08-26
公開日2022-12-07
最終更新日2022-12-14
実験手法ELECTRON MICROSCOPY (3.38 Å)
主引用文献Structural insights into assembly and function of GluN1-2C, GluN1-2A-2C, and GluN1-2D NMDARs.
Mol.Cell, 82, 2022
8JTP
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BU of 8jtp by Molmil
Crystal structure of apo Enoyl-Acyl Carrier Protein Reductase (FabI) from Klebsiella pneumoniae
分子名称: Enoyl-[acyl-carrier-protein] reductase [NADH], HEXAETHYLENE GLYCOL
著者Biswas, S, Kushwaha, G.S, Suar, M.
登録日2023-06-22
公開日2023-12-06
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structural and Biochemical Studies on Klebsiella Pneumoniae Enoyl-ACP Reductase (FabI) Suggest Flexible Substrate Binding Site.
Protein J., 43, 2024
6CJ9
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Crystal structure of lectin from Dioclea lasiophylla seeds (DlyL) complexed with X-Man
分子名称: 5-bromo-4-chloro-1H-indol-3-yl alpha-D-mannopyranoside, CALCIUM ION, Lectin, ...
著者Pinto-Junior, V.R, Santiago, M.Q, Osterne, V.J.S, Araripe, D.A, Neco, A.H.B, Silva-Filho, J.C, Leal, R.B, Rocha, C.R.C, Nascimento, K.S, Cavada, B.S.
登録日2018-02-26
公開日2018-03-07
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structure of DlyL, a mannose-specific lectin from Dioclea lasiophylla Mart. Ex Benth seeds that display cytotoxic effects against C6 glioma cells.
Int. J. Biol. Macromol., 114, 2018
1TVX
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BU of 1tvx by Molmil
NEUTROPHIL ACTIVATING PEPTIDE-2 VARIANT FORM M6L WITH FIVE ADDITIONAL AMINO TERMINAL RESIDUES (DSDLY)
分子名称: NEUTROPHIL ACTIVATING PEPTIDE 2 VARIANT
著者Malkowski, M.G, Edwards, B.F.P.
登録日1996-11-05
公開日1997-01-11
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献The amino-terminal residues in the crystal structure of connective tissue activating peptide-III (des10) block the ELR chemotactic sequence.
J.Mol.Biol., 266, 1997
1KEV
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BU of 1kev by Molmil
STRUCTURE OF NADP-DEPENDENT ALCOHOL DEHYDROGENASE
分子名称: NADP-DEPENDENT ALCOHOL DEHYDROGENASE, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ZINC ION
著者Korkhin, Y, Frolow, F.
登録日1996-10-21
公開日1997-10-22
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Crystalline alcohol dehydrogenases from the mesophilic bacterium Clostridium beijerinckii and the thermophilic bacterium Thermoanaerobium brockii: preparation, characterization and molecular symmetry.
Acta Crystallogr.,Sect.D, 52, 1996
8R79
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The D2 domain of human DTX3L
分子名称: E3 ubiquitin-protein ligase DTX3L, SULFATE ION
著者Vela-Rodriguez, C, Lehtio, L, Maksimainen, M, Duman, R, Wagner, A, Glumoff, T.
登録日2023-11-24
公開日2023-12-27
実験手法X-RAY DIFFRACTION (2.18 Å)
主引用文献Oligomerisation mediated by the D2 domain of DTX3L is critical for DTX3L-PARP9 reading function of mono-ADP-ribosylated androgen receptor.
Biorxiv, 2023
8EVK
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BU of 8evk by Molmil
Crystal structure of Helicobacter pylori dihydroneopterin aldolase (DHNA)
分子名称: 1,2-ETHANEDIOL, Dihydroneopterin aldolase, PTERINE
著者Shaw, G.X, Cherry, S, Tropea, J.E, Ji, X.
登録日2022-10-20
公開日2023-03-01
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (1.49 Å)
主引用文献Structure of Helicobacter pylori dihydroneopterin aldolase suggests a fragment-based strategy for isozyme-specific inhibitor design.
Curr Res Struct Biol, 5, 2023
2OIE
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BU of 2oie by Molmil
Crystal structure of RS21-C6 core segment RSCUT
分子名称: RS21-C6, SULFATE ION
著者Wu, B, Liu, Y, Zhao, Q, Liao, S, Zhang, J, Bartlam, M, Chen, W, Rao, Z.
登録日2007-01-10
公開日2007-03-06
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal Structure of RS21-C6, Involved in Nucleoside Triphosphate Pyrophosphohydrolysis
J.Mol.Biol., 367, 2007
7LVT
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BU of 7lvt by Molmil
Structure of full-length GluK1 with L-Glu
分子名称: Isoform Glur5-2 of Glutamate receptor ionotropic, kainate 1
著者Meyerson, J.R, Selvakumar, P.
