3ERK
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![BU of 3erk by Molmil](/molmil-images/mine/3erk) | THE COMPLEX STRUCTURE OF THE MAP KINASE ERK2/SB220025 | 分子名称: | 4-(4-FLUOROPHENYL)-1-(4-PIPERIDINYL)-5-(2-AMINO-4-PYRIMIDINYL)-IMIDAZOLE, EXTRACELLULAR REGULATED KINASE 2 | 著者 | Wang, Z, Canagarajah, B, Boehm, J.C, Cobb, M.H, Young, P.R, Abdel-Meguid, S, Adams, J.L, Goldsmith, E.J. | 登録日 | 1998-07-09 | 公開日 | 1999-07-22 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structural basis of inhibitor selectivity in MAP kinases. Structure, 6, 1998
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1Y0J
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![BU of 1y0j by Molmil](/molmil-images/mine/1y0j) | Zinc fingers as protein recognition motifs: structural basis for the GATA-1/Friend of GATA interaction | 分子名称: | Erythroid transcription factor, ZINC ION, Zinc-finger protein ush | 著者 | Liew, C.K, Simpson, R.J.Y, Kwan, A.H.Y, Crofts, L.A, Loughlin, F.E, Matthews, J.M, Crossley, M, Mackay, J.P. | 登録日 | 2004-11-15 | 公開日 | 2005-01-25 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Zinc fingers as protein recognition motifs: Structural basis for the GATA-1/Friend of GATA interaction Proc.Natl.Acad.Sci.Usa, 102, 2005
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7E29
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![BU of 7e29 by Molmil](/molmil-images/mine/7e29) | Crystal Structure of Saccharomyces cerevisiae Ioc4 PWWP domain fused with MBP | 分子名称: | Maltose/maltodextrin-binding periplasmic protein,ISWI one complex protein 4, alpha-D-glucopyranose-(1-4)-alpha-D-glucopyranose | 著者 | Li, J, Smolle, M, Liang, H, Liu, Y. | 登録日 | 2021-02-05 | 公開日 | 2022-02-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.303 Å) | 主引用文献 | H3K36 methylation and DNA-binding both promote Ioc4 recruitment and Isw1b remodeler function. Nucleic Acids Res., 50, 2022
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1TRU
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6FIC
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![BU of 6fic by Molmil](/molmil-images/mine/6fic) | Bivalent Inhibitor UNC4512 Bound to the TAF1 Bromodomain Tandem | 分子名称: | 3-azanyl-2-[3-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[2-[[3-azanyl-1-[[2-[[3-methyl-6-[4-methyl-3-(methylsulfonyl-$l^{2}-azanyl)cyclohexa-1,3,5-trien-1-yl]-[1,2,4]triazolo[4,3-b]pyridazin-8-yl]-$l^{2}-azanyl]-2-oxidanylidene-ethyl]amino]-1-oxidanylidene-propan-2-yl]amino]-2-oxidanylidene-ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-~{N}-[3-[[3-methyl-6-[4-methyl-3-(methylsulfonylamino)phenyl]-[1,2,4]triazolo[4,3-b]pyridazin-8-yl]amino]-3-oxidanylidene-propyl]propanamide, Transcription initiation factor TFIID subunit 1 | 著者 | Mathea, S, Suh, J.L, Salah, E, Tallant, C, Siejka, P, Pike, A.C.W, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, James, L.I, Frye, S.V, Knapp, S. | 登録日 | 2018-01-17 | 公開日 | 2018-01-31 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2.18 Å) | 主引用文献 | Bivalent Inhibitor UNC4512 Bound to the TAF1 Bromodomain Tandem To Be Published
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1TRW
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1TRV
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6F07
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![BU of 6f07 by Molmil](/molmil-images/mine/6f07) | CBF3 Core Complex | 分子名称: | Centromere DNA-binding protein complex CBF3 subunit B, Suppressor of kinetochore protein 1, ZINC ION | 著者 | Leber, V, Singleton, M.R. | 登録日 | 2017-11-17 | 公開日 | 2017-12-13 | 最終更新日 | 2019-12-11 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Structural basis for assembly of the CBF3 kinetochore complex. EMBO J., 37, 2018
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4HC9
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![BU of 4hc9 by Molmil](/molmil-images/mine/4hc9) | DNA binding by GATA transcription factor-complex 3 | 分子名称: | DNA (5'-D(*AP*AP*GP*GP*TP*TP*AP*TP*CP*TP*CP*TP*GP*AP*TP*TP*TP*AP*GP*G)-3'), DNA (5'-D(*TP*TP*CP*CP*TP*AP*AP*AP*TP*CP*AP*GP*AP*GP*AP*TP*AP*AP*CP*C)-3'), Trans-acting T-cell-specific transcription factor GATA-3, ... | 著者 | Chen, Y, Bates, D.L, Dey, R, Chen, L. | 登録日 | 2012-09-28 | 公開日 | 2012-12-05 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | DNA Binding by GATA Transcription Factor Suggests Mechanisms of DNA Looping and Long-Range Gene Regulation. Cell Rep, 2, 2012
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6C16
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1ERW
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![BU of 1erw by Molmil](/molmil-images/mine/1erw) | HUMAN THIOREDOXIN DOUBLE MUTANT WITH CYS 32 REPLACED BY SER AND CYS 35 REPLACED BY SER | 分子名称: | THIOREDOXIN | 著者 | Weichsel, A, Gasdaska, J.R, Powis, G, Montfort, W.R. | 登録日 | 1996-02-07 | 公開日 | 1996-10-14 | 最終更新日 | 2021-11-03 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystal structures of reduced, oxidized, and mutated human thioredoxins: evidence for a regulatory homodimer. Structure, 4, 1996
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1ERV
