4YGV
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![BU of 4ygv by Molmil](/molmil-images/mine/4ygv) | Reversal Agent for Dabigatran | 分子名称: | GLYCEROL, aDabi-Fab2a heavy chain, aDabi-Fab2a light chain | 著者 | Schiele, F, Nar, H. | 登録日 | 2015-02-26 | 公開日 | 2015-06-17 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.76 Å) | 主引用文献 | Structure-guided residence time optimization of a dabigatran reversal agent. Mabs, 7, 2015
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5NJD
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![BU of 5njd by Molmil](/molmil-images/mine/5njd) | Structure of Interleukin 23 in complex with Briakinumab FAb | 分子名称: | Briakinumab FAb Heavy chain, Briakinumab FAb Light chain, Interleukin-12 subunit beta, ... | 著者 | Bloch, Y, Savvides, S.N. | 登録日 | 2017-03-28 | 公開日 | 2018-01-03 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (3.9 Å) | 主引用文献 | Structural Activation of Pro-inflammatory Human Cytokine IL-23 by Cognate IL-23 Receptor Enables Recruitment of the Shared Receptor IL-12R beta 1. Immunity, 48, 2018
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4YHM
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![BU of 4yhm by Molmil](/molmil-images/mine/4yhm) | Reversal Agent for Dabigatran | 分子名称: | N-[(2-{[(4-carbamimidoylphenyl)amino]methyl}-1-methyl-1H-benzimidazol-5-yl)carbonyl]-N-pyridin-2-yl-beta-alanine, aDabi-Fab2b heavy chain, aDabi-Fab2b light chain | 著者 | Schiele, F, Nar, H. | 登録日 | 2015-02-27 | 公開日 | 2016-01-13 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.16 Å) | 主引用文献 | Structure-guided residence time optimization of a dabigatran reversal agent. Mabs, 7, 2015
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4YHI
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![BU of 4yhi by Molmil](/molmil-images/mine/4yhi) | Reversal Agent for Dabigatran | 分子名称: | N-[(2-{[(4-carbamimidoylphenyl)amino]methyl}-1-methyl-1H-benzimidazol-5-yl)carbonyl]-N-pyridin-2-yl-beta-alanine, aDabi-Fab2a heavy chain, aDabi-Fab2a light chain | 著者 | Schiele, F, Nar, H. | 登録日 | 2015-02-27 | 公開日 | 2016-01-13 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure-guided residence time optimization of a dabigatran reversal agent. Mabs, 7, 2015
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4YHN
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![BU of 4yhn by Molmil](/molmil-images/mine/4yhn) | Dabigatran Reversal Agent | 分子名称: | aDabi-Fab3 heavy chain, aDabi-Fab3 light chain | 著者 | Schiele, F, Nar, H. | 登録日 | 2015-02-27 | 公開日 | 2016-02-10 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.31 Å) | 主引用文献 | Structure-guided residence time optimization of a dabigatran reversal agent. Mabs, 7, 2015
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4YC3
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![BU of 4yc3 by Molmil](/molmil-images/mine/4yc3) | CDK1/CyclinB1/CKS2 Apo | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, Cyclin-dependent kinase 1, Cyclin-dependent kinases regulatory subunit 2, ... | 著者 | Brown, N.R, Korolchuk, S, Martin, M.P, Stanley, W, Moukhametzianov, R, Noble, M.E.M, Endicott, J.A. | 登録日 | 2015-02-19 | 公開日 | 2016-04-20 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | CDK1 structures reveal conserved and unique features of the essential cell cycle CDK. Nat Commun, 6, 2015
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4YHO
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![BU of 4yho by Molmil](/molmil-images/mine/4yho) | Reversal Agent for Dabigatran | 分子名称: | N-[(2-{[(4-carbamimidoylphenyl)amino]methyl}-1-methyl-1H-benzimidazol-5-yl)carbonyl]-N-pyridin-2-yl-beta-alanine, aDabi-Fab3 heavy chain, aDabi-Fab3 light chain | 著者 | Schiele, F, Nar, H. | 登録日 | 2015-02-27 | 公開日 | 2016-01-13 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.82 Å) | 主引用文献 | Structure-guided residence time optimization of a dabigatran reversal agent. Mabs, 7, 2015
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4YHK
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![BU of 4yhk by Molmil](/molmil-images/mine/4yhk) | Reversal Agent for Dabigatran | 分子名称: | GLYCEROL, N-[(2-{[(4-carbamimidoylphenyl)amino]methyl}-1-methyl-1H-benzimidazol-5-yl)carbonyl]-N-pyridin-2-yl-beta-alanine, aDabi-Fab2a heavy chain, ... | 著者 | Schiele, F, Nar, H. | 登録日 | 2015-02-27 | 公開日 | 2016-01-13 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.21 Å) | 主引用文献 | Structure-guided residence time optimization of a dabigatran reversal agent. Mabs, 7, 2015
