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2JJI
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Endothiapepsin in complex with a gem-diol inhibitor.
分子名称: ENDOTHIAPEPSIN, N~2~-[(2R)-2-benzyl-3-(tert-butylsulfonyl)propanoyl]-N-{(1R)-1-(cyclohexylmethyl)-3,3-difluoro-2,2-dihydroxy-4-[(2-morpholin-4-ylethyl)amino]-4-oxobutyl}-3-(1H-imidazol-3-ium-4-yl)-L-alaninamide, SULFATE ION
著者Coates, L, Tuan, H.-F, Tomanicek, S.J, Kovalevsky, A, Mustyakimov, M, Erskine, P, Cooper, J.
登録日2008-04-09
公開日2008-05-27
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.57 Å)
主引用文献The Catalytic Mechanism of an Aspartic Proteinase Explored with Neutron and X-Ray Diffraction
J.Am.Chem.Soc., 130, 2008
2JJJ
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Endothiapepsin in complex with a gem-diol inhibitor.
分子名称: ENDOTHIAPEPSIN, N~2~-[(2R)-2-benzyl-3-(tert-butylsulfonyl)propanoyl]-N-{(1R)-1-(cyclohexylmethyl)-3,3-difluoro-2,2-dihydroxy-4-[(2-morpholin-4-ylethyl)amino]-4-oxobutyl}-3-(1H-imidazol-3-ium-4-yl)-L-alaninamide, SULFATE ION
著者Coates, L, Tuan, H.-F, Tomanicek, S.J, Kovalevsky, A, Mustyakimov, M, Erskine, P, Cooper, J.
登録日2008-04-09
公開日2008-05-27
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1 Å)
主引用文献The Catalytic Mechanism of an Aspartic Proteinase Explored with Neutron and X-Ray Diffraction
J.Am.Chem.Soc., 130, 2008
2JJK
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FRUCTOSE-1,6-BISPHOSPHATASE(D-FRUCTOSE-1,6-BISPHOSPHATE -1- PHOSPHOHYDROLASE) (E.C.3.1.3.11) COMPLEXED WITH A DUAL BINDING AMP SITE INHIBITOR
分子名称: FRUCTOSE-1,6-BISPHOSPHATASE 1, N,N'-(heptane-1,7-diyldicarbamoyl)bis(3-chlorobenzenesulfonamide)
著者Ruf, A, Joseph, C, Benz, J, Fol, B, Tetaz, T, Hebeisen, P.
登録日2008-04-09
公開日2008-07-22
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Allosteric Fbpase Inhibitors Gain 10(5) Times in Potency When Simultaneously Binding Two Neighboring AMP Sites.
Bioorg.Med.Chem.Lett., 18, 2008
2JJL
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Structure of avian reovirus sigmaC117-326, P321 crystal form
分子名称: CHLORIDE ION, SIGMA-C CAPSID PROTEIN, SULFATE ION, ...
著者Guardado-Calvo, P, Fox, G.C, Llamas-Saiz, A.L, Benavente, J, van Raaij, M.J.
登録日2008-04-14
公開日2009-01-13
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystallographic structure of the alpha-helical triple coiled-coil domain of avian reovirus S1133 fibre.
J. Gen. Virol., 90, 2009
2JJM
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Crystal Structure of a family GT4 glycosyltransferase from Bacillus anthracis ORF BA1558.
分子名称: GLYCOSYL TRANSFERASE, GROUP 1 FAMILY PROTEIN
著者Ruane, K.M, Davies, G.J, Martinez-Fleites, C.
登録日2008-04-15
公開日2008-08-05
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Crystal Structure of a Family Gt4 Glycosyltransferase from Bacillus Anthracis Orf Ba1558.
Proteins, 73, 2008
2JJN
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Structure of closed cytochrome P450 EryK
分子名称: CYTOCHROME P450 113A1, PROTOPORPHYRIN IX CONTAINING FE, SULFATE ION
著者Savino, C, Sciara, G, Miele, A.E, Kendrew, S.G, Vallone, B.
登録日2008-04-15
公開日2009-07-14
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.59 Å)
主引用文献Investigating the Structural Plasticity of a Cytochrome P450: Three-Dimensional Structures of P450 Eryk and Binding to its Physiological Substrate.
J.Biol.Chem., 284, 2009
2JJO
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Structure of cytochrome P450 EryK in complex with its natural substrate erD
分子名称: CYTOCHROME P450 113A1, Erythromycin D, PROTOPORPHYRIN IX CONTAINING FE
著者Savino, C, Sciara, G, Miele, A.E, Kendrew, S.G, Vallone, B.
登録日2008-04-15
公開日2009-07-14
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Investigating the Structural Plasticity of a Cytochrome P450: Three-Dimensional Structures of P450 Eryk and Binding to its Physiological Substrate.
J.Biol.Chem., 284, 2009
2JJP
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Structure of cytochrome P450 EryK in complex with inhibitor ketoconazole (KC)
分子名称: 1-ACETYL-4-(4-{[(2S,4R)-2-(2,4-DICHLOROPHENYL)-2-(1H-IMIDAZOL-1-YLMETHYL)-1,3-DIOXOLAN-4-YL]METHOXY}PHENYL)PIPERAZINE, CYTOCHROME P450 113A1, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Savino, C, Sciara, G, Miele, A.E, Kendrew, S.G, Vallone, B.
