7RK9
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6K2Y
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![BU of 6k2y by Molmil](/molmil-images/mine/6k2y) | Human Galectin-14 | 分子名称: | Placental protein 13-like | 著者 | Su, J. | 登録日 | 2019-05-15 | 公開日 | 2020-06-17 | 最終更新日 | 2021-03-10 | 実験手法 | X-RAY DIFFRACTION (1.57 Å) | 主引用文献 | Structure-function studies of galectin-14, an important effector molecule in embryology. Febs J., 288, 2021
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3QLU
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3QLT
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3OLZ
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4V8M
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![BU of 4v8m by Molmil](/molmil-images/mine/4v8m) | High-resolution cryo-electron microscopy structure of the Trypanosoma brucei ribosome | 分子名称: | 18S RRNA OF THE SMALL RIBOSOMAL SUBUNIT, 40S RIBOSOMAL PROTEIN S10, PUTATIVE, ... | 著者 | Hashem, Y, des Georges, A, Fu, J, Buss, S.N, Jossinet, F, Jobe, A, Zhang, Q, Liao, H.Y, Grassucci, R.A, Bajaj, C, Westhof, E, Madison-Antenucci, S, Frank, J. | 登録日 | 2012-12-09 | 公開日 | 2014-07-09 | 最終更新日 | 2019-12-11 | 実験手法 | ELECTRON MICROSCOPY (5.57 Å) | 主引用文献 | High-Resolution Cryo-Electron Microscopy Structure of the Trypanosoma Brucei Ribosome. Nature, 494, 2013
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8SCB
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![BU of 8scb by Molmil](/molmil-images/mine/8scb) | Terminating ribosome with SRI-41315 | 分子名称: | (2S,4aS)-2-cyclobutyl-10-methyl-3-phenyl-2,10-dihydropyrimido[4,5-b]quinoline-4,5(3H,4aH)-dione, 18S_rRNA, 28S_rRNA, ... | 著者 | Yip, M.C.J, Coelho, J.P.L, Oltion, K, Tauton, J, Shao, S. | 登録日 | 2023-04-05 | 公開日 | 2023-12-27 | 最終更新日 | 2024-07-17 | 実験手法 | ELECTRON MICROSCOPY (2.5 Å) | 主引用文献 | The eRF1 degrader SRI-41315 acts as a molecular glue at the ribosomal decoding center. Nat.Chem.Biol., 20, 2024
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8R6F
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![BU of 8r6f by Molmil](/molmil-images/mine/8r6f) | CryoEM structure of wheat 40S ribosomal subunit, body domain | 分子名称: | 30S ribosomal protein S11, chloroplastic, 30S ribosomal protein S4, ... | 著者 | Kravchenko, O.V, Baymukhametov, T.N, Afonina, Z.A, Vasilenko, K.S. | 登録日 | 2023-11-22 | 公開日 | 2023-12-27 | 最終更新日 | 2024-04-24 | 実験手法 | ELECTRON MICROSCOPY (2.34 Å) | 主引用文献 | High-Resolution Structure and Internal Mobility of a Plant 40S Ribosomal Subunit. Int J Mol Sci, 24, 2023
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3FB4
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1VAX
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![BU of 1vax by Molmil](/molmil-images/mine/1vax) | Crystal Structure of Uricase from Arthrobacter globiformis | 分子名称: | Uric acid oxidase | 著者 | Hossain, M.T, Suzuki, K, Yamamoto, T, Imamura, S, Sekiguchi, T, Takenaka, A. | 登録日 | 2004-02-19 | 公開日 | 2005-06-28 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.99 Å) | 主引用文献 | Crystal Structure of Uricase from Arthrobacter globiformis To be Published
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7YSJ
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6YV7
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8DMB
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![BU of 8dmb by Molmil](/molmil-images/mine/8dmb) | Structure of Desulfovirgula thermocuniculi IsrB (DtIsrB) in complex with omega RNA and target DNA | 分子名称: | MAGNESIUM ION, Ubiquitin-like protein SMT3,IsrB protein,monomeric superfolder Green Fluorescent Protein, non-target DNA, ... | 著者 | Seiichi, H, Kappel, K, Zhang, F. | 登録日 | 2022-07-08 | 公開日 | 2022-10-19 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Structure of the OMEGA nickase IsrB in complex with omega RNA and target DNA. Nature, 610, 2022
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6YV9
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5H7H
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![BU of 5h7h by Molmil](/molmil-images/mine/5h7h) | Crystal structure of the BCL6 BTB domain in complex with F1324(10-13) | 分子名称: | 1,2-ETHANEDIOL, B-cell lymphoma 6 protein, F1324 peptide residues 10-13 | 著者 | Sogabe, S, Ida, K, Lane, W, Snell, G. | 登録日 | 2016-11-18 | 公開日 | 2016-12-07 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Discovery of high-affinity BCL6-binding peptide and its structure-activity relationship. Biochem. Biophys. Res. Commun., 482, 2017
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5H8O
