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4NA7
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Factor XIA in complex with the inhibitor 3'-[(2S,4R)-6-carbamimidoyl-4-methyl-4-phenyl-1,2,3,4-tetrahydroquinolin-2-yl]-4-carbamoyl-5'-[(3-methylbutanoyl)amino]biphenyl-2-carboxylic acid
分子名称: 3'-[(2S,4R)-6-carbamimidoyl-4-methyl-4-phenyl-1,2,3,4-tetrahydroquinolin-2-yl]-4-carbamoyl-5'-[(3-methylbutanoyl)amino]biphenyl-2-carboxylic acid, Coagulation factor XI, SULFATE ION
著者Wei, A.
登録日2013-10-21
公開日2014-02-12
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Tetrahydroquinoline Derivatives as Potent and Selective Factor XIa Inhibitors.
J.Med.Chem., 57, 2014
7UY5
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Tetrahymena telomerase with CST
分子名称: Telomerase La-related protein p65, Telomerase RNA, Telomerase associated protein p50, ...
著者He, Y, Song, H, Chan, H, Wang, Y, Liu, B, Susac, L, Zhou, Z.H, Feigon, J.
登録日2022-05-06
公開日2022-07-13
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Structure of Tetrahymena telomerase-bound CST with polymerase alpha-primase.
Nature, 608, 2022
7TH4
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T. thermophilus methylenetetrahydrofolate reductase complex with 5-formyltetrahydrofolate
分子名称: ACETATE ION, CHLORIDE ION, FLAVIN-ADENINE DINUCLEOTIDE, ...
著者Yamada, K, Koutmos, M.
登録日2022-01-10
公開日2023-01-18
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献5-Formyltetrahydrofolate promotes conformational remodeling in a methylenetetrahydrofolate reductase active site and inhibits its activity.
J.Biol.Chem., 299, 2022
7UY7
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Tetrahymena CST with Polymerase alpha-Primase
分子名称: DNA polymerase, Telomerase associated protein p50, Telomerase-associated protein of 19 kDa, ...
著者He, Y, Song, H, Chan, H, Wang, Y, Liu, B, Susac, L, Zhou, Z.H, Feigon, J.
登録日2022-05-06
公開日2022-07-13
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (4.2 Å)
主引用文献Structure of Tetrahymena telomerase-bound CST with polymerase alpha-primase.
Nature, 608, 2022
7UY6
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Tetrahymena telomerase at 2.9 Angstrom resolution
分子名称: Telomerase La-related protein p65, Telomerase RNA, Telomerase associated protein p50, ...
著者He, Y, Song, H, Chan, H, Wang, Y, Liu, B, Susac, L, Zhou, Z.H, Feigon, J.
登録日2022-05-06
公開日2022-07-13
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献Structure of Tetrahymena telomerase-bound CST with polymerase alpha-primase.
Nature, 608, 2022
2CFI
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The hydrolase domain of human 10-FTHFD in complex with 6- formyltetrahydropterin
分子名称: 10-FORMYLTETRAHYDROFOLATE DEHYDROGENASE, 6-FORMYLTETRAHYDROPTERIN, SULFATE ION
著者Kursula, P, Stenmark, P, Arrowsmith, C, Edwards, A, Ehn, M, Graslund, S, Hammarstrom, M, Hallberg, M, Kotenyova, T, Nilsson-Ehle, P, Nordlund, P, Ogg, D.J, Persson, C, Sagemark, J, Schuler, H, Sundstrom, M, Thorsell, A, Weigelt, J.
登録日2006-02-21
公開日2006-03-14
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Structures of the Hydrolase Domain of Human 10-Formyltetrahydrofolate Dehydrogenase and its Complex with a Substrate Analogue.