登録日2008-04-15
公開日2009-07-14
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Azole Drugs Trap Cytochrome P450 Eryk in Alternative Conformational States.
Biochemistry, 49, 2010
2JJQ
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The crystal structure of Pyrococcus abyssi tRNA (uracil-54, C5)- methyltransferase in complex with S-adenosyl-L-homocysteine
分子名称: GLYCEROL, S-ADENOSYL-L-HOMOCYSTEINE, UNCHARACTERIZED RNA METHYLTRANSFERASE PYRAB10780
著者Walbott, H, Leulliot, N, Grosjean, H, Golinelli-Pimpaneau, B.
登録日2008-04-17
公開日2008-08-05
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献The Crystal Structure of Pyrococcus Abyssi tRNA (Uracil-54, C5)-Methyltransferase Provides Insights Into its tRNA Specificity.
Nucleic Acids Res., 36, 2008
2JJR
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V232K, N236D-trichosanthin
分子名称: DI(HYDROXYETHYL)ETHER, RIBOSOME-INACTIVATING PROTEIN ALPHA-TRICHOSANTHIN, SULFATE ION, ...
著者Too, P.H, Ma, M.K, Mak, A.N, Tung, C.K, Zhu, G, Au, S.W, Wong, K.B, Shaw, P.C.
登録日2008-04-21
公開日2008-12-30
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献The C-Terminal Fragment of the Ribosomal P Protein Complexed to Trichosanthin Reveals the Interaction between the Ribosome-Inactivating Protein and the Ribosome.
Nucleic Acids Res., 37, 2009
2JJS
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Structure of human CD47 in complex with human signal regulatory protein (SIRP) alpha
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, IODIDE ION, LEUKOCYTE SURFACE ANTIGEN CD47, ...
著者Hatherley, D, Graham, S.C, Turner, J, Harlos, K, Stuart, D.I, Barclay, A.N.
登録日2008-04-22
公開日2008-08-05
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Paired receptor specificity explained by structures of signal regulatory proteins alone and complexed with CD47.
Mol. Cell, 31, 2008
2JJT
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Structure of human CD47 in complex with human signal regulatory protein (SIRP) alpha
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, LEUKOCYTE SURFACE ANTIGEN CD47, TYROSINE-PROTEIN PHOSPHATASE NON-RECEPTOR TYPE SUBSTRATE 1
著者Hatherley, D, Graham, S.C, Turner, J, Harlos, K, Stuart, D.I, Barclay, A.N.
登録日2008-04-22
公開日2008-08-05
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Paired receptor specificity explained by structures of signal regulatory proteins alone and complexed with CD47.
Mol. Cell, 31, 2008
2JJU
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Structure of human signal regulatory protein (sirp) beta
分子名称: CHLORIDE ION, SIGNAL REGULATORY PROTEIN BETA-1, SULFATE ION
著者Hatherley, D, Graham, S.C, Turner, J, Harlos, K, Stuart, D.I, Barclay, A.N.
登録日2008-04-22
公開日2008-08-05
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.19 Å)
主引用文献Paired Receptor Specificity Explained by Structures of Signal Regulatory Proteins Alone and Complexed with Cd47.
Mol.Cell, 31, 2008
2JJV
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Structure of human signal regulatory protein (sirp) beta(2)
分子名称: CHLORIDE ION, SIGNAL-REGULATORY PROTEIN BETA 1., SULFATE ION
著者Hatherley, D, Graham, S.C, Turner, J, Harlos, K, Stuart, D.I, Barclay, A.N.
登録日2008-04-22
公開日2008-08-05
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Paired Receptor Specificity Explained by Structures of Signal Regulatory Proteins Alone and Complexed with Cd47.
Mol.Cell, 31, 2008
2JJW
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Structure of human signal regulatory protein (sirp) gamma
分子名称: SIGNAL REGULATORY PROTEIN GAMMA
著者Hatherley, D, Graham, S.C, Turner, J, Harlos, K, Stuart, D.I, Barclay, A.N.
登録日2008-04-22
公開日2008-08-05
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Paired Receptor Specificity Explained by Structures of Signal Regulatory Proteins Alone and Complexed with Cd47.
Mol.Cell, 31, 2008
2JJX
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THE CRYSTAL STRUCTURE OF UMP KINASE FROM BACILLUS ANTHRACIS (BA1797)
分子名称: ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, URIDYLATE KINASE
著者Meier, C, Carter, L.G, Mancini, E.J, Owens, R.J, Stuart, D.I, Esnouf, R.M, Oxford Protein Production Facility (OPPF), Structural Proteomics in Europe (SPINE)
登録日2008-04-23
公開日2008-07-29
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.82 Å)
主引用文献The Crystal Structure of Ump Kinase from Bacillus Anthracis (Ba1797) Reveals an Allosteric Nucleotide-Binding Site.
