3BSW
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3BSS
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![BU of 3bss by Molmil](/molmil-images/mine/3bss) | PglD from Campylobacter jejuni, NCTC 11168, with native substrate | 分子名称: | Acetyltransferase, UDP-2-acetamido-4-amino-2,4,6-trideoxy-alpha-D-glucopyranose | 著者 | Olivier, N.B, Imperiali, B. | 登録日 | 2007-12-26 | 公開日 | 2008-07-22 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal structure and catalytic mechanism of PglD from Campylobacter jejuni. J.Biol.Chem., 283, 2008
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3CDZ
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![BU of 3cdz by Molmil](/molmil-images/mine/3cdz) | Crystal structure of human factor VIII | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ... | 著者 | Ngo, J.C, Huang, M, Roth, D.A, Furie, B.C, Furie, B. | 登録日 | 2008-02-27 | 公開日 | 2008-04-01 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (3.98 Å) | 主引用文献 | Crystal structure of human factor VIII: implications for the formation of the factor IXa-factor VIIIa complex. Structure, 16, 2008
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3SJM
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3TB2
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![BU of 3tb2 by Molmil](/molmil-images/mine/3tb2) | 1-Cys peroxidoxin from Plasmodium Yoelli | 分子名称: | 1,2-ETHANEDIOL, 1-Cys peroxiredoxin, GLYCEROL, ... | 著者 | Qiu, W, Artz, J.D, Vedadi, M, Sharma, S, Houston, S, Lew, J, Wasney, G, Amani, M, Xu, X, Bray, J, Sundstrom, M, Arrowsmith, C, Edwards, A, Hui, R, Bochkarev, A, Structural Genomics Consortium (SGC) | 登録日 | 2011-08-04 | 公開日 | 2011-10-19 | 最終更新日 | 2018-01-31 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Genome-scale protein expression and structural biology of Plasmodium falciparum and related Apicomplexan organisms. Mol.Biochem.Parasitol., 151, 2007
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3S8Y
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![BU of 3s8y by Molmil](/molmil-images/mine/3s8y) | Bromide soaked structure of an esterase from the oil-degrading bacterium Oleispira antarctica | 分子名称: | BROMIDE ION, Esterase APC40077 | 著者 | Petit, P, Dong, A, Kagan, O, Savchenko, A, Yakunin, A.F. | 登録日 | 2011-05-31 | 公開日 | 2011-06-15 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structure and activity of the cold-active and anion-activated carboxyl esterase OLEI01171 from the oil-degrading marine bacterium Oleispira antarctica. Biochem.J., 445, 2012
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3V62
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![BU of 3v62 by Molmil](/molmil-images/mine/3v62) | Structure of the S. cerevisiae Srs2 C-terminal domain in complex with PCNA conjugated to SUMO on lysine 164 | 分子名称: | ATP-dependent DNA helicase SRS2, N-ETHYLMALEIMIDE, Proliferating cell nuclear antigen, ... | 著者 | Armstrong, A.A, Mohideen, F, Lima, C.D. | 登録日 | 2011-12-18 | 公開日 | 2012-02-29 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Recognition of SUMO-modified PCNA requires tandem receptor motifs in Srs2. Nature, 483, 2012
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3BSY
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3CLD
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![BU of 3cld by Molmil](/molmil-images/mine/3cld) | Ligand binding domain of the glucocorticoid receptor complexed with fluticazone furoate | 分子名称: | (6alpha,11alpha,14beta,16alpha,17alpha)-6,9-difluoro-17-{[(fluoromethyl)sulfanyl]carbonyl}-11-hydroxy-16-methyl-3-oxoan drosta-1,4-dien-17-yl furan-2-carboxylate, Glucocorticoid receptor, Tif2 coactivator motif | 著者 | Shewchuk, L.M, McLay, I, Stewart, E, Biggadike, K.B, Hassell, A.M, Bledsoe, R.K. | 登録日 | 2008-03-18 | 公開日 | 2008-06-24 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.84 Å) | 主引用文献 | X-ray crystal structure of the novel enhanced-affinity glucocorticoid agonist fluticasone furoate in the glucocorticoid receptor-ligand binding domain. J.Med.Chem., 51, 2008
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3DT3
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3DKI
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3DRY
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3DRX
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3DRZ
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1W5R
