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1EZX
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CRYSTAL STRUCTURE OF A SERPIN:PROTEASE COMPLEX
分子名称: ALPHA-1-ANTITRYPSIN, TRYPSIN
著者Huntington, J.A, Carrell, R.W.
登録日2000-05-12
公開日2000-10-25
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structure of a serpin-protease complex shows inhibition by deformation.
Nature, 407, 2000
2IEZ
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Crystal Structure of mouse Rab27b bound to GDP in monoclinic space group
分子名称: CALCIUM ION, GUANOSINE-5'-DIPHOSPHATE, Ras-related protein Rab-27B
著者Chavas, L.M.G, Torii, S, Kamikubo, H, Kawasaki, M, Ihara, K, Kato, R, Kataoka, M, Izumi, T, Wakatsuki, S.
登録日2006-09-19
公開日2007-05-01
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure of the small GTPase Rab27b shows an unexpected swapped dimer
Acta Crystallogr.,Sect.D, 63, 2007
1F5L
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UROKINASE PLASMINOGEN ACTIVATOR B-CHAIN-AMILORIDE COMPLEX
分子名称: 3,5-DIAMINO-N-(AMINOIMINOMETHYL)-6-CHLOROPYRAZINECARBOXAMIDE, SULFATE ION, UROKINASE-TYPE PLASMINOGEN ACTIVATOR
著者Zeslawska, E, Schweinitz, A, Karcher, A, Sondermann, P, Sperl, S, Sturzebecher, J, Jacob, U.
登録日2000-06-15
公開日2001-06-15
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystals of the urokinase type plasminogen activator variant beta(c)-uPAin complex with small molecule inhibitors open the way towards structure-based drug design.
J.Mol.Biol., 301, 2000
1F0P
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MYCOBACTERIUM TUBERCULOSIS ANTIGEN 85B WITH TREHALOSE
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, ANTIGEN 85-B, ...
著者Anderson, D.H, Harth, G, Horwitz, M.A, Eisenberg, D, TB Structural Genomics Consortium (TBSGC)
登録日2000-05-16
公開日2001-01-24
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献An interfacial mechanism and a class of inhibitors inferred from two crystal structures of the Mycobacterium tuberculosis 30 kDa major secretory protein (Antigen 85B), a mycolyl transferase.
J.Mol.Biol., 307, 2001
1SJ4
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Crystal structure of a C75U mutant Hepatitis Delta Virus ribozyme precursor, in Cu2+ solution
分子名称: precursor form of the Hepatitis Delta virus ribozyme, small nuclear ribonucleoprotein A
著者Ke, A, Zhou, K, Ding, F, Cate, J.H, Doudna, J.A.
登録日2004-03-02
公開日2004-05-18
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献A Conformational Switch controls hepatitis delta virus ribozyme catalysis
Nature, 429, 2004
2I7B
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Structure of the naturally occuring mutant of human ABO(H) Blood group B glycosyltransferase: GTB/A268T
分子名称: MERCURY (II) ION, alpha 1-3-galactosyltransferase
著者Letts, J.A, Evans, S.V.
登録日2006-08-30
公開日2007-05-22
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Structural basis for red cell phenotypic changes in newly identified, naturally occurring subgroup mutants of the human blood group B glycosyltransferase.
Transfusion, 47, 2007
1F0N
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MYCOBACTERIUM TUBERCULOSIS ANTIGEN 85B
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, ANTIGEN 85B
著者Anderson, D.H, Harth, G, Horwitz, M.A, Eisenberg, D, TB Structural Genomics Consortium (TBSGC)
登録日2000-05-16
公開日2001-01-24
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献An interfacial mechanism and a class of inhibitors inferred from two crystal structures of the Mycobacterium tuberculosis 30 kDa major secretory protein (Antigen 85B), a mycolyl transferase.
J.Mol.Biol., 307, 2001
2HNT
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CRYSTALLOGRAPHIC STRUCTURE OF HUMAN GAMMA-THROMBIN
分子名称: GAMMA-THROMBIN
著者Tulinsky, A.
登録日1994-08-23
公開日1994-11-30
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystallographic structure of human gamma-thrombin.
J.Biol.Chem., 269, 1994
2IHE
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Crystal structure of wild-type single-stranded DNA binding protein from Thermus aquaticus
分子名称: Single-stranded DNA-binding protein
著者Fedorov, R, Witte, G, Urbanke, C, Manstein, D.J, Curth, U.
登録日2006-09-26
公開日2007-01-02
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献3D structure of Thermus aquaticus single-stranded DNA-binding protein gives insight into the functioning of SSB proteins.
