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3E2H
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Structure of the m67 high-affinity mutant of the 2C TCR in complex with Ld/QL9
分子名称: H-2 class I histocompatibility antigen, L-D alpha chain, M67 TCR beta chain, ...
著者Colf, L.A, Garcia, K.C.
登録日2008-08-05
公開日2008-11-04
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献Distinct CDR3 Conformations in TCRs Determine the Level of Cross-Reactivity for Diverse Antigens, but Not the Docking Orientation
J.Immunol., 181, 2008
3E46
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Crystal structure of ubiquitin-conjugating enzyme E2-25kDa (Huntington interacting protein 2) M172A mutant
分子名称: CALCIUM ION, Ubiquitin-conjugating enzyme E2-25 kDa
著者Hughes, R.C, Wilson, R.C, Flatt, J.W, Meehan, E.J, Ng, J.D, Twigg, P.D.
登録日2008-08-09
公開日2008-08-26
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献Structure of full-length ubiquitin-conjugating enzyme E2-25K (huntingtin-interacting protein 2).
Acta Crystallogr.,Sect.F, 65, 2009
3E28
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H. influenzae beta-carbonic anhydrase, variant Y181F
分子名称: Carbonic anhydrase 2, SULFATE ION, ZINC ION
著者Rowlett, R.S, Lee, J.
登録日2008-08-05
公開日2009-06-02
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Allosteric site variants of Haemophilus influenzae beta-carbonic anhydrase.
Biochemistry, 48, 2009
3E2U
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Crystal structure of the zink-knuckle 2 domain of human CLIP-170 in complex with CAP-Gly domain of human dynactin-1 (p150-GLUED)
分子名称: CAP-Gly domain-containing linker protein 1, Dynactin subunit 1, ZINC ION
著者Weisbrich, A, Honnappa, S, Capitani, G, Steinmetz, M.O.
登録日2008-08-06
公開日2008-08-19
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structure-function relationship of CAP-Gly domains
Nat.Struct.Mol.Biol., 14, 2007
3E3T
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Structure of porcine pancreatic elastase with the magic triangle I3C
分子名称: 5-amino-2,4,6-triiodobenzene-1,3-dicarboxylic acid, Elastase-1, IODIDE ION, ...
著者Beck, T, Gruene, T, Sheldrick, G.M.
登録日2008-08-08
公開日2008-10-28
最終更新日2012-04-11
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献A magic triangle for experimental phasing of macromolecules
Acta Crystallogr.,Sect.D, 64, 2008
3E6L
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BU of 3e6l by Molmil
Structure of murine INOS oxygenase domain with inhibitor AR-C132283
分子名称: 5,6,7,8-TETRAHYDROBIOPTERIN, ETHYL 4-[(4-CHLOROPYRIDIN-2-YL)AMINO]PIPERIDINE-1-CARBOXYLATE, Nitric oxide synthase, ...
著者Garcin, E.D, Arvai, A.S, Rosenfeld, R.J, Kroeger, M.D, Crane, B.R, Andersson, G, Andrews, G, Hamley, P.J, Mallinder, P.R, Nicholls, D.J, St-Gallay, S.A, Tinker, A.C, Gensmantel, N.P, Mete, A, Cheshire, D.R, Connolly, S, Stueh, D.J, Aberg, A, Wallace, A.V, Tainer, J.A, Getzoff, E.D.
登録日2008-08-15
公開日2008-10-07
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Anchored plasticity opens doors for selective inhibitor design in nitric oxide synthase.
Nat.Chem.Biol., 4, 2008
3E3Z
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BU of 3e3z by Molmil
Crystal structure of bovine coupling Factor B bound with phenylarsine oxide
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ATP synthase subunit s, mitochondrial, ...
著者Stroud, R.M, Lee, J.K, Belogrudov, G.I.
登録日2008-08-08
公開日2008-08-26
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structure of bovine mitochondrial factor B at 0.96-A resolution.
Proc.Natl.Acad.Sci.Usa, 105, 2008
3E74
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Crystal structure of E. coli allantoinase with iron ions at the metal center
分子名称: Allantoinase, FE (III) ION
著者Kim, K.
登録日2008-08-17
公開日2009-02-24
最終更新日2021-11-10
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystal structure of metal-dependent allantoinase from Escherichia coli
J.Mol.Biol., 387, 2009
3E45
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Q138F HincII bound to Noncognate DNA (GTGCAC) and Ca2+
分子名称: 5'-D(*DGP*DCP*DCP*DGP*DGP*DTP*DGP*DCP*DAP*DCP*DCP*DGP*DGP*DC)-3', CALCIUM ION, SODIUM ION, ...
著者Horton, N.C, Babic, A.C, Little, E.J, Manohar, V.M.
