8D8F
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8D8C
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8D8B
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8A3Q
| Human Plasma Kallekrein in complex with 14W | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, Plasma kallikrein, ... | 著者 | McEwan, P.A. | 登録日 | 2022-06-08 | 公開日 | 2022-11-02 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.801 Å) | 主引用文献 | Sebetralstat (KVD900): A Potent and Selective Small Molecule Plasma Kallikrein Inhibitor Featuring a Novel P1 Group as a Potential Oral On-Demand Treatment for Hereditary Angioedema. J.Med.Chem., 65, 2022
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8D80
| Cereblon~DDB1 bound to Iberdomide and Ikaros ZF1-2-3 | 分子名称: | (3S)-3-[4-({4-[(morpholin-4-yl)methyl]phenyl}methoxy)-1-oxo-1,3-dihydro-2H-isoindol-2-yl]piperidine-2,6-dione, DNA damage-binding protein 1, DNA-binding protein Ikaros, ... | 著者 | Watson, E.R, Lander, G.C. | 登録日 | 2022-06-07 | 公開日 | 2022-07-20 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Molecular glue CELMoD compounds are regulators of cereblon conformation. Science, 378, 2022
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8D74
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8D7R
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8D7E
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8D7H
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8D82
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8D85
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8D7M
| Human Casein kinase 1 delta in complex with phosphorylated human PERIOD2 FASP peptide | 分子名称: | Casein kinase I isoform delta, Period circadian protein homolog 2 peptide | 著者 | Philpott, J.M, Freeberg, A.M, Tripathi, S.M, Partch, C.L. | 登録日 | 2022-06-07 | 公開日 | 2023-05-17 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | PERIOD phosphorylation leads to feedback inhibition of CK1 activity to control circadian period. Mol.Cell, 83, 2023
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8D7O
| Human Casein kinase 1 delta in complex with phosphorylated human PERIOD2 FASP peptide | 分子名称: | Casein kinase I isoform delta, Period circadian protein homolog 2 peptide | 著者 | Philpott, J.M, Freeberg, A.M, Tripathi, S.M, Partch, C.L. | 登録日 | 2022-06-07 | 公開日 | 2023-05-17 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | PERIOD phosphorylation leads to feedback inhibition of CK1 activity to control circadian period. Mol.Cell, 83, 2023
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8D7P
| Human Casein kinase 1 delta in complex with phosphorylated Drosophila PERIOD peptide | 分子名称: | Casein kinase I isoform delta, Period circadian protein peptide | 著者 | Philpott, J.M, Freeberg, A.M, Tripathi, S.M, Partch, C.L. | 登録日 | 2022-06-07 | 公開日 | 2023-05-17 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | PERIOD phosphorylation leads to feedback inhibition of CK1 activity to control circadian period. Mol.Cell, 83, 2023
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8D7N
| Human Casein kinase 1 delta in complex with phosphorylated human PERIOD2 FASP peptide | 分子名称: | Casein kinase I isoform delta, Period circadian protein homolog 2 peptide | 著者 | Philpott, J.M, Freeberg, A.M, Tripathi, S.M, Partch, C.L. | 登録日 | 2022-06-07 | 公開日 | 2023-05-17 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.66 Å) | 主引用文献 | PERIOD phosphorylation leads to feedback inhibition of CK1 activity to control circadian period. Mol.Cell, 83, 2023
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8D7Z
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8D7L
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8D77
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8D7Q
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8D75
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8D7A
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8D7J
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8D7D
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8D7B
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8D7C
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