5K8V
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![BU of 5k8v by Molmil](/molmil-images/mine/5k8v) | Crystal Structure of Mus musculus Protein Arginine Methyltransferase 4 (CARM1 130-487) with CP1 | 分子名称: | 1,2-DIMETHOXYETHANE, 1,2-ETHANEDIOL, 1-(2-METHOXY-ETHOXY)-2-{2-[2-(2-METHOXY-ETHOXY]-ETHOXY}-ETHANE, ... | 著者 | Cura, V, Marechal, N, Mailliot, J, Troffer-Charlier, N, Hassenboehler, P, Wurtz, J.M, Bonnefond, L, Cavarelli, J. | 登録日 | 2016-05-31 | 公開日 | 2016-11-09 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Structural studies of protein arginine methyltransferase 2 reveal its interactions with potential substrates and inhibitors. FEBS J., 284, 2017
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1B1J
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![BU of 1b1j by Molmil](/molmil-images/mine/1b1j) | CRYSTAL STRUCTURE OF HUMAN ANGIOGENIN VARIANT H13A. | 分子名称: | HYDROLASE ANGIOGENIN | 著者 | Leonidas, D.D, Acharya, K.R. | 登録日 | 1998-11-20 | 公開日 | 1999-04-02 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Refined crystal structures of native human angiogenin and two active site variants: implications for the unique functional properties of an enzyme involved in neovascularisation during tumour growth. J.Mol.Biol., 285, 1999
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5KEW
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![BU of 5kew by Molmil](/molmil-images/mine/5kew) | Vibrio parahaemolyticus VtrA/VtrC complex bound to the bile salt taurodeoxycholate | 分子名称: | 1,2-ETHANEDIOL, ACETATE ION, SULFATE ION, ... | 著者 | Tomchick, D.R, Orth, K, Rivera-Cancel, G. | 登録日 | 2016-06-10 | 公開日 | 2016-07-20 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (2.103 Å) | 主引用文献 | Bile salt receptor complex activates a pathogenic type III secretion system. Elife, 5, 2016
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5KHO
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![BU of 5kho by Molmil](/molmil-images/mine/5kho) | Rasip1 RA domain in complex with Rap1B | 分子名称: | GLYCEROL, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER, ... | 著者 | Gingras, A.R. | 登録日 | 2016-06-15 | 公開日 | 2016-10-19 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.78 Å) | 主引用文献 | Structural Basis of Dimeric Rasip1 RA Domain Recognition of the Ras Subfamily of GTP-Binding Proteins. Structure, 24, 2016
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5UIH
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5VAY
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4X3R
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1RJK
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![BU of 1rjk by Molmil](/molmil-images/mine/1rjk) | crystal structure of the rat vitamin D receptor ligand binding domain complexed with 2MD and a synthetic peptide containing the NR2 box of DRIP 205 | 分子名称: | 5-{2-[1-(5-HYDROXY-1,5-DIMETHYL-HEXYL)-7A-METHYL-OCTAHYDRO-INDEN-4-YLIDENE]-ETHYLIDENE}-2-METHYLENE-CYCLOHEXANE-1,3-DIO L, Peroxisome proliferator-activated receptor binding protein, Vitamin D3 receptor | 著者 | Vanhooke, J.L, Benning, M.M, Bauer, C.B, Pike, J.W, DeLuca, H.F. | 登録日 | 2003-11-19 | 公開日 | 2004-04-13 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.99 Å) | 主引用文献 | Molecular Structure of the Rat Vitamin D Receptor Ligand Binding Domain Complexed with 2-Carbon-Substituted Vitamin D(3) Hormone Analogues and a LXXLL-Containing Coactivator Peptide Biochemistry, 43, 2004
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1AQY
