5SZG
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![BU of 5szg by Molmil](/molmil-images/mine/5szg) | Structure of the bMERB domain of Mical-3 | 分子名称: | DI(HYDROXYETHYL)ETHER, Protein-methionine sulfoxide oxidase MICAL3 | 著者 | Rai, A, Oprisko, A, Campos, J, Fu, Y, Friese, T, Itzen, A, Goody, R.S, Gazdag, E.M, Mueller, M.P. | 登録日 | 2016-08-14 | 公開日 | 2016-08-24 | 最終更新日 | 2017-09-06 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | bMERB domains are bivalent Rab8 family effectors evolved by gene duplication. Elife, 5, 2016
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4YHT
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![BU of 4yht by Molmil](/molmil-images/mine/4yht) | bRaf complexed with an inhibitor | 分子名称: | 3-[(5-chloro-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-N-methyl-4-(morpholin-4-yl)benzenesulfonamide, GLYCEROL, Serine/threonine-protein kinase B-raf | 著者 | Shewchuk, L.M, Lawhorn, B.G. | 登録日 | 2015-02-27 | 公開日 | 2016-03-16 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (3.05 Å) | 主引用文献 | GSK114: A selective inhibitor for elucidating the biological role of TNNI3K. Bioorg.Med.Chem.Lett., 26, 2016
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5JTI
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1SXR
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![BU of 1sxr by Molmil](/molmil-images/mine/1sxr) | Drosophila Peptidoglycan Recognition Protein (PGRP)-SA | 分子名称: | 1,2-ETHANEDIOL, Peptidoglycan recognition protein SA CG11709-PA, SULFATE ION | 著者 | Reiser, J.B, Teyton, L, Wilson, I.A. | 登録日 | 2004-03-31 | 公開日 | 2004-06-29 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.56 Å) | 主引用文献 | Crystal structure of the Drosophila peptidoglycan recognition protein (PGRP)-SA at 1.56 A resolution J.Mol.Biol., 340, 2004
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5SZV
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5T0R
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5JOU
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![BU of 5jou by Molmil](/molmil-images/mine/5jou) | Bacteroides ovatus Xyloglucan PUL GH31 | 分子名称: | 1,2-ETHANEDIOL, Alpha-xylosidase BoGH31A, NICKEL (II) ION | 著者 | Thompson, A.J, Hemsworth, G.R, Stepper, J, Sobala, L.F, Coyle, T, Larsbrink, J, Spadiut, O, Stubbs, K.A, Brumer, H, Davies, G.J. | 登録日 | 2016-05-03 | 公開日 | 2016-08-10 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structural dissection of a complex Bacteroides ovatus gene locus conferring xyloglucan metabolism in the human gut. Open Biology, 6, 2016
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4YOM
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![BU of 4yom by Molmil](/molmil-images/mine/4yom) | Structure of SAD kinase | 分子名称: | 1,2-ETHANEDIOL, Serine/threonine-protein kinase BRSK2 | 著者 | Wu, J.X, Wang, J, Chen, L, Wang, Z.X, Wu, J.W. | 登録日 | 2015-03-12 | 公開日 | 2015-12-16 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.49 Å) | 主引用文献 | Structural insight into the mechanism of synergistic autoinhibition of SAD kinases Nat Commun, 6, 2015
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5JSF
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![BU of 5jsf by Molmil](/molmil-images/mine/5jsf) | Crystal structure of 17beta-hydroxysteroid dehydrogenase 14 S205 variant in complex with NAD. | 分子名称: | 17-beta-hydroxysteroid dehydrogenase 14, CHLORIDE ION, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ... | 著者 | Bertoletti, N, Marchais-Oberwinkler, S, Heine, A, Klebe, G. | 登録日 | 2016-05-08 | 公開日 | 2016-07-13 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.842 Å) | 主引用文献 | New Insights into Human 17 beta-Hydroxysteroid Dehydrogenase Type 14: First Crystal Structures in Complex with a Steroidal Ligand and with a Potent Nonsteroidal Inhibitor. J.Med.Chem., 59, 2016
