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3CJO
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Crystal structure of KSP in complex with inhibitor 30
分子名称: (2S)-4-(2,5-difluorophenyl)-N-[(3R,4S)-3-fluoro-1-methylpiperidin-4-yl]-2-(hydroxymethyl)-N-methyl-2-phenyl-2,5-dihydro-1H-pyrrole-1-carboxamide, ADENOSINE-5'-DIPHOSPHATE, Kinesin-like protein KIF11, ...
著者Yan, Y.
登録日2008-03-13
公開日2008-07-01
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.28 Å)
主引用文献Kinesin spindle protein (KSP) inhibitors. 9. Discovery of (2S)-4-(2,5-difluorophenyl)-n-[(3R,4S)-3-fluoro-1-methylpiperidin-4-yl]-2-(hydroxymethyl)-N-methyl-2-phenyl-2,5-dihydro-1H-pyrrole-1-carboxamide (MK-0731) for the treatment of taxane-refractory cancer.
J.Med.Chem., 51, 2008
2VVG
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Crystal Structure of the G.intestinalis Kinesin 2 GiKIN2a Motor Domain
分子名称: ADENOSINE-5'-DIPHOSPHATE, KINESIN-2, MAGNESIUM ION
著者Hoeng, J.C, Loewe, J, Dawson, S.C, Cande, W.Z, Sagolla, M.S, Mancuso, J.J.
登録日2008-06-08
公開日2008-07-08
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献High-Resolution Crystal Structure and in Vivo Function of a Kinesin-2 Homologue in Giardia Intestinalis.
Mol.Biol.Cell, 19, 2008
2P4N
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BU of 2p4n by Molmil
Human Monomeric Kinesin (1BG2) and Bovine Tubulin (1JFF) Docked into the 9-Angstrom Cryo-EM Map of Nucleotide-Free Kinesin Complexed to the Microtubule
分子名称: ADENOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ...
著者Sindelar, C.V, Downing, K.H.
登録日2007-03-12
公開日2008-07-08
最終更新日2024-02-21
実験手法ELECTRON MICROSCOPY (9 Å)
主引用文献The beginning of kinesin's force-generating cycle visualized at 9-A resolution.
J.Cell Biol., 177, 2007
2ZFJ
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BU of 2zfj by Molmil
Crystal Structure of the Kif1A Motor Domain during Mg release: Mg-releasing Transition-1
分子名称: ADENOSINE-5'-DIPHOSPHATE, Kinesin-like protein KIF1A, Kinesin heavy chain isoform 5C, ...
著者Nitta, R, Okada, Y, Hirokawa, N.
登録日2008-01-08
公開日2008-09-23
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Structural model for strain-dependent microtubule activation of Mg-ADP release from kinesin.
Nat.Struct.Mol.Biol., 15, 2008
2ZFI
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Crystal Structure of the Kif1A Motor Domain Before Mg Release
分子名称: ADENOSINE-5'-DIPHOSPHATE, Kinesin-like protein KIF1A, Kinesin heavy chain isoform 5C, ...
著者Nitta, R, Okada, Y, Hirokawa, N.
登録日2008-01-07
公開日2008-09-23
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Structural model for strain-dependent microtubule activation of Mg-ADP release from kinesin.
Nat.Struct.Mol.Biol., 15, 2008
2ZFK
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Crystal Structure of the Kif1A Motor Domain during Mg release: Mg-releasing Transition-2
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ADENOSINE-5'-DIPHOSPHATE, Kinesin-like protein KIF1A, ...
著者Nitta, R, Okada, Y, Hirokawa, N.
登録日2008-01-08
公開日2008-09-23
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (3.61 Å)
主引用文献Structural model for strain-dependent microtubule activation of Mg-ADP release from kinesin.
Nat.Struct.Mol.Biol., 15, 2008
2ZFL
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BU of 2zfl by Molmil
Crystal Structure of the Kif1A Motor Domain during Mg release: Mg-releasing Transition-3
分子名称: ADENOSINE-5'-DIPHOSPHATE, Kinesin-like protein KIF1A, Kinesin heavy chain isoform 5C
著者Nitta, R, Okada, Y, Hirokawa, N.
