7M2F
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7m2f by Molmil](/molmil-images/mine/7m2f) | CDK2 with compound 14 inhibitor with carboxylate | 分子名称: | Cyclin-dependent kinase 2, [(1r,4r)-4-{4-[4-(5-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]-3,6-dihydropyridin-1(2H)-yl}cyclohexyl]acetic acid | 著者 | Longenecker, K.L, Qiu, W, Korepanova, A, Tong, Y. | 登録日 | 2021-03-16 | 公開日 | 2021-07-07 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.632 Å) | 主引用文献 | Balancing Properties with Carboxylates: A Lead Optimization Campaign for Selective and Orally Active CDK9 Inhibitors. Acs Med.Chem.Lett., 12, 2021
|
|
7M20
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7m20 by Molmil](/molmil-images/mine/7m20) | 18-mer HeLa-tubulin rings in complex with Cryptophycin 1 | 分子名称: | Cryptophycin 1, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ... | 著者 | Eren, E. | 登録日 | 2021-03-15 | 公開日 | 2021-09-08 | 最終更新日 | 2024-05-29 | 実験手法 | ELECTRON MICROSCOPY (3.84 Å) | 主引用文献 | Conformational changes in tubulin upon binding cryptophycin-52 reveal its mechanism of action. J.Biol.Chem., 297, 2021
|
|
7EDD
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7edd by Molmil](/molmil-images/mine/7edd) | |
7NVR
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7nvr by Molmil](/molmil-images/mine/7nvr) | Human Mediator with RNA Polymerase II Pre-initiation complex | 分子名称: | CDK-activating kinase assembly factor MAT1, Cyclin-H, Cyclin-dependent kinase 7, ... | 著者 | Rengachari, S, Schilbach, S, Aibara, S, Cramer, P. | 登録日 | 2021-03-15 | 公開日 | 2021-05-05 | 最終更新日 | 2024-07-10 | 実験手法 | ELECTRON MICROSCOPY (4.5 Å) | 主引用文献 | Structures of mammalian RNA polymerase II pre-initiation complexes. Nature, 594, 2021
|
|
7NVQ
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7nvq by Molmil](/molmil-images/mine/7nvq) | |
7NUY
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7nuy by Molmil](/molmil-images/mine/7nuy) | |
7NUZ
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7nuz by Molmil](/molmil-images/mine/7nuz) | Proteinase K structure at atomic resolution from crystals grown in agarose gel | 分子名称: | GLYCEROL, MAGNESIUM ION, NITRATE ION, ... | 著者 | Gavira, J.A, Artusio, F, Castellvi, A, Pisano, R. | 登録日 | 2021-03-15 | 公開日 | 2022-01-19 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.09 Å) | 主引用文献 | Tuning Transport Phenomena in Agarose Gels for the Control of Protein Nucleation Density and Crystal Form Crystals, 2021
|
|
7NVN
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7nvn by Molmil](/molmil-images/mine/7nvn) | Human TRiC complex in closed state with nanobody and tubulin bound | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ALUMINUM FLUORIDE, MAGNESIUM ION, ... | 著者 | Kelly, J.J, Chi, G, Bulawa, C, Paavilainen, V.O, Bountra, C, Huiskonen, J.T, Yue, W. | 登録日 | 2021-03-15 | 公開日 | 2022-03-02 | 最終更新日 | 2022-06-01 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Snapshots of actin and tubulin folding inside the TRiC chaperonin. Nat.Struct.Mol.Biol., 29, 2022
|
|
7NVM
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7nvm by Molmil](/molmil-images/mine/7nvm) | Human TRiC complex in closed state with nanobody Nb18, actin and PhLP2A bound | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, ALUMINUM FLUORIDE, Actin, ... | 著者 | Kelly, J.J, Chi, G, Bulawa, C, Paavilainen, V.O, Bountra, C, Huiskonen, J.T, Yue, W, Structural Genomics Consortium (SGC) | 登録日 | 2021-03-15 | 公開日 | 2022-03-02 | 最終更新日 | 2022-06-01 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Snapshots of actin and tubulin folding inside the TRiC chaperonin. Nat.Struct.Mol.Biol., 29, 2022
