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1DPF
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CRYSTAL STRUCTURE OF A MG-FREE FORM OF RHOA COMPLEXED WITH GDP
分子名称: GUANOSINE-5'-DIPHOSPHATE, RHOA
著者Shimizu, T, Ihara, K, Maesaki, R, Kuroda, S, Kaibuchi, K, Hakoshima, T.
登録日1999-12-27
公開日2000-06-21
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献An open conformation of switch I revealed by the crystal structure of a Mg2+-free form of RHOA complexed with GDP. Implications for the GDP/GTP exchange mechanism.
J.Biol.Chem., 275, 2000
1E0G
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LYSM Domain from E.coli MLTD
分子名称: Membrane-bound lytic murein transglycosylase D
著者Bateman, A, Bycroft, M.
登録日2000-03-27
公開日2000-06-21
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献The Structure of a Lysm Domain from E.Coli Membrane Bound Lytic Murein Transglycosylase D (Mltd)
J.Mol.Biol., 299, 2000
1E1D
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Hybrid Cluster Protein from Desulfovibrio vulgaris
分子名称: HYDROXYLAMINE REDUCTASE, IRON/SULFUR CLUSTER, IRON/SULFUR/OXYGEN HYBRID CLUSTER
著者Arendsen, A.F, Cooper, S.J, Bailey, S, Garner, C.D, Hagen, W.R, Lindley, P.F.
登録日2000-05-02
公開日2000-06-21
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.72 Å)
主引用文献Hybrid-Cluster Protein (Hcp) from Desulfovibrio Vulgaris (Hildenborough) at 1.6 A Resolution.
Biochemistry, 39, 2000
1QR3
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Structure of porcine pancreatic elastase in complex with FR901277, a novel macrocyclic inhibitor of elastases at 1.6 angstrom resolution
分子名称: CALCIUM ION, Chymotrypsin-like elastase family member 1, FR901277 Inhibitor, ...
著者Nakanishi, I, Kinoshita, T, Sato, A, Tada, T.
登録日1999-06-18
公開日2000-06-21
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structure of porcine pancreatic elastase complexed with FR901277, a novel macrocyclic inhibitor of elastases, at 1.6 A resolution.
Biopolymers, 53, 2000
1F4D
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CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE C146S, L143C COVALENTLY MODIFIED AT C143 WITH N-[TOSYL-D-PROLINYL]AMINO-ETHANETHIOL
分子名称: GLYCEROL, N-[TOSYL-D-PROLINYL]AMINO-ETHANETHIOL, SULFATE ION, ...
著者Erlanson, D.A, Braisted, A.C, Raphael, D.R, Randal, M, Stroud, R.M, Gordon, E, Wells, J.A.
登録日2000-06-07
公開日2000-06-22
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Site-directed ligand discovery.
Proc.Natl.Acad.Sci.USA, 97, 2000
1F4F
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CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE COMPLEXED WITH SP-722
分子名称: 4-[[GLUTAMIC ACID]-CARBONYL]-BENZENE-SULFONYL-D-PROLINE, SULFATE ION, THYMIDYLATE SYNTHASE
著者Erlanson, D.A, Braisted, A.C, Raphael, D.R, Randal, M, Stroud, R.M, Gordon, E, Wells, J.A.
登録日2000-06-07
公開日2000-06-22
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Site-directed ligand discovery.
Proc.Natl.Acad.Sci.USA, 97, 2000
1F4G
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CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE COMPLEXED WITH SP-876
分子名称: GLYCEROL, N-[4-[[GLUTAMIC ACID]-CARBONYL]-BENZENE-SULFONYL-D-PROLINYL]-3-AMINO-PROPANOIC ACID, SULFATE ION, ...
著者Erlanson, D.A, Braisted, A.C, Raphael, D.R, Randal, M, Stroud, R.M, Gordon, E, Wells, J.A.
登録日2000-06-07
公開日2000-06-22
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Site-directed ligand discovery.
Proc.Natl.Acad.Sci.USA, 97, 2000
1F4C
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CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE COVALENTLY MODIFIED AT C146 WITH N-[TOSYL-D-PROLINYL]AMINO-ETHANETHIOL
分子名称: GLYCEROL, N-[TOSYL-D-PROLINYL]AMINO-ETHANETHIOL, SULFATE ION, ...
著者Erlanson, D.A, Braisted, A.C, Raphael, D.R, Randal, M, Stroud, R.M, Gordon, E, Wells, J.A.
登録日2000-06-07
公開日2000-06-22
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Site-directed ligand discovery.
Proc.Natl.Acad.Sci.USA, 97, 2000
1F4B
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CRYSTAL STRUCTURE OF ESCHERICHIA COLI THYMIDYLATE SYNTHASE
分子名称: GLYCEROL, SULFATE ION, THYMIDYLATE SYNTHASE
著者Erlanson, D.A, Braisted, A.C, Raphael, D.R, Randal, M, Stroud, R.M, Gordon, E, Wells, J.A.
