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2DE9
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Crystal structure of porcine pancreatic elastase complexed with Tris after soaking a tris-free solution
分子名称: Elastase-1, SULFATE ION
著者Kinoshita, T, Tada, T.
登録日2006-02-09
公開日2006-07-11
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Tris(hydroxymethyl)aminomethane induces conformational change and crystal-packing contraction of porcine pancreatic elastase.
Acta Crystallogr.,Sect.F, 62, 2006
1VLZ
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BU of 1vlz by Molmil
UNCOUPLED PHOSPHORYLATION AND ACTIVATION IN BACTERIAL CHEMOTAXIS: THE 2.1 ANGSTROM STRUCTURE OF A THREONINE TO ISOLEUCINE MUTANT AT POSITION 87 OF CHEY
分子名称: CHEY
著者Ganguli, S, Wang, H, Matsumura, P, Volz, K.
登録日1995-04-21
公開日1995-07-10
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Uncoupled phosphorylation and activation in bacterial chemotaxis. The 2.1-A structure of a threonine to isoleucine mutant at position 87 of CheY.
J.Biol.Chem., 270, 1995
1VMC
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BU of 1vmc by Molmil
STROMA CELL-DERIVED FACTOR-1ALPHA (SDF-1ALPHA)
分子名称: Stromal cell-derived factor 1
著者Gozansky, E.K, Clore, G.M.
登録日2004-09-20
公開日2005-03-01
最終更新日2023-12-27
実験手法SOLUTION NMR
主引用文献Mapping the binding of the N-terminal extracellular tail of the CXCR4 receptor to stromal cell-derived factor-1alpha.
J.Mol.Biol., 345, 2005
1JTP
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BU of 1jtp by Molmil
Degenerate interfaces in antigen-antibody complexes
分子名称: FORMIC ACID, LYSOZYME C, SODIUM ION, ...
著者Decanniere, K, Transue, T.R, Desmyter, A, Maes, D, Muyldermans, S, Wyns, L.
登録日2001-08-21
公開日2001-12-05
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Degenerate interfaces in antigen-antibody complexes.
J.Mol.Biol., 313, 2001
1JV8
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BU of 1jv8 by Molmil
NMR Structure of BPTI Mutant G37A
分子名称: TRYPSIN INHIBITOR
著者Battiste, J.L, Li, R, Woodward, C.
登録日2001-08-28
公開日2001-09-12
最終更新日2021-10-27
実験手法SOLUTION NMR
主引用文献A highly destabilizing mutation, G37A, of the bovine pancreatic trypsin inhibitor retains the average native conformation but greatly increases local flexibility
Biochemistry, 41, 2002
2DH8
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BU of 2dh8 by Molmil
Solution structure of the N-terminal RNA binding domain in DAZ-associated protein 1
分子名称: DAZ-associated protein 1
著者Arai, S, Tsuda, K, Muto, Y, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-03-23
公開日2006-09-23
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the N-terminal RNA binding domain in DAZ-associated protein 1
To be Published
2DI2
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BU of 2di2 by Molmil
NMR structure of the HIV-2 nucleocapsid protein
分子名称: Nucleocapsid protein p7, ZINC ION
著者Matsui, T, Kodera, Y, Endoh, H, Miyauchi, E, Komatsu, H, Sato, K, Tanaka, T, Kohno, T, Maeda, T.
登録日2006-03-27
公開日2007-03-13
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献RNA Recognition Mechanism of the Minimal Active Domain of the Human Immunodeficiency Virus Type-2 Nucleocapsid Protein
J.Biochem.(Tokyo), 141, 2007
1VEB
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BU of 1veb by Molmil
Crystal Structure of Protein Kinase A in Complex with Azepane Derivative 5
分子名称: (3R,4R)-N-{4-[4-(2-FLUORO-6-HYDROXY-3-METHOXY-BENZOYL)-BENZYLOXY]-AZEPAN-3-YL}-ISONICOTINAMIDE, cAMP-dependent protein kinase inhibitor, alpha form, ...
著者Breitenlechner, C.B, Wegge, T, Berillon, L, Graul, K, Marzenell, K, Friebe, W.-G, Thomas, U, Schumacher, R, Huber, R, Engh, R.A, Masjost, B.
登録日2004-03-29
公開日2005-03-29
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.89 Å)
主引用文献Structure-based optimization of novel azepane derivatives as PKB inhibitors
J.Med.Chem., 47, 2004
1JWN
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BU of 1jwn by Molmil
Crystal Structure of Scapharca inaequivalvis HbI, I114F Mutant Ligated to Carbon Monoxide.
分子名称: CARBON MONOXIDE, Globin I - Ark Shell, PROTOPORPHYRIN IX CONTAINING FE
著者Knapp, J.E, Gibson, Q.H, Cushing, L, Royer Jr, W.E.