登録日2008-08-08
公開日2008-08-26
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.78 Å)
主引用文献DNA distortion and specificity in a sequence-specific endonuclease.
J.Mol.Biol., 383, 2008
3E4G
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Crystal structure of bovine coupling Factor B, G28E mutant
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ATP synthase subunit s, mitochondrial, ...
著者Stroud, R.M, Lee, J.K, Belogrudov, G.I.
登録日2008-08-11
公開日2008-08-26
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (0.96 Å)
主引用文献Crystal structure of bovine mitochondrial factor B at 0.96-A resolution.
Proc.Natl.Acad.Sci.Usa, 105, 2008
3E83
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Crystal Structure of the the open NaK channel pore
分子名称: CESIUM ION, Potassium channel protein, SODIUM ION
著者Jiang, Y, Alam, A.
登録日2008-08-19
公開日2008-12-23
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural analysis of ion selectivity in the NaK channel
Nat.Struct.Mol.Biol., 16, 2009
3E88
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Crystal structures of the kinase domain of AKT2 in complex with ATP-competitive inhibitors
分子名称: 4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-6-{[(2R)-2-amino-3-phenylpropyl]oxy}-1-ethyl-1H-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol, Glycogen synthase kinase-3 beta peptide, RAC-beta serine/threonine-protein kinase
著者Concha, N.O, Elkins, P.A, Smallwood, A, Ward, P.
登録日2008-08-19
公開日2008-10-14
最終更新日2021-10-20
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Aminofurazans as potent inhibitors of AKT kinase
Bioorg.Med.Chem.Lett., 19, 2009
3E5H
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BU of 3e5h by Molmil
Crystal Structure of Rab28 GTPase in the Active (GppNHp-bound) Form
分子名称: GLYCEROL, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER, ...
著者Lee, S.H, Baek, K, Li, Y, Dominguez, R.
登録日2008-08-13
公開日2008-08-26
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.499 Å)
主引用文献Large nucleotide-dependent conformational change in Rab28.
Febs Lett., 582, 2008
3E8O
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CRYSTAL STRUCTURE OF A PUTATIVE ANTIBIOTIC BIOSYNTHESIS MONOOXYGENASE (DR_2100) FROM DEINOCOCCUS RADIODURANS AT 1.40 A RESOLUTION
分子名称: 1,2-ETHANEDIOL, UNKNOWN LIGAND, uncharacterized protein with ferredoxin-like fold
著者Joint Center for Structural Genomics (JCSG)
登録日2008-08-20
公開日2008-09-09
最終更新日2023-02-01
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Crystal structure of protein of unknown function with ferredoxin-like fold (NP_295823.1) from DEINOCOCCUS RADIODURANS at 1.40 A resolution
To be published
3E8W
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Crystal Structure of Epiphyas postvittana Takeout 1
分子名称: Takeout-like protein 1, Ubiquinone-8
著者Hamiaux, C, Stanley, D, Greenwood, D.R, Baker, E.N, Newcomb, R.D.
登録日2008-08-20
公開日2008-12-09
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of Epiphyas postvittana takeout 1 with bound ubiquinone supports a role as ligand carriers for takeout proteins in insects
J.Biol.Chem., 284, 2009
3E92
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Crystal Structure of P38 Kinase in Complex with A Biaryl Amide Inhibitor
分子名称: GLYCEROL, Mitogen-activated protein kinase 14, N-cyclopropyl-2',6-dimethyl-4'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-3-carboxamide
著者Somers, D.O, Patel, S.
登録日2008-08-21
公開日2008-09-30
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Kinase array design, back to front: Biaryl amides
Bioorg.Med.Chem.Lett., 18, 2008
3E7I
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BU of 3e7i by Molmil
Structure of murine inos oxygenase domain with inhibitor AR-C94864
分子名称: (2R)-5-FLUORO-2-(2-THIENYL)-1,2-DIHYDROQUINAZOLIN-4-AMINE, 5,6,7,8-TETRAHYDROBIOPTERIN, Nitric oxide synthase, ...
著者Garcin, E.D, Arvai, A.S, Rosenfeld, R.J, Kroeger, M.D, Crane, B.R, Andersson, G, Andrews, G, Hamley, P.J, Mallinder, P.R, Nicholls, D.J, St-Gallay, S.A, Tinker, A.C, Gensmantel, N.P, Mete, A, Cheshire, D.R, Connolly, S, Stuehr, D.J, Aberg, A, Wallace, A.V, Tainer, J.A, Getzoff, E.D.
登録日2008-08-18
公開日2008-10-07
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Anchored plasticity opens doors for selective inhibitor design in nitric oxide synthase.