|
|
7M1P
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7m1p by Molmil](/molmil-images/mine/7m1p) | Human ABCA4 structure in the unbound state | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Retinal-specific phospholipid-transporting ATPase ABCA4, ... | 著者 | Scortecci, J.F, Van Petegem, F, Molday, R.S. | 登録日 | 2021-03-14 | 公開日 | 2021-09-08 | 最終更新日 | 2021-10-20 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Cryo-EM structures of the ABCA4 importer reveal mechanisms underlying substrate binding and Stargardt disease. Nat Commun, 12, 2021
|
|
7M1Q
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7m1q by Molmil](/molmil-images/mine/7m1q) | Human ABCA4 structure in complex with N-ret-PE | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, MAGNESIUM ION, Retinal-specific phospholipid-transporting ATPase ABCA4, ... | 著者 | Scortecci, J.F, Van Petegem, F, Molday, R.S. | 登録日 | 2021-03-14 | 公開日 | 2021-09-08 | 最終更新日 | 2021-10-20 | 実験手法 | ELECTRON MICROSCOPY (2.92 Å) | 主引用文献 | Cryo-EM structures of the ABCA4 importer reveal mechanisms underlying substrate binding and Stargardt disease. Nat Commun, 12, 2021
|
|
7M1K
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7m1k by Molmil](/molmil-images/mine/7m1k) | Crystal structure of dehaloperoxidase B in complex with 2,6-difluorophenol | 分子名称: | 2,6-DIFLUOROPHENOL, Dehaloperoxidase B, GLYCEROL, ... | 著者 | Ghiladi, R.A, de Serrano, V.S, Malewschik, T. | 登録日 | 2021-03-13 | 公開日 | 2022-08-31 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.795 Å) | 主引用文献 | Bridging the functional gap between reactivity and inhibition in dehaloperoxidase B from Amphitrite ornata: Mechanistic and structural studies with 2,4- and 2,6-dihalophenols. J.Inorg.Biochem., 236, 2022
|
|
7M1J
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7m1j by Molmil](/molmil-images/mine/7m1j) | Crystal structure of dehaloperoxidase B in complex with 2,6-dibromophenol | 分子名称: | 2,6-bis(bromanyl)phenol, Dehaloperoxidase B, GLYCEROL, ... | 著者 | Ghiladi, R.A, de Serrano, V.S, Malewschik, T. | 登録日 | 2021-03-13 | 公開日 | 2022-08-31 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.554 Å) | 主引用文献 | Bridging the functional gap between reactivity and inhibition in dehaloperoxidase B from Amphitrite ornata: Mechanistic and structural studies with 2,4- and 2,6-dihalophenols. J.Inorg.Biochem., 236, 2022
|
|
7M1I
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7m1i by Molmil](/molmil-images/mine/7m1i) | Crystal structure of dehaloperoxidase B in complex with 2,6-dichlorophenol | 分子名称: | 2,6-dichlorophenol, Dehaloperoxidase B, GLYCEROL, ... | 著者 | Ghiladi, R.A, de Serrano, V.S, Malewschik, T. | 登録日 | 2021-03-13 | 公開日 | 2022-08-17 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.66 Å) | 主引用文献 | Bridging the functional gap between reactivity and inhibition in dehaloperoxidase B from Amphitrite ornata: Mechanistic and structural studies with 2,4- and 2,6-dihalophenols. J.Inorg.Biochem., 236, 2022
|
|
7ECY
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7ecy by Molmil](/molmil-images/mine/7ecy) | EV-D68 in complex with 2H12 Fab (State 3) | 分子名称: | Capsid protein VP1, Capsid protein VP2, Capsid protein VP3, ... | 著者 | Xu, C, Cong, Y. | 登録日 | 2021-03-13 | 公開日 | 2021-03-31 | 最終更新日 | 2021-06-02 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Functional and structural characterization of a two-MAb cocktail for delayed treatment of enterovirus D68 infections. Nat Commun, 12, 2021
|
|
7M18
