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4UX2
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Cryo-EM structure of antagonist-bound E2P gastric H,K-ATPase (SCH.E2. MgF)
分子名称: POTASSIUM-TRANSPORTING ATPASE ALPHA CHAIN 1, POTASSIUM-TRANSPORTING ATPASE SUBUNIT BETA
著者Abe, K, Tani, K, Fujiyoshi, Y.
登録日2014-08-18
公開日2014-09-17
最終更新日2014-11-12
実験手法ELECTRON CRYSTALLOGRAPHY (7 Å)
主引用文献Systematic Comparison of Molecular Conformations of H+,K+-ATPase Reveals an Important Contribution of the A-M2 Linker for the Luminal Gating.
J.Biol.Chem., 289, 2014
5NCQ
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Structure of the (SR) Ca2+-ATPase bound to a Tetrahydrocarbazole and TNP-ATP
分子名称: (1~{S})-~{N}-[(4-bromophenyl)methyl]-7-(trifluoromethyloxy)-2,3,4,9-tetrahydro-1~{H}-carbazol-1-amine, 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, POTASSIUM ION, ...
著者Bublitz, M, Kjellerup, L, O'Hanlon Cohrt, K, Gordon, S, Mortensen, A.L, Clausen, J.D, Pallin, D, Hansen, J.B, Brown, W.D, Fuglsang, A, Winther, A.-M.L.
登録日2017-03-06
公開日2018-01-10
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Tetrahydrocarbazoles are a novel class of potent P-type ATPase inhibitors with antifungal activity.
PLoS ONE, 13, 2018
4HQJ
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Crystal structure of Na+,K+-ATPase in the Na+-bound state
分子名称: ADENOSINE-5'-DIPHOSPHATE, CHOLESTEROL, MAGNESIUM ION, ...
著者Nyblom, M, Reinhard, L, Gourdon, P, Nissen, P.
登録日2012-10-25
公開日2013-10-02
最終更新日2014-09-10
実験手法X-RAY DIFFRACTION (4.3 Å)
主引用文献Crystal structure of Na+, K(+)-ATPase in the Na(+)-bound state.
Science, 342, 2013
4HYT
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Na,K-ATPase in the E2P state with bound ouabain and Mg2+ in the cation-binding site
分子名称: 1-O-decanoyl-beta-D-tagatofuranosyl beta-D-allopyranoside, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Laursen, M, Yatime, L, Nissen, P, Fedosova, N.U.
登録日2012-11-14
公開日2013-06-26
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (3.404 Å)
主引用文献Crystal structure of the high-affinity Na+,K+-ATPase-ouabain complex with Mg2+ bound in the cation binding site.
Proc.Natl.Acad.Sci.USA, 110, 2013
4H1W
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E1 structure of the (SR) Ca2+-ATPase in complex with Sarcolipin
分子名称: MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, POTASSIUM ION, ...
著者Bublitz, M, Winther, A.-M.L, Karlsen, J, Moller, J.V, Hansen, J.B, Buch-Pedersen, M.J, Nissen, P.
登録日2012-09-11
公開日2013-03-06
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献The sarcolipin-bound calcium pump stabilizes calcium sites exposed to the cytoplasm.
Nature, 495, 2013
6XMU
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Structure of P5A-ATPase Spf1, endogenous substrate-bound
分子名称: BERYLLIUM TRIFLUORIDE ION, MAGNESIUM ION, P5A-type ATPase, ...
著者Park, E, Sim, S.I.
登録日2020-06-30
公開日2020-09-23
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献The endoplasmic reticulum P5A-ATPase is a transmembrane helix dislocase.
Science, 369, 2020
6XMS
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Structure of P5A-ATPase Spf1, AlF4-bound form
分子名称: MAGNESIUM ION, P5A-type ATPase, TETRAFLUOROALUMINATE ION
著者Park, E, Sim, S.I.
登録日2020-06-30
公開日2020-09-23
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献The endoplasmic reticulum P5A-ATPase is a transmembrane helix dislocase.
Science, 369, 2020
7FJQ
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Cryo EM structure of lysosomal ATPase
分子名称: Polyamine-transporting ATPase 13A2, SPERMINE
著者Zhang, S.S.
登録日2021-08-04
公開日2023-03-08
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Cryo-EM structures and transport mechanism of human P5B type ATPase ATP13A2.
Cell Discov, 7, 2021
7FJP
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Cryo EM structure of lysosomal ATPase
分子名称: ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, PHOSPHATE ION, ...
