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4H6Z
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Tubulin acetyltransferase
分子名称: ACETYL COENZYME *A, Alpha-tubulin N-acetyltransferase, PHOSPHATE ION
著者Kizub, L, Szyk, A, Piszczek, G, Roll-Mecak, A.
登録日2012-09-19
公開日2012-11-07
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (2.701 Å)
主引用文献Crystal structures of tubulin acetyltransferase reveal a conserved catalytic core and the plasticity of the essential N terminus.
J.Biol.Chem., 287, 2012
3B3Q
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Crystal structure of a synaptic adhesion complex
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ...
著者Chen, X, Liu, H, Shim, A, Focia, P, He, X.
登録日2007-10-22
公開日2008-01-15
最終更新日2024-10-09
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural basis for synaptic adhesion mediated by neuroligin-neurexin interactions.
Nat.Struct.Mol.Biol., 15, 2008
3B5G
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Crystal Structure of the Unstable and Highly Fibrillogenic PRO7SER Mutant of the Recombinant Variable Domain 6AJL2
分子名称: ACETATE ION, AMYLOID LAMBDA 6 LIGHT CHAIN VARIABLE REGION PIP, GLYCEROL, ...
著者Hernandez-Santoyo, A, Rodriguez-Romero, A.
登録日2007-10-25
公開日2008-11-04
最終更新日2024-10-16
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献A single mutation at the sheet switch region results in conformational changes favoring lambda6 light-chain fibrillogenesis.
J.Mol.Biol., 396, 2010
1R0O
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Crystal Structure of the Heterodimeric Ecdysone Receptor DNA-binding Complex
分子名称: Ecdysone Response Element, Ecdysone receptor, Ultraspiracle protein, ...
著者Devarakonda, S, Harp, J.M, Kim, Y, Ozyhar, A, Rastinejad, F.
登録日2003-09-22
公開日2003-10-21
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.24 Å)
主引用文献Structure of the Heterodimeric Ecdysone Receptor DNA-binding Complex
Embo J., 22, 2003
5DO2
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Complex structure of MERS-RBD bound with 4C2 antibody
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 4C2 heavy chain, 4C2 light chain, ...
著者Li, Y, Wan, Y, Liu, P, Zhao, J, Lu, G, Qi, J, Wang, Q, Lu, X, Wu, Y, Liu, W, Yuen, K.Y, Perlman, S, Gao, G.F, Yan, J.
登録日2015-09-10
公開日2015-10-14
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.409 Å)
主引用文献A humanized neutralizing antibody against MERS-CoV targeting the receptor-binding domain of the spike protein.
Cell Res., 25, 2015
3GQB
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Crystal Structure of the A3B3 complex from V-ATPase
分子名称: V-type ATP synthase alpha chain, V-type ATP synthase beta chain
著者Meher, M, Akimoto, S, Iwata, M, Nagata, K, Hori, Y, Yoshida, M, Yokoyama, S, Iwata, S, Yokoyama, K.
登録日2009-03-24
公開日2009-11-24
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal structure of A(3)B(3) complex of V-ATPase from Thermus thermophilus.
Embo J., 28, 2009
4N5D
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Tailoring Small Molecules for an Allosteric Site on Procaspase-6: Cpd1
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 6-amino-2,8-dimethylpyrido[2,3-d]pyrimidin-7(8H)-one, Caspase-6, ...
著者Murray, J.M, Steffek, M.
登録日2013-10-09
公開日2013-12-18
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.06 Å)
主引用文献Tailoring small molecules for an allosteric site on procaspase-6.
Chemmedchem, 9, 2014
4NBN
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Tailoring Small Molecules for an Allosteric Site on Procaspase-6
分子名称: 2,2'-[pyrimidine-4,6-diylbis(iminomethanediyl)]diphenol, Caspase-6, PHOSPHATE ION
著者Murray, J.M, Steffek, M.
登録日2013-10-23
公開日2013-12-18
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Tailoring small molecules for an allosteric site on procaspase-6.
Chemmedchem, 9, 2014
2ZQY
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T-state structure of allosteric L-lactate dehydrogenase from Lactobacillus casei
分子名称: L-lactate dehydrogenase, NITRATE ION
著者Arai, K, Ishimitsu, T, Fushinobu, S, Uchikoba, H, Matsuzawa, H, Taguchi, H.
