3DQ2
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![BU of 3dq2 by Molmil](/molmil-images/mine/3dq2) | |
3DQC
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![BU of 3dqc by Molmil](/molmil-images/mine/3dqc) | |
3DPW
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![BU of 3dpw by Molmil](/molmil-images/mine/3dpw) | |
3DQ4
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![BU of 3dq4 by Molmil](/molmil-images/mine/3dq4) | |
3DQF
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![BU of 3dqf by Molmil](/molmil-images/mine/3dqf) | |
3DQO
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![BU of 3dqo by Molmil](/molmil-images/mine/3dqo) | |
3DPX
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![BU of 3dpx by Molmil](/molmil-images/mine/3dpx) | |
3DQ5
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![BU of 3dq5 by Molmil](/molmil-images/mine/3dq5) | |
3DQE
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![BU of 3dqe by Molmil](/molmil-images/mine/3dqe) | |
3DQI
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![BU of 3dqi by Molmil](/molmil-images/mine/3dqi) | |
3DQU
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![BU of 3dqu by Molmil](/molmil-images/mine/3dqu) | |
3DQJ
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![BU of 3dqj by Molmil](/molmil-images/mine/3dqj) | |
3DQ7
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![BU of 3dq7 by Molmil](/molmil-images/mine/3dq7) | |
3DQK
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![BU of 3dqk by Molmil](/molmil-images/mine/3dqk) | |
3DPZ
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![BU of 3dpz by Molmil](/molmil-images/mine/3dpz) | |
3DQ8
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![BU of 3dq8 by Molmil](/molmil-images/mine/3dq8) | |
1LL9
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![BU of 1ll9 by Molmil](/molmil-images/mine/1ll9) | Crystal Structure Of AmpC beta-Lactamase From E. Coli In Complex With Amoxicillin | 分子名称: | 2-{1-[2-AMINO-2-(4-HYDROXY-PHENYL)-ACETYLAMINO]-2-OXO-ETHYL}-5,5-DIMETHYL-THIAZOLIDINE-4-CARBOXYLIC ACID, beta-lactamase | 著者 | Trehan, I, Morandi, F, Blaszczak, L.C, Shoichet, B.K. | 登録日 | 2002-04-26 | 公開日 | 2002-10-02 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | Using steric hindrance to design new inhibitors of class C beta-lactamases. Chem.Biol., 9, 2002
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2HGW
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![BU of 2hgw by Molmil](/molmil-images/mine/2hgw) | |
2HDK
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![BU of 2hdk by Molmil](/molmil-images/mine/2hdk) | |
8CDQ
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![BU of 8cdq by Molmil](/molmil-images/mine/8cdq) | Plasmodium falciparum Myosin A full-length, post-rigor state complexed to the inhibitor KNX-002 and Mg.ATP-gamma-S | 分子名称: | 1,2-ETHANEDIOL, 1-(4-methoxyphenyl)-~{N}-[(3-thiophen-2-yl-1~{H}-pyrazol-4-yl)methyl]cyclopropan-1-amine, GLYCEROL, ... | 著者 | Moussaoui, D, Robblee, J.P, Robert-Paganin, J, Auguin, D, Fisher, F, Fagnant, P.M, MacFarlane, J.E, Schaletzky, J, Wehri, E, Mueller-Dieckmann, C, Baum, J, Trybus, K.M, Houdusse, A. | 登録日 | 2023-01-31 | 公開日 | 2023-06-21 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.21 Å) | 主引用文献 | Mechanism of small molecule inhibition of Plasmodium falciparum myosin A informs antimalarial drug design. Nat Commun, 14, 2023
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7Z3U
