8OKM
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![BU of 8okm by Molmil](/molmil-images/mine/8okm) | Crystal structure of F2F-2020197-00X bound to the main protease (3CLpro/Mpro) of SARS-CoV-2. | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 1,2-ETHANEDIOL, 3C-like proteinase nsp5, ... | 著者 | Costanzi, E, Demitri, N, Storici, P. | 登録日 | 2023-03-28 | 公開日 | 2023-05-03 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.66 Å) | 主引用文献 | Broad-spectrum coronavirus 3C-like protease peptidomimetic inhibitors effectively block SARS-CoV-2 replication in cells: Design, synthesis, biological evaluation, and X-ray structure determination. Eur.J.Med.Chem., 253, 2023
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8OKN
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![BU of 8okn by Molmil](/molmil-images/mine/8okn) | Crystal structure of F2F-2020198-00X bound to the main protease (3CLpro/Mpro) of SARS-CoV-2. | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 1,2-ETHANEDIOL, 3C-like proteinase nsp5, ... | 著者 | Costanzi, E, Demitri, N, Storici, P. | 登録日 | 2023-03-28 | 公開日 | 2023-05-03 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | Broad-spectrum coronavirus 3C-like protease peptidomimetic inhibitors effectively block SARS-CoV-2 replication in cells: Design, synthesis, biological evaluation, and X-ray structure determination. Eur.J.Med.Chem., 253, 2023
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6HER
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![BU of 6her by Molmil](/molmil-images/mine/6her) | Mouse prion protein in complex with Nanobody 484 | 分子名称: | GLYCEROL, Major prion protein, Nanobody 484, ... | 著者 | Soror, S.H, Abskharon, R, Wohlkonig, A. | 登録日 | 2018-08-20 | 公開日 | 2019-12-04 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.199 Å) | 主引用文献 | Structural evidence for the critical role of the prion protein hydrophobic region in forming an infectious prion. Plos Pathog., 15, 2019
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3MK9
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![BU of 3mk9 by Molmil](/molmil-images/mine/3mk9) | |
4WPB
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![BU of 4wpb by Molmil](/molmil-images/mine/4wpb) | Vascular endothelial growth factor in complex with alpha/beta-VEGF-1 | 分子名称: | Vascular endothelial growth factor A, alpha/beta-VEGF-1 | 著者 | Kreitler, D.F, Checco, J.W, Gellman, S.H, Forest, K.T. | 登録日 | 2014-10-17 | 公開日 | 2015-04-15 | 最終更新日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (3.11 Å) | 主引用文献 | Targeting diverse protein-protein interaction interfaces with alpha / beta-peptides derived from the Z-domain scaffold. Proc.Natl.Acad.Sci.USA, 112, 2015
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8P5F
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![BU of 8p5f by Molmil](/molmil-images/mine/8p5f) | Human wild-type GAPDH,orthorhombic form | 分子名称: | ACETATE ION, Glyceraldehyde-3-phosphate dehydrogenase, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ... | 著者 | Samygina, V.R, Muronetz, V.I, Schmalhausen, E.V. | 登録日 | 2023-05-24 | 公開日 | 2023-07-05 | 最終更新日 | 2023-07-12 | 実験手法 | X-RAY DIFFRACTION (1.82 Å) | 主引用文献 | S-nitrosylation and S-glutathionylation of GAPDH: Similarities, differences, and relationships. Biochim Biophys Acta Gen Subj, 1867, 2023
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5KHY
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![BU of 5khy by Molmil](/molmil-images/mine/5khy) | |
1E8T
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![BU of 1e8t by Molmil](/molmil-images/mine/1e8t) | Structure of the multifunctional paramyxovirus hemagglutinin-neuraminidase | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ... | 著者 | Crennell, S, Takimoto, T, Portner, A, Taylor, G. | 登録日 | 2000-10-01 | 公開日 | 2001-04-03 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal Structure of the Multifunctional Paramyxovirus Hemagglutinin-Neuraminidase Nat.Struct.Biol., 7, 2000
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4WYJ
