4Y46
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4y46 by Molmil](/molmil-images/mine/4y46) | |
4Y5H
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4y5h by Molmil](/molmil-images/mine/4y5h) | |
5LW1
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5lw1 by Molmil](/molmil-images/mine/5lw1) | Crystal structure of DARPin-DARPin rigid fusion, variant DD_232_11_D12 in complex JNK1a1 and JIP1 peptide | 分子名称: | ADENOSINE, C-Jun-amino-terminal kinase-interacting protein 1, DD_232_11_D12, ... | 著者 | Wu, Y, Batyuk, A, Mittl, P.R, Honegger, A, Plueckthun, A. | 登録日 | 2016-09-15 | 公開日 | 2017-12-13 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (3.2 Å) | 主引用文献 | Structural Basis for the Selective Inhibition of c-Jun N-Terminal Kinase 1 Determined by Rigid DARPin-DARPin Fusions. J.Mol.Biol., 430, 2018
|
|
5VPD
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5vpd by Molmil](/molmil-images/mine/5vpd) | Transcription factor FosB/JunD bZIP domain in its oxidized form, type-III crystal | 分子名称: | CHLORIDE ION, Protein fosB, SODIUM ION, ... | 著者 | Yin, Z, Machius, M, Rudenko, G. | 登録日 | 2017-05-04 | 公開日 | 2017-09-06 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.79 Å) | 主引用文献 | Activator Protein-1: redox switch controlling structure and DNA-binding. Nucleic Acids Res., 45, 2017
|
|
5VPE
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5vpe by Molmil](/molmil-images/mine/5vpe) | Transcription factor FosB/JunD bZIP domain in complex with cognate DNA, type-I crystal | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, DNA (5'-D(*CP*GP*TP*CP*GP*GP*TP*GP*AP*CP*TP*CP*AP*CP*CP*GP*AP*CP*G)-3'), ... | 著者 | Yin, Z, Machius, M, Rudenko, G. | 登録日 | 2017-05-04 | 公開日 | 2017-09-06 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.053 Å) | 主引用文献 | Activator Protein-1: redox switch controlling structure and DNA-binding. Nucleic Acids Res., 45, 2017
|
|
5VPC
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5vpc by Molmil](/molmil-images/mine/5vpc) | Transcription factor FosB/JunD bZIP domain in its oxidized form, type-II crystal | 分子名称: | CHLORIDE ION, Protein fosB, SODIUM ION, ... | 著者 | Yin, Z, Machius, M.C, Rudenko, G. | 登録日 | 2017-05-04 | 公開日 | 2017-09-06 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.498 Å) | 主引用文献 | Activator Protein-1: redox switch controlling structure and DNA-binding. Nucleic Acids Res., 45, 2017
|
|
5VPB
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5vpb by Molmil](/molmil-images/mine/5vpb) | Transcription factor FosB/JunD bZIP domain in its oxidized form, type-I crystal | 分子名称: | CHLORIDE ION, Protein fosB, Transcription factor jun-D | 著者 | Yin, Z, Machius, M, Rudenko, G. | 登録日 | 2017-05-04 | 公開日 | 2017-09-06 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.691 Å) | 主引用文献 | Activator Protein-1: redox switch controlling structure and DNA-binding. Nucleic Acids Res., 45, 2017
|
|
5VPA
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5vpa by Molmil](/molmil-images/mine/5vpa) | Transcription factor FosB/JunD bZIP domain | 分子名称: | CHLORIDE ION, Protein fosB, SODIUM ION, ... | 著者 | Yin, Z, Machius, M, Rudenko, G. | 登録日 | 2017-05-04 | 公開日 | 2017-09-06 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.83 Å) | 主引用文献 | Activator Protein-1: redox switch controlling structure and DNA-binding. Nucleic Acids Res., 45, 2017
|
|
5VPF
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5vpf by Molmil](/molmil-images/mine/5vpf) | Transcription factor FosB/JunD bZIP domain in complex with cognate DNA, type-II crystal | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, DNA (5'-D(*CP*GP*TP*CP*GP*GP*TP*GP*AP*CP*TP*CP*AP*CP*CP*GP*AP*CP*G)-3'), ... | 著者 | Yin, Z, Rudenko, G, Machius, M. | 登録日 | 2017-05-04 | 公開日 | 2017-09-06 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.694 Å) | 主引用文献 | Activator Protein-1: redox switch controlling structure and DNA-binding. Nucleic Acids Res., 45, 2017
|
|
5VKT