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![BU of 1w5r by Molmil](/molmil-images/mine/1w5r) | X-ray crystallographic structure of a C70Q Mycobacterium smegmatis N- arylamine Acetyltransferase | 分子名称: | ARYLAMINE N-ACETYLTRANSFERASE | 著者 | Holton, S.J, Sandy, J, Rodrigues-Lima, F, Dupret, J.-M, Bhakta, S, Noble, M.E.M, Sim, E. | 登録日 | 2004-08-09 | 公開日 | 2005-05-11 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Investigation of the Catalytic Triad of Arylamine N-Acetyltransferases: Essential Residues Required for Acetyl Transfer to Arylamines. Biochem.J., 390, 2005
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1WBU
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![BU of 1wbu by Molmil](/molmil-images/mine/1wbu) | Fragment based lead discovery using crystallography | 分子名称: | 5-AMINO-1H-PYRIMIDINE-2,4-DIONE, RIBONUCLEASE | 著者 | Cleasby, A, Hartshorn, M.J, Murray, C.W, Jhoti, H, Tickle, I.J. | 登録日 | 2004-11-05 | 公開日 | 2005-01-27 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Fragment-Based Lead Discovery Using X-Ray Crystallography J.Med.Chem., 48, 2005
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1WAX
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![BU of 1wax by Molmil](/molmil-images/mine/1wax) | Protein tyrosine phosphatase 1B with active site inhibitor | 分子名称: | MAGNESIUM ION, PROTEIN-TYROSINE PHOSPHATASE, [[4-(AMINOMETHYL)PHENYL]AMINO]OXO-ACETIC ACID, | 著者 | Hartshorn, M.J, Murray, C.W, Cleasby, A, Frederickson, M, Tickle, I.J, Jhoti, H. | 登録日 | 2004-10-28 | 公開日 | 2005-01-27 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Fragment-Based Lead Discovery Using X-Ray Crystallography J.Med.Chem., 48, 2005
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1W7H
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![BU of 1w7h by Molmil](/molmil-images/mine/1w7h) | p38 Kinase crystal structure in complex with small molecule inhibitor | 分子名称: | 3-(BENZYLOXY)PYRIDIN-2-AMINE, MITOGEN-ACTIVATED PROTEIN KINASE 14 | 著者 | Jhoti, H, Gill, A, Cleasby, A, Devine, L. | 登録日 | 2004-09-02 | 公開日 | 2005-02-08 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.214 Å) | 主引用文献 | Fragment-Based Lead Discovery Using X-Ray Crystallography J.Med.Chem., 48, 2005
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1WCC
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![BU of 1wcc by Molmil](/molmil-images/mine/1wcc) | Screening for fragment binding by X-ray crystallography | 分子名称: | 2-AMINO-6-CHLOROPYRAZINE, CELL DIVISION PROTEIN KINASE 2 | 著者 | Cleasby, A, O'Reilly, M, Hartshorn, M.J, Murray, C.W, Tickle, I.J, Jhoti, H, Frederickson, M. | 登録日 | 2004-11-12 | 公開日 | 2005-01-27 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Fragment-Based Lead Discovery Using X-Ray Crystallography J.Med.Chem., 48, 2005
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1WBO
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![BU of 1wbo by Molmil](/molmil-images/mine/1wbo) | fragment based p38 inhibitors | 分子名称: | 2-CHLOROPHENOL, MITOGEN-ACTIVATED PROTEIN KINASE 14 | 著者 | Cleasby, A, Devine, L, Gill, A, Jhoti, H. | 登録日 | 2004-11-04 | 公開日 | 2005-01-27 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.16 Å) | 主引用文献 | Fragment-Based Lead Discovery Using X-Ray Crystallography J.Med.Chem., 48, 2005
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1VHH
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![BU of 1vhh by Molmil](/molmil-images/mine/1vhh) | A POTENTIAL CATALYTIC SITE WITHIN THE AMINO-TERMINAL SIGNALLING DOMAIN OF SONIC HEDGEHOG | 分子名称: | SONIC HEDGEHOG, SULFATE ION, ZINC ION | 著者 | Hall, T.M.T, Porter, J.A, Beachy, P.A, Leahy, D.J. | 登録日 | 1995-10-03 | 公開日 | 1996-01-29 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | A potential catalytic site revealed by the 1.7-A crystal structure of the amino-terminal signalling domain of Sonic hedgehog. Nature, 378, 1995
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1TMR
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![BU of 1tmr by Molmil](/molmil-images/mine/1tmr) | THE STRUCTURE OF A 19 RESIDUE FRAGMENT FROM THE C-LOOP OF THE FOURTH EPIDERMAL GROWTH FACTOR-LIKE DOMAIN OF THROMBOMODULIN | 分子名称: | THROMBOMODULIN PRECURSOR | 著者 | Adler, M, Seto, M, Nitecki, D, Light, D.R, Morser, J. | 登録日 | 1994-05-20 | 公開日 | 1995-06-08 | 最終更新日 | 2022-03-02 | 実験手法 | SOLUTION NMR | 主引用文献 | The structure of a 19-residue fragment from the C-loop of the fourth epidermal growth factor-like domain of thrombomodulin. J.Biol.Chem., 270, 1995
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1UUA
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1U5F
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1UUB
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