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![BU of 1aqy by Molmil](/molmil-images/mine/1aqy) | ESTROGEN SULFOTRANSFERASE WITH PAP | 分子名称: | ADENOSINE-3'-5'-DIPHOSPHATE, ESTROGEN SULFOTRANSFERASE | 著者 | Kakuta, Y, Pedersen, L.G, Carter, C.W, Negishi, M, Pedersen, L.C. | 登録日 | 1997-08-04 | 公開日 | 1998-10-28 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Crystal structure of estrogen sulphotransferase. Nat.Struct.Biol., 4, 1997
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1B7V
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![BU of 1b7v by Molmil](/molmil-images/mine/1b7v) | Structure of the C-553 cytochrome from Bacillus pasteruii to 1.7 A resolution | 分子名称: | HEME C, PROTEIN (CYTOCHROME C-553) | 著者 | Gonzalez, A, Benini, S, Rypniewski, W.R, Wilson, K.S, Ciurli, S. | 登録日 | 1999-01-22 | 公開日 | 2000-03-27 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Crystal structure of oxidized Bacillus pasteurii cytochrome c553 at 0.97-A resolution. Biochemistry, 39, 2000
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5KHM
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![BU of 5khm by Molmil](/molmil-images/mine/5khm) | The first BET bromodomain of BRD4 bound to compound 13 in a bivalent manner | 分子名称: | (3~{R})-4-[2-[4-[1-(3-methoxy-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)piperidin-4-yl]phenoxy]ethyl]-1,3-dimethyl-piperazin-2-one, Bromodomain-containing protein 4, GLYCEROL | 著者 | Patel, J. | 登録日 | 2016-06-15 | 公開日 | 2016-09-21 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.48 Å) | 主引用文献 | Optimization of a Series of Bivalent Triazolopyridazine Based Bromodomain and Extraterminal Inhibitors: The Discovery of (3R)-4-[2-[4-[1-(3-Methoxy-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)-4-piperidyl]phenoxy]ethyl]-1,3-dimethyl-piperazin-2-one (AZD5153). J.Med.Chem., 59, 2016
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3K2A
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![BU of 3k2a by Molmil](/molmil-images/mine/3k2a) | Crystal structure of the homeobox domain of human homeobox protein Meis2 | 分子名称: | ACETATE ION, CHLORIDE ION, Homeobox protein Meis2 | 著者 | Lam, R, Soloveychik, M, Battaile, K.P, Romanov, V, Lam, K, Beletskaya, I, Gordon, E, Pai, E.F, Chirgadze, N.Y. | 登録日 | 2009-09-29 | 公開日 | 2010-10-13 | 最終更新日 | 2017-11-01 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Crystal structure of the homeobox domain of human homeobox protein Meis2 To be Published
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5VCC
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5KB5
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![BU of 5kb5 by Molmil](/molmil-images/mine/5kb5) | Crystal structure of the adenosine kinase from Mus musculus in complex with adenosine and adenosine-diphosphate | 分子名称: | ADENOSINE, ADENOSINE-5'-DIPHOSPHATE, Adenosine kinase, ... | 著者 | Oliveira, R.R, Neto, R.M, Polo, C.C, Tonoli, C.C.C, Murakami, M.T, Franchini, K.G. | 登録日 | 2016-06-02 | 公開日 | 2017-06-07 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystal structure of the adenosine kinase from Mus musculus in complex with adenosine and adenosine-diphosphate To Be Published
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5UIY
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![BU of 5uiy by Molmil](/molmil-images/mine/5uiy) | Structure of Bromodomain from human BAZ1A | 分子名称: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Bromodomain adjacent to zinc finger domain protein 1A | 著者 | Oppikofer, M, Sudhamsu, J. | 登録日 | 2017-01-16 | 公開日 | 2017-07-12 | 最終更新日 | 2024-03-06 | 実験手法 | X-RAY DIFFRACTION (1.687 Å) | 主引用文献 | Non-canonical reader modules of BAZ1A promote recovery from DNA damage. Nat Commun, 8, 2017
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5KD4