著者Zhang, S.S.
登録日2021-08-04
公開日2023-03-08
実験手法ELECTRON MICROSCOPY (3 Å)
主引用文献Cryo-EM structures and transport mechanism of human P5B type ATPase ATP13A2.
Cell Discov, 7, 2021
7OP1
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Cryo-EM structure of P5B-ATPase E2PiAlF/SPM
分子名称: Cation-transporting ATPase, MAGNESIUM ION, SPERMINE, ...
著者Li, P, Gourdon, P.
登録日2021-05-28
公開日2021-06-30
最終更新日2021-09-01
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献Structure and transport mechanism of P5B-ATPases.
Nat Commun, 12, 2021
7OP8
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Cryo-EM structure of P5B-ATPase E2Pinhibit
分子名称: BERYLLIUM TRIFLUORIDE ION, Cation-transporting ATPase, MAGNESIUM ION
著者Li, P, Gourdon, P.
登録日2021-05-31
公開日2021-06-30
最終更新日2021-09-01
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Structure and transport mechanism of P5B-ATPases.
Nat Commun, 12, 2021
7OP3
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Cryo-EM structure of P5B-ATPase E2PiSPM
分子名称: Cation-transporting ATPase, SPERMINE
著者Li, P, Gronberg, C, Wang, K.T, Salustros, N, Gourdon, P.E.
登録日2021-05-28
公開日2021-06-30
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Structure and transport mechanism of P5B-ATPases.
Nat Commun, 12, 2021
7OP5
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Cryo-EM structure of P5B-ATPase E2P
分子名称: BERYLLIUM TRIFLUORIDE ION, MAGNESIUM ION, P5B-ATPase
著者Li, P, Gourdon, P.
登録日2021-05-29
公開日2021-06-30
最終更新日2021-09-01
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献Structure and transport mechanism of P5B-ATPases.
Nat Commun, 12, 2021
6YAA
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Structure of the (SR) Ca2+-ATPase bound to the inhibitor compound CAD204520 and TNP-ATP
分子名称: 4-[2-[(2~{R})-2-[3-propyl-6-(trifluoromethyloxy)-1~{H}-indol-2-yl]piperidin-1-yl]ethyl]morpholine, POTASSIUM ION, SPIRO(2,4,6-TRINITROBENZENE[1,2A]-2O',3O'-METHYLENE-ADENINE-TRIPHOSPHATE, ...
著者Heit, S, Marchesini, M, Gherli, A, Montanaro, A, Patrizi, L, Sorrentino, C, Pagliaro, L, Rompietti, C, Kitara, S, Olesen, C.E, Moller, J.V, Savi, M, Bocchi, L, Vilella, R, Rizzi, F, Baglione, M, Rastelli, G, Loiacona, C, La Starza, R, Mecucci, C, Stegmair, K, Aversa, F, Stilli, D, Lund Winther, A.M, Sportoletti, P, Dalby-Brown, W, Roti, G, Bublitz, M.
登録日2020-03-11
公開日2020-05-20
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (3.4 Å)
主引用文献Blockade of Oncogenic NOTCH1 with the SERCA Inhibitor CAD204520 in T Cell Acute Lymphoblastic Leukemia.
Cell Chem Biol, 27, 2020
6YSO
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Crystal structure of the (SR) Ca2+-ATPase solved by vanadium SAD phasing
分子名称: CHLORIDE ION, MAGNESIUM ION, OCTANOIC ACID [3S-[3ALPHA, ...
著者El Omari, K, Mohamad, N, Bountra, K, Duman, R, Romano, M, Schlegel, K, Kwong, H, Mykhaylyk, V, Olesen, C.E, Moller, J.V, Bublitz, M, Beis, K, Wagner, A.
登録日2020-04-22
公開日2020-11-04
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (3.13 Å)
主引用文献Experimental phasing with vanadium and application to nucleotide-binding membrane proteins.
Iucrj, 7, 2020
1SU4
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Crystal structure of calcium ATPase with two bound calcium ions
分子名称: CALCIUM ION, SODIUM ION, Sarcoplasmic/endoplasmic reticulum calcium ATPase 1
著者Toyoshima, C, Nakasako, M, Nomura, H, Ogawa, H.
登録日2004-03-26
公開日2004-05-04
最終更新日2017-10-11
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal structure of the calcium pump of sarcoplasmic reticulum at 2.6 A resolution
Nature, 405, 2000
1T5S
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Structure of the (SR)Ca2+-ATPase Ca2-E1-AMPPCP form
分子名称: CALCIUM ION, MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, ...