J.Mol.Biol., 381, 2008
2JJY
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Crystal structure of Francisella tularensis enoyl reductase (ftFabI) with bound NAD
分子名称: ENOYL-[ACYL-CARRIER-PROTEIN] REDUCTASE, NICOTINAMIDE-ADENINE-DINUCLEOTIDE
著者Luckner, S.R, Lu, H, Truglio, J.J, Tonge, P.J, Kisker, C.
登録日2008-04-25
公開日2009-02-24
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Slow-Onset Inhibition of the Fabi Enoyl Reductase from Francisella Tularensis: Residence Time and in Vivo Activity
Acs Chem.Biol., 4, 2009
2JJZ
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Crystal Structure of Human Iba2, orthorhombic crystal form
分子名称: ACETATE ION, CHLORIDE ION, IONIZED CALCIUM-BINDING ADAPTER MOLECULE 2, ...
著者Schulze, J.O, Quedenau, C, Roske, Y, Turnbull, A, Mueller, U, Heinemann, U, Buessow, K.
登録日2008-05-15
公開日2009-07-14
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Structural and Functional Characterization of Human Iba Proteins.
FEBS J., 275, 2008
2JK0
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Structural and functional insights into Erwinia carotovora L- asparaginase
分子名称: ASPARTIC ACID, L-ASPARAGINASE
著者Papageorgiou, A.C, Posypanova, G.A, Andersson, C.S, Sokolov, N.N, Krasotkina, J.
登録日2008-05-23
公開日2008-08-05
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural and Functional Insights Into Erwinia Carotovora L-Asparaginase.
FEBS J., 275, 2008
2JK1
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Crystal structure of the wild-type HupR receiver domain
分子名称: HYDROGENASE TRANSCRIPTIONAL REGULATORY PROTEIN HUPR1, MAGNESIUM ION
著者Davies, K.M, Lowe, E.D, Venien-Bryan, C, Johnson, L.N.
登録日2008-05-26
公開日2008-11-11
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献The Hupr Receiver Domain Crystal Structure in its Nonphospho and Inhibitory Phospho States.
J.Mol.Biol., 385, 2009
2JK2
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STRUCTURAL BASIS OF HUMAN TRIOSEPHOSPHATE ISOMERASE DEFICIENCY. CRYSTAL STRUCTURE OF THE WILD TYPE ENZYME.
分子名称: TRIOSEPHOSPHATE ISOMERASE
著者Rodriguez-Almazan, C, Arreola-Alemon, R, Rodriguez-Larrea, D, Aguirre-Lopez, B, De Gomez-Puyou, M.T, Perez-Montfort, R, Costas, M, Gomez-Puyou, A, Torres-Larios, A.
登録日2008-06-22
公開日2008-07-01
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural Basis of Human Triosephosphate Isomerase Deficiency: Mutation E104D is Related to Alterations of a Conserved Water Network at the Dimer Interface.
J.Biol.Chem., 283, 2008
2JK3
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CRYSTAL STRUCTURE OF THE HLYIIR MUTANT PROTEIN WITH RESIDUES 169-186 SUBSTITUTED BY GSSGSSG LINKER
分子名称: HEMOLYSIN II REGULATORY PROTEIN, SULFATE ION
著者Kovalevskiy, O.V, Solonin, A.S, Antson, A.A.
登録日2008-08-11
公開日2008-08-19
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural Investigation of Transcriptional Regulator Hlyiir: Influence of a Disordered Region on Protein Fold and Dimerization.
Proteins, 78, 2010
2JK4
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Structure of the human voltage-dependent anion channel
分子名称: VOLTAGE-DEPENDENT ANION-SELECTIVE CHANNEL PROTEIN 1
著者Bayrhuber, M, Meins, T, Habeck, M, Becker, S, Giller, K, Villinger, S, Vonrhein, C, Griesinger, C, Zweckstetter, M, Zeth, K.
登録日2008-08-15
公開日2008-10-14
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (4.1 Å)
主引用文献Structure of the Human Voltage-Dependent Anion Channel.
Proc.Natl.Acad.Sci.USA, 105, 2008
2JK5
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Potassium Channel KcsA in complex with Tetrabutylammonium in high K
分子名称: (2S)-3-HYDROXY-2-(NONANOYLOXY)PROPYL LAURATE, ANTIBODY FAB FRAGMENT HEAVY CHAIN, ANTIBODY FAB FRAGMENT LIGHT CHAIN, ...
著者Lenaeus, M.J, Focia, P.J, Wagner, T, Gross, A.
登録日2008-08-15
公開日2009-11-17
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structures of Kcsa in Complex with Symmetrical Quaternary Ammonium Compounds Reveal a Hydrophobic Binding Site.
Biochemistry, 53, 2014
2JK6
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Structure of Trypanothione Reductase from Leishmania infantum
分子名称: FLAVIN-ADENINE DINUCLEOTIDE, SULFATE ION, TRYPANOTHIONE REDUCTASE
著者Baiocco, P, Colotti, G, Franceschini, S, Ilari, A.
登録日2008-08-21
公開日2009-04-28
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Molecular Basis of Antimony Treatment in Leishmaniasis.
J.Med.Chem., 52, 2009

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