登録日2008-01-08
公開日2008-09-23
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structural model for strain-dependent microtubule activation of Mg-ADP release from kinesin.
Nat.Struct.Mol.Biol., 15, 2008
2ZFM
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BU of 2zfm by Molmil
Crystal Structure of the Kif1A Motor Domain After Mg Release
分子名称: ADENOSINE-5'-DIPHOSPHATE, Kinesin-like protein KIF1A, Kinesin heavy chain isoform 5C
著者Nitta, R, Okada, Y, Hirokawa, N.
登録日2008-01-08
公開日2008-09-23
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.31 Å)
主引用文献Structural model for strain-dependent microtubule activation of Mg-ADP release from kinesin.
Nat.Struct.Mol.Biol., 15, 2008
3EDL
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BU of 3edl by Molmil
Kinesin13-Microtubule Ring complex
分子名称: 2-MERCAPTO-N-[1,2,3,10-TETRAMETHOXY-9-OXO-5,6,7,9-TETRAHYDRO-BENZO[A]HEPTALEN-7-YL]ACETAMIDE, Beta tubulin, GUANOSINE-5'-DIPHOSPHATE, ...
著者Tan, D, Rice, W.J, Sosa, H.
登録日2008-09-03
公開日2009-01-20
最終更新日2024-02-21
実験手法ELECTRON MICROSCOPY (28 Å)
主引用文献Structure of the kinesin13-microtubule ring complex.
Structure, 16, 2008
3DC4
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BU of 3dc4 by Molmil
Crystal structure of the Drosophila kinesin family member NOD in complex with ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, Kinesin-like protein Nod, MAGNESIUM ION
著者Cochran, J.C, Mulko, N.K, Kull, F.J.
登録日2008-06-03
公開日2009-02-10
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献ATPase cycle of the nonmotile kinesin NOD allows microtubule end tracking and drives chromosome movement.
Cell(Cambridge,Mass.), 136, 2009
3DCO
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BU of 3dco by Molmil
Drosophila NOD (3DC4) and Bovine Tubulin (1JFF) Docked into the 11-Angstrom Cryo-EM Map of Nucleotide-Free NOD Complexed to the Microtubule
分子名称: ADENOSINE-5'-DIPHOSPHATE, Bovine Alpha Tubulin, Bovine Beta Tubulin, ...
著者Sindelar, C.V, Cochran, J.C, Kull, F.J.
登録日2008-06-04
公開日2009-02-10
最終更新日2024-02-21
実験手法ELECTRON MICROSCOPY (11 Å)
主引用文献ATPase cycle of the nonmotile kinesin NOD allows microtubule end tracking and drives chromosome movement.
Cell(Cambridge,Mass.), 136, 2009
3DCB
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BU of 3dcb by Molmil
Crystal structure of the Drosophila kinesin family member NOD in complex with AMPPNP
分子名称: Kinesin-like protein Nod, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER
著者Cochran, J.C, Mulko, N.K, Kull, F.J.
登録日2008-06-03
公開日2009-02-10
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献ATPase cycle of the nonmotile kinesin NOD allows microtubule end tracking and drives chromosome movement.
Cell(Cambridge,Mass.), 136, 2009
3GBJ
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BU of 3gbj by Molmil
Crystal structure of the motor domain of kinesin KIF13B bound with ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, KIF13B protein, MAGNESIUM ION, ...
著者Tong, Y, Shen, L, Shen, Y, Tempel, W, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC)
登録日2009-02-19
公開日2009-03-03
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.102 Å)
主引用文献Crystal structure of the motor domain of kinesin KIF13B bound with ADP
To be Published
2WBE
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BU of 2wbe by Molmil
Kinesin-5-Tubulin Complex with AMPPNP
分子名称: BIPOLAR KINESIN KRP-130, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ...