著者Sorensen, T.L.-M, Moller, J.V, Nissen, P.
登録日2004-05-05
公開日2004-06-15
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Phosphoryl transfer and calcium ion occlusion in the calcium pump.
Science, 304, 2004
7LC3
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CryoEM Structure of KdpFABC in E1-ATP state
分子名称: (2R)-3-(((2-aminoethoxy)(hydroxy)phosphoryl)oxy)-2-(palmitoyloxy)propyl (E)-octadec-9-enoate, MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, ...
著者Sweet, M.E, Larsen, C, Pedersen, B.P, Stokes, D.L.
登録日2021-01-09
公開日2021-01-27
最終更新日2024-05-29
実験手法ELECTRON MICROSCOPY (3.23 Å)
主引用文献Structural basis for potassium transport in prokaryotes by KdpFABC.
Proc.Natl.Acad.Sci.USA, 118, 2021
7LC6
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Cryo-EM Structure of KdpFABC in E2-P state with BeF3
分子名称: (2R)-3-(((2-aminoethoxy)(hydroxy)phosphoryl)oxy)-2-(palmitoyloxy)propyl (E)-octadec-9-enoate, MAGNESIUM ION, POTASSIUM ION, ...
著者Sweet, M.E, Larsen, C, Pedersen, B.P, Stokes, D.L.
登録日2021-01-09
公開日2021-01-27
最終更新日2024-05-29
実験手法ELECTRON MICROSCOPY (3.7 Å)
主引用文献Structural basis for potassium transport in prokaryotes by KdpFABC.
Proc.Natl.Acad.Sci.USA, 118, 2021
1VFP
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Crystal structure of the SR CA2+-ATPase with bound AMPPCP
分子名称: CALCIUM ION, MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, ...
著者Toyoshima, C, Mizutani, T.
登録日2004-04-18
公開日2004-07-06
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal structure of the calcium pump with a bound ATP analogue.
Nature, 430, 2004
1T5T
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Structure of the (SR)Ca2+-ATPase Ca2-E1-ADP:AlF4- form
分子名称: ADENOSINE-5'-DIPHOSPHATE, CALCIUM ION, MAGNESIUM ION, ...
著者Sorensen, T.L.-M, Moller, J.V, Nissen, P.
登録日2004-05-05
公開日2004-06-15
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Phosphoryl transfer and calcium ion occlusion in the calcium pump.
Science, 304, 2004
5XAA
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Complete structure factors and an atomic model of the calcium pump (SERCA1A) and associated phospholipids in the E2-ALF-(TG) crystals of P21212 symmetry
分子名称: 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, MAGNESIUM ION, OCTANOIC ACID [3S-[3ALPHA, ...
著者Norimatsu, Y, Hasegawa, K, Shimizu, N, Toyoshima, C.
登録日2017-03-11
公開日2017-05-24
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Protein-phospholipid interplay revealed with crystals of a calcium pump.
Nature, 545, 2017
5XA8
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Complete structure factors and an atomic model of the calcium pump (SERCA1A) and associated phospholipids in the E1-ALF4-ADP-2CA2+ crystals
分子名称: 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, ADENOSINE-5'-DIPHOSPHATE, CALCIUM ION, ...
著者Norimatsu, Y, Hasegawa, K, Shimizu, N, Toyoshima, C.
登録日2017-03-11
公開日2017-05-17
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Protein-phospholipid interplay revealed with crystals of a calcium pump.
Nature, 545, 2017
5XA9
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Complete structure factors and an atomic model of the calcium pump (SERCA1A) and associated phospholipids in the E2-ALF-(TG) crystals of C2 symmetry
分子名称: 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, MAGNESIUM ION, OCTANOIC ACID [3S-[3ALPHA, ...
著者Norimatsu, Y, Hasegawa, K, Shimizu, N, Toyoshima, C.
登録日2017-03-11
公開日2017-06-14
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Protein-phospholipid interplay revealed with crystals of a calcium pump.
Nature, 545, 2017
5XA7
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Complete structure factors and an atomic model of the calcium pump (SERCA1A) and associated phospholipids in the E1-2CA2+ crystals
分子名称: 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, CALCIUM ION, SODIUM ION, ...
著者Norimatsu, Y, Hasegawa, K, Shimizu, N, Toyoshima, C.
登録日2017-03-11
公開日2017-05-17
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Protein-phospholipid interplay revealed with crystals of a calcium pump.
Nature, 545, 2017

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