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![BU of 1erv by Molmil](/molmil-images/mine/1erv) | HUMAN THIOREDOXIN MUTANT WITH CYS 73 REPLACED BY SER (REDUCED FORM) | 分子名称: | THIOREDOXIN | 著者 | Weichsel, A, Gasdaska, J.R, Powis, G, Montfort, W.R. | 登録日 | 1996-02-07 | 公開日 | 1996-10-14 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Crystal structures of reduced, oxidized, and mutated human thioredoxins: evidence for a regulatory homodimer. Structure, 4, 1996
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1ERT
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![BU of 1ert by Molmil](/molmil-images/mine/1ert) | HUMAN THIOREDOXIN (REDUCED FORM) | 分子名称: | THIOREDOXIN | 著者 | Weichsel, A, Gasdaska, J.R, Powis, G, Montfort, W.R. | 登録日 | 1996-02-07 | 公開日 | 1996-10-14 | 最終更新日 | 2018-04-18 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Crystal structures of reduced, oxidized, and mutated human thioredoxins: evidence for a regulatory homodimer. Structure, 4, 1996
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3EZG
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1ERU
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![BU of 1eru by Molmil](/molmil-images/mine/1eru) | HUMAN THIOREDOXIN (OXIDIZED FORM) | 分子名称: | THIOREDOXIN | 著者 | Weichsel, A, Gasdaska, J.R, Powis, G, Montfort, W.R. | 登録日 | 1996-02-07 | 公開日 | 1996-08-01 | 最終更新日 | 2018-04-18 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Crystal structures of reduced, oxidized, and mutated human thioredoxins: evidence for a regulatory homodimer. Structure, 4, 1996
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1TRS
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6W9E
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![BU of 6w9e by Molmil](/molmil-images/mine/6w9e) | Crystal Structure of Human CDK9/cyclinT1 in complex with MC180295 | 分子名称: | (4-amino-2-{[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanone, (4-amino-2-{[(1S,2S,4R)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanone, Cyclin-T1, ... | 著者 | Zhang, P, Wu, J. | 登録日 | 2020-03-22 | 公開日 | 2021-09-01 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Comparative Modeling of CDK9 Inhibitors to Explore Selectivity and Structure-Activity Relationships To Be Published
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6WJ3
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2HSH
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8EU9
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![BU of 8eu9 by Molmil](/molmil-images/mine/8eu9) | Class1 of the INO80-Nucleosome complex | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, Actin-related protein 5, Chromatin-remodeling ATPase INO80, ... | 著者 | Wu, H, Munoz, E, Gourdet, M, Cheng, Y.F, Narlikar, G. | 登録日 | 2022-10-18 | 公開日 | 2023-07-12 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (3.48 Å) | 主引用文献 | Reorientation of INO80 on hexasomes reveals basis for mechanistic versatility. Science, 381, 2023
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8ETU
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![BU of 8etu by Molmil](/molmil-images/mine/8etu) | Class2 of the INO80-Hexasome complex | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, Actin-related protein 5, Chromatin-remodeling ATPase INO80, ... | 著者 | Wu, H, Munoz, E, Gourdet, M, Cheng, Y.F, Narlikar, G. | 登録日 | 2022-10-17 | 公開日 | 2023-07-19 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (2.8 Å) | 主引用文献 | Reorientation of INO80 on hexasomes reveals basis for mechanistic versatility. Science, 381, 2023
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8ETW
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![BU of 8etw by Molmil](/molmil-images/mine/8etw) | Class3 of INO80-Hexasome complex | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, Actin-related protein 5, Chromatin-remodeling ATPase INO80, ... | 著者 | Wu, H, Munoz, E, Gourdet, M, Narlikar, G, Cheng, Y.F. | 登録日 | 2022-10-17 | 公開日 | 2023-07-19 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (2.64 Å) | 主引用文献 | Reorientation of INO80 on hexasomes reveals basis for mechanistic versatility. Science, 381, 2023
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8ETS
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![BU of 8ets by Molmil](/molmil-images/mine/8ets) | Class1 of the INO80-Hexasome complex | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, Actin-related protein 5, Chromatin-remodeling ATPase INO80, ... | 著者 | Wu, H, Munoz, E, Gourdet, M, Cheng, Y.F, Narlikar, G. | 登録日 | 2022-10-17 | 公開日 | 2023-07-19 | 最終更新日 | 2024-06-19 | 実験手法 | ELECTRON MICROSCOPY (3.04 Å) | 主引用文献 | Reorientation of INO80 on hexasomes reveals basis for mechanistic versatility. Science, 381, 2023
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6WJ2
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![BU of 6wj2 by Molmil](/molmil-images/mine/6wj2) | CryoEM structure of the SLC38A9-RagA-RagC-Ragulator complex in the pre-GAP state | 分子名称: | 9-{5-O-[(S)-hydroxy{[(R)-hydroxy(thiophosphonooxy)phosphoryl]oxy}phosphoryl]-alpha-L-arabinofuranosyl}-3,9-dihydro-1H-purine-2,6-dione, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ... | 著者 | Fromm, S.A, Hurley, J.H. | 登録日 | 2020-04-11 | 公開日 | 2020-09-02 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (3.2 Å) | 主引用文献 | Structural mechanism for amino acid-dependent Rag GTPase nucleotide state switching by SLC38A9. Nat.Struct.Mol.Biol., 27, 2020
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2HXK
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