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8ETI
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BU of 8eti by Molmil
Fkbp39 associated 60S nascent ribosome State 1
分子名称: 60S ribosomal protein L13, 60S ribosomal protein L14, 60S ribosomal protein L15-A, ...
著者Zhou, X, Bilokapic, S, Deshmukh, A.A, Halic, M.
登録日2022-10-17
公開日2022-11-30
最終更新日2024-06-19
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献Chromatin localization of nucleophosmin organizes ribosome biogenesis.
Mol.Cell, 82, 2022
8ETH
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BU of 8eth by Molmil
Ytm1 associated 60S nascent ribosome State 1B
分子名称: 60S ribosomal protein L13, 60S ribosomal protein L14, 60S ribosomal protein L15-A, ...
著者Zhou, X, Bilokapic, S, Deshmukh, A.A, Halic, M.
登録日2022-10-17
公開日2022-11-30
最終更新日2024-06-19
実験手法ELECTRON MICROSCOPY (3.8 Å)
主引用文献Chromatin localization of nucleophosmin organizes ribosome biogenesis.
Mol.Cell, 82, 2022
8EUP
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BU of 8eup by Molmil
Ytm1 associated 60S nascent ribosome State 1A
分子名称: 60S ribosomal protein L13, 60S ribosomal protein L14, 60S ribosomal protein L15-A, ...
著者Zhou, X, Bilokapic, S, Deshmukh, A.A, Halic, M.
登録日2022-10-19
公開日2022-11-30
最終更新日2024-06-19
実験手法ELECTRON MICROSCOPY (3.1 Å)
主引用文献Chromatin localization of nucleophosmin organizes ribosome biogenesis.
Mol.Cell, 82, 2022
8EV3
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BU of 8ev3 by Molmil
Ytm1 associated 60S nascent ribosome (-Fkbp39) State 1B
分子名称: 60S ribosomal protein L13, 60S ribosomal protein L14, 60S ribosomal protein L15-A, ...
著者Zhou, X, Bilokapic, S, Deshmukh, A.A, Halic, M.
登録日2022-10-19
公開日2022-11-30
最終更新日2024-06-19
実験手法ELECTRON MICROSCOPY (3 Å)
主引用文献Chromatin localization of nucleophosmin organizes ribosome biogenesis.
Mol.Cell, 82, 2022
3KKU
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BU of 3kku by Molmil
Cruzain in complex with a non-covalent ligand
分子名称: 1,2-ETHANEDIOL, Cruzipain, N-[2-(1H-benzimidazol-2-yl)ethyl]-2-(2-bromophenoxy)acetamide, ...
著者Ferreira, R.S, Eidam, O, Shoichet, B.K.
登録日2009-11-06
公開日2010-07-07
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.28 Å)
主引用文献Complementarity between a docking and a high-throughput screen in discovering new cruzain inhibitors.
J.Med.Chem., 53, 2010
3N8X
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BU of 3n8x by Molmil
Crystal Structure of Cyclooxygenase-1 in Complex with Nimesulide
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 4-NITRO-2-PHENOXYMETHANESULFONANILIDE, ...
著者Lee, J.Y.
登録日2010-05-28
公開日2010-07-28
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Comparison of Cyclooxygenase-1 Crystal Structures: Cross-Talk between Monomers Comprising Cyclooxygenase-1 Homodimers
Biochemistry, 49, 2010
3PH7
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BU of 3ph7 by Molmil
Crystal structure of Plasmodium vivax putative polyprenyl pyrophosphate synthase in complex with geranylgeranyl diphosphate
分子名称: Farnesyl pyrophosphate synthase, GERANYLGERANYL DIPHOSPHATE
著者Wernimont, A.K, Dunford, J, Lew, J, Zhao, Y, Kozieradzki, I, Cossar, D, Schapiro, M, Bochkarev, A, Arrowsmith, C.H, Bountra, C, Weigelt, J, Edwards, A.M, Hui, R, Artz, J.D, Structural Genomics Consortium (SGC)
登録日2010-11-03
公開日2010-11-17
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Molecular characterization of a novel geranylgeranyl pyrophosphate synthase from Plasmodium parasites.
J.Biol.Chem., 286, 2011
3PHV
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BU of 3phv by Molmil
X-RAY ANALYSIS OF HIV-1 PROTEINASE AT 2.7 ANGSTROMS RESOLUTION CONFIRMS STRUCTURAL HOMOLOGY AMONG RETROVIRAL ENZYMES
分子名称: UNLIGANDED HIV-1 PROTEASE
著者Lapatto, R, Blundell, T.L, Hemmings, A, Wilderspin, A, Wood, S.P, Danley, D.E, Geoghegan, K.F, Hawrylik, S.J, Hobart, P.M.
登録日1991-11-04
公開日1992-01-15
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献X-ray analysis of HIV-1 proteinase at 2.7 A resolution confirms structural homology among retroviral enzymes.