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7m18 by Molmil](/molmil-images/mine/7m18) | HeLa-tubulin in complex with cryptophycin 1 | 分子名称: | Cryptophycin 1, GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, ... | 著者 | Eren, E. | 登録日 | 2021-03-12 | 公開日 | 2021-09-08 | 最終更新日 | 2024-05-29 | 実験手法 | ELECTRON MICROSCOPY (3.38 Å) | 主引用文献 | Conformational changes in tubulin upon binding cryptophycin-52 reveal its mechanism of action. J.Biol.Chem., 297, 2021
|
|
7NUM
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7num by Molmil](/molmil-images/mine/7num) | |
7NUO
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7nuo by Molmil](/molmil-images/mine/7nuo) | Rhinovirus 14 empty particle at pH 6.2 | 分子名称: | Genome polyprotein, P1 | 著者 | Hrebik, D, Plevka, P. | 登録日 | 2021-03-12 | 公開日 | 2021-05-19 | 最終更新日 | 2024-07-10 | 実験手法 | ELECTRON MICROSCOPY (3.9 Å) | 主引用文献 | ICAM-1 induced rearrangements of capsid and genome prime rhinovirus 14 for activation and uncoating. Proc.Natl.Acad.Sci.USA, 118, 2021
|
|
7NUL
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7nul by Molmil](/molmil-images/mine/7nul) | |
7NUQ
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7nuq by Molmil](/molmil-images/mine/7nuq) | Rhinovirus 14 virion-like at pH 6.2 | 分子名称: | Genome polyprotein, Octanucleotide | 著者 | Hrebik, D, Plevka, P. | 登録日 | 2021-03-12 | 公開日 | 2021-05-19 | 最終更新日 | 2024-07-10 | 実験手法 | ELECTRON MICROSCOPY (2.8 Å) | 主引用文献 | ICAM-1 induced rearrangements of capsid and genome prime rhinovirus 14 for activation and uncoating. Proc.Natl.Acad.Sci.USA, 118, 2021
|
|
7NUN
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7nun by Molmil](/molmil-images/mine/7nun) | |
7NUF
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7nuf by Molmil](/molmil-images/mine/7nuf) | Vaccinia virus protein 018 in complex with STAT1 | 分子名称: | ACETYL GROUP, SULFATE ION, Signal transducer and activator of transcription 1-alpha/beta, ... | 著者 | Pantelejevs, T, Talbot-Cooper, C, Smith, G.L, Hyvonen, M. | 登録日 | 2021-03-12 | 公開日 | 2021-07-28 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.0004015 Å) | 主引用文献 | Poxviruses and paramyxoviruses use a conserved mechanism of STAT1 antagonism to inhibit interferon signaling. Cell Host Microbe, 30, 2022
|
|
7M0S
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7m0s by Molmil](/molmil-images/mine/7m0s) | |
7EBT
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7ebt by Molmil](/molmil-images/mine/7ebt) | Crystal structure of Aedes aegypti Noppera-bo, glutathione S-transferase epsilon 8, in glutathione-bound form | 分子名称: | CALCIUM ION, GLUTATHIONE, Glutathione transferase | 著者 | Inaba, K, Koiwai, K, Senda, M, Senda, T, Niwa, R. | 登録日 | 2021-03-11 | 公開日 | 2022-01-26 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.51 Å) | 主引用文献 | Molecular action of larvicidal flavonoids on ecdysteroidogenic glutathione S-transferase Noppera-bo in Aedes aegypti. Bmc Biol., 20, 2022
|
|
7EBW
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7ebw by Molmil](/molmil-images/mine/7ebw) | Crystal structure of Aedes aegypti Noppera-bo, glutathione S-transferase epsilon 8, in desmethylglycitein and glutathione-bound form | 分子名称: | 6,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one, CALCIUM ION, GLUTATHIONE, ... | 著者 | Inaba, K, Koiwai, K, Senda, M, Senda, T, Niwa, R. | 登録日 | 2021-03-11 | 公開日 | 2022-01-26 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Molecular action of larvicidal flavonoids on ecdysteroidogenic glutathione S-transferase Noppera-bo in Aedes aegypti. Bmc Biol., 20, 2022
|
|