登録日2000-06-07
公開日2000-06-22
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Site-directed ligand discovery.
Proc.Natl.Acad.Sci.USA, 97, 2000
1F4E
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CRYSTAL STRUCTURE OF E. COLI THYMIDYLATE SYNTHASE COMPLEXED WITH TOSYL-D-PROLINE
分子名称: GLYCEROL, SULFATE ION, THYMIDYLATE SYNTHASE, ...
著者Erlanson, D.A, Braisted, A.C, Raphael, D.R, Randal, M, Stroud, R.M, Gordon, E, Wells, J.A.
登録日2000-06-07
公開日2000-06-22
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Site-directed ligand discovery.
Proc.Natl.Acad.Sci.USA, 97, 2000
1DZQ
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LECTIN UEA-II COMPLEXED WITH GALACTOSE
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, LECTIN II, ...
著者Loris, R, De Greve, H, Dao-Thi, M.-H, Messens, J, Imberty, A, Wyns, L.
登録日2000-03-07
公開日2000-06-22
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Structural Basis of Carbohydrate Recognition by Lectin II from Ulex Europaeus, a Protein with a Promiscuous Carbohydrate Binding Site
J.Mol.Biol., 301, 2000
1QJ6
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Novel Covalent Active Site Thrombin Inhibitors
分子名称: 6-CARBAMIMIDOYL-2-[2-HYDROXY-5-(3-METHOXY-PHENYL)-INDAN-1-YL]-HEXANOIC ACID, HIRUGEN, THROMBIN
著者Jhoti, H, Cleasby, A.
登録日1999-06-22
公開日2000-06-22
最終更新日2018-05-30
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal Structures of Thrombin Complexed to a Novel Series of Synthetic Inhibitors Containing a 5,5-Trans-Lactone Template
Biochemistry, 38, 1999
1QJ7
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Novel Covalent Active Site Thrombin Inhibitors
分子名称: 6-CARBAMIMIDOYL-2-[5-(3-DIETHYLCARBAMOYL-PHENYL)-2-HYDROXY-INDAN-1-YL]-HEXANOIC ACID, HIRUGEN, THROMBIN
著者Jhoti, H, Cleasby, A.
登録日1999-06-22
公開日2000-06-22
最終更新日2018-05-30
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal Structures of Thrombin Complexed to a Novel Series of Synthetic Inhibitors Containing a 5,5-Trans-Lactone Template
Biochemistry, 38, 1999
1QJ3
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Crystal structure of 7,8-diaminopelargonic acid synthase in complex with 7-keto-8-aminopelargonic acid
分子名称: 7,8-DIAMINOPELARGONIC ACID SYNTHASE, 7-KETO-8-AMINOPELARGONIC ACID, PYRIDOXAL-5'-PHOSPHATE, ...
著者Kaeck, H, Sandmark, J, Gibson, K.J, Lindqvist, Y, Schneider, G.
登録日1999-06-21
公開日2000-06-22
最終更新日2019-05-08
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Crystal Structure of Diaminopelargonic Acid Synthase; Evolutionary Relationships between Pyridoxal-5'-Phosphate Dependent Enzymes
J.Mol.Biol., 291, 1999
1QJ5
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Crystal structure of 7,8-diaminopelargonic acid synthase
分子名称: 7,8-DIAMINOPELARGONIC ACID SYNTHASE, POTASSIUM ION, PYRIDOXAL-5'-PHOSPHATE
著者Kack, H, Sandmark, J, Gibson, K.J, Lindqvist, Y, Schneider, G.
登録日1999-06-21
公開日2000-06-22
最終更新日2019-07-24
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal Structure of Diaminopelargonic Acid Synthase; Evolutionary Relationships between Pyridoxal-5'-Phosphate Dependent Enzymes
J.Mol.Biol., 291, 1999
1QJ1
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BU of 1qj1 by Molmil
Novel Covalent Active Site Thrombin Inhibitors
分子名称: 6-CARBAMIMIDOYL-2-[2-HYDROXY-6-(4-HYDROXY-PHENYL)-INDAN-1-YL]-HEXANOIC ACID, HIRUGEN, THROMBIN
著者Jhoti, H, Cleasby, A.
登録日1999-06-21
公開日2000-06-22
最終更新日2018-05-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal Structures of Thrombin Complexed to a Novel Series of Synthetic Inhibitors Containing a 5,5-Trans-Lactone Template
Biochemistry, 38, 1999
1EZU
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ECOTIN Y69F, D70P BOUND TO D102N TRYPSIN
分子名称: CALCIUM ION, ECOTIN, TRYPSIN II, ...