Nature, 342, 1989
4F3T
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BU of 4f3t by Molmil
Human Argonaute-2 - miR-20a complex
分子名称: PHENOL, Protein argonaute-2, RNA (5'-R(P*UP*AP*AP*AP*GP*UP*GP*CP*UP*UP*AP*UP*AP*GP*UP*G*CP*AP*GP*G)-3')
著者Elkayam, E, Kuhn, C.-D, Tocilj, A, Joshua-Tor, L.
登録日2012-05-09
公開日2012-05-30
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献The Structure of Human Argonaute-2 in Complex with miR-20a.
Cell(Cambridge,Mass.), 150, 2012
6WTH
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BU of 6wth by Molmil
Full-length human ENaC ECD
分子名称: 10D4 Fab, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Posert, R, Baconguis, I, Noreng, S, Bharadwaj, A, Houser, A.
登録日2020-05-02
公開日2020-08-12
実験手法ELECTRON MICROSCOPY (3.06 Å)
主引用文献Molecular principles of assembly, activation, and inhibition in epithelial sodium channel.
Elife, 9, 2020
6WM3
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BU of 6wm3 by Molmil
Human V-ATPase in state 2 with SidK and ADP
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, ADENOSINE-5'-DIPHOSPHATE, Renin receptor, ...
著者Wang, L, Wu, H, Fu, T.M.
登録日2020-04-20
公開日2020-11-11
最終更新日2020-11-18
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Structures of a Complete Human V-ATPase Reveal Mechanisms of Its Assembly.
Mol.Cell, 80, 2020
3RC9
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BU of 3rc9 by Molmil
Crystal Structure of the K102A mutant of KijD10, a 3-ketoreductase from Actinomadura kijaniata in complex with TDP-benzene and NADP
分子名称: 5'-O-[(S)-hydroxy{[(S)-hydroxy(phenoxy)phosphoryl]oxy}phosphoryl]thymidine, CHLORIDE ION, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ...
著者Holden, H.M, Kubiak, R.L.
登録日2011-03-30
公開日2011-06-08
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.91 Å)
主引用文献Combined Structural and Functional Investigation of a C-3''-Ketoreductase Involved in the Biosynthesis of dTDP-l-Digitoxose.
Biochemistry, 50, 2011
1EZU
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BU of 1ezu by Molmil
ECOTIN Y69F, D70P BOUND TO D102N TRYPSIN
分子名称: CALCIUM ION, ECOTIN, TRYPSIN II, ...
著者Gillmor, S.A, Takeuchi, T, Yang, S.Q, Craik, C.S, Fletterick, R.J.
登録日2000-05-11
公開日2000-06-23
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Compromise and accommodation in ecotin, a dimeric macromolecular inhibitor of serine proteases.
J.Mol.Biol., 299, 2000
1EZS
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BU of 1ezs by Molmil
CRYSTAL STRUCTURE OF ECOTIN MUTANT M84R, W67A, G68A, Y69A, D70A BOUND TO RAT ANIONIC TRYPSIN II
分子名称: CALCIUM ION, ECOTIN, TRYPSIN II, ...
著者Gillmor, S.A, Takeuchi, T, Yang, S.Q, Craik, C.S, Fletterick, R.J.
登録日2000-05-11
公開日2000-06-23
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Compromise and accommodation in ecotin, a dimeric macromolecular inhibitor of serine proteases.
J.Mol.Biol., 299, 2000
7S4G
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BU of 7s4g by Molmil
Fab fragment bound to the Cter peptide of Ly6G6D
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, GLYCEROL, Lymphocyte antigen 6 complex locus protein G6d, ...
著者Rouge, L, Lupardus, P.
登録日2021-09-08
公開日2022-04-13
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Novel Anti-LY6G6D/CD3 T-Cell-Dependent Bispecific Antibody for the Treatment of Colorectal Cancer.
Mol.Cancer Ther., 21, 2022
8I9P
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BU of 8i9p by Molmil
Cryo-EM structure of a Chaetomium thermophilum pre-60S ribosomal subunit - State Mak16
分子名称: 60S ribosomal protein L13, 60S ribosomal protein L14-like protein, 60S ribosomal protein L16-like protein, ...
著者Lau, B, Huang, Z, Beckmann, R, Hurt, E, Cheng, J.
登録日2023-02-07
公開日2023-05-17
最終更新日2024-05-29
実験手法ELECTRON MICROSCOPY (3 Å)
主引用文献Mechanism of 5S RNP recruitment and helicase-surveilled rRNA maturation during pre-60S biogenesis.
Embo Rep., 24, 2023
7SH4
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BU of 7sh4 by Molmil
CD1a-phosphatidylglycerol binary structure
分子名称: (21R,24R,27S)-24,27,28-trihydroxy-18,24-dioxo-19,23,25-trioxa-24lambda~5~-phosphaoctacosan-21-yl (9Z)-octadec-9-enoate, 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, ...
著者Wegrecki, M, Rossjohn, J.
登録日2021-10-07
公開日2022-10-05
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Staphylococcal phosphatidylglycerol antigens activate human T cells via CD1a.