登録日2008-08-22
公開日2009-09-08
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Active and inactive state structures of unliganded Lactobacillus casei allosteric L-lactate dehydrogenase.
Proteins, 78, 2010
4N7J
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Tailoring Small Molecules for an Allosteric Site on Procaspase-6
分子名称: 3-(pyrrolidin-1-yl)isoquinolin-1(2H)-one, Caspase-6, PHOSPHATE ION
著者Murray, J.M, Steffek, M.
登録日2013-10-15
公開日2013-12-18
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.673 Å)
主引用文献Tailoring small molecules for an allosteric site on procaspase-6.
Chemmedchem, 9, 2014
3E3B
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Crystal structure of catalytic subunit of human protein kinase CK2alpha prime with a potent indazole-derivative inhibitor
分子名称: Casein kinase II subunit alpha', [1-(6-{6-[(1-methylethyl)amino]-1H-indazol-1-yl}pyrazin-2-yl)-1H-pyrrol-3-yl]acetic acid
著者Kinoshita, T, Nakaniwa, T, Tada, T.
登録日2008-08-07
公開日2009-03-03
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structure of human protein kinase CK2alpha2 with a potent indazole-derivative inhibitor
Acta Crystallogr.,Sect.F, 65, 2009
4NBL
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Tailoring Small Molecules for an Allosteric Site on Procaspase-6
分子名称: 5-fluoro-2-({[3-(pyrimidin-2-yl)pyridin-2-yl]amino}methyl)phenol, Caspase-6, PHOSPHATE ION
著者Murray, J.M, Steffek, M.
登録日2013-10-23
公開日2014-01-01
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.756 Å)
主引用文献Tailoring small molecules for an allosteric site on procaspase-6.
Chemmedchem, 9, 2014
1I9A
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STRUCTURAL STUDIES OF CHOLESTEROL BIOSYNTHESIS: MEVALONATE 5-DIPHOSPHATE DECARBOXYLASE AND ISOPENTENYL DIPHOSPHATE ISOMERASE
分子名称: ISOPENTENYL-DIPHOSPHATE DELTA-ISOMERASE, MANGANESE (II) ION
著者Bonanno, J.B, Edo, C, Eswar, N, Pieper, U, Romanowski, M.J, Ilyin, V, Gerchman, S.E, Kycia, H, Studier, F.W, Sali, A, Burley, S.K, New York SGX Research Center for Structural Genomics (NYSGXRC)
登録日2001-03-18
公開日2001-03-28
最終更新日2021-02-03
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural genomics of enzymes involved in sterol/isoprenoid biosynthesis.
Proc.Natl.Acad.Sci.USA, 98, 2001
2GA5
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yeast frataxin
分子名称: Frataxin homolog, mitochondrial
著者He, Y, Alam, S.L, Proteasa, S.V, Zhang, Y, Lesuisse, E, Dancis, A.
登録日2006-03-07
公開日2006-03-21
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Yeast Frataxin Solution Structure, Iron Binding and Ferrochelatase Interaction
Biochemistry, 43, 2004
4LD0
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T. thermophilus RuvC in complex with Holliday junction substrate
分子名称: Crossover junction endodeoxyribonuclease RuvC, DNA 11-MER, DNA 13-MER, ...
著者Gorecka, K.M, Komorowska, W, Nowotny, M.
登録日2013-06-24
公開日2013-09-04
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.75 Å)
主引用文献Crystal structure of RuvC resolvase in complex with Holliday junction substrate.
Nucleic Acids Res., 41, 2013
4PMI
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Crystal structure of Rev and Rev-response-element RNA complex
分子名称: PHOSPHATE ION, Protein Rev, Rev-Response-Element RNA
著者Jayaraman, B, Crosby, D.C, Homer, C, Ribeiro, I, Mavor, D, Frankel, A.D.
登録日2014-05-21
公開日2014-12-24
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献RNA-directed remodeling of the HIV-1 protein Rev orchestrates assembly of the Rev-Rev response element complex.
Elife, 4, 2014
3WLV
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Thermostable urate oxidase from Bacillus sp. TB-90
分子名称: 8-AZAXANTHINE, CHLORIDE ION, POTASSIUM ION, ...
著者Hibi, T, Hayashi, Y, Itoh, T.
登録日2013-11-14
公開日2014-06-18
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.747 Å)
主引用文献Intersubunit salt bridges with a sulfate anion control subunit dissociation and thermal stabilization of Bacillus sp. TB-90 urate oxidase.