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![BU of 7z3u by Molmil](/molmil-images/mine/7z3u) | Crystal structure of SARS-CoV-2 Main Protease after incubation with Sulfo-Calpeptin | 分子名称: | 3C-like proteinase nsp5, CHLORIDE ION, Calpetin, ... | 著者 | Reinke, P.Y.A, Falke, S, Lieske, J, Ewert, W, Loboda, J, Rahmani Mashhour, A, Hauser, M, Karnicar, K, Usenik, A, Lindic, N, Lach, M, Boehler, H, Beck, T, Cox, R, Chapman, H.N, Hinrichs, W, Turk, D, Guenther, S, Meents, A. | 登録日 | 2022-03-02 | 公開日 | 2023-03-22 | 最終更新日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (1.72 Å) | 主引用文献 | Calpeptin is a potent cathepsin inhibitor and drug candidate for SARS-CoV-2 infections. Commun Biol, 6, 2023
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8SS4
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![BU of 8ss4 by Molmil](/molmil-images/mine/8ss4) | Structure of LBD-TMD of AMPA receptor GluA2 in complex with auxiliary subunits TARP gamma-5 and cornichon-2 (apo state) | 分子名称: | Glutamate receptor 2, Voltage-dependent calcium channel gamma-5 subunit chimera, Protein cornichon homolog 2, ... | 著者 | Yen, L.Y, Gangwar, S.P, Yelshanskaya, M.V, Sobolevsky, A.I. | 登録日 | 2023-05-08 | 公開日 | 2023-09-06 | 最終更新日 | 2023-11-01 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | Modulation of GluA2-gamma 5 synaptic complex desensitization, polyamine block and antiepileptic perampanel inhibition by auxiliary subunit cornichon-2. Nat.Struct.Mol.Biol., 30, 2023
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8SS8
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![BU of 8ss8 by Molmil](/molmil-images/mine/8ss8) | Structure of AMPA receptor GluA2 complex with auxiliary subunit TARP gamma-5 bound to competitive antagonist ZK and antiepileptic drug perampanel (closed state) | 分子名称: | 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 2-(6'-oxo-1'-phenyl[1',6'-dihydro[2,3'-bipyridine]]-5'-yl)benzonitrile, CHOLESTEROL, ... | 著者 | Gangwar, S.P, Yen, L.Y, Yelshanskaya, M.V, Sobolevsky, A.I. | 登録日 | 2023-05-08 | 公開日 | 2023-09-06 | 最終更新日 | 2023-10-25 | 実験手法 | ELECTRON MICROSCOPY (2.81 Å) | 主引用文献 | Modulation of GluA2-gamma 5 synaptic complex desensitization, polyamine block and antiepileptic perampanel inhibition by auxiliary subunit cornichon-2. Nat.Struct.Mol.Biol., 30, 2023
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8SSA
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![BU of 8ssa by Molmil](/molmil-images/mine/8ssa) | Structure of AMPA receptor GluA2 complex with auxiliary subunits TARP gamma-5 and cornichon-2 bound to glutamate and channel blocker spermidine (desensitized state) | 分子名称: | 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, GLUTAMIC ACID, Glutamate receptor 2, ... | 著者 | Gangwar, S.P, Yen, L.Y, Yelshanskaya, M.V, Sobolevsky, A.I. | 登録日 | 2023-05-08 | 公開日 | 2023-09-06 | 最終更新日 | 2023-11-01 | 実験手法 | ELECTRON MICROSCOPY (3.88 Å) | 主引用文献 | Modulation of GluA2-gamma 5 synaptic complex desensitization, polyamine block and antiepileptic perampanel inhibition by auxiliary subunit cornichon-2. Nat.Struct.Mol.Biol., 30, 2023
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8SS5
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![BU of 8ss5 by Molmil](/molmil-images/mine/8ss5) | Structure of LBD-TMD of AMPA receptor GluA2 in complex with auxiliary subunit TARP gamma-5 (apo state) | 分子名称: | Glutamate receptor 2, Voltage-dependent calcium channel gamma-5 subunit chimera, SODIUM ION | 著者 | Yen, L.Y, Gangwar, S.P, Yelshanskaya, M.V, Sobolevsky, A.I. | 登録日 | 2023-05-08 | 公開日 | 2023-09-06 | 最終更新日 | 2023-10-25 | 実験手法 | ELECTRON MICROSCOPY (3.56 Å) | 主引用文献 | Modulation of GluA2-gamma 5 synaptic complex desensitization, polyamine block and antiepileptic perampanel inhibition by auxiliary subunit cornichon-2. Nat.Struct.Mol.Biol., 30, 2023
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