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![BU of 4wyj by Molmil](/molmil-images/mine/4wyj) | Adenovirus 3 head domain mutant V239D | 分子名称: | Fiber protein, SULFATE ION | 著者 | Lieber, A, Zubieta, C, Fender, P. | 登録日 | 2014-11-17 | 公開日 | 2015-07-01 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.65 Å) | 主引用文献 | Preclinical safety and efficacy studies with an affinity-enhanced epithelial junction opener and PEGylated liposomal doxorubicin. Mol Ther Methods Clin Dev, 2, 2015
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3RRC
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![BU of 3rrc by Molmil](/molmil-images/mine/3rrc) | |
5KA6
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![BU of 5ka6 by Molmil](/molmil-images/mine/5ka6) | |
8Q93
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![BU of 8q93 by Molmil](/molmil-images/mine/8q93) | Crystal structure of the SARS-COV-2 RBD with neutralizing-VHHs Re30H02 and Re21D01 | 分子名称: | Nanobody Re21D01, Nanobody Re30H02, Spike protein S1 | 著者 | Aksu, M, Guttler, T, Rymarenko, O, Gorlich, D. | 登録日 | 2023-08-19 | 公開日 | 2023-12-20 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Nanobodies to multiple spike variants and inhalation of nanobody-containing aerosols neutralize SARS-CoV-2 in cell culture and hamsters. Antiviral Res., 221, 2023
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8Q95
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![BU of 8q95 by Molmil](/molmil-images/mine/8q95) | Crystal structure of the SARS-CoV-2 BA.1 RBD with neutralizing-VHHs Ma16B06 and Ma3F05 | 分子名称: | Nanobody Ma16B06, Nanobody Ma3F05, Spike protein S1 | 著者 | Aksu, M, Rymarenko, O, Guttler, T, Gorlich, D. | 登録日 | 2023-08-19 | 公開日 | 2023-12-20 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Nanobodies to multiple spike variants and inhalation of nanobody-containing aerosols neutralize SARS-CoV-2 in cell culture and hamsters. Antiviral Res., 221, 2023
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8Q94
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4FHQ
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![BU of 4fhq by Molmil](/molmil-images/mine/4fhq) | Crystal Structure of HVEM | 分子名称: | Tumor necrosis factor receptor superfamily member 14 | 著者 | Liu, W, Zhan, C, Patskovsky, Y, Bhosle, R.C, Nathenson, S.G, Almo, S.C, Atoms-to-Animals: The Immune Function Network (IFN), New York Structural Genomics Research Consortium (NYSGRC) | 登録日 | 2012-06-06 | 公開日 | 2012-07-18 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.251 Å) | 主引用文献 | Increased Heterologous Protein Expression in Drosophila S2 Cells for Massive Production of Immune Ligands/Receptors and Structural Analysis of Human HVEM. Mol Biotechnol, 57, 2015
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1O7Q
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![BU of 1o7q by Molmil](/molmil-images/mine/1o7q) | Roles of Individual Residues of Alpha-1,3 Galactosyltransferases in Substrate Binding and Catalysis | 分子名称: | GLYCEROL, MANGANESE (II) ION, N-ACETYLLACTOSAMINIDE ALPHA-1,3-GALACTOSYLTRANSFERASE, ... | 著者 | Zhang, Y, Swaminathan, G.J, Deshpande, A, Natesh, R, Xie, Z, Acharya, K.R, Brew, K. | 登録日 | 2002-11-12 | 公開日 | 2003-11-06 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Roles of Individual Enzyme-Substrate Interactions by Alpha-1,3-Galactosyltransferase in Catalysis and Specificity. Biochemistry, 42, 2003
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3U3Y
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![BU of 3u3y by Molmil](/molmil-images/mine/3u3y) | Mouse TREX1 D200H mutant | 分子名称: | 1,4-BUTANEDIOL, 5'-D(*GP*AP*CP*G)-3', CALCIUM ION, ... | 著者 | Bailey, S.L, Harvey, S, Perrino, F.W, Hollis, T. | 登録日 | 2011-10-06 | 公開日 | 2011-12-28 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.28 Å) | 主引用文献 | Defects in DNA degradation revealed in crystal structures of TREX1 exonuclease mutations linked to autoimmune disease. Dna Repair, 11, 2012
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4GN4
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![BU of 4gn4 by Molmil](/molmil-images/mine/4gn4) | |
3UL7
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![BU of 3ul7 by Molmil](/molmil-images/mine/3ul7) | Crystal structure of the TV3 mutant F63W | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, SULFATE ION, Toll-like receptor 4, ... | 著者 | Kim, H.J, Cheong, H.K, Jeon, Y.H. | 登録日 | 2011-11-10 | 公開日 | 2012-04-04 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.37 Å) | 主引用文献 | Structure-Based Rational Design of a Toll-like Receptor 4 (TLR4) Decoy Receptor with High Binding Affinity for a Target Protein. Plos One, 7, 2012
