4HFQ
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![BU of 4hfq by Molmil](/molmil-images/mine/4hfq) | Crystal structure of UDP-X diphosphatase | 分子名称: | 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, DI(HYDROXYETHYL)ETHER, ... | 著者 | Duong-Ly, K.C, Amzel, L.M, Gabelli, S.B. | 登録日 | 2012-10-05 | 公開日 | 2013-08-07 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.39 Å) | 主引用文献 | A UDP-X diphosphatase from Streptococcus pneumoniae hydrolyzes precursors of peptidoglycan biosynthesis. Plos One, 8, 2013
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4DYW
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![BU of 4dyw by Molmil](/molmil-images/mine/4dyw) | |
4C9X
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![BU of 4c9x by Molmil](/molmil-images/mine/4c9x) | Crystal structure of NUDT1 (MTH1) with S-crizotinib | 分子名称: | 3-[(1S)-1-(2,6-DICHLORO-3-FLUOROPHENYL)ETHOXY]-5-(1-PIPERIDIN-4-YLPYRAZOL-4-YL)PYRIDIN-2-AMINE, 7,8-DIHYDRO-8-OXOGUANINE TRIPHOSPHATASE, CHLORIDE ION, ... | 著者 | Elkins, J.M, Salah, E, Huber, K, Superti-Furga, G, Abdul Azeez, K.R, Krojer, T, von Delft, F, Bountra, C, Edwards, A, Knapp, S. | 登録日 | 2013-10-03 | 公開日 | 2014-04-02 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.2 Å) | 主引用文献 | Stereospecific Targeting of Mth1 by (S)-Crizotinib as an Anticancer Strategy. Nature, 508, 2014
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4C9W
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![BU of 4c9w by Molmil](/molmil-images/mine/4c9w) | Crystal structure of NUDT1 (MTH1) with R-crizotinib | 分子名称: | 3-[(1R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1H-pyrazol-4-yl)pyridin-2-amine, 7,8-DIHYDRO-8-OXOGUANINE TRIPHOSPHATASE, CHLORIDE ION, ... | 著者 | Elkins, J.M, Salah, E, Huber, K, Superti-Furga, G, Abdul Azeez, K.R, Raynor, J, Krojer, T, von Delft, F, Bountra, C, Edwards, A, Knapp, S. | 登録日 | 2013-10-03 | 公開日 | 2014-04-02 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Stereospecific Targeting of Mth1 by (S)-Crizotinib as an Anticancer Strategy. Nature, 508, 2014
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3ZR1
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![BU of 3zr1 by Molmil](/molmil-images/mine/3zr1) | Crystal structure of human MTH1 | 分子名称: | 7,8-DIHYDRO-8-OXOGUANINE TRIPHOSPHATASE, ACETATE ION, SULFATE ION | 著者 | Svensson, L.M, Jemth, A, Desroses, M, Loseva, O, Helleday, T, Hogbom, M, Stenmark, P. | 登録日 | 2011-06-13 | 公開日 | 2011-07-27 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal Structure of Human Mth1 and the 8-Oxo-Dgmp Product Complex. FEBS Lett., 585, 2011
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3ZR0
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![BU of 3zr0 by Molmil](/molmil-images/mine/3zr0) | Crystal structure of human MTH1 in complex with 8-oxo-dGMP | 分子名称: | 7,8-DIHYDRO-8-OXOGUANINE TRIPHOSPHATASE, 8-OXO-2'-DEOXY-GUANOSINE-5'-MONOPHOSPHATE, SULFATE ION | 著者 | Svensson, L.M, Jemth, A, Desroses, M, Loseva, O, Helleday, T, Hogbom, M, Stenmark, P. | 登録日 | 2011-06-13 | 公開日 | 2011-07-27 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystal Structure of Human Mth1 and the 8-Oxo-Dgmp Product Complex. FEBS Lett., 585, 2011
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3X0S
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![BU of 3x0s by Molmil](/molmil-images/mine/3x0s) | ADP ribose pyrophosphatase from Thermus thermophilus HB8 in E'-state at reaction time of 50 min | 分子名称: | ADP-ribose pyrophosphatase, GLYCEROL, MANGANESE (II) ION, ... | 著者 | Furuike, Y, Akita, Y, Miyahara, I, Kamiya, N. | 登録日 | 2014-10-17 | 公開日 | 2016-04-27 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.1 Å) | 主引用文献 | ADP-Ribose Pyrophosphatase Reaction in Crystalline State Conducted by Consecutive Binding of Two Manganese(II) Ions as Cofactors Biochemistry, 55, 2016