Acta Crystallogr.,Sect.D, 62, 2006
1V3X
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Factor Xa in complex with the inhibitor 1-[6-methyl-4,5,6,7-tetrahydrothiazolo(5,4-c)pyridin-2-yl] carbonyl-2-carbamoyl-4-(6-chloronaphth-2-ylsulphonyl)piperazine
分子名称: (2R)-4-[(6-CHLORO-2-NAPHTHYL)SULFONYL]-1-[(5-METHYL-4,5,6,7-TETRAHYDRO[1,3]THIAZOLO[5,4-C]PYRIDIN-2-YL)CARBONYL]PIPERAZ INE-2-CARBOXAMIDE, CALCIUM ION, Coagulation factor X, ...
著者Suzuki, M.
登録日2003-11-07
公開日2004-11-07
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Synthesis and conformational analysis of a non-amidine factor Xa inhibitor that incorporates 5-methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine as S4 binding element
J.Med.Chem., 47, 2004
1QJC
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Phosphopantetheine Adenylyltransferase from Escherichia coli in complex with 4'-phosphopantetheine
分子名称: 4'-PHOSPHOPANTETHEINE, PHOSPHOPANTETHEINE ADENYLYLTRANSFERASE, SULFATE ION
著者Izard, T.
登録日1999-06-23
公開日2001-06-27
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.63 Å)
主引用文献The Crystal Structures of Phosphopantetheine Adenylyltransferase with Bound Substrates Reveal the Enzyme'S Catalytic Mechanism
J.Mol.Biol., 315, 2001
1UZI
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C3 EXOENZYME FROM CLOSTRIDIUM BOTULINUM, TETRAGONAL FORM
分子名称: CYCLO-TETRAMETAVANADATE, GLYCEROL, MONO-ADP-RIBOSYLTRANSFERASE C3, ...
著者Evans, H.R, Holloway, D.E, Sutton, J.M, Ayriss, J, Shone, C.C, Acharya, K.R.
登録日2004-03-12
公開日2004-07-29
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.89 Å)
主引用文献C3 Exoenzyme from Clostridium Botulinum: Structure of a Tetragonal Crystal Form and a Reassessment of Nad-Induced Flexure
Acta Crystallogr.,Sect.D, 60, 2004
1H1T
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PHOSPHOPANTETHEINE ADENYLYLTRANSFERASE IN COMPLEX WITH Coenzyme A FROM ESCHERICHIA COLI
分子名称: 4'-PHOSPHOPANTETHEINE, COENZYME A, PHOSPHOPANTETHEINE ADENYLYLTRANSFERASE, ...
著者Izard, T.
登録日2002-07-21
公開日2003-07-07
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.78 Å)
主引用文献A Novel Adenylate Binding Site Confers Phosphopantetheine Adenylyltransferase Interactions with Coenzyme A
J.Bacteriol., 185, 2003
1YYN
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A common binding site for disialyllactose and a tri-peptide in the C-fragment of tetanus neurotoxin
分子名称: N-acetyl-alpha-neuraminic acid-(2-8)-N-acetyl-alpha-neuraminic acid-(2-3)-alpha-D-galactopyranose-(1-4)-beta-D-glucopyranose, Tetanus toxin
著者Seetharaman, J, Eswaramoorthy, S, Kumaran, D, Swaminathan, S.
登録日2005-02-25
公開日2005-03-15
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Common binding site for disialyllactose and tri-peptide in C-fragment of tetanus neurotoxin
Proteins, 61, 2005
1YXW
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A common binding site for disialyllactose and a tri-peptide in the C-fragment of tetanus neurotoxin
分子名称: GLUTAMIC ACID, TRYPTOPHAN, TYROSINE, ...
著者Jayaraman, S, Eswaramoorthy, S, Kumaran, D, Swaminathan, S.
登録日2005-02-22
公開日2005-03-15
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Common binding site for disialyllactose and tri-peptide in C-fragment of tetanus neurotoxin
Proteins, 61, 2005
4X8I
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de novo crystal structure of the Pyrococcus Furiosus TET3 aminopeptidase
分子名称: 10-((2R)-2-HYDROXYPROPYL)-1,4,7,10-TETRAAZACYCLODODECANE 1,4,7-TRIACETIC ACID, CHLORIDE ION, COBALT (II) ION, ...