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5vkt by Molmil](/molmil-images/mine/5vkt) | Cinnamyl alcohol dehydrogenases (SbCAD4) from Sorghum bicolor (L.) Moench | 分子名称: | ACETATE ION, Cinnamyl alcohol dehydrogenases (SbCAD4), D-MALATE, ... | 著者 | Walker, A.M, Jun, S.Y, Kang, C. | 登録日 | 2017-04-22 | 公開日 | 2017-08-09 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.827 Å) | 主引用文献 | The Enzyme Activity and Substrate Specificity of Two Major Cinnamyl Alcohol Dehydrogenases in Sorghum (Sorghum bicolor), SbCAD2 and SbCAD4. Plant Physiol., 174, 2017
|
|
7UCC
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7ucc by Molmil](/molmil-images/mine/7ucc) | Transcription factor FosB/JunD bZIP domain in the reduced form | 分子名称: | CHLORIDE ION, ETHANOL, Protein fosB, ... | 著者 | Kumar, A, Machius, M.C, Rudenko, G. | 登録日 | 2022-03-16 | 公開日 | 2023-01-25 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Chemically targeting the redox switch in AP1 transcription factor Delta FOSB. Nucleic Acids Res., 50, 2022
|
|
7UCD
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7ucd by Molmil](/molmil-images/mine/7ucd) | Transcription factor FosB/JunD bZIP domain covalently modified with the cysteine-targeting alpha-haloketone compound Z2159931480 | 分子名称: | 7-acetyl-4-methoxy-1-benzofuran-3(2H)-one, CHLORIDE ION, Protein fosB, ... | 著者 | Kumar, A, Machius, M.C, Rudenko, G. | 登録日 | 2022-03-16 | 公開日 | 2023-01-25 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (3.21 Å) | 主引用文献 | Chemically targeting the redox switch in AP1 transcription factor Delta FOSB. Nucleic Acids Res., 50, 2022
|
|
2G01
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 2g01 by Molmil](/molmil-images/mine/2g01) | Pyrazoloquinolones as Novel, Selective JNK1 inhibitors | 分子名称: | 6-CHLORO-9-HYDROXY-1,3-DIMETHYL-1,9-DIHYDRO-4H-PYRAZOLO[3,4-B]QUINOLIN-4-ONE, C-jun-amino-terminal kinase-interacting protein 1, Mitogen-activated protein kinase 8, ... | 著者 | Abad-Zapatero, C. | 登録日 | 2006-02-10 | 公開日 | 2006-04-18 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | Synthesis and SAR of 1,9-dihydro-9-hydroxypyrazolo[3,4-b]quinolin-4-ones as novel, selective c-Jun N-terminal kinase inhibitors. Bioorg.Med.Chem.Lett., 16, 2006
|
|
1JNM
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 1jnm by Molmil](/molmil-images/mine/1jnm) | Crystal Structure of the Jun/CRE Complex | 分子名称: | 5'-D(*CP*GP*TP*CP*GP*AP*TP*GP*AP*CP*GP*TP*CP*AP*TP*CP*GP*AP*CP*G)-3', PROTO-ONCOGENE C-JUN | 著者 | Kim, Y, Podust, L.M. | 登録日 | 2001-07-24 | 公開日 | 2003-06-03 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Crystal Structure of the Jun bZIP homodimer complexed with CRE To be Published
|
|
5EN2
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5en2 by Molmil](/molmil-images/mine/5en2) | Molecular basis for antibody-mediated neutralization of New World hemorrhagic fever mammarenaviruses | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, ... | 著者 | Mahmutovic, S, Clark, L, Levis, S, Briggiler, A, Enria, D, Harrison, S.C, Abraham, J. | 登録日 | 2015-11-09 | 公開日 | 2015-12-30 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.821 Å) | 主引用文献 | Molecular Basis for Antibody-Mediated Neutralization of New World Hemorrhagic Fever Mammarenaviruses. Cell Host Microbe, 18, 2015
|
|
6XJF
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 6xjf by Molmil](/molmil-images/mine/6xjf) | |
3VUD
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3vud by Molmil](/molmil-images/mine/3vud) | Crystal structure of a cysteine-deficient mutant M1 in MAP kinase JNK1 | 分子名称: | Mitogen-activated protein kinase 8, Peptide from C-Jun-amino-terminal kinase-interacting protein 1, SULFATE ION | 著者 | Nakaniwa, T, Kinoshita, T, Inoue, T. | 登録日 | 2012-06-28 | 公開日 | 2013-02-13 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (3.5 Å) | 主引用文献 | Seven cysteine-deficient mutants depict the interplay between thermal and chemical stabilities of individual cysteine residues in mitogen-activated protein kinase c-Jun N-terminal kinase 1 Biochemistry, 51, 2012
|
|
3VUM