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4YHL
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![BU of 4yhl by Molmil](/molmil-images/mine/4yhl) | Reversal Agent for Dabigatran | 分子名称: | aDabi-Fab2b heavy chain, aDabi-Fab2b light chain | 著者 | Schiele, F, Nar, H. | 登録日 | 2015-02-27 | 公開日 | 2016-01-13 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.09 Å) | 主引用文献 | Structure-guided residence time optimization of a dabigatran reversal agent. Mabs, 7, 2015
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5QCK
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![BU of 5qck by Molmil](/molmil-images/mine/5qck) | FACTOR XIA IN COMPLEX WITH THE INHIBITOR 4-[[(2~{S},3~{R})-1-[(~{E})-3-[5-chloranyl-2-(1,2,3,4-tetrazol-1-yl)phenyl]prop-2-enoyl]-3-phenyl-pyrrolidin-2-yl]carbonylamino]benzoic acid | 分子名称: | 1,2-ETHANEDIOL, 4-[[(2~{S},3~{R})-1-[(~{E})-3-[5-chloranyl-2-(1,2,3,4-tetrazol-1-yl)phenyl]prop-2-enoyl]-3-phenyl-pyrrolidin-2-yl]carbonylamino]benzoic acid, Coagulation factor XI, ... | 著者 | Sheriff, S. | 登録日 | 2017-08-10 | 公開日 | 2017-11-08 | 最終更新日 | 2018-02-21 | 実験手法 | X-RAY DIFFRACTION (2.64 Å) | 主引用文献 | Discovery of a Parenteral Small Molecule Coagulation Factor XIa Inhibitor Clinical Candidate (BMS-962212). J. Med. Chem., 60, 2017
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5QCM
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![BU of 5qcm by Molmil](/molmil-images/mine/5qcm) | FACTOR XIA IN COMPLEX WITH THE INHIBITOR methyl ~{N}-[4-[[(1~{S})-2-[(~{E})-3-[3-chloranyl-2-fluoranyl-6-(1,2,3,4-tetrazol-1-yl)phenyl]prop-2-enoyl]-3,4-dihydro-1~{H}-isoquinolin-1-yl]carbonylamino]phenyl]carbamate | 分子名称: | 1,2-ETHANEDIOL, Coagulation factor XI, SULFATE ION, ... | 著者 | Sheriff, S. | 登録日 | 2017-08-10 | 公開日 | 2017-11-08 | 最終更新日 | 2018-02-21 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Discovery of a Parenteral Small Molecule Coagulation Factor XIa Inhibitor Clinical Candidate (BMS-962212). J. Med. Chem., 60, 2017
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8B0H
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![BU of 8b0h by Molmil](/molmil-images/mine/8b0h) | 2C9, C5b9-CD59 cryoEM structure | 分子名称: | CD59 glycoprotein, Complement C5, Complement component C6, ... | 著者 | Couves, E.C, Gardner, S, Bubeck, D. | 登録日 | 2022-09-07 | 公開日 | 2023-02-22 | 最終更新日 | 2023-03-01 | 実験手法 | ELECTRON MICROSCOPY (3.3 Å) | 主引用文献 | Structural basis for membrane attack complex inhibition by CD59. Nat Commun, 14, 2023
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9EOQ
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![BU of 9eoq by Molmil](/molmil-images/mine/9eoq) | Cryo-EM Structure of a 1033 Scaffold Base DNA Origami Nanostructure V4 and TBA | 分子名称: | DNA (42-MER), DNA (5'-D(P*AP*TP*AP*TP*AP*GP*CP*GP*TP*GP*GP*AP*AP*GP*T)-3') | 著者 | Ali, K, Georg, K, Volodymyr, M, Johanna, G, Maximilian, N.H, Lukas, K, Simone, C, Hendrik, D. | 登録日 | 2024-03-15 | 公開日 | 2024-04-24 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (7.5 Å) | 主引用文献 | Designing Rigid DNA Origami Templates for Molecular Visualization Using Cryo-EM. Nano Lett., 24, 2024
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9B55
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![BU of 9b55 by Molmil](/molmil-images/mine/9b55) | |
9B58
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![BU of 9b58 by Molmil](/molmil-images/mine/9b58) | |
9B5D
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![BU of 9b5d by Molmil](/molmil-images/mine/9b5d) | |
9B59
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![BU of 9b59 by Molmil](/molmil-images/mine/9b59) | |
9B57
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![BU of 9b57 by Molmil](/molmil-images/mine/9b57) | |
9B5C
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![BU of 9b5c by Molmil](/molmil-images/mine/9b5c) | |
9B5A
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![BU of 9b5a by Molmil](/molmil-images/mine/9b5a) | |
9FEB
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![BU of 9feb by Molmil](/molmil-images/mine/9feb) | |
9B56
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![BU of 9b56 by Molmil](/molmil-images/mine/9b56) | |
9B5B
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![BU of 9b5b by Molmil](/molmil-images/mine/9b5b) | |
9FE6
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![BU of 9fe6 by Molmil](/molmil-images/mine/9fe6) | |
8AW0
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![BU of 8aw0 by Molmil](/molmil-images/mine/8aw0) | |