登録日2001-09-04
公開日2001-12-18
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Restricting the ligand-linked heme movement in Scapharca dimeric hemoglobin reveals tight coupling between distal and proximal contributions to cooperativity.
Biochemistry, 40, 2001
2DIV
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BU of 2div by Molmil
Solution structure of the RRM domain of TRNA selenocysteine associated protein
分子名称: TRNA selenocysteine associated protein
著者Dang, W, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-03-30
公開日2006-09-30
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the RRM domain of TRNA selenocysteine associated protein
To be Published
1JDO
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BU of 1jdo by Molmil
SPERM WHALE MYOGLOBIN (FERROUS, NITRIC OXIDE BOUND)
分子名称: MYOGLOBIN, NITRIC OXIDE, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Brucker, E.A, Phillips Jr, G.N.
登録日1998-02-10
公開日1998-05-27
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Nitric oxide myoglobin: crystal structure and analysis of ligand geometry.
Proteins, 30, 1998
2XCK
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BU of 2xck by Molmil
Crystal structure of PDK1 in complex with a pyrazoloquinazoline inhibitor
分子名称: 1-METHYL-8-{[4-(4-METHYLPIPERAZIN-1-YL)PHENYL]AMINO}-N-[(2-METHYLPYRIDIN-4-YL)METHYL]-4,5-DIHYDRO-1H-PYRAZOLO[4,3-H]QUINAZOLINE-3-CARBOXAMIDE, 3-PHOSPHOINOSITIDE DEPENDENT PROTEIN KINASE 1, GLYCEROL, ...
著者Angiolini, M, Banfi, P, Casale, E, Casuscelli, F, Fiorelli, C, Saccardo, M.B, Silvagni, M, Zuccotto, F.
登録日2010-04-23
公開日2010-07-28
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structure-Based Optimization of Potent Pdk1 Inhibitors.
Bioorg.Med.Chem.Lett., 20, 2010
1K1A
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BU of 1k1a by Molmil
Crystal structure of the ankyrin repeat domain of Bcl-3: a unique member of the IkappaB protein family
分子名称: B-cell lymphoma 3-encoded protein
著者Michel, F, Soler-Lopez, M, Petosa, C, Cramer, P, Siebenlist, U, Mueller, C.W.
登録日2001-09-24
公開日2001-11-21
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献Crystal structure of the ankyrin repeat domain of Bcl-3: a unique member of the IkappaB protein family.
EMBO J., 20, 2001
1JAH
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BU of 1jah by Molmil
H-RAS P21 PROTEIN MUTANT G12P, COMPLEXED WITH GUANOSINE-5'-[BETA,GAMMA-METHYLENE] TRIPHOSPHATE AND MAGNESIUM
分子名称: C-HA-RAS, MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID GUANYLATE ESTER
著者Schweins, T, Scheffzek, K, Assheuer, R, Wittinghofer, A.
登録日1996-12-15
公開日1997-07-23
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献The role of the metal ion in the p21ras catalysed GTP-hydrolysis: Mn2+ versus Mg2+.
J.Mol.Biol., 266, 1997
2V7O
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BU of 2v7o by Molmil
Crystal structure of human calcium-calmodulin-dependent protein kinase II gamma
分子名称: 1,2-ETHANEDIOL, BISINDOLYLMALEIMIDE IX, CALCIUM/CALMODULIN-DEPENDENT PROTEIN KINASE TYPE II GAMMA CHAIN
著者Pike, A.C.W, Rellos, P, Fedorov, O, Burgess-Brown, N, Shrestha, L, Ugochukwu, E, Pilka, E.S, von Delft, F, Edwards, A, Weigelt, J, Arrowsmith, C.H, Sundstrom, M, Knapp, S.
登録日2007-07-31
公開日2007-09-11
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Structure of the Camkiidelta/Calmodulin Complex Reveals the Molecular Mechanism of Camkii Kinase Activation.
Plos Biol., 8, 2010
2DMO
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BU of 2dmo by Molmil
Refined solution structure of the 1st SH3 domain from human Neutrophil cytosol factor 2 (NCF-2)
分子名称: Neutrophil cytosol factor 2
著者Tochio, N, Chikayama, E, Koshiba, S, Inoue, M, Kigawa, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-04-22
公開日2006-05-02
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the 1st SH3 domain from human Neutrophil cytosol factor 2 (NCF-2)
To be Published
2DMU
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BU of 2dmu by Molmil
Solution structure of the homeobox domain of Homeobox protein goosecoid
分子名称: Homeobox protein goosecoid
著者Ohnishi, S, Sato, M, Koshiba, S, Inoue, M, Kigawa, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-04-24
公開日2006-10-24
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the homeobox domain of Homeobox protein goosecoid
To be Published
1JAI
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BU of 1jai by Molmil
H-RAS P21 PROTEIN MUTANT G12P, COMPLEXED WITH GUANOSINE-5'-[BETA,GAMMA-METHYLENE] TRIPHOSPHATE AND MANGANESE
分子名称: C-HA-RAS, MANGANESE (II) ION, PHOSPHOMETHYLPHOSPHONIC ACID GUANYLATE ESTER
著者Schweins, T, Scheffzek, K, Assheuer, R, Wittinghofer, A.
