PDB: 672 件ウェブページステータス検索Chemie searchBIRD

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1S50	X-ray structure of the GluR6 ligand binding core (S1S2A) in complex with glutamate at 1.65 A resolution 分子名称: GLUTAMIC ACID, Glutamate Receptor 6 著者 Mayer, M.L. 登録日 2004-01-19 公開日 2005-02-08 最終更新日 2023-08-23 実験手法 X-RAY DIFFRACTION (1.65 Å) 主引用文献 Crystal structures of the GluR5 and GluR6 ligand binding cores: Molecular mechanisms underlying kainate receptor selectivity Neuron, 45, 2005
1S7Y	Crystal structure of the GluR6 ligand binding core in complex with glutamate at 1.75 A resolution orthorhombic form 分子名称: GLUTAMIC ACID, Glutamate receptor, ionotropic kainate 2 precursor 著者 Mayer, M.L. 登録日 2004-01-30 公開日 2005-02-08 最終更新日 2024-02-14 実験手法 X-RAY DIFFRACTION (1.75 Å) 主引用文献 Crystal structures of the GluR5 and GluR6 ligand binding cores: Molecular mechanisms underlying kainate receptor selectivity Neuron, 45, 2005
1S9T	Crystal structure of the GLUR6 ligand binding core in complex with quisqualate at 1.8A resolution 分子名称: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, CHLORIDE ION, Glutamate receptor, ... 著者 Mayer, M.L. 登録日 2004-02-05 公開日 2005-02-08 最終更新日 2023-10-25 実験手法 X-RAY DIFFRACTION (1.8 Å) 主引用文献 Crystal structures of the GluR5 and GluR6 ligand binding cores: molecular mechanisms underlying kainate receptor selectivity. Neuron, 45, 2005
1SD3	Crystal structure of the GLUR6 ligand binding core in complex with 2S,4R-4-methylglutamate at 1.8 Angstrom resolution 分子名称: 2S,4R-4-METHYLGLUTAMATE, Glutamate receptor, ionotropic kainate 2 著者 Mayer, M.L. 登録日 2004-02-12 公開日 2005-02-15 最終更新日 2023-10-25 実験手法 X-RAY DIFFRACTION (1.8 Å) 主引用文献 Crystal structures of the GluR5 and GluR6 ligand binding cores: molecular mechanisms underlying kainate receptor selectivity. Neuron, 45, 2005
1SYI	X-RAY STRUCTURE OF THE Y702F MUTANT OF THE GLUR2 LIGAND-BINDING CORE (S1S2J) IN COMPLEX WITH (S)-CPW399 AT 2.1 A RESOLUTION. 分子名称: (S)-2-AMINO-3-(1,3,5,7-PENTAHYDRO-2,4-DIOXO-CYCLOPENTA[E]PYRIMIDIN-1-YL) PROIONIC ACID, Glutamate receptor 2 著者 Frandsen, A, Pickering, D.S, Vestergaard, B, Kasper, C, Nielsen, B.B, Greenwood, J.R, Campiani, G, Gajhede, M, Schousboe, A, Kastrup, J.S. 登録日 2004-04-01 公開日 2005-03-22 最終更新日 2023-08-23 実験手法 X-RAY DIFFRACTION (2.1 Å) 主引用文献 Tyr702 Is an Important Determinant of Agonist Binding and Domain Closure of the Ligand-Binding Core of GluR2. Mol.Pharmacol., 67, 2005
1SYH	X-RAY STRUCTURE OF THE GLUR2 LIGAND-BINDING CORE (S1S2J) IN COMPLEX WITH (S)-CPW399 AT 1.85 A RESOLUTION. 分子名称: (S)-2-AMINO-3-(1,3,5,7-PENTAHYDRO-2,4-DIOXO-CYCLOPENTA[E]PYRIMIDIN-1-YL) PROIONIC ACID, Glutamate receptor 2 著者 Frandsen, A, Pickering, D.S, Vestergaard, B, Kasper, C, Nielsen, B.B, Greenwood, J.R, Campiani, G, Gajhede, M, Schousboe, A, Kastrup, J.S. 登録日 2004-04-01 公開日 2005-03-22 最終更新日 2023-08-23 実験手法 X-RAY DIFFRACTION (1.8 Å) 主引用文献 Tyr702 Is an Important Determinant of Agonist Binding and Domain Closure of the Ligand-Binding Core of GluR2. Mol.Pharmacol., 67, 2005