Nat.Immunol., 24, 2023
2R63
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BU of 2r63 by Molmil
STRUCTURAL ROLE OF A BURIED SALT BRIDGE IN THE 434 REPRESSOR DNA-BINDING DOMAIN, NMR, 20 STRUCTURES
分子名称: REPRESSOR PROTEIN FROM BACTERIOPHAGE 434
著者Pervushin, K.V, Billeter, M, Siegal, G, Wuthrich, K.
登録日1996-11-13
公開日1997-06-16
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Structural role of a buried salt bridge in the 434 repressor DNA-binding domain.
J.Mol.Biol., 264, 1996
3J7P
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BU of 3j7p by Molmil
Structure of the 80S mammalian ribosome bound to eEF2
分子名称: 18S ribosomal RNA, 28S ribosomal RNA, 5.8S ribosomal RNA, ...
著者Voorhees, R.M, Fernandez, I.S, Scheres, S.H.W, Hegde, R.S.
登録日2014-08-01
公開日2014-09-03
最終更新日2018-07-18
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Structure of the Mammalian ribosome-sec61 complex to 3.4 a resolution.
Cell(Cambridge,Mass.), 157, 2014
7EKV
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BU of 7ekv by Molmil
Crystal Structure of human Pin1 complexed with a covalent inhibitor
分子名称: 3,6,9,12,15,18,21-HEPTAOXATRICOSANE-1,23-DIOL, 8-(2-chloroacetyl)-4-((5-phenylfuran-2-yl)methyl)-1-thia-4,8-diazaspiro[4.5]decan-3-one, Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1
著者Liu, L, Li, J.
登録日2021-04-06
公開日2022-02-16
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Computational and Structure-Based Development of High Potent Cell-Active Covalent Inhibitor Targeting the Peptidyl-Prolyl Isomerase NIMA-Interacting-1 (Pin1).
J.Med.Chem., 65, 2022
7EFJ
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BU of 7efj by Molmil
Crystal Structure Analysis of human PIN1
分子名称: 3,6,9,12,15,18,21-HEPTAOXATRICOSANE-1,23-DIOL, 8-(2-chloroacetyl)-4-(furan-2-ylmethyl)-1-thia-4,8-diazaspiro[4.5]decan-3-one, Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1
著者Liu, L, Li, J.
登録日2021-03-21
公開日2022-02-16
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.992 Å)
主引用文献Computational and Structure-Based Development of High Potent Cell-Active Covalent Inhibitor Targeting the Peptidyl-Prolyl Isomerase NIMA-Interacting-1 (Pin1).
J.Med.Chem., 65, 2022
7SUT
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BU of 7sut by Molmil
Light harvesting phycobiliprotein HaPE645 from the cryptophyte Hemiselmis andersenii CCMP644
分子名称: (15,16)-DIHYDROBILIVERDIN (SINGLY LINKED), 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, ...
著者Rathbone, H.W, Michie, K.A, Laos, A.L, Curmi, P.M.G.
登録日2021-11-18
公開日2023-10-25
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.49 Å)
主引用文献Molecular dissection of the soluble photosynthetic antenna from the cryptophyte alga Hemiselmis andersenii.
Commun Biol, 6, 2023
7F0M
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BU of 7f0m by Molmil
Crystal Structure of human Pin1 complexed with a potent covalent inhibitor
分子名称: 3,6,9,12,15,18-HEXAOXAICOSANE-1,20-DIOL, 8-(2-chloranylethanoyl)-4-[(5-naphthalen-1-ylfuran-2-yl)methyl]-1-thia-4,8-diazaspiro[4.5]decan-3-one, Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1
著者Liu, L, Li, J.
登録日2021-06-05
公開日2022-02-16
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Computational and Structure-Based Development of High Potent Cell-Active Covalent Inhibitor Targeting the Peptidyl-Prolyl Isomerase NIMA-Interacting-1 (Pin1).
J.Med.Chem., 65, 2022
3ZMB
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BU of 3zmb by Molmil
Native structure of Farnesyl Pyrophosphate Synthase from Pseudomonas aeruginosa PA01, with bound fragment SPB02696.
分子名称: 3-(2-oxo-1,3-benzoxazol-3(2H)-yl)propanoic acid, CHLORIDE ION, DIMETHYL SULFOXIDE, ...
著者Schmidberger, J.W, Schnell, R, Schneider, G.
登録日2013-02-07
公開日2014-02-26
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural Characterization of Substrate and Inhibitor Binding to Farnesyl Pyrophosphate Synthase from Pseudomonas Aeruginosa
Acta Crystallogr.,Sect.D, 71, 2015
8FKZ
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BU of 8fkz by Molmil
Human nucleolar pre-60S ribosomal subunit (State G)
分子名称: 28S rRNA, 5.8S rRNA, 60S ribosomal protein L12, ...
著者Vanden Broeck, A, Klinge, S.
登録日2022-12-21
公開日2023-07-12
最終更新日2024-06-19
実験手法ELECTRON MICROSCOPY (3.04 Å)
主引用文献Principles of human pre-60 S biogenesis.
Science, 381, 2023

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件を2024-08-14に公開中

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