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5FBQ

PI4KB in complex with Rab11 and the MI358 Inhibitor

Summary for 5FBQ
Entry DOI10.2210/pdb5fbq/pdb
DescriptorPhosphatidylinositol 4-kinase beta,Phosphatidylinositol 4-kinase beta, Ras-related protein Rab-11A, ~{N}-[2-[[6-chloranyl-3-[3-[4-(hydroxymethyl)piperidin-1-yl]sulfonyl-4-methoxy-phenyl]-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamide, ... (4 entities in total)
Functional Keywordsinhibitor, complex, kinase, lipid, transferase
Biological sourceHomo sapiens (Human)
More
Cellular locationEndomembrane system: Q9UBF8
Cell membrane ; Lipid-anchor : P62491
Total number of polymer chains2
Total formula weight91087.00
Authors
Chalupska, D.,Mejdrova, I.,Nencka, R.,Boura, E. (deposition date: 2015-12-14, release date: 2016-12-28, Last modification date: 2024-01-10)
Primary citationChalupska, D.,Mejdrova, I.,Nencka, R.,Boura, E.
PI4KB in complex with Rab11 and the MI358 Inhibitor
To Be Published,
Experimental method
X-RAY DIFFRACTION (3.789 Å)
Structure validation

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PDB entries from 2024-04-10

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