1TT1	CRYSTAL STRUCTURE OF THE GLUR6 LIGAND BINDING CORE IN COMPLEX WITH KAINATE 1.93 A RESOLUTION 分子名称: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, Glutamate receptor, ionotropic kainate 2 著者 Mayer, M.L. 登録日 2004-06-21 公開日 2005-02-08 最終更新日 2023-08-23 実験手法 X-RAY DIFFRACTION (1.93 Å) 主引用文献 Crystal structures of the GluR5 and GluR6 ligand binding cores: Molecular mechanisms underlying kainate receptor selectivity Neuron, 45, 2005
1TXF	CRYSTAL STRUCTURE OF THE GLUR5 LIGAND BINDING CORE IN COMPLEX WITH GLUTAMATE AT 2.1 ANGSTROM RESOLUTION 分子名称: GLUTAMIC ACID, Glutamate receptor, ionotropic kainate 1 著者 Mayer, M.L. 登録日 2004-07-04 公開日 2005-02-08 最終更新日 2023-08-23 実験手法 X-RAY DIFFRACTION (2.1 Å) 主引用文献 Crystal structures of the GluR5 and GluR6 ligand binding cores: Molecular mechanisms underlying kainate receptor selectivity Neuron, 45, 2005
1XHY	X-ray structure of the Y702F mutant of the GluR2 ligand-binding core (S1S2J) in complex with kainate at 1.85 A resolution 分子名称: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, Glutamate receptor, SULFATE ION 著者 Frandsen, A, Pickering, D.S, Vestergaard, B, Kasper, C, Nielsen, B.B, Greenwood, J.R, Campiani, G, Gajhede, M, Schousboe, A, Kastrup, J.S. 登録日 2004-09-21 公開日 2005-03-22 最終更新日 2023-08-23 実験手法 X-RAY DIFFRACTION (1.85 Å) 主引用文献 Tyr702 Is an Important Determinant of Agonist Binding and Domain Closure of the Ligand-Binding Core of GluR2. Mol.Pharmacol., 67, 2005
1Y1M	Crystal structure of the NR1 ligand binding core in complex with cycloleucine 分子名称: 1-AMINOCYCLOPENTANECARBOXYLIC ACID, Glutamate [NMDA] receptor subunit zeta 1 著者 Inanobe, A, Gouaux, E. 登録日 2004-11-18 公開日 2005-07-12 最終更新日 2017-07-26 実験手法 X-RAY DIFFRACTION (1.8 Å) 主引用文献 Mechanism of Partial Agonist Action at the NR1 Subunit of NMDA Receptors. Neuron, 47, 2005
1Y1Z	Crystal structure of the NR1 ligand binding core in complex with ACBC 分子名称: 1-AMINOCYCLOBUTANECARBOXLIC ACID, Glutamate [NMDA] receptor subunit zeta 1 著者 Inanobe, A, Gouaux, E. 登録日 2004-11-19 公開日 2005-07-12 最終更新日 2017-07-26 実験手法 X-RAY DIFFRACTION (1.5 Å) 主引用文献 Mechanism of Partial Agonist Action at the NR1 Subunit of NMDA Receptors. Neuron, 47, 2005
1Y20	Crystal structure of the NR1 ligand-binding core in complex with ACPC 分子名称: 1-AMINOCYCLOPROPANECARBOXYLIC ACID, Glutamate [NMDA] receptor subunit zeta 1 著者 Inanobe, A, Gouaux, E. 登録日 2004-11-19 公開日 2005-07-12 最終更新日 2017-07-26 実験手法 X-RAY DIFFRACTION (1.4 Å) 主引用文献 Mechanism of Partial Agonist Action at the NR1 Subunit of NMDA Receptors. Neuron, 47, 2005
1WVJ	Exploring the GluR2 ligand-binding core in complex with the bicyclic AMPA analogue (S)-4-AHCP 分子名称: 3-(3-HYDROXY-7,8-DIHYDRO-6H-CYCLOHEPTA[D]ISOXAZOL-4-YL)-L-ALANINE, GLYCEROL, SULFATE ION, ... 著者 Nielsen, B.B, Pickering, D.S, Greenwood, J.R, Brehm, L, Gajhede, M, Schousboe, A, Kastrup, J.S. 登録日 2004-12-15 公開日 2005-04-26 最終更新日 2023-10-25 実験手法 X-RAY DIFFRACTION (1.75 Å) 主引用文献 Exploring the GluR2 ligand-binding core in complex with the bicyclical AMPA analogue (S)-4-AHCP FEBS J., 272, 2005