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3X0R
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![BU of 3x0r by Molmil](/molmil-images/mine/3x0r) | DP ribose pyrophosphatase from Thermus thermophilus HB8 in E'-state at reaction time of 30 min | 分子名称: | ADP-ribose pyrophosphatase, GLYCEROL, MANGANESE (II) ION, ... | 著者 | Furuike, Y, Akita, Y, Miyahara, I, Kamiya, N. | 登録日 | 2014-10-17 | 公開日 | 2016-04-27 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.15 Å) | 主引用文献 | ADP-Ribose Pyrophosphatase Reaction in Crystalline State Conducted by Consecutive Binding of Two Manganese(II) Ions as Cofactors Biochemistry, 55, 2016
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3X0Q
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![BU of 3x0q by Molmil](/molmil-images/mine/3x0q) | ADP ribose pyrophosphatase from Thermus thermophilus HB8 in ESMM-state at reaction time of 20 min | 分子名称: | ADP-ribose pyrophosphatase, GLYCEROL, MANGANESE (II) ION, ... | 著者 | Furuike, Y, Akita, Y, Miyahara, I, Kamiya, N. | 登録日 | 2014-10-17 | 公開日 | 2016-04-27 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.14 Å) | 主引用文献 | ADP-Ribose Pyrophosphatase Reaction in Crystalline State Conducted by Consecutive Binding of Two Manganese(II) Ions as Cofactors Biochemistry, 55, 2016
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3X0P
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![BU of 3x0p by Molmil](/molmil-images/mine/3x0p) | ADP ribose pyrophosphatase from Thermus thermophilus HB8 in ESMM-state at reaction time of 15 min | 分子名称: | ADP-ribose pyrophosphatase, GLYCEROL, MANGANESE (II) ION, ... | 著者 | Furuike, Y, Akita, Y, Miyahara, I, Kamiya, N. | 登録日 | 2014-10-17 | 公開日 | 2016-04-27 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.22 Å) | 主引用文献 | ADP-Ribose Pyrophosphatase Reaction in Crystalline State Conducted by Consecutive Binding of Two Manganese(II) Ions as Cofactors Biochemistry, 55, 2016
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3X0O
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![BU of 3x0o by Molmil](/molmil-images/mine/3x0o) | ADP ribose pyrophosphatase from Thermus thermophilus HB8 in ESMM-state at reaction time of 10 min | 分子名称: | ADP-ribose pyrophosphatase, GLYCEROL, MANGANESE (II) ION, ... | 著者 | Furuike, Y, Akita, Y, Miyahara, I, Kamiya, N. | 登録日 | 2014-10-17 | 公開日 | 2016-04-27 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.09 Å) | 主引用文献 | ADP-Ribose Pyrophosphatase Reaction in Crystalline State Conducted by Consecutive Binding of Two Manganese(II) Ions as Cofactors Biochemistry, 55, 2016
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3X0N
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![BU of 3x0n by Molmil](/molmil-images/mine/3x0n) | ADP ribose pyrophosphatase from Thermus thermophilus HB8 in ESM-state at reaction time of 6 min | 分子名称: | ADP-ribose pyrophosphatase, GLYCEROL, MANGANESE (II) ION, ... | 著者 | Furuike, Y, Akita, Y, Miyahara, I, Kamiya, N. | 登録日 | 2014-10-17 | 公開日 | 2016-04-27 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.12 Å) | 主引用文献 | ADP-Ribose Pyrophosphatase Reaction in Crystalline State Conducted by Consecutive Binding of Two Manganese(II) Ions as Cofactors Biochemistry, 55, 2016
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3X0M
