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8K2C
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BU of 8k2c by Molmil
Cryo-EM structure of the human 80S ribosome with Tigecycline
分子名称: 18S rRNA, 28S rRNA, 40S ribosomal protein S10, ...
著者Li, X, Wang, M, Cheng, J.
登録日2023-07-12
公開日2024-07-10
実験手法ELECTRON MICROSCOPY (2.4 Å)
主引用文献Structural basis for differential inhibition of eukaryotic ribosomes by tigecycline.
Nat Commun, 15, 2024
6XJP
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BU of 6xjp by Molmil
Crystal Structure of KPT-185 bound to CRM1 (537-DLTVK-541 to GLCEQ)
分子名称: Exportin-1, GTP-binding nuclear protein Ran, MAGNESIUM ION, ...
著者Baumhardt, J.M, Chook, Y.M.
登録日2020-06-24
公開日2021-01-27
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.802 Å)
主引用文献Recurrent XPO1 mutations alter pathogenesis of chronic lymphocytic leukemia.
J Hematol Oncol, 14, 2021
6XJT
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BU of 6xjt by Molmil
Crystal Structure of KPT-8602 bound to CRM1 (537-DLTVK-541 to GLCEQ)
分子名称: (2R)-3-{3-[3,5-bis(trifluoromethyl)phenyl]-1H-1,2,4-triazol-1-yl}-2-(pyrimidin-5-yl)propanamide, Exportin-1, GTP-binding nuclear protein Ran, ...
著者Baumhardt, J.M, Chook, Y.M.
登録日2020-06-24
公開日2021-01-27
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.406 Å)
主引用文献Recurrent XPO1 mutations alter pathogenesis of chronic lymphocytic leukemia.
J Hematol Oncol, 14, 2021
8J07
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BU of 8j07 by Molmil
96nm repeat of human respiratory doublet microtubule and associated axonemal complexes
分子名称: ACTA2, Axonemal dynein light intermediate polypeptide 1, Calaxin, ...
著者Gui, M, Brown, A.
登録日2023-04-09
公開日2023-07-26
最終更新日2023-08-02
実験手法ELECTRON MICROSCOPY (4.1 Å)
主引用文献Axonemal structures reveal mechanoregulatory and disease mechanisms.
Nature, 618, 2023
6F1Z
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BU of 6f1z by Molmil
Roadblock-1 region of the dynein tail/dynactin/BICDR1 complex
分子名称: Cytoplasmic dynein 1 intermediate chain 2, Dynein light chain roadblock-type 1
著者Urnavicius, L, Lau, C.K, Elshenawy, M.M, Morales-Rios, E, Motz, C, Yildiz, A, Carter, A.P.
登録日2017-11-23
公開日2018-01-17
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Cryo-EM shows how dynactin recruits two dyneins for faster movement.
Nature, 554, 2018
4UJ5
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BU of 4uj5 by Molmil
Crystal structure of human Rab11-Rabin8-FIP3
分子名称: MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER, RAB-3A-INTERACTING PROTEIN, ...
著者Vetter, M, Lorentzen, E.
登録日2015-04-08
公開日2015-08-12
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.604 Å)
主引用文献Structure of Rab11-Fip3-Rabin8 Reveals Simultaneous Binding of Fip3 and Rabin8 Effectors to Rab11.
Nat.Struct.Mol.Biol., 22, 2015
4UJ4
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BU of 4uj4 by Molmil
Crystal structure of human Rab11-Rabin8-FIP3
分子名称: MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER, Rab-3A-interacting protein, ...
著者Vetter, M, Lorentzen, E.
登録日2015-04-08
公開日2015-08-12
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (4.2 Å)
主引用文献Structure of Rab11-FIP3-Rabin8 reveals simultaneous binding of FIP3 and Rabin8 effectors to Rab11.
Nat. Struct. Mol. Biol., 22, 2015
4UJ3
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BU of 4uj3 by Molmil
Crystal structure of human Rab11-Rabin8-FIP3
分子名称: MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER, RAB-3A-INTERACTING PROTEIN, ...
著者Vetter, M, Lorentzen, E.
登録日2015-04-08
公開日2015-08-12
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structure of Rab11-Fip3-Rabin8 Reveals Simultaneous Binding of Fip3 and Rabin8 Effectors to Rab11.