著者Colombo, M.
登録日2014-12-10
公開日2016-02-10
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Tuned by metals: the TET peptidase activity is controlled by 3 metal binding sites.
Sci Rep, 6, 2016
6WG9
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Crystal structure of tetracycline destructase Tet(X7)
分子名称: FLAVIN-ADENINE DINUCLEOTIDE, Tetracycline destructase Tet(X7)
著者Kumar, H, Tolia, N.H.
登録日2020-04-05
公開日2021-02-10
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献Tetracycline-inactivating enzymes from environmental, human commensal, and pathogenic bacteria cause broad-spectrum tetracycline resistance.
Commun Biol, 3, 2020
7NE6
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Human TET2 in complex with unfavourable DNA substrate.
分子名称: 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, DNA (5'-D(*AP*CP*AP*GP*GP*(5CM)P*GP*CP*CP*TP*G)-3'), ...
著者Rafalski, D, Bochtler, M.
登録日2021-02-03
公開日2022-03-02
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Pronounced sequence specificity of the TET enzyme catalytic domain guides its cellular function.
Sci Adv, 8, 2022
7NE3
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Human TET2 in complex with favourable DNA substrate.
分子名称: 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, DNA (5'-D(*AP*CP*AP*GP*GP*(5CM)P*GP*CP*CP*TP*G)-3'), ...
著者Rafalski, D, Bochtler, M.
登録日2021-02-03
公開日2022-03-02
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.26 Å)
主引用文献Pronounced sequence specificity of the TET enzyme catalytic domain guides its cellular function.
Sci Adv, 8, 2022
4ABZ
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TetR(D) in Complex with Tigecycline and Magnesium, co-crystallized
分子名称: CHLORIDE ION, MAGNESIUM ION, TIGECYCLINE, ...
著者Volkers, G, Hinrichs, W.
登録日2011-12-12
公開日2012-12-26
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.886 Å)
主引用文献TetR(D) in Complex with Tigecycline and Magnesium
To be Published
2NS7
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How an in vitro selected peptide mimics the antibiotic tetracycline to induce TET repressor
分子名称: Tetracycline repressor protein
著者Luckner, S.R, Klotzsche, M, Berens, C, Hillen, W, Muller, Y.A.
登録日2006-11-03
公開日2007-07-24
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献How an agonist peptide mimics the antibiotic tetracycline to induce Tet-repressor
J.Mol.Biol., 368, 2007
4MC9
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HIV protease in complex with AA74
分子名称: (3S)-tetrahydrofuran-3-yl {(2S,3R)-4-[(4R)-7-fluoro-1,1-dioxido-4-(propan-2-yl)-4,5-dihydro-1,2-benzothiazepin-2(3H)-yl]-3-hydroxy-1-phenylbutan-2-yl}carbamate, 1,2-ETHANEDIOL, CHLORIDE ION, ...
著者Ganguly, A.K, Alluri, S.S, Wang, C, Antropow, A, White, A, Caroccia, D, Biswas, D, Kang, E, Zhang, L, Carroll, S.S, Burlein, C, Munshi, V, Orth, P, Strickland, C.
登録日2013-08-21
公開日2014-04-02
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.19 Å)
主引用文献Structural Optimization of Cyclic Sulfonamide based Novel HIV-1 Protease Inhibitors to Pico Molar Affinities guided by X-ray Crystallographic Analysis
Tetrahedron, 2014
4NM6
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Crystal structure of TET2-DNA complex
分子名称: 5'-D(*AP*CP*CP*AP*CP*(5CM)P*GP*GP*TP*GP*GP*T)-3', FE (II) ION, Methylcytosine dioxygenase TET2, ...