1YAE	Structure of the Kainate Receptor Subunit GluR6 Agonist Binding Domain Complexed with Domoic Acid 分子名称: (2S,3S,4S)-2-CARBOXY-4-[(1Z,3E,5R)-5-CARBOXY-1-METHYL-1,3-HEXADIENYL]-3-PYRROLIDINEACETIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor, ... 著者 Nanao, M.H, Green, T, Stern-Bach, Y, Heinemann, S.F, Choe, S. 登録日 2004-12-17 公開日 2005-02-01 最終更新日 2023-08-23 実験手法 X-RAY DIFFRACTION (3.11 Å) 主引用文献 Structure of the kainate receptor subunit GluR6 agonist-binding domain complexed with domoic acid. Proc.Natl.Acad.Sci.USA, 102, 2005
1YCJ	Crystal structure of the kainate receptor GluR5 ligand-binding core in complex with (S)-glutamate 分子名称: GLUTAMIC ACID, Ionotropic glutamate receptor 5, SULFATE ION 著者 Naur, P, Vestergaard, B, Skov, L.K, Egebjerg, J, Gajhede, M, Kastrup, J.S. 登録日 2004-12-22 公開日 2005-02-01 最終更新日 2023-10-25 実験手法 X-RAY DIFFRACTION (1.95 Å) 主引用文献 Crystal structure of the kainate receptor GluR5 ligand-binding core in complex with (S)-glutamate Febs Lett., 579, 2005
2A5S	Crystal Structure Of The NR2A Ligand Binding Core In Complex With Glutamate 分子名称: GLUTAMIC ACID, N-methyl-D-aspartate receptor NMDAR2A subunit 著者 Furukawa, H, Singh, S.K, Mancusso, R, Gouaux, E. 登録日 2005-06-30 公開日 2005-11-15 最終更新日 2017-07-26 実験手法 X-RAY DIFFRACTION (1.7 Å) 主引用文献 Subunit arrangement and function in NMDA receptors Nature, 438, 2005
2A5T	Crystal Structure Of The NR1/NR2A ligand-binding cores complex 分子名称: GLUTAMIC ACID, GLYCINE, N-methyl-D-aspartate receptor NMDAR1-4a subunit, ... 著者 Furukawa, H, Singh, S.K, Mancusso, R, Gouaux, E. 登録日 2005-06-30 公開日 2005-11-15 最終更新日 2017-07-26 実験手法 X-RAY DIFFRACTION (2 Å) 主引用文献 Subunit arrangement and function in NMDA receptors Nature, 438, 2005
2AIX	X-ray structure of the GLUR2 ligand-binding core (S1S2J) in complex with (s)-thio-atpa at 2.2 a resolution. 分子名称: (S)-2-AMINO-3-(3-HYDROXY-5-TERT-BUTYLISOTHIAZOL-4-YL) PROPRIONIC ACID, Glutamate receptor 2 著者 Kastrup, J.S. 登録日 2005-08-01 公開日 2005-08-09 最終更新日 2023-08-23 実験手法 X-RAY DIFFRACTION (2.17 Å) 主引用文献 Distinct kinetics of ionotropic glutamate receptor 2 splice variants characterized by fast agonist application and crystallization of a receptor-ligand complex. To be Published
2AL4	CRYSTAL STRUCTURE OF THE GLUR2 LIGAND BINDING CORE (S1S2J) IN COMPLEX WITH quisqualate and CX614. 分子名称: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, 2,3,6A,7,8,9-HEXAHYDRO-11H-[1,4]DIOXINO[2,3-G]PYRROLO[2,1-B][1,3]BENZOXAZIN-11-ONE, Glutamate receptor 2, ... 著者 Jin, R, Clark, S, Weeks, A.M, Dudman, J.T, Gouaux, E, Partin, K.M. 登録日 2005-08-04 公開日 2005-10-25 最終更新日 2023-08-23 実験手法 X-RAY DIFFRACTION (1.7 Å) 主引用文献 Mechanism of positive allosteric modulators acting on AMPA receptors. J.Neurosci., 25, 2005