著者Bodey, A.J, Kikkawa, M, Moores, C.A.
登録日2009-02-26
公開日2009-03-24
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (9.4 Å)
主引用文献9-Angstrom Structure of a Microtubule-Bound Mitotic Motor.
J.Mol.Biol., 388, 2009
3H4S
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BU of 3h4s by Molmil
Structure of the complex of a mitotic kinesin with its calcium binding regulator
分子名称: ADENOSINE-5'-DIPHOSPHATE, CALCIUM ION, KCBP interacting Ca2+-binding protein, ...
著者Vinogradova, M.V.
登録日2009-04-20
公開日2009-05-19
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structure of the complex of a mitotic kinesin with its calcium binding regulator.
Proc.Natl.Acad.Sci.USA, 106, 2009
3K5E
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BU of 3k5e by Molmil
The structure of human kinesin-like motor protein Kif11/KSP/Eg5 in complex with ADP and enastrol.
分子名称: (4S,5R)-5-hydroxy-4-(3-hydroxyphenyl)-3,4,5,6,7,8-hexahydroquinazoline-2(1H)-thione, ADENOSINE-5'-DIPHOSPHATE, Kinesin-like protein KIF11, ...
著者Crawley, L, Cheng, R.K.Y, Wood, M, Barker, J, Felicetti, B, Whittaker, M.
登録日2009-10-07
公開日2009-10-20
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献The structure of human kinesin-like motor protein Kif11/KSP/Eg5 in complex with ADP and enastrol.
To be Published
3HQD
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BU of 3hqd by Molmil
Human kinesin Eg5 motor domain in complex with AMPPNP and Mg2+
分子名称: Kinesin-like protein KIF11, MAGNESIUM ION, PHOSPHATE ION, ...
著者Parke, C.L, Wojcik, E.J, Kim, S, Worthylake, D.K.
登録日2009-06-05
公開日2009-12-08
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.19 Å)
主引用文献ATP Hydrolysis in Eg5 Kinesin Involves a Catalytic Two-water Mechanism.
J.Biol.Chem., 285, 2010
3K3B
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BU of 3k3b by Molmil
Co-crystal structure of the human kinesin Eg5 with a novel tetrahydro-beta-carboline
分子名称: 3-[(1R)-2-acetyl-6-methyl-2,3,4,9-tetrahydro-1H-beta-carbolin-1-yl]phenol, ADENOSINE-5'-DIPHOSPHATE, CHLORIDE ION, ...
著者Bussiere, D.E, Bellamacina, C, Le, V.
登録日2009-10-02
公開日2009-12-15
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The discovery of tetrahydro-beta-carbolines as inhibitors of the kinesin Eg5.
Bioorg.Med.Chem.Lett., 20, 2010
3L9H
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BU of 3l9h by Molmil
X-ray structure of mitotic kinesin-5 (KSP, KIF11, Eg5)in complex with the hexahydro-2H-pyrano[3,2-c]quinoline EMD 534085
分子名称: 1-[2-(dimethylamino)ethyl]-3-{[(2R,4aS,5R,10bS)-5-phenyl-9-(trifluoromethyl)-3,4,4a,5,6,10b-hexahydro-2H-pyrano[3,2-c]quinolin-2-yl]methyl}urea, ADENOSINE-5'-DIPHOSPHATE, Kinesin-like protein KIF11
著者Knoechel, T.
登録日2010-01-05
公開日2010-03-02
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The discovery and optimization of hexahydro-2H-pyrano[3,2-c]quinolines (HHPQs) as potent and selective inhibitors of the mitotic kinesin-5.
Bioorg.Med.Chem.Lett., 20, 2010
3KEN
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Human Eg5 in complex with S-trityl-L-cysteine
分子名称: ADENOSINE-5'-DIPHOSPHATE, Kinesin-like protein KIF11, MAGNESIUM ION, ...
著者Parke, C.L, Wojcik, E.J, Kim, S, Worthylake, D.K.