著者Hu, L, Li, Z, Cheng, J, Rao, Q, Gong, W, Liu, M, Wang, P, Xu, Y.
登録日2013-11-14
公開日2013-12-18
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.026 Å)
主引用文献Crystal Structure of TET2-DNA Complex: Insight into TET-Mediated 5mC Oxidation.
Cell(Cambridge,Mass.), 155, 2013
2XGC
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Crystal structure of a designed heterodimeric variant T-A(I)B of the tetracycline repressor
分子名称: TETRACYCLINE REPRESSOR PROTEIN CLASS B FROM TRANSPOSON TN10, TETRACYCLINE REPRESSOR PROTEIN CLASS D
著者Stiebritz, M.T, Wengrzik, S, Richter, J.P, Muller, Y.A.
登録日2010-06-03
公開日2010-09-22
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Computational Design of a Chain-Specific Tetracycline Repressor Heterodimer.
J.Mol.Biol., 403, 2010
4MC2
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HIV protease in complex with SA525P
分子名称: (3S)-tetrahydrofuran-3-yl {(2S,3R)-4-[(4R)-4-tert-butyl-7-fluoro-1,1-dioxido-4,5-dihydro-1,2-benzothiazepin-2(3H)-yl]-3-hydroxy-1-phenylbutan-2-yl}carbamate, CHLORIDE ION, Protease
著者Ganguly, A.K, Alluri, S.S, Wang, C, Caroccia, D, Biswas, D, Kang, E, Zhang, L, Carroll, S.S, Burlein, C, Munshi, V, Orth, P, Strickland, C.
登録日2013-08-21
公開日2014-04-02
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献Structural Optimization of Cyclic Sulfonamide based Novel HIV-1 Protease Inhibitors to Pico Molar Affinities guided by X-ray Crystallographic Analysis
Tetrahedron, 2014
4MC1
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HIV protease in complex with SA526P
分子名称: (3S)-tetrahydrofuran-3-yl {(2S,3R)-4-[(4S)-4-tert-butyl-7-fluoro-1,1-dioxido-4,5-dihydro-1,2-benzothiazepin-2(3H)-yl]-3-hydroxy-1-phenylbutan-2-yl}carbamate, CHLORIDE ION, Protease
著者Ganguly, A.K, Alluri, S.S, Wang, C, Antropow, A, White, A, Caroccia, D, Biswas, D, Kang, E, Zhang, L, Carroll, S.S, Burlein, C, Munshi, V, Orth, P, Strickland, C.
登録日2013-08-21
公開日2014-04-02
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.39 Å)
主引用文献Structural Optimization of Cyclic Sulfonamide based Novel HIV-1 Protease Inhibitors to Pico Molar Affinities guided by X-ray Crystallographic Analysis
Tetrahedron, 2014
1ZP4
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Glu28Gln mutant of E. coli Methylenetetrahydrofolate Reductase (oxidized) complex with Methyltetrahydrofolate
分子名称: 5,10-methylenetetrahydrofolate reductase, 5-METHYL-5,6,7,8-TETRAHYDROFOLIC ACID, FLAVIN-ADENINE DINUCLEOTIDE, ...
著者Pejchal, R, Sargeant, R, Ludwig, M.L.
登録日2005-05-16
公開日2005-08-09
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Structures of NADH and CH(3)-H(4)Folate Complexes of Escherichia coli Methylenetetrahydrofolate Reductase Reveal a Spartan Strategy for a Ping-Pong Reaction
Biochemistry, 44, 2005
5FKL
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TetR(D) H100A mutant in complex with anhydrotetracycline and magnesium
分子名称: 5A,6-ANHYDROTETRACYCLINE, CHLORIDE ION, MAGNESIUM ION, ...
著者Werten, S, Schneider, J, Palm, G.J, Hinrichs, W.
登録日2015-10-17
公開日2016-04-06
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Modular Organisation of Inducer Recognition and Allostery in the Tetracycline Repressor
FEBS J., 283, 2016

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