登録日2021-02-26
公開日2021-11-03
最終更新日2021-11-10
実験手法ELECTRON MICROSCOPY (4.6 Å)
主引用文献Structural and compositional diversity in the kainate receptor family.
Cell Rep, 37, 2021
1QHX
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CHLORAMPHENICOL PHOSPHOTRANSFERASE IN COMPLEX WITH ATP FROM STREPTOMYCES VENEZUELAE
分子名称: ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, PROTEIN (CHLORAMPHENICOL PHOSPHOTRANSFERASE)
著者Izard, T.
登録日1999-05-31
公開日2000-06-01
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The Crystal Structures of Chloramphenicol Phosphotransferase Reveal a Novel Inactivation Mechanism
Embo J., 19, 2000
8QUD
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BU of 8qud by Molmil
Cryo-EM Structure of Human Kv3.1 in Complex with Modulator AUT5
分子名称: (5R)-5-ethyl-3-(6-spiro[2H-1-benzofuran-3,1'-cyclopropane]-4-yloxypyridin-3-yl)imidazolidine-2,4-dione, 1,2-DIACYL-SN-GLYCERO-3-PHOSHOCHOLINE, CHOLESTEROL HEMISUCCINATE, ...
著者Chi, G, Mckinley, G, Marsden, B, Pike, A.C.W, Ye, M, Brooke, L.M, Bakshi, S, Lakshminarayana, B, Pilati, N, Marasco, A, Gunthorpe, M, Alvaro, G.S, Large, C.H, Williams, E, Sauer, D.B.
登録日2023-10-16
公開日2024-04-03
実験手法ELECTRON MICROSCOPY (2.5 Å)
主引用文献The binding and mechanism of a positive allosteric modulator of Kv3 channels.
Nat Commun, 15, 2024
5AO2
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Crystal structure of human SAMHD1 (amino acid residues 115-583) R164A variant bound to dGTP
分子名称: 2'-DEOXYGUANOSINE-5'-TRIPHOSPHATE, DEOXYNUCLEOSIDE TRIPHOSPHATE TRIPHOSPHOHYDROLASE SAMHD1, FE (III) ION
著者Schwefel, D, Taylor, I.A.
登録日2015-09-09
公開日2015-10-14
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.966 Å)
主引用文献Phospho-Dependent Regulation of Samhd1 Oligomerisation Couples Catalysis and Restriction.
Plos Pathog., 11, 2015
3TUU
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BU of 3tuu by Molmil
Structure of dihydrodipicolinate synthase from the common grapevine
分子名称: BROMIDE ION, CHLORIDE ION, dihydrodipicolinate synthase
著者Perugini, M.A, Dobson, R.C, Atkinson, S.C.
登録日2011-09-19
公開日2012-07-25
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal, Solution and In silico Structural Studies of Dihydrodipicolinate Synthase from the Common Grapevine.
Plos One, 7, 2012
6R66
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Crystal structure of transthyretin in complex with CHF5075, a flurbiprofen analogue
分子名称: 1-[4-[3,5-bis(chloranyl)phenyl]-3-fluoranyl-phenyl]cyclopropane-1-carboxylic acid, Transthyretin
著者Loconte, V, Menozzi, I, Ferrari, A, Berni, R, Zanotti, G.
登録日2019-03-26
公開日2019-09-11
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Structure-activity relationships of flurbiprofen analogues as stabilizers of the amyloidogenic protein transthyretin.
J.Struct.Biol., 208, 2019
1THA
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BU of 1tha by Molmil
MECHANISM OF MOLECULAR RECOGNITION. STRUCTURAL ASPECTS OF 3,3'-DIIODO-L-THYRONINE BINDING TO HUMAN SERUM TRANSTHYRETIN
分子名称: 3,3'-DEIODO-THYROXINE, TRANSTHYRETIN
著者Wojtczak, A, Luft, J, Cody, V.
登録日1991-11-21
公開日1994-01-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Mechanism of molecular recognition. Structural aspects of 3,3'-diiodo-L-thyronine binding to human serum transthyretin.
J.Biol.Chem., 267, 1992
1QHN
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BU of 1qhn by Molmil
CHLORAMPHENICOL PHOSPHOTRANSFERASE FROM STREPTOMYCES VENEZUELAE
分子名称: CHLORAMPHENICOL PHOSPHOTRANSFERASE, SULFATE ION
著者Izard, T.
登録日1999-05-23
公開日2000-06-07
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献The Crystal Structures of Chloramphenicol Phosphotransferase Reveal a Novel Inactivation Mechanism
Embo J., 19, 2000
5DT5
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BU of 5dt5 by Molmil
Crystal structure of the GH1 beta-glucosidase from Exiguobacterium antarcticum B7 in space group P21
分子名称: Beta-glucosidase, SULFATE ION
著者Zanphorlin, L.M, Giuseppe, P.O, Tonoli, C.C.C, Murakami, M.T.