Nat.Struct.Mol.Biol., 22, 2015
5EZ5
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BU of 5ez5 by Molmil
Crystal structure of active Rab11A (S20V) in complex with GTP
分子名称: GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, Ras-related protein Rab-11A
著者Shin, Y.-C, Yoon, J.H, Park, H.H.
登録日2015-11-26
公開日2016-12-07
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal structure of active Rab11A (S20V) in complex with GTP
To Be Published
6A3A
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BU of 6a3a by Molmil
MVM NES mutant Nm2 in complex with CRM1-Ran-RanBP1
分子名称: 1,2-ETHANEDIOL, Exportin-1, GLYCEROL, ...
著者Sun, Q, Li, Y.
登録日2018-06-15
公開日2019-06-19
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Cancer Therapy with Nanoparticle-Medicated Intracellular Expression of Peptide CRM1-Inhibitor.
Int J Nanomedicine, 16, 2021
6A3E
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BU of 6a3e by Molmil
MVM NES mutant Nm15 in complex with CRM1-Ran-RanBP1
分子名称: Exportin-1, GTP-binding nuclear protein Ran, GUANOSINE-5'-TRIPHOSPHATE, ...
著者Sun, Q, Li, Y.
登録日2018-06-15
公開日2019-06-19
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Cancer Therapy with Nanoparticle-Medicated Intracellular Expression of Peptide CRM1-Inhibitor.
Int J Nanomedicine, 16, 2021
5FBW
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BU of 5fbw by Molmil
PI4KB in complex with Rab11 and the MI369 Inhibitor
分子名称: 5'-GUANOSINE-DIPHOSPHATE-MONOTHIOPHOSPHATE, Phosphatidylinositol 4-kinase beta,Phosphatidylinositol 4-kinase beta, Ras-related protein Rab-11A, ...
著者Chalupska, D, Mejdrova, I, Nencka, R, Boura, E.
登録日2015-12-14
公開日2016-12-28
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (3.487 Å)
主引用文献PI4KB in complex with Rab11 and the MI369 Inhibitor
To Be Published
6A3C
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BU of 6a3c by Molmil
MVM NES mutant Nm12 in complex with CRM1-Ran-RanBP1
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, Exportin-1, ...
著者Sun, Q, Li, Y.
登録日2018-06-15
公開日2019-06-19
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Cancer Therapy with Nanoparticle-Medicated Intracellular Expression of Peptide CRM1-Inhibitor.
Int J Nanomedicine, 16, 2021
6A38
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BU of 6a38 by Molmil
MVM NS2 NES in complex with CRM1-Ran-RanBP1
分子名称: 1,2-ETHANEDIOL, Exportin-1, GLYCEROL, ...
著者Sun, Q, Li, Y.
登録日2018-06-15
公開日2019-06-19
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.69 Å)
主引用文献Cancer Therapy with Nanoparticle-Medicated Intracellular Expression of Peptide CRM1-Inhibitor.
Int J Nanomedicine, 16, 2021
6A3B
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BU of 6a3b by Molmil
MVM NES mutant Nm13 in complex with CRM1-Ran-RanBP1
分子名称: 1,2-ETHANEDIOL, Exportin-1, GLYCEROL, ...
著者Sun, Q, Li, Y.
登録日2018-06-15
公開日2019-06-19
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.51 Å)
主引用文献Cancer Therapy with Nanoparticle-Medicated Intracellular Expression of Peptide CRM1-Inhibitor.
Int J Nanomedicine, 16, 2021
2IV8
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BU of 2iv8 by Molmil
beta appendage in complex with b-arrestin peptide
分子名称: AP-2 COMPLEX SUBUNIT BETA-1, BETA-ARRESTIN-1
著者Ford, M.G.J, Schmid, E.M, McMahon, H.T.
登録日2006-06-08
公開日2007-06-12
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Role of the Ap2 Beta-Appendage Hub in Recruiting Partners for Clathrin-Coated Vesicle Assembly.
Plos Biol., 4, 2006
2JJU
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BU of 2jju by Molmil
Structure of human signal regulatory protein (sirp) beta
分子名称: CHLORIDE ION, SIGNAL REGULATORY PROTEIN BETA-1, SULFATE ION
著者Hatherley, D, Graham, S.C, Turner, J, Harlos, K, Stuart, D.I, Barclay, A.N.
登録日2008-04-22
公開日2008-08-05
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.19 Å)
主引用文献Paired Receptor Specificity Explained by Structures of Signal Regulatory Proteins Alone and Complexed with Cd47.