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8OPN
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![BU of 8opn by Molmil](/molmil-images/mine/8opn) | Human Coronavirus HKU1 spike glycoprotein in complex with an alpha2,8-linked 9-O-acetylated disialoside (1-up state) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 9-O-acetyl-5-acetamido-3,5-dideoxy-D-glycero-alpha-D-galacto-non-2-ulopyranosonic acid-(2-8)-N-acetyl-alpha-neuraminic acid, ... | 著者 | Pronker, M.F, Creutznacher, R, Hurdiss, D.L. | 登録日 | 2023-04-07 | 公開日 | 2023-08-02 | 最終更新日 | 2023-12-13 | 実験手法 | ELECTRON MICROSCOPY (4.7 Å) | 主引用文献 | Sialoglycan binding triggers spike opening in a human coronavirus. Nature, 624, 2023
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8OPO
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![BU of 8opo by Molmil](/molmil-images/mine/8opo) | Human Coronavirus HKU1 spike glycoprotein in complex with an alpha2,8-linked 9-O-acetylated disialoside (3-up state) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 9-O-acetyl-5-acetamido-3,5-dideoxy-D-glycero-alpha-D-galacto-non-2-ulopyranosonic acid-(2-8)-N-acetyl-alpha-neuraminic acid, ... | 著者 | Pronker, M.F, Creutznacher, R, Hurdiss, D.L. | 登録日 | 2023-04-07 | 公開日 | 2023-08-02 | 最終更新日 | 2023-12-13 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Sialoglycan binding triggers spike opening in a human coronavirus. Nature, 624, 2023
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8OPM
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![BU of 8opm by Molmil](/molmil-images/mine/8opm) | Human Coronavirus HKU1 spike glycoprotein in complex with an alpha2,8-linked 9-O-acetylated disialoside (closed state) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 9-O-acetyl-5-acetamido-3,5-dideoxy-D-glycero-alpha-D-galacto-non-2-ulopyranosonic acid-(2-8)-N-acetyl-alpha-neuraminic acid, ... | 著者 | Pronker, M.F, Creutznacher, R, Hurdiss, D.L. | 登録日 | 2023-04-07 | 公開日 | 2023-08-02 | 最終更新日 | 2023-12-13 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | Sialoglycan binding triggers spike opening in a human coronavirus. Nature, 624, 2023
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1N1I
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![BU of 1n1i by Molmil](/molmil-images/mine/1n1i) | The structure of MSP-1(19) from Plasmodium knowlesi | 分子名称: | HISTIDINE, IMIDAZOLE, Merozoite surface protein-1 | 著者 | Garman, S.C, Simcoke, W.N, Stowers, A.W, Garboczi, D.N. | 登録日 | 2002-10-17 | 公開日 | 2003-02-25 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structure of the C-terminal domains of merozoite surface protein-1 from
Plasmodium knowlesi reveals a novel histidine binding site J.Biol.Chem., 278, 2003
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6HHD
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![BU of 6hhd by Molmil](/molmil-images/mine/6hhd) | Mouse Prion Protein in complex with Nanobody 484 | 分子名称: | CHLORIDE ION, GLYCEROL, Major prion protein, ... | 著者 | Soror, S, Abskharon, R, Wohlkonig, A. | 登録日 | 2018-08-28 | 公開日 | 2019-12-11 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.102 Å) | 主引用文献 | Structural evidence for the critical role of the prion protein hydrophobic region in forming an infectious prion. Plos Pathog., 15, 2019
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3QII
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![BU of 3qii by Molmil](/molmil-images/mine/3qii) | Crystal structure of tudor domain 2 of human PHD finger protein 20 | 分子名称: | PHD finger protein 20, UNKNOWN ATOM OR ION | 著者 | Li, Z, Tempel, W, Wernimont, A.K, Chao, X, Bian, C, Lam, R, Crombet, L, Bountra, C, Weigelt, J, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Min, J, Structural Genomics Consortium (SGC) | 登録日 | 2011-01-27 | 公開日 | 2011-02-09 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Crystal structures of the Tudor domains of human PHF20 reveal novel structural variations on the Royal Family of proteins. Febs Lett., 586, 2012
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