Nucleic Acids Res., 34, 2006
1F16
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SOLUTION STRUCTURE OF A PRO-APOPTOTIC PROTEIN BAX
分子名称: PROTEIN (APOPTOSIS REGULATOR BAX, MEMBRANE ISOFORM ALPHA)
著者Suzuki, M, Youle, R.J, Tjandra, N.
登録日2000-05-18
公開日2000-11-22
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Structure of Bax: coregulation of dimer formation and intracellular localization.
Cell(Cambridge,Mass.), 103, 2000
1F61
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CRYSTAL STRUCTURE OF ISOCITRATE LYASE FROM MYCOBACTERIUM TUBERCULOSIS
分子名称: ISOCITRATE LYASE, MAGNESIUM ION
著者Sharma, V, Sharma, S, Hoener zu Bentrup, K.H, McKinney, J.D, Russell, D.G, Jacobs Jr, W.R, Sacchettini, J.C, TB Structural Genomics Consortium (TBSGC)
登録日2000-06-19
公開日2000-08-30
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure of isocitrate lyase, a persistence factor of Mycobacterium tuberculosis.
Nat.Struct.Biol., 7, 2000
1SSD
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Understanding protein lids: Structural analysis of active hinge mutants in triosephosphate isomerase
分子名称: SULFATE ION, Triosephosphate isomerase
著者Kursula, I, Salin, M, Sun, J, Norledge, B.V, Haapalainen, A.M, Sampson, N.S, Wierenga, R.K.
登録日2004-03-24
公開日2004-08-24
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Understanding protein lids: structural analysis of active hinge mutants in triosephosphate isomerase
Protein Eng.Des.Sel., 17, 2004
2HBY
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Crystal structure of human caspase-1 (Glu390->Ala) in complex with 3-[2-(2-benzyloxycarbonylamino-3-methyl-butyrylamino)-propionylamino]-4-oxo-pentanoic acid (z-VAD-FMK)
分子名称: Caspase-1, N-[(benzyloxy)carbonyl]-L-valyl-N-[(2S)-1-carboxy-4-fluoro-3-oxobutan-2-yl]-L-alaninamide
著者Scheer, J.M, Wells, J.A, Romanowski, M.J.
登録日2006-06-14
公開日2006-06-27
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献A Common Allosteric Site and Mechanism in Caspases
Proc.Natl.Acad.Sci.USA, 103, 2006
2HDM
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Solution structure of V21C/V59C Lymphotactin/XCL1
分子名称: Lymphotactin
著者Volkman, B.F, Tuinstra, R.L, Peterson, F.C, Elgin, E.S.
登録日2006-06-20
公開日2007-05-01
最終更新日2021-10-20
実験手法SOLUTION NMR
主引用文献An engineered second disulfide bond restricts lymphotactin/XCL1 to a chemokine-like conformation with XCR1 agonist activity
Biochemistry, 46, 2007
1TDH
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Crystal structure of human endonuclease VIII-like 1 (NEIL1)
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, nei endonuclease VIII-like 1
著者Doublie, S, Bandaru, V, Bond, J.P, Wallace, S.S.
登録日2004-05-22
公開日2004-07-20
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The crystal structure of human endonuclease VIII-like 1 (NEIL1) reveals a zincless finger motif required for glycosylase activity.
Proc.Natl.Acad.Sci.USA, 101, 2004
1F7Z
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RAT TRYPSINOGEN K15A COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR
分子名称: CALCIUM ION, PANCREATIC TRYPSIN INHIBITOR, SULFATE ION, ...
著者Pasternak, A, White, A, Jeffery, C.J, Medina, N, Cahoon, M, Ringe, D, Hedstrom, L.
登録日2000-06-28
公開日2001-07-04
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献The energetic cost of induced fit catalysis: Crystal structures of trypsinogen mutants with enhanced activity and inhibitor affinity.
Protein Sci., 10, 2001
2J61
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L-ficolin complexed to N-acetylglucosamine (forme C)
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, FICOLIN-2
著者Garlatti, V, Gaboriaud, C.
登録日2006-09-21
公開日2007-01-23
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structural Insights Into the Innate Immune Recognition Specificities of L- and H-Ficolins.
Embo J., 26, 2007
1FG7
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CRYSTAL STRUCTURE OF L-HISTIDINOL PHOSPHATE AMINOTRANSFERASE WITH PYRIDOXAL-5'-PHOSPHATE
分子名称: 4'-DEOXY-4'-AMINOPYRIDOXAL-5'-PHOSPHATE, HISTIDINOL PHOSPHATE AMINOTRANSFERASE
著者Sivaraman, J, Cygler, M, Montreal-Kingston Bacterial Structural Genomics Initiative (BSGI)
登録日2000-07-28
公開日2001-08-22
最終更新日2017-10-04
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Crystal structure of histidinol phosphate aminotransferase (HisC) from Escherichia coli, and its covalent complex with pyridoxal-5'-phosphate and l-histidinol phosphate.