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3vum by Molmil](/molmil-images/mine/3vum) | Crystal structure of a cysteine-deficient mutant M7 in MAP kinase JNK1 | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Mitogen-activated protein kinase 8, Peptide from C-Jun-amino-terminal kinase-interacting protein 1, ... | 著者 | Nakaniwa, T, Kinoshita, T, Inoue, T. | 登録日 | 2012-07-02 | 公開日 | 2013-02-13 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.69 Å) | 主引用文献 | Seven cysteine-deficient mutants depict the interplay between thermal and chemical stabilities of individual cysteine residues in mitogen-activated protein kinase c-Jun N-terminal kinase 1 Biochemistry, 51, 2012
|
|
3VUH
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3vuh by Molmil](/molmil-images/mine/3vuh) | Crystal structure of a cysteine-deficient mutant M3 in MAP kinase JNK1 | 分子名称: | GLYCEROL, Mitogen-activated protein kinase 8, Peptide from C-Jun-amino-terminal kinase-interacting protein 1, ... | 著者 | Nakaniwa, T, Kinoshita, T, Inoue, T. | 登録日 | 2012-06-28 | 公開日 | 2013-02-13 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Seven cysteine-deficient mutants depict the interplay between thermal and chemical stabilities of individual cysteine residues in mitogen-activated protein kinase c-Jun N-terminal kinase 1 Biochemistry, 51, 2012
|
|
3VUL
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3vul by Molmil](/molmil-images/mine/3vul) | |
3VUK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3vuk by Molmil](/molmil-images/mine/3vuk) | Crystal structure of a cysteine-deficient mutant M5 in MAP kinase JNK1 | 分子名称: | Mitogen-activated protein kinase 8, Peptide from C-Jun-amino-terminal kinase-interacting protein 1, SULFATE ION | 著者 | Nakaniwa, T, Kinoshita, T, Inoue, T. | 登録日 | 2012-07-02 | 公開日 | 2013-02-13 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.95 Å) | 主引用文献 | Seven cysteine-deficient mutants depict the interplay between thermal and chemical stabilities of individual cysteine residues in mitogen-activated protein kinase c-Jun N-terminal kinase 1 Biochemistry, 51, 2012
|
|
3VUG
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3vug by Molmil](/molmil-images/mine/3vug) | Crystal structure of a cysteine-deficient mutant M2 in MAP kinase JNK1 | 分子名称: | Mitogen-activated protein kinase 8, Peptide from C-Jun-amino-terminal kinase-interacting protein 1, SULFATE ION | 著者 | Nakaniwa, T, Kinoshita, T, Inoue, T. | 登録日 | 2012-06-28 | 公開日 | 2013-02-13 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (3.24 Å) | 主引用文献 | Seven cysteine-deficient mutants depict the interplay between thermal and chemical stabilities of individual cysteine residues in mitogen-activated protein kinase c-Jun N-terminal kinase 1 Biochemistry, 51, 2012
|
|
3VUI
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3vui by Molmil](/molmil-images/mine/3vui) | Crystal structure of a cysteine-deficient mutant M2 in MAP kinase JNK1 | 分子名称: | Mitogen-activated protein kinase 8, Peptide from C-Jun-amino-terminal kinase-interacting protein 1, SULFATE ION | 著者 | Nakaniwa, T, Kinoshita, T, Inoue, T. | 登録日 | 2012-06-28 | 公開日 | 2013-02-13 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Seven cysteine-deficient mutants depict the interplay between thermal and chemical stabilities of individual cysteine residues in mitogen-activated protein kinase c-Jun N-terminal kinase 1 Biochemistry, 51, 2012
|
|
4GKL
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 4gkl by Molmil](/molmil-images/mine/4gkl) | |
3OOB
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 3oob by Molmil](/molmil-images/mine/3oob) | Structural and functional insights of directly targeting Pin1 by Epigallocatechin-3-gallate | 分子名称: | (2R,3R)-5,7-dihydroxy-2-(3,4,5-trihydroxyphenyl)-3,4-dihydro-2H-chromen-3-yl 3,4,5-trihydroxybenzoate, 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1, ... | 著者 | Urusova, D.V, Shim, J.-H, Kim, D.-J, Jung, S.K, Zykova, T.A, Bode, A.M, Dong, Z. | 登録日 | 2010-08-30 | 公開日 | 2011-08-17 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (1.89 Å) | 主引用文献 | Epigallocatechin-gallate suppresses tumorigenesis by directly targeting Pin1. Cancer Prev Res (Phila), 4, 2011
|
|