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3L6C
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![BU of 3l6c by Molmil](/molmil-images/mine/3l6c) | X-ray crystal structure of rat serine racemase in complex with malonate a potent inhibitor | 分子名称: | MALONATE ION, MANGANESE (II) ION, PYRIDOXAL-5'-PHOSPHATE, ... | 著者 | Smith, M.A, Mack, V, Ebneth, A, Moraes, I, Felicetti, B, Wood, M, Schonfeld, D, Mather, O, Cesura, A, Barker, J. | 登録日 | 2009-12-23 | 公開日 | 2010-01-26 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | The structure of mammalian serine racemase: evidence for conformational changes upon inhibitor binding. J.Biol.Chem., 285, 2010
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5SZY
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![BU of 5szy by Molmil](/molmil-images/mine/5szy) | Novel Structural Insights into GDP-Mediated Regulation of Acyl-CoA Thioesterases | 分子名称: | Acyl-CoA hydrolase, CHLORIDE ION, COENZYME A, ... | 著者 | Khandokar, Y.B, Srivastava, P, Forwood, J.K. | 登録日 | 2016-08-15 | 公開日 | 2016-09-14 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structural insights into GDP-mediated regulation of a bacterial acyl-CoA thioesterase. J. Biol. Chem., 292, 2017
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1T2L
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![BU of 1t2l by Molmil](/molmil-images/mine/1t2l) | Three Crystal Structures of Human Coactosin-like Protein | 分子名称: | Coactosin-like protein | 著者 | Liu, L, Wei, Z, Chen, Z, Wang, Y, Gong, W. | 登録日 | 2004-04-22 | 公開日 | 2004-11-23 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Crystal Structure of Human Coactosin-like Protein J.Mol.Biol., 344, 2004
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3LRE
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5T0S
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![BU of 5t0s by Molmil](/molmil-images/mine/5t0s) | Synaptotagmin 1 C2B domain, cadmium-bound | 分子名称: | CADMIUM ION, SODIUM ION, Synaptotagmin-1 | 著者 | Taylor, A.B, Hart, P.J, Igumenova, T.I. | 登録日 | 2016-08-16 | 公開日 | 2017-06-14 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.42 Å) | 主引用文献 | Non-Native Metal Ion Reveals the Role of Electrostatics in Synaptotagmin 1-Membrane Interactions. Biochemistry, 56, 2017
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5K4L
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5JPO
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1T66
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![BU of 1t66 by Molmil](/molmil-images/mine/1t66) | The structure of FAB with intermediate affinity for fluorescein. | 分子名称: | 2-(6-HYDROXY-3-OXO-3H-XANTHEN-9-YL)-BENZOIC ACID, immunoglobulin heavy chain, immunoglobulin light chain | 著者 | Terzyan, S, Ramsland, P.A, Voss Jr, E.W, Herron, J.N, Edmundson, A.B. | 登録日 | 2004-05-05 | 公開日 | 2004-05-18 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Three-dimensional Structures of Idiotypically Related Fabs with Intermediate and High Affinity for Fluorescein. J.Mol.Biol., 339, 2004
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5T4Y
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![BU of 5t4y by Molmil](/molmil-images/mine/5t4y) | Crystal structure of BT1762-1763 | 分子名称: | MAGNESIUM ION, SusC homolog, SusD homolog | 著者 | van den Berg, B. | 登録日 | 2016-08-30 | 公開日 | 2016-12-14 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Structural basis for nutrient acquisition by dominant members of the human gut microbiota. Nature, 541, 2017
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5JTJ