Mol.Cell, 31, 2008
5FBR
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BU of 5fbr by Molmil
PI4KB in complex with Rab11 and the MI359 Inhibitor
分子名称: 5'-GUANOSINE-DIPHOSPHATE-MONOTHIOPHOSPHATE, Phosphatidylinositol 4-kinase beta,Phosphatidylinositol 4-kinase beta, Ras-related protein Rab-11A, ...
著者Chalupska, D, Mejdrova, I, Nencka, R, Boura, E.
登録日2015-12-14
公開日2016-12-28
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (3.28 Å)
主引用文献PI4KB in complex with Rab11 and the MI359 Inhibitor
To Be Published
5ET1
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BU of 5et1 by Molmil
Crystal structure of Myo3b-ARB1 in complex with Espin1-AR
分子名称: Espin, GLYCEROL, Myosin-IIIb
著者Liu, H, Li, J, liu, W, Zhang, M.
登録日2015-11-17
公開日2016-02-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Myosin III-mediated cross-linking and stimulation of actin bundling activity of Espin
Elife, 5, 2016
5EUQ
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BU of 5euq by Molmil
Crystal structure of an engineered construct of phosphatidylinositol 4 kinase III beta with a potent and selective inhibitor in complex with GDP loaded Rab11
分子名称: GUANOSINE-5'-DIPHOSPHATE, Phosphatidylinositol 4-kinase beta, Ras-related protein Rab-11A, ...
著者Burke, J.E, Fowler, M.L.
登録日2015-11-19
公開日2016-02-24
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Design and Structural Characterization of Potent and Selective Inhibitors of Phosphatidylinositol 4 Kinase III beta.
J.Med.Chem., 59, 2016
4GMX
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BU of 4gmx by Molmil
Crystal structure of KPT185 in complex with CRM1-Ran-RanBP1
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, Exportin-1, ...
著者Sun, Q, Chook, Y.M.
登録日2012-08-16
公開日2012-10-17
最終更新日2012-12-12
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Selective inhibitors of nuclear export show that CRM1/XPO1 is a target in chronic lymphocytic leukemia.
Blood, 120, 2012
5FBQ
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BU of 5fbq by Molmil
PI4KB in complex with Rab11 and the MI358 Inhibitor
分子名称: GUANOSINE-5'-DIPHOSPHATE, Phosphatidylinositol 4-kinase beta,Phosphatidylinositol 4-kinase beta, Ras-related protein Rab-11A, ...
著者Chalupska, D, Mejdrova, I, Nencka, R, Boura, E.
登録日2015-12-14
公開日2016-12-28
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (3.789 Å)
主引用文献PI4KB in complex with Rab11 and the MI358 Inhibitor
To Be Published
5FBL
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BU of 5fbl by Molmil
PI4KB in complex with Rab11 and the MI356 Inhibitor
分子名称: 5'-GUANOSINE-DIPHOSPHATE-MONOTHIOPHOSPHATE, Phosphatidylinositol 4-kinase beta,Phosphatidylinositol 4-kinase beta, Ras-related protein Rab-11A, ...
著者Chalupska, D, Mejdrova, I, Nencka, R, Boura, E.
登録日2015-12-14
公開日2016-12-28
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (3.372 Å)
主引用文献PI4KB in complex with Rab11 and the MI356 Inhibitor
To Be Published
5FBV
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BU of 5fbv by Molmil
PI4KB in complex with Rab11 and the MI364 Inhibitor
分子名称: 5'-GUANOSINE-DIPHOSPHATE-MONOTHIOPHOSPHATE, Phosphatidylinositol 4-kinase beta,Phosphatidylinositol 4-kinase beta, Ras-related protein Rab-11A, ...
著者Chalupska, D, Mejdrova, I, Nencka, R, Boura, E.
登録日2015-12-14
公開日2016-12-28
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (3.285 Å)
主引用文献PI4KB in complex with Rab11 and the MI364 Inhibitor
To Be Published
2F9M
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BU of 2f9m by Molmil
3D structure of active human Rab11b GTPase
分子名称: MAGNESIUM ION, NICKEL (II) ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER, ...
著者Scapin, S.M.N, Guimaraes, B.G, Zanchin, N.I.T.
登録日2005-12-06
公開日2006-04-04
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献The crystal structure of the small GTPase Rab11b reveals critical differences relative to the Rab11a isoform.
J.Struct.Biol., 154, 2006

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