登録日1996-12-15
公開日1997-07-23
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献The role of the metal ion in the p21ras catalysed GTP-hydrolysis: Mn2+ versus Mg2+.
J.Mol.Biol., 266, 1997
1VG8
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BU of 1vg8 by Molmil
GPPNHP-Bound Rab7
分子名称: MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER, Ras-related protein Rab-7
著者Rak, A, Pylypenko, O, Niculae, A, Pyatkov, K, Goody, R.S, Alexandrov, K.
登録日2004-04-23
公開日2004-07-20
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structure of the Rab7:REP-1 complex: insights into the mechanism of Rab prenylation and choroideremia disease
Cell(Cambridge,Mass.), 117, 2004
2DNU
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BU of 2dnu by Molmil
Solution structure of RSGI RUH-061, a SH3 domain from human
分子名称: SH3 multiple domains 1
著者Ohashi, W, Hirota, H, Nagashima, T, Kurosaki, C, Hayashi, F, Yoshida, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2006-04-26
公開日2006-10-26
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of RSGI RUH-061, a SH3 domain from human
to be published
8K5C
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BU of 8k5c by Molmil
Cryo-EM structure of Acipimox bound human hydroxy-carboxylic acid receptor 2 (Local refinement)
分子名称: 5-methyl-4-oxidanyl-pyrazin-4-ium-2-carboxylic acid, Human hydroxycarboxylic acid receptor 2
著者Park, J.H, Ishimoto, N, Park, S.Y.
登録日2023-07-21
公開日2023-11-22
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.13 Å)
主引用文献Structural basis for ligand recognition and signaling of hydroxy-carboxylic acid receptor 2.
Nat Commun, 14, 2023
8K5D
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BU of 8k5d by Molmil
Cryo-EM structure of GSK256073 bound human hydroxy-carboxylic acid receptor 2 (Local refinement)
分子名称: 8-chloranyl-3-pentyl-7H-purine-2,6-dione, Human hydroxycarboxylic acid receptor 2
著者Park, J.H, Ishimoto, N, Park, S.Y.
登録日2023-07-21
公開日2023-11-22
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.74 Å)
主引用文献Structural basis for ligand recognition and signaling of hydroxy-carboxylic acid receptor 2.
Nat Commun, 14, 2023
8K5B
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BU of 8k5b by Molmil
Cryo-EM structure of niacin bound human hydroxy-carboxylic acid receptor 2 (Local refinement)
分子名称: Human Hydroxycarboxylic acid receptor 2, NICOTINIC ACID
著者Park, J.H, Ishimoto, N, Park, S.Y.
登録日2023-07-21
公開日2023-11-22
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.43 Å)
主引用文献Structural basis for ligand recognition and signaling of hydroxy-carboxylic acid receptor 2.
Nat Commun, 14, 2023
1JSA
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BU of 1jsa by Molmil
MYRISTOYLATED RECOVERIN WITH TWO CALCIUMS BOUND, NMR, 24 STRUCTURES
分子名称: CALCIUM ION, MYRISTIC ACID, RECOVERIN
著者Ames, J.B, Ishima, R, Tanaka, T, Gordon, J.I, Stryer, L, Ikura, M.
登録日1997-06-04
公開日1997-10-15
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献Molecular mechanics of calcium-myristoyl switches.
Nature, 389, 1997
2XBJ
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BU of 2xbj by Molmil
Crystal Structure of Chk2 in complex with an inhibitor
分子名称: 4-FLUORO-2-(4-{[(3S,4R)-4-(1-HYDROXY-1-METHYLETHYL)PYRROLIDIN-3-YL]AMINO}-6,7-DIMETHOXYQUINAZOLIN-2-YL)PHENOL, MAGNESIUM ION, NITRATE ION, ...
著者Anderson, V.E, Walton, M.I, Eve, P.D, Caldwell, J.J, Pearl, L.H, Oliver, A.W, Collins, I, Garrett, M.D.
登録日2010-04-12
公開日2011-01-12
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structure-Based Design of Potent and Selective 2-(Quinazolin-2-Yl)Phenol Inhibitors of Checkpoint Kinase 2.
J.Med.Chem., 54, 2011

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