J.Mol.Biol., 311, 2001
2ILN
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Crystal structure of the Bowman-Birk inhibitor from snail medic seeds in complex with bovine trypsin
分子名称: Bowman-Birk type proteinase inhibitor, Cationic trypsin
著者Capaldi, S, Perduca, M, Faggion, B, Carrizo, M.E, Tava, A, Ragona, L, Monaco, H.L.
登録日2006-10-03
公開日2007-04-10
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of the anticarcinogenic Bowman-Birk inhibitor from snail medic (Medicago scutellata) seeds complexed with bovine trypsin
J.Struct.Biol., 158, 2007
1TJG
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Crystal Structure of the broadly neutralizing anti-HIV-1 antibody 2F5 in complex with a gp41 7mer epitope
分子名称: 1,2-ETHANEDIOL, Envelope glycoprotein GP41, FAB 2F5 Heavy Chain, ...
著者Ofek, G, Tang, M, Sambor, A, Katinger, H, Mascola, J.R, Wyatt, R, Kwong, P.D.
登録日2004-06-04
公開日2004-10-05
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure and mechanistic analysis of the Anti-Human Immunodeficiency Virus Type 1 antibody 2F5 in complex with its gp41 epitope
J.Virol., 78, 2004
2IF0
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Crystal Structure of mouse Rab27b bound to GDP in monoclinic space group
分子名称: GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Ras-related protein Rab-27B
著者Chavas, L.M.G, Torii, S, Kamikubo, H, Kawasaki, M, Ihara, K, Kato, R, Kataoka, M, Izumi, T, Wakatsuki, S.
登録日2006-09-19
公開日2007-05-01
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure of the small GTPase Rab27b shows an unexpected swapped dimer
Acta Crystallogr.,Sect.D, 63, 2007
1TON
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RAT SUBMAXILLARY GLAND SERINE PROTEASE, TONIN. STRUCTURE SOLUTION AND REFINEMENT AT 1.8 ANGSTROMS RESOLUTION
分子名称: TONIN, ZINC ION
著者Fujinaga, M, James, M.N.G.
登録日1987-06-03
公開日1988-01-16
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Rat submaxillary gland serine protease, tonin. Structure solution and refinement at 1.8 A resolution.
J.Mol.Biol., 195, 1987
1U53
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Novel X-Ray Structure of Na-ASP-2, a PR-1 protein from the nematode parasite Necator americanus and a vaccine antigen for human hookworm infection
分子名称: secreted protein ASP-2
著者Asojo, O.A, Goud, G, Dhar, K, Loukas, A, Zhan, B, Deumic, V, Liu, S, Borgstahl, G.E.O, Hotez, P.J.
登録日2004-07-26
公開日2005-02-01
最終更新日2017-10-11
実験手法X-RAY DIFFRACTION (1.56 Å)
主引用文献X-ray structure of Na-ASP-2, a pathogenesis-related-1 protein from the nematode parasite, Necator americanus, and a vaccine antigen for human hookworm infection.
J.Mol.Biol., 346, 2005
1F92
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UROKINASE PLASMINOGEN ACTIVATOR B CHAIN-UKI-1D COMPLEX
分子名称: SULFATE ION, UROKINASE-TYPE PLASMINOGEN ACTIVATOR, [2,4,6-TRIISOPROPYL-PHENYLSULFONYL-L-[3-AMIDINO-PHENYLALANINYL]]-N'-BETA-ALANINYL-PIPERAZINE
著者Zeslawska, E, Schweinitz, A, Karcher, A, Sondermann, P, Sperl, S, Sturzebecher, J, Jacob, U.
登録日2000-07-06
公開日2001-07-06
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Crystals of the urokinase type plasminogen activator variant beta(c)-uPAin complex with small molecule inhibitors open the way towards structure-based drug design.
J.Mol.Biol., 301, 2000
2IWM
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precursor mutant Cys1Ser of Penicillin V Acylase from Bacillus sphaericus
分子名称: PENICILLIN ACYLASE
著者Chandra, P.M, Dodson, G, Suresh, C.G.
登録日2006-07-01
公開日2007-08-07
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Precursor Mutant Cys1Ser of Penicillin V Acylase from Bacilus Sphaericus
To be Published

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