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1QR3

Structure of porcine pancreatic elastase in complex with FR901277, a novel macrocyclic inhibitor of elastases at 1.6 angstrom resolution

Summary for 1QR3
Entry DOI10.2210/pdb1qr3/pdb
Related PRD IDPRD_000561
DescriptorChymotrypsin-like elastase family member 1, FR901277 Inhibitor, CALCIUM ION, ... (5 entities in total)
Functional Keywordsprotease, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor
Biological sourceSus scrofa (Pig)
More
Total number of polymer chains2
Total formula weight27080.27
Authors
Nakanishi, I.,Kinoshita, T.,Sato, A.,Tada, T. (deposition date: 1999-06-18, release date: 2000-06-21, Last modification date: 2023-11-15)
Primary citationNakanishi, I.,Kinoshita, T.,Sato, A.,Tada, T.
Structure of porcine pancreatic elastase complexed with FR901277, a novel macrocyclic inhibitor of elastases, at 1.6 A resolution.
Biopolymers, 53:434-445, 2000
Cited by
PubMed: 10738204
DOI: 10.1002/(SICI)1097-0282(20000415)53:5<434::AID-BIP7>3.0.CO;2-5
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.6 Å)
Structure validation

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