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![BU of 5h8o by Molmil](/molmil-images/mine/5h8o) | Crystal structure of an ASC-binding nanobody in complex with the CARD domain of ASC | 分子名称: | Apoptosis-associated speck-like protein containing a CARD, VHH nanobody | 著者 | Lu, A, Schmidt, F.I, Ruan, J, Tang, C, Wu, H, Ploegh, H.L. | 登録日 | 2015-12-23 | 公開日 | 2016-04-06 | 最終更新日 | 2016-05-18 | 実験手法 | X-RAY DIFFRACTION (4.206 Å) | 主引用文献 | A single domain antibody fragment that recognizes the adaptor ASC defines the role of ASC domains in inflammasome assembly. J.Exp.Med., 213, 2016
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5H7G
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![BU of 5h7g by Molmil](/molmil-images/mine/5h7g) | Crystal structure of the BCL6 BTB domain in complex with F1324 | 分子名称: | B-cell lymphoma 6 protein, F1324 peptide, SULFATE ION | 著者 | Sogabe, S, Ida, K, Lane, W, Snell, G. | 登録日 | 2016-11-18 | 公開日 | 2016-12-07 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Discovery of high-affinity BCL6-binding peptide and its structure-activity relationship. Biochem. Biophys. Res. Commun., 482, 2017
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5H8D
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![BU of 5h8d by Molmil](/molmil-images/mine/5h8d) | Crystal structure of an ASC binding nanobody | 分子名称: | VHH nanobody | 著者 | Lu, A, Schmidt, F.I, Ruan, J, Tang, C, Wu, H, Ploegh, H.L. | 登録日 | 2015-12-23 | 公開日 | 2016-04-06 | 最終更新日 | 2016-05-18 | 実験手法 | X-RAY DIFFRACTION (1.89 Å) | 主引用文献 | A single domain antibody fragment that recognizes the adaptor ASC defines the role of ASC domains in inflammasome assembly. J.Exp.Med., 213, 2016
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6EI3
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![BU of 6ei3 by Molmil](/molmil-images/mine/6ei3) | Crystal structure of auto inhibited POT family peptide transporter | 分子名称: | (2S)-2,3-DIHYDROXYPROPYL(7Z)-PENTADEC-7-ENOATE, Proton-dependent oligopeptide transporter family protein | 著者 | Newstead, S, Brinth, A, Vogeley, L, Caffrey, M. | 登録日 | 2017-09-17 | 公開日 | 2017-11-22 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Proton movement and coupling in the POT family of peptide transporters. Proc. Natl. Acad. Sci. U.S.A., 114, 2017
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6F62
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6F64
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![BU of 6f64 by Molmil](/molmil-images/mine/6f64) | Crystal structure of the SYCP1 C-terminal back-to-back assembly | 分子名称: | ACETATE ION, Synaptonemal complex protein 1 | 著者 | Dunce, J.M, Millan, C, Uson, I, Davies, O.R. | 登録日 | 2017-12-04 | 公開日 | 2018-06-06 | 最終更新日 | 2020-04-22 | 実験手法 | X-RAY DIFFRACTION (2.493 Å) | 主引用文献 | Structural basis of meiotic chromosome synapsis through SYCP1 self-assembly. Nat. Struct. Mol. Biol., 25, 2018
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6F5X
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7TGR
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![BU of 7tgr by Molmil](/molmil-images/mine/7tgr) | Structure of SARS-CoV-2 main protease in complex with GC376 | 分子名称: | (1R,2S)-2-({N-[(benzyloxy)carbonyl]-L-leucyl}amino)-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonic acid, (1S,2S)-2-({N-[(benzyloxy)carbonyl]-L-leucyl}amino)-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonic acid, 1,2-ETHANEDIOL, ... | 著者 | Esler, M.A, Shi, K, Aihara, H, Harris, R.S. | 登録日 | 2022-01-09 | 公開日 | 2022-05-04 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.68 Å) | 主引用文献 | Gain-of-Signal Assays for Probing Inhibition of SARS-CoV-2 M pro /3CL pro in Living Cells. Mbio, 13, 2022
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4JQ7
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![BU of 4jq7 by Molmil](/molmil-images/mine/4jq7) | Crystal structure of EGFR kinase domain in complex with compound 2a | 分子名称: | (2S)-2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]-2-phenylethanol, Epidermal growth factor receptor | 著者 | Peng, Y.H, Wu, J.S. | 登録日 | 2013-03-20 | 公開日 | 2013-06-19 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.73 Å) | 主引用文献 | Protein Kinase Inhibitor Design by Targeting the Asp-Phe-Gly (DFG) Motif: The Role of the DFG Motif in the Design of Epidermal Growth Factor Receptor Inhibitors J.Med.Chem., 56, 2013
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4JRV
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![BU of 4jrv by Molmil](/molmil-images/mine/4jrv) | Crystal structure of EGFR kinase domain in complex with compound 4c | 分子名称: | 4-(dimethylamino)-N-[3-(4-{[(1S)-2-hydroxy-1-phenylethyl]amino}-6-phenylfuro[2,3-d]pyrimidin-5-yl)phenyl]butanamide, Epidermal growth factor receptor | 著者 | Peng, Y.H, Wu, J.S. | 登録日 | 2013-03-22 | 公開日 | 2013-06-19 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Protein Kinase Inhibitor Design by Targeting the Asp-Phe-Gly (DFG) Motif: The Role of the DFG Motif in the Design of Epidermal Growth Factor Receptor Inhibitors J.Med.Chem., 56, 2013
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