登録日2009-10-26
公開日2010-03-16
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Allosteric drug discrimination is coupled to mechanochemical changes in the kinesin-5 motor core.
J.Biol.Chem., 285, 2010
2X7E
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Crystal structure of human kinesin Eg5 in complex with (R)-fluorastrol
分子名称: (4R)-5-[(S)-(3,4-DIFLUOROPHENYL)(HYDROXY)METHYL]-4-(3-HYDROXYPHENYL)-1,6-DIMETHYL-3,4-DIHYDROPYRIMIDINE-2(1H)-THIONE, ADENOSINE-5'-DIPHOSPHATE, KINESIN-LIKE PROTEIN KIF11, ...
著者Kaan, H.Y.K, Ulaganathan, V, Rath, O, Laggner, C, Prokopcova, H, Dallinger, D, Kappe, C.O, Kozielski, F.
登録日2010-02-26
公開日2010-07-14
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural Basis for Inhibition of Eg5 by Dihydropyrimidines: Stereoselectivity of Antimitotic Inhibitors Enastron, Dimethylenastron and Fluorastrol.
J.Med.Chem., 53, 2010
2X7C
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BU of 2x7c by Molmil
Crystal structure of human kinesin Eg5 in complex with (S)-enastron
分子名称: (S)-4-(3-HYDROXYPHENYL)-2-THIOXO-1,2,3,4,7,8-HEXAHYDROQUINAZOLIN-5(6H)-ONE, ADENOSINE-5'-DIPHOSPHATE, KINESIN-LIKE PROTEIN KIF11, ...
著者Kaan, H.Y.K, Ulaganathan, V, Rath, O, Laggner, C, Prokopcova, H, Dallinger, D, Kappe, C.O, Kozielski, F.
登録日2010-02-26
公開日2010-07-14
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural Basis for Inhibition of Eg5 by Dihydropyrimidines: Stereoselectivity of Antimitotic Inhibitors Enastron, Dimethylenastron and Fluorastrol.
J.Med.Chem., 53, 2010
2X7D
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Crystal structure of human kinesin Eg5 in complex with (S)-dimethylenastron
分子名称: (4S)-4-(3-HYDROXYPHENYL)-7,7-DIMETHYL-2-THIOXO-2,3,4,6,7,8-HEXAHYDROQUINAZOLIN-5(1H)-ONE, ADENOSINE-5'-DIPHOSPHATE, KINESIN-LIKE PROTEIN KIF11, ...
著者Kaan, H.Y.K, Ulaganathan, V, Rath, O, Laggner, C, Prokopcova, H, Dallinger, D, Kappe, C.O, Kozielski, F.
登録日2010-02-26
公開日2010-07-14
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural Basis for Inhibition of Eg5 by Dihydropyrimidines: Stereoselectivity of Antimitotic Inhibitors Enastron, Dimethylenastron and Fluorastrol.
J.Med.Chem., 53, 2010
3NWN
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BU of 3nwn by Molmil
Crystal structure of the human KIF9 motor domain in complex with ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, CHLORIDE ION, Kinesin-like protein KIF9, ...
著者Zhu, H, Tempel, W, He, H, Shen, Y, Wang, J, Brothers, G, Landry, R, Arrowsmith, C.H, Edwards, A.M, Sundstrom, M, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC)
登録日2010-07-09
公開日2010-07-21
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of the human KIF9 motor domain in complex with ADP
To be Published
2WOG
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Intermediate and final states of human kinesin Eg5 in complex with S-trityl-L-cysteine
分子名称: ADENOSINE-5'-DIPHOSPHATE, KINESIN-LIKE PROTEIN KIF11, MAGNESIUM ION, ...
著者Kaan, H.Y.K, Ulaganathan, V, Hackney, D.D, Kozielski, F.
登録日2009-07-23
公開日2010-08-04
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献An Allosteric Transition Trapped in an Intermediate State of a New Kinesin-Inhibitor Complex.
Biochem.J., 425, 2010

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