Biochemistry, 53, 2014
2C78
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EF-Tu complexed with a GTP analog and the antibiotic pulvomycin
分子名称: (1S,2S,3E,5E,7E,10S,11S,12S)-12-[(2R,4E,6E,8Z,10R,12E,14E,16Z,18S,19Z)-10,18-DIHYDROXY-12,16,19-TRIMETHYL-11,22-DIOXOOX ACYCLODOCOSA-4,6,8,12,14,16,19-HEPTAEN-2-YL]-2,11-DIHYDROXY-1,10-DIMETHYL-9-OXOTRIDECA-3,5,7-TRIEN-1-YL 6-DEOXY-2,4-DI-O-METHYL-BETA-L-GALACTOPYRANOSIDE, ELONGATION FACTOR TU-A, MAGNESIUM ION, ...
著者Parmeggiani, A, Krab, I.M, Okamura, S, Nielsen, R.C, Nyborg, J, Nissen, P.
登録日2005-11-18
公開日2006-03-16
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Structural basis of the action of pulvomycin and GE2270 A on elongation factor Tu.
Biochemistry, 45, 2006
4N6G
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Tailoring Small Molecules for an Allosteric Site on Procaspase-6
分子名称: 3-(pyrrolidin-1-yl)isoquinolin-1(2H)-one, Caspase-6, PHOSPHATE ION
著者Murray, J.M, Steffek, M.
登録日2013-10-11
公開日2014-01-01
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.142 Å)
主引用文献Tailoring small molecules for an allosteric site on procaspase-6.
Chemmedchem, 9, 2014
4NBK
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Tailoring Small Molecules for an Allosteric Site on Procaspase-6
分子名称: 2-{[(3-methylpyridin-2-yl)amino]methyl}phenol, Caspase-6, PHOSPHATE ION
著者Murray, J.M, Steffek, M.
登録日2013-10-23
公開日2014-01-01
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.936 Å)
主引用文献Tailoring small molecules for an allosteric site on procaspase-6.
Chemmedchem, 9, 2014
2EVZ
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Structure of RNA Binding Domains 3 and 4 of Polypyrimidine Tract Binding Protein
分子名称: Polypyrimidine tract-binding protein 1
著者Allain, F.H, Auweter, S.D.
登録日2005-11-01
公開日2006-01-17
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Structure of the two most C-terminal RNA recognition motifs of PTB using segmental isotope labeling
Embo J., 25, 2006
3TNF
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LidA from Legionella in complex with active Rab8a
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, LidA, MAGNESIUM ION, ...
著者Schoebel, S, Cichy, A.L, Goody, R.S, Itzen, A.
登録日2011-09-01
公開日2011-11-02
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Protein LidA from Legionella is a Rab GTPase supereffector.
Proc.Natl.Acad.Sci.USA, 108, 2011
5E6X
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Re-refinement of the Crystal Structure of the Plexin-Semaphorin-Integrin Domain/Hybrid Domain/I-EGF1 Segment from the Human Integrin b2 Subunit
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Integrin beta-2
著者Springer, T.A, Sen, M.
登録日2015-10-10
公開日2016-03-02
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Leukocyte integrin alpha L beta 2 headpiece structures: The alpha I domain, the pocket for the internal ligand, and concerted movements of its loops.
Proc.Natl.Acad.Sci.USA, 113, 2016
5E6R
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Structures of leukocyte integrin aLb2: The aI domain, the headpiece, and the pocket for the internal ligand
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, Integrin alpha-L, ...
著者Sen, M, Springer, T.A.
登録日2015-10-10
公開日2016-03-02
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.901 Å)
主引用文献Leukocyte integrin alpha L beta 2 headpiece structures: The alpha I domain, the pocket for the internal ligand, and concerted movements of its loops.
Proc.Natl.Acad.Sci.USA, 113, 2016
1I9B
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X-RAY STRUCTURE OF ACETYLCHOLINE BINDING PROTEIN (ACHBP)
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ACETYLCHOLINE BINDING PROTEIN, CALCIUM ION
著者Brejc, K, van Dijk, W.J, Klaassen, R, Schuurmans, M, van der Oost, J, Smit, A.B, Sixma, T.K.
登録日2001-03-18
公開日2001-05-16
最終更新日2018-03-07
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal structure of an ACh-binding protein reveals the ligand-binding domain of nicotinic receptors.
Nature, 411, 2001

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