登録日2015-09-17
公開日2016-04-13
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.24 Å)
主引用文献Oligomerization as a strategy for cold adaptation: Structure and dynamics of the GH1 beta-glucosidase from Exiguobacterium antarcticum B7.
Sci Rep, 6, 2016
1SY7
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Crystal structure of the catalase-1 from Neurospora crassa, native structure at 1.75A resolution.
分子名称: CIS-HEME D HYDROXYCHLORIN GAMMA-SPIROLACTONE, Catalase 1, PROTOPORPHYRIN IX CONTAINING FE
著者Diaz, A, Horjales, E, Rudino-Pinera, E, Arreola, R, Hansberg, W.
登録日2004-04-01
公開日2004-10-12
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Unusual Cys-Tyr covalent bond in a large catalase
J.Mol.Biol., 342, 2004
2H95
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Structure of the Amantadine-Blocked Influenza A M2 Proton Channel Trans-membrane Domain by Solid-state NMR spectroscopy
分子名称: Matrix protein 2
著者Hu, J, Asbury, T, Cross, T.A.
登録日2006-06-08
公開日2007-04-24
最終更新日2024-05-29
実験手法SOLID-STATE NMR
主引用文献Backbone structure of the amantadine-blocked trans-membrane domain m2 proton channel from influenza a virus.
Biophys.J., 92, 2007
1QHS
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BU of 1qhs by Molmil
CHLORAMPHENICOL PHOSPHOTRANSFERASE IN COMPLEX WITH CHLORAMPHENICOL FROM STREPTOMYCES VENEZUELAE
分子名称: CHLORAMPHENICOL, PROTEIN (CHLORAMPHENICOL PHOSPHOTRANSFERASE), SULFATE ION
著者Izard, T.
登録日1999-05-28
公開日2000-06-01
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The Crystal Structures of Chloramphenicol Phosphotransferase Reveal a Novel Inactivation Mechanism
Embo J., 19, 2000
1QHY
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CHLORAMPHENICOL PHOSPHOTRANSFERASE FROM STREPTOMYCES VENEZUELAE IN COMPLEX WITH ATPGAMMAS AND CHLORAMPHENICOL
分子名称: CHLORAMPHENICOL, CHLORAMPHENICOL PHOSPHOTRANSFERASE, MAGNESIUM ION, ...
著者Izard, T.
登録日1999-06-01
公開日2000-06-07
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献The Crystal Structures of Chloramphenicol Phosphotransferase Reveal a Novel Inactivation Mechanism
Embo J., 19, 2000
1DSX
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BU of 1dsx by Molmil
KV1.2 T1 DOMAIN, RESIDUES 33-119, T46V MUTANT
分子名称: PROTEIN (KV1.2 VOLTAGE-GATED POTASSIUM CHANNEL)
著者Minor Jr, D.L, Lin, Y.-F, Mobley, B.C, Avelar, A, Jan, Y.N, Jan, L.Y, Berger, J.M.
登録日2000-01-10
公開日2000-09-20
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献The polar T1 interface is linked to conformational changes that open the voltage-gated potassium channel.
Cell(Cambridge,Mass.), 102, 2000
1M3S
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Crystal structure of YckF from Bacillus subtilis
分子名称: Hypothetical protein yckf
著者Sanishvili, R, Wu, R, Kim, D.E, Collart, F, Joachimiak, A, Midwest Center for Structural Genomics (MCSG)
登録日2002-06-28
公開日2003-01-21
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Crystal structure of Bacillus subtilis YckF: structural and functional evolution.
J.Struct.Biol., 148, 2004
4FXF
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Structure of M2 pyruvate kinase in complex with phenylalanine
分子名称: 1,6-di-O-phosphono-beta-D-fructofuranose, ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
著者Walkinshaw, M.D, Morgan, H.P.
登録日2012-07-03
公開日2013-03-27
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献M2 pyruvate kinase provides a mechanism for nutrient sensing and regulation of cell proliferation.
Proc.Natl.Acad.Sci.USA, 110, 2013
4FXJ
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Structure of M2 pyruvate kinase in complex with phenylalanine
分子名称: PHENYLALANINE, PHOSPHATE ION, Pyruvate kinase isozymes M1/M2
著者Walkinshaw, M.D, Morgan, H.P.
登録日2012-07-03
公開日2013-03-27
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献M2 pyruvate kinase provides a mechanism for nutrient sensing and regulation of cell proliferation.
Proc.Natl.Acad.Sci.USA, 110, 2013

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