Nat.Chem.Biol., 4, 2008
3E7T
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BU of 3e7t by Molmil
Structure of murine iNOS oxygenase domain with inhibitor AR-C102222
分子名称: 1-(6-CYANO-3-PYRIDYLCARBONYL)-5',8'-DIFLUOROSPIRO[PIPERIDINE-4,2'(1'H)-QUINAZOLINE]-4'-AMINE, 7,8-DIHYDROBIOPTERIN, Nitric oxide synthase, ...
著者Garcin, E.D, Arvai, A.S, Rosenfeld, R.J, Kroeger, M.D, Crane, B.R, Andersson, G, Andrews, G, Hamley, P.J, Mallinder, P.R, Nicholls, D.J, St-Gallay, S.A, Tinker, A.C, Gensmantel, N.P, Mete, A, Cheshire, D.R, Connolly, S, Stuehr, D.J, Aberg, A, Wallace, A.V, Tainer, J.A, Getzoff, E.D.
登録日2008-08-18
公開日2008-10-07
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Anchored plasticity opens doors for selective inhibitor design in nitric oxide synthase.
Nat.Chem.Biol., 4, 2008
3E8H
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Crystal Structure of the the open NaK channel-K+ complex
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, POTASSIUM ION, Potassium channel protein
著者Jiang, Y, Alam, A.
登録日2008-08-19
公開日2008-12-23
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural analysis of ion selectivity in the NaK channel
Nat.Struct.Mol.Biol., 16, 2009
3E8V
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Crystal structure of a possible transglutaminase-family protein proteolytic fragment from Bacteroides fragilis
分子名称: Possible transglutaminase-family protein, UNKNOWN LIGAND
著者Bonanno, J.B, Rutter, M, Bain, K.T, Hu, S, Romero, R, Smith, D, Wasserman, S, Sauder, J.M, Burley, S.K, Almo, S.C, New York SGX Research Center for Structural Genomics (NYSGXRC)
登録日2008-08-20
公開日2008-09-02
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal structure of a possible transglutaminase-family protein proteolytic fragment from Bacteroides fragilis
To be Published
3E93
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Crystal Structure of P38 Kinase in Complex with A Biaryl Amide Inhibitor
分子名称: 4-methyl-N-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamide, GLYCEROL, Mitogen-activated protein kinase 14
著者Somers, D.O, Patel, S.
登録日2008-08-21
公開日2008-09-30
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Kinase array design, back to front: Biaryl amides
Bioorg.Med.Chem.Lett., 18, 2008
3EC2
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BU of 3ec2 by Molmil
Crystal structure of the DnaC helicase loader
分子名称: ADENOSINE-5'-DIPHOSPHATE, DNA replication protein DnaC, MAGNESIUM ION
著者Mott, M.L, Erzberger, J.P, Coons, M.M, Berger, J.M.
登録日2008-08-28
公開日2008-11-25
最終更新日2017-10-25
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structural synergy and molecular crosstalk between bacterial helicase loaders and replication initiators.
Cell(Cambridge,Mass.), 135, 2008
3ECL
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BU of 3ecl by Molmil
Carbonmonoxy Sperm Whale Myoglobin at 40 K: Laser on
分子名称: CARBON MONOXIDE, Myoglobin, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Tomita, A, Sato, T, Ichiyanagi, K, Nozawa, S, Ichikawa, H, Chollet, M, Kawai, F, Park, S.-Y, Koshihara, S, Adachi, S.
登録日2008-09-01
公開日2009-02-24
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.21 Å)
主引用文献Visualizing breathing motion of internal cavities in concert with ligand migration in myoglobin
Proc.Natl.Acad.Sci.USA, 106, 2009
3EDA
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BU of 3eda by Molmil
Carbonmonoxy Sperm Whale Myoglobin at 100 K: Laser on [150 min]
分子名称: CARBON MONOXIDE, Myoglobin, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Tomita, A, Sato, T, Ichiyanagi, K, Nozawa, S, Ichikawa, H, Chollet, M, Kawai, F, Park, S.-Y, Koshihara, S, Adachi, S.
登録日2008-09-03
公開日2009-02-24
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.21 Å)
主引用文献Visualizing breathing motion of internal cavities in concert with ligand migration in myoglobin
Proc.Natl.Acad.Sci.USA, 106, 2009
3EBU
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Replacement of Val3 in Human Thymidylate Synthase Affects Its Kinetic Properties and Intracellular Stability
分子名称: 1,2-ETHANEDIOL, SULFATE ION, Thymidylate synthase
著者Huang, X, Gibson, L.M, Bell, B.J, Lovelace, L.L, Pena, M.M, Berger, F.G, Berger, S.H.
登録日2008-08-28
公開日2010-03-02
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Replacement of Val3 in human thymidylate synthase affects its kinetic properties and intracellular stability .
Biochemistry, 49, 2010

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