2AL5	Crystal structure of the GluR2 ligand binding core (S1S2J) in complex with fluoro-willardiine and aniracetam 分子名称: 1-(4-METHOXYBENZOYL)-2-PYRROLIDINONE, 2-AMINO-3-(5-FLUORO-2,4-DIOXO-3,4-DIHYDRO-2H-PYRIMIDIN-1-YL)-PROPIONIC ACID, Glutamate receptor 2 著者 Jin, R, Clark, S, Weeks, A.M, Dudman, J.T, Gouaux, E, Partin, K.M. 登録日 2005-08-04 公開日 2005-10-25 最終更新日 2023-08-23 実験手法 X-RAY DIFFRACTION (1.65 Å) 主引用文献 Mechanism of positive allosteric modulators acting on AMPA receptors. J.Neurosci., 25, 2005
2ANJ	Crystal Structure of the Glur2 Ligand Binding Core (S1S2J-Y450W) Mutant in Complex With the Partial Agonist Kainic Acid at 2.1 A Resolution 分子名称: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, Glutamate receptor 2 著者 Holm, M.M, Naur, P, Vestergaard, B, Geballe, M.T, Gajhede, M, Kastrup, J.S, Traynelis, S.F, Egebjerg, J. 登録日 2005-08-11 公開日 2005-08-30 最終更新日 2023-08-23 実験手法 X-RAY DIFFRACTION (2.1 Å) 主引用文献 A Binding Site Tyrosine Shapes Desensitization Kinetics and Agonist Potency at GluR2: a mutagenic, kinetic, and crystallographic study J.Biol.Chem., 280, 2005
2F36	Crystal Structure of the GluR5 Ligand Binding Core Dimer with Glutamate At 2.1 Angstroms Resolution 分子名称: GLUTAMATE RECEPTOR, IONOTROPIC KAINATE 1, GLUTAMIC ACID, ... 著者 Mayer, M.L. 登録日 2005-11-18 公開日 2006-04-04 最終更新日 2023-08-23 実験手法 X-RAY DIFFRACTION (2.11 Å) 主引用文献 Crystal structures of the kainate receptor GluR5 ligand binding core dimer with novel GluR5-selective antagonists. J.Neurosci., 26, 2006
2F34	Crystal Structure of the GluR5 Ligand Binding Core Dimer with UBP310 At 1.74 Angstroms Resolution 分子名称: (S)-1-(2-AMINO-2-CARBOXYETHYL)-3(2-CARBOXYTHIOPHENE-3-YL-METHYL)-5-METHYLPYRIMIDINE-2,4-DIONE, CHLORIDE ION, GLUTAMATE RECEPTOR, ... 著者 Mayer, M.L. 登録日 2005-11-18 公開日 2006-04-04 最終更新日 2023-08-23 実験手法 X-RAY DIFFRACTION (1.74 Å) 主引用文献 Crystal structures of the kainate receptor GluR5 ligand binding core dimer with novel GluR5-selective antagonists. J.Neurosci., 26, 2006
2F35	Crystal Structure of the GluR5 Ligand Binding Core with UBP302 At 1.87 Angstroms Resolution 分子名称: (S)-1-(2-AMINO-2-CARBOXYETHYL)-3-(2-CARBOXYBENZYL)PYRIMIDINE-2,4-DIONE, CHLORIDE ION, GLUTAMATE RECEPTOR, ... 著者 Mayer, M.L. 登録日 2005-11-18 公開日 2006-04-04 最終更新日 2024-04-03 実験手法 X-RAY DIFFRACTION (1.87 Å) 主引用文献 Crystal structures of the kainate receptor GluR5 ligand binding core dimer with novel GluR5-selective antagonists. J.Neurosci., 26, 2006
2GFE	Crystal structure of the GluR2 A476E S673D Ligand Binding Core Mutant at 1.54 Angstroms Resolution 分子名称: GLUTAMIC ACID, Glutamate receptor 2, ZINC ION 著者 Mayer, M.L. 登録日 2006-03-21 公開日 2006-08-22 最終更新日 2023-08-30 実験手法 X-RAY DIFFRACTION (1.54 Å) 主引用文献 Interdomain interactions in AMPA and kainate receptors regulate affinity for glutamate. J.Neurosci., 26, 2006

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