著者Gillmor, S.A, Takeuchi, T, Yang, S.Q, Craik, C.S, Fletterick, R.J.
登録日2000-05-11
公開日2000-06-23
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Compromise and accommodation in ecotin, a dimeric macromolecular inhibitor of serine proteases.
J.Mol.Biol., 299, 2000
1EZS
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CRYSTAL STRUCTURE OF ECOTIN MUTANT M84R, W67A, G68A, Y69A, D70A BOUND TO RAT ANIONIC TRYPSIN II
分子名称: CALCIUM ION, ECOTIN, TRYPSIN II, ...
著者Gillmor, S.A, Takeuchi, T, Yang, S.Q, Craik, C.S, Fletterick, R.J.
登録日2000-05-11
公開日2000-06-23
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Compromise and accommodation in ecotin, a dimeric macromolecular inhibitor of serine proteases.
J.Mol.Biol., 299, 2000
1GFW
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THE 2.8 ANGSTROM CRYSTAL STRUCTURE OF CASPASE-3 (APOPAIN OR CPP32)IN COMPLEX WITH AN ISATIN SULFONAMIDE INHIBITOR.
分子名称: 1-METHYL-5-(2-PHENOXYMETHYL-PYRROLIDINE-1-SULFONYL)-1H-INDOLE-2,3-DIONE, CASPASE-3 (APOPAIN, P10), ...
著者Concha, N.O, Janson, C.A.
登録日2000-06-16
公開日2000-06-23
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Potent and selective nonpeptide inhibitors of caspases 3 and 7 inhibit apoptosis and maintain cell functionality.
J.Biol.Chem., 275, 2000
1EGK
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CRYSTAL STRUCTURE OF A NUCLEIC ACID FOUR-WAY JUNCTION
分子名称: 10-23 DNA ENZYME, MAGNESIUM ION, RNA (5'-R(*AP*GP*GP*AP*GP*AP*GP*AP*GP*AP*UP*GP*GP*GP*UP*GP*CP*GP*AP*G)-3')
著者Nowakowski, J, Shim, P.J, Stout, C.D, Joyce, G.F.
登録日2000-02-15
公開日2000-06-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Alternative conformations of a nucleic acid four-way junction.
J.Mol.Biol., 300, 2000
1F5H
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The G7(syn)-G4(anti) structure of r(GCAGGCGUGC)2
分子名称: 5'-R(*GP*CP*AP*GP*GP*CP*GP*UP*GP*C)-3'
著者Burkard, M.E, Turner, D.H.
登録日2000-06-14
公開日2000-06-26
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献NMR structures of r(GCAGGCGUGC)2 and determinants of stability for single guanosine-guanosine base pairs
Biochemistry, 39, 2000
1F5G
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The G7(syn)-G4(anti) structure of r(GCAGGCGUGC)2
分子名称: 5'-R(*GP*CP*AP*GP*GP*CP*GP*UP*GP*C)-3'
著者Burkard, M.E, Turner, D.H.
登録日2000-06-14
公開日2000-06-26
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献NMR structures of r(GCAGGCGUGC)2 and determinants of stability for single guanosine-guanosine base pairs
Biochemistry, 39, 2000
1EQ7
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CORE STRUCTURE OF THE OUTER MEMBRANE LIPOPROTEIN FROM ESCHERICHIA COLI AT 1.9 ANGSTROM RESOLUTION
分子名称: OUTER MEMBRANE LIPOPROTEIN
著者Shu, W, Liu, J, Ji, H, Lu, M.
登録日2000-04-03
公開日2000-06-28
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Core structure of the outer membrane lipoprotein from Escherichia coli at 1.9 A resolution.
J.Mol.Biol., 299, 2000
1F5B
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CRYSTAL STRUCTURE OF F2H FERREDOXIN 1 MUTANT FROM AZOTOBACTER VINELANDII AT 1.75 ANGSTROM RESOLUTION
分子名称: FE3-S4 CLUSTER, FERREDOXIN 1, IRON/SULFUR CLUSTER
著者Chen, K, Bonagura, C.A, Tilley, G.J, Jung, Y.S, Armstrong, F.A, Stout, C.D, Burgess, B.K.
登録日2000-06-13
公開日2000-06-28
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.62 Å)
主引用文献Crystal structures of ferredoxin variants exhibiting large changes in [Fe-S] reduction potential.
Nat.Struct.Biol., 9, 2002
1F1Z
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TNSA, a catalytic component of the TN7 transposition system
分子名称: CHLORIDE ION, MAGNESIUM ION, TNSA ENDONUCLEASE
著者Hickman, A.B, Li, Y, Mathew, S.V, May, E.W, Craig, N.L, Dyda, F.
登録日2000-05-21
公開日2000-06-28
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Unexpected structural diversity in DNA recombination: the restriction endonuclease connection.
Mol.Cell, 5, 2000

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