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![BU of 3x0m by Molmil](/molmil-images/mine/3x0m) | ADP ribose pyrophosphatase from Thermus thermophilus HB8 in ESM-state at reaction time of 3 min | 分子名称: | ADP-ribose pyrophosphatase, GLYCEROL, MANGANESE (II) ION, ... | 著者 | Furuike, Y, Akita, Y, Miyahara, I, Kamiya, N. | 登録日 | 2014-10-17 | 公開日 | 2016-04-27 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.15 Å) | 主引用文献 | ADP-Ribose Pyrophosphatase Reaction in Crystalline State Conducted by Consecutive Binding of Two Manganese(II) Ions as Cofactors Biochemistry, 55, 2016
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3X0L
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![BU of 3x0l by Molmil](/molmil-images/mine/3x0l) | ADP ribose pyrophosphatase from Thermus thermophilus HB8 in ES-state at 1.00 angstrom resolution | 分子名称: | ADP-ribose pyrophosphatase, [(2R,3S,4R,5R)-5-(6-AMINOPURIN-9-YL)-3,4-DIHYDROXY-OXOLAN-2-YL]METHYL [HYDROXY-[[(2R,3S,4R,5S)-3,4,5-TRIHYDROXYOXOLAN-2-YL]METHOXY]PHOSPHORYL] HYDROGEN PHOSPHATE | 著者 | Furuike, Y, Akita, Y, Miyahara, I, Kamiya, N. | 登録日 | 2014-10-17 | 公開日 | 2016-04-27 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1 Å) | 主引用文献 | ADP-Ribose Pyrophosphatase Reaction in Crystalline State Conducted by Consecutive Binding of Two Manganese(II) Ions as Cofactors Biochemistry, 55, 2016
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3X0K
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![BU of 3x0k by Molmil](/molmil-images/mine/3x0k) | ADP ribose pyrophosphatase from Thermus thermophilus HB8 in ES-state at 0.97 angstrom resolution | 分子名称: | ADP-ribose pyrophosphatase, GLYCEROL, [(2R,3S,4R,5R)-5-(6-AMINOPURIN-9-YL)-3,4-DIHYDROXY-OXOLAN-2-YL]METHYL [HYDROXY-[[(2R,3S,4R,5S)-3,4,5-TRIHYDROXYOXOLAN-2-YL]METHOXY]PHOSPHORYL] HYDROGEN PHOSPHATE | 著者 | Furuike, Y, Akita, Y, Miyahara, I, Kamiya, N. | 登録日 | 2014-10-16 | 公開日 | 2016-04-27 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (0.97 Å) | 主引用文献 | ADP-Ribose Pyrophosphatase Reaction in Crystalline State Conducted by Consecutive Binding of Two Manganese(II) Ions as Cofactors Biochemistry, 55, 2016
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3X0J
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![BU of 3x0j by Molmil](/molmil-images/mine/3x0j) | ADP ribose pyrophosphatase from Thermus thermophilus HB8 in apo state at 0.92 angstrom resolution | 分子名称: | ADP-ribose pyrophosphatase, GLYCEROL, SULFATE ION | 著者 | Furuike, Y, Akita, Y, Miyahara, I, Kamiya, N. | 登録日 | 2014-10-16 | 公開日 | 2016-04-27 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (0.92 Å) | 主引用文献 | ADP-Ribose Pyrophosphatase Reaction in Crystalline State Conducted by Consecutive Binding of Two Manganese(II) Ions as Cofactors Biochemistry, 55, 2016
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3X0I
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![BU of 3x0i by Molmil](/molmil-images/mine/3x0i) | ADP ribose pyrophosphatase in apo state at 0.91 angstrom resolution | 分子名称: | ADP-ribose pyrophosphatase, GLYCEROL, SULFATE ION | 著者 | Furuike, Y, Akita, Y, Miyahara, I, Kamiya, N. | 登録日 | 2014-10-16 | 公開日 | 2016-04-27 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (0.91 Å) | 主引用文献 | ADP-Ribose Pyrophosphatase Reaction in Crystalline State Conducted by Consecutive Binding of Two Manganese(II) Ions as Cofactors Biochemistry, 55, 2016
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3WHW
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![BU of 3whw by Molmil](/molmil-images/mine/3whw) | MTH1 in complex with Ruthenium-based inhibitor | 分子名称: | 7,8-dihydro-8-oxoguanine triphosphatase, SULFATE ION, [4-amino-2-methyl-6-(pyridin-2-yl-kappaN)quinazolin-7-yl-kappaC~7~](carbonyl){1-[(2,6-dimethoxyphenoxy)carbonyl]cyclopenta-2,4-dien-1-yl}ruthenium | 著者 | Streib, M, Kraeling, K, Richter, K, Steuber, H, Meggers, E. | 登録日 | 2013-09-03 | 公開日 | 2014-02-12 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.701 Å) | 主引用文献 | An Organometallic Inhibitor for the Human Repair Enzyme 7,8-Dihydro-8-oxoguanosine Triphosphatase. Angew.Chem.Int.Ed.Engl., 53, 2014