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![BU of 5jtj by Molmil](/molmil-images/mine/5jtj) | USP7CD-CTP in complex with Ubiquitin | 分子名称: | CALCIUM ION, Polyubiquitin-B, Ubiquitin carboxyl-terminal hydrolase 7,Ubiquitin carboxyl-terminal hydrolase 7 | 著者 | Murray, J.M, Rouge, L. | 登録日 | 2016-05-09 | 公開日 | 2016-08-10 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (3.321 Å) | 主引用文献 | Molecular Understanding of USP7 Substrate Recognition and C-Terminal Activation. Structure, 24, 2016
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1TDH
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![BU of 1tdh by Molmil](/molmil-images/mine/1tdh) | Crystal structure of human endonuclease VIII-like 1 (NEIL1) | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, nei endonuclease VIII-like 1 | 著者 | Doublie, S, Bandaru, V, Bond, J.P, Wallace, S.S. | 登録日 | 2004-05-22 | 公開日 | 2004-07-20 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | The crystal structure of human endonuclease VIII-like 1 (NEIL1) reveals a zincless finger motif required for glycosylase activity. Proc.Natl.Acad.Sci.USA, 101, 2004
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5JTV
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![BU of 5jtv by Molmil](/molmil-images/mine/5jtv) | USP7CD-UBL45 in complex with Ubiquitin | 分子名称: | Polyubiquitin-B, Ubiquitin carboxyl-terminal hydrolase 7 | 著者 | Murray, J.M, Rouge, L. | 登録日 | 2016-05-09 | 公開日 | 2016-10-12 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (3.312 Å) | 主引用文献 | Molecular Understanding of USP7 Substrate Recognition and C-Terminal Activation. Structure, 24, 2016
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1AK2
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![BU of 1ak2 by Molmil](/molmil-images/mine/1ak2) | ADENYLATE KINASE ISOENZYME-2 | 分子名称: | ADENYLATE KINASE ISOENZYME-2, SULFATE ION | 著者 | Schlauderer, G.J, Schulz, G.E. | 登録日 | 1995-12-29 | 公開日 | 1996-06-10 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.92 Å) | 主引用文献 | The structure of bovine mitochondrial adenylate kinase: comparison with isoenzymes in other compartments. Protein Sci., 5, 1996
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3L6Y
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![BU of 3l6y by Molmil](/molmil-images/mine/3l6y) | Crystal structure of p120 catenin in complex with E-cadherin | 分子名称: | Catenin delta-1, E-cadherin | 著者 | Ishiyama, N, Lee, S.-H, Liu, S, Li, G.-Y, Smith, M.J, Reichardt, L.F, Ikura, M. | 登録日 | 2009-12-27 | 公開日 | 2010-04-21 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Dynamic and static interactions between p120 catenin and E-cadherin regulate the stability of cell-cell adhesion. Cell(Cambridge,Mass.), 141, 2010
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5UER
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![BU of 5uer by Molmil](/molmil-images/mine/5uer) | BRD4_BD2_A-1359930 | 分子名称: | Bromodomain-containing protein 4, N-[3-(3-methyl-4-oxo-4,5,6,7-tetrahydro-2H-isoindol-1-yl)-4-phenoxyphenyl]methanesulfonamide | 著者 | Park, C.H. | 登録日 | 2017-01-03 | 公開日 | 2017-06-14 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | Complex structure of BRD4_BD2_A-1359930 To Be Published
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5UEW
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![BU of 5uew by Molmil](/molmil-images/mine/5uew) | BRD2 Bromodomain2 with A-1360579 | 分子名称: | Bromodomain-containing protein 2, N-[3-(4-methoxy-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-4-phenoxyphenyl]methanesulfonamide | 著者 | Park, C.H. | 登録日 | 2017-01-03 | 公開日 | 2017-05-10 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.83 Å) | 主引用文献 | Fragment-Based, Structure-Enabled Discovery of Novel Pyridones and Pyridone Macrocycles as Potent Bromodomain and Extra-Terminal Domain (BET) Family Bromodomain Inhibitors. J. Med. Chem., 60, 2017
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