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![BU of 5kd4 by Molmil](/molmil-images/mine/5kd4) | Crystal Structure of Murine MHC-I H-2Dd in complex with Murine Beta2-Microglobulin and a Variant of Peptide (PVI10) of HIV gp120 MN Isolate (IGPGRAFYVI) | 分子名称: | Beta-2-microglobulin, H-2 class I histocompatibility antigen, D-D alpha chain, ... | 著者 | Jiang, J, Natarajan, K, Margulies, D. | 登録日 | 2016-06-07 | 公開日 | 2017-10-11 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (3.05 Å) | 主引用文献 | Effects of Cross-Presentation, Antigen Processing, and Peptide Binding in HIV Evasion of T Cell Immunity. J. Immunol., 200, 2018
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1RTF
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5ULF
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3JV3
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1BSA
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3K45
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![BU of 3k45 by Molmil](/molmil-images/mine/3k45) | Alternate Binding Modes Observed for the E- and Z-isomers of 2,4-Diaminofuro[2,3d]pyrimidines as Ternary Complexes with NADPH and Mouse Dihydrofolate Reductase | 分子名称: | 5-[(1Z)-2-(2-methoxyphenyl)prop-1-en-1-yl]furo[2,3-d]pyrimidine-2,4-diamine, Dihydrofolate reductase, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE | 著者 | Cody, V. | 登録日 | 2009-10-05 | 公開日 | 2009-10-13 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Design, synthesis, and X-ray crystal structures of 2,4-diaminofuro[2,3-d]pyrimidines as multireceptor tyrosine kinase and dihydrofolate reductase inhibitors. Bioorg.Med.Chem., 17, 2009
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1BUY
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![BU of 1buy by Molmil](/molmil-images/mine/1buy) | HUMAN ERYTHROPOIETIN, NMR MINIMIZED AVERAGE STRUCTURE | 分子名称: | PROTEIN (ERYTHROPOIETIN) | 著者 | Cheetham, J.C, Smith, D.M, Aoki, K.H, Stevenson, J.L, Hoeffel, T.J, Syed, R.S, Egrie, J, Harvey, T.S. | 登録日 | 1998-09-08 | 公開日 | 1999-09-10 | 最終更新日 | 2023-12-27 | 実験手法 | SOLUTION NMR | 主引用文献 | NMR structure of human erythropoietin and a comparison with its receptor bound conformation. Nat.Struct.Biol., 5, 1998
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1BNJ
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![BU of 1bnj by Molmil](/molmil-images/mine/1bnj) | BARNASE WILDTYPE STRUCTURE AT PH 9.0 | 分子名称: | BARNASE | 著者 | Cameron, A, Henrick, K, Fersht, A.R, Dodson, G, Buckle, A.M. | 登録日 | 1995-05-17 | 公開日 | 1995-09-15 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Crystal structural analysis of mutations in the hydrophobic cores of barnase. J.Mol.Biol., 234, 1993
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5UOY
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![BU of 5uoy by Molmil](/molmil-images/mine/5uoy) | Crystal structure of human PDE1B catalytic domain in complex with inhibitor 16j (6-(4-Methoxybenzyl)-9-((tetrahydro-2H-pyran-4-yl)methyl)-8,9,10,11-tetrahydropyrido[4',3':4,5]thieno[3,2-e][1,2,4]triazolo[1,5-c]pyrimidin-5(6H)-one) | 分子名称: | 6-[(4-methoxyphenyl)methyl]-9-[(oxan-4-yl)methyl]-8,9,10,11-tetrahydropyrido[4',3':4,5]thieno[3,2-e][1,2,4]triazolo[1,5-c]pyrimidin-5(6H)-one, Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B, MAGNESIUM ION, ... | 著者 | Cedervall, E.P, Allerston, C.K, Xu, R, Sridhar, V, Barker, R, Aertgeerts, K. | 登録日 | 2017-02-01 | 公開日 | 2017-04-26 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.82 Å) | 主引用文献 | Discovery of Selective Phosphodiesterase 1 Inhibitors with Memory Enhancing Properties. J. Med. Chem., 60, 2017
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4WFX
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