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3U53
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![BU of 3u53 by Molmil](/molmil-images/mine/3u53) | Crystal structure of human Ap4A hydrolase | 分子名称: | Bis(5'-nucleosyl)-tetraphosphatase [asymmetrical], GLYCEROL, SULFATE ION | 著者 | Ge, H.H, Teng, M.K. | 登録日 | 2011-10-10 | 公開日 | 2012-10-10 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.705 Å) | 主引用文献 | Crystal structure of wild-type and mutant human Ap4A hydrolase Biochem.Biophys.Res.Commun., 432, 2013
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3SMD
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![BU of 3smd by Molmil](/molmil-images/mine/3smd) | |
3SHD
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![BU of 3shd by Molmil](/molmil-images/mine/3shd) | |
3QSJ
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![BU of 3qsj by Molmil](/molmil-images/mine/3qsj) | Crystal structure of NUDIX hydrolase from Alicyclobacillus acidocaldarius | 分子名称: | CALCIUM ION, GLYCEROL, NUDIX hydrolase | 著者 | Michalska, K, Wu, R, Bearden, J, Joachimiak, A, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2011-02-21 | 公開日 | 2011-04-13 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Crystal structure of NUDIX hydrolase from Alicyclobacillus acidocaldarius To be Published
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3Q93
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![BU of 3q93 by Molmil](/molmil-images/mine/3q93) | Crystal Structure of Human 8-oxo-dGTPase (MTH1) | 分子名称: | 7,8-dihydro-8-oxoguanine triphosphatase, GLYCEROL, IMIDAZOLE, ... | 著者 | Tresaugues, L, Siponen, M.I, Arrowsmith, C.H, Berglund, H, Bountra, C, Collins, R, Edwards, A.M, Ekblad, T, Flodin, S, Flores, A, Graslund, S, Hammarstrom, M, Johansson, I, Karlberg, T, Kol, S, Kotenyova, T, Kouznetsova, E, Moche, M, Nyman, T, Persson, C, Schuler, H, Schutz, P, Thorsell, A.G, Van Der Berg, S, Wahlberg, E, Weigelt, J, Welin, M, Nordlund, P, Structural Genomics Consortium (SGC) | 登録日 | 2011-01-07 | 公開日 | 2011-03-02 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystal Structure of Human 8-oxo-dGTPase (MTH1) To be Published
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3Q4I
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![BU of 3q4i by Molmil](/molmil-images/mine/3q4i) | Crystal structure of CDP-Chase in complex with Gd3+ | 分子名称: | GADOLINIUM ION, Phosphohydrolase (MutT/nudix family protein) | 著者 | Duong-Ly, K.C, Gabelli, S.B, Amzel, L.M. | 登録日 | 2010-12-23 | 公開日 | 2011-07-13 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | The Nudix Hydrolase CDP-Chase, a CDP-Choline Pyrophosphatase, Is an Asymmetric Dimer with Two Distinct Enzymatic Activities. J.Bacteriol., 193, 2011
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3Q1P
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![BU of 3q1p by Molmil](/molmil-images/mine/3q1p) | Crystal structure of CDP-Chase | 分子名称: | Phosphohydrolase (MutT/nudix family protein), SULFATE ION | 著者 | Duong-Ly, K.C, Gabelli, S.B, Amzel, L.M. | 登録日 | 2010-12-17 | 公開日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | The Nudix Hydrolase CDP-Chase, a CDP-Choline Pyrophosphatase, Is an Asymmetric Dimer with Two Distinct Enzymatic Activities. J.Bacteriol., 193, 2011
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