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1E7U
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Structure determinants of phosphoinositide 3-kinase inhibition by wortmannin, LY294002, quercetin, myricetin and staurosporine
分子名称: (1S,6BR,9AS,11R,11BR)-9A,11B-DIMETHYL-1-[(METHYLOXY)METHYL]-3,6,9-TRIOXO-1,6,6B,7,8,9,9A,10,11,11B-DECAHYDRO-3H-FURO[4, 3,2-DE]INDENO[4,5-H][2]BENZOPYRAN-11-YL ACETATE, PHOSPHATIDYLINOSITOL 3-KINASE CATALYTIC SUBUNIT
著者Walker, E.H, Perisic, O, Ried, C, Stephens, L, Williams, R.L.
登録日2000-09-08
公開日2000-11-17
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural Determinations of Phosphoinositide 3-Kinase Inhibition by Wortmannin, Ly294002, Quercetin, Myricetin and Staurosporine
Mol.Cell, 6, 2000
1E6L
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Two-component signal transduction system D13A mutant of CheY
分子名称: Chemotaxis protein CheY
著者Sola, M, Lopez-Hernandez, E, Cronet, P, Lacroix, E, Serrano, L, Coll, M, Parraga, A.
登録日2000-08-18
公開日2001-03-05
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Towards understanding a molecular switch mechanism: thermodynamic and crystallographic studies of the signal transduction protein CheY.
J.Mol.Biol., 303, 2000
1E55
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Crystal structure of the inactive mutant Monocot (Maize ZMGlu1) beta-glucosidase ZMGluE191D in complex with the competitive inhibitor dhurrin
分子名称: (2S)-HYDROXY(4-HYDROXYPHENYL)ETHANENITRILE, BETA-GLUCOSIDASE, beta-D-glucopyranose
著者Czjzek, M, Cicek, M, Bevan, D.R, Zamboni, V, Henrissat, B, Esen, A.
登録日2000-07-18
公開日2000-12-11
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The mechanism of substrate (aglycone) specificity in beta-glucosidases is revealed by crystal structures of mutant maize beta-glucosidase-DIMBOA, -DIMBOAGlc, and -dhurrin complexes.
Proc. Natl. Acad. Sci. U.S.A., 97, 2000
5H8J
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Crystal structure of Medicago truncatula N-carbamoylputrescine amidohydrolase (MtCPA) in complex with cadaverine
分子名称: 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, GLYCEROL, ...
著者Sekula, B, Ruszkowski, M, Malinska, M, Dauter, Z.
登録日2015-12-23
公開日2016-04-20
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.19 Å)
主引用文献Structural Investigations of N-carbamoylputrescine Amidohydrolase from Medicago truncatula: Insights into the Ultimate Step of Putrescine Biosynthesis in Plants.
Front Plant Sci, 7, 2016
1E63
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Ferredoxin:NADP+ Reductase Mutant with LYS 75 Replaced by SER (K75S)
分子名称: FERREDOXIN-NADP+ REDUCTASE, FLAVIN-ADENINE DINUCLEOTIDE, SULFATE ION
著者Hermoso, J.A, Mayoral, T, Medina, M, Gomez-Moreno, C.
登録日2000-08-07
公開日2001-05-25
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural Analysis of Interactions for Complex Formation between Ferredoxin-Nadp+ Reductase and its Protein Partners.
Proteins, 59, 2005
2YJK
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Structure of Dps from MICROBACTERIUM ARBORESCENS in the high iron form
分子名称: AFP, FE (III) ION, Iron(II) oxide
著者Zeth, K, Buecheler, R, Boland, W.
登録日2011-05-19
公開日2011-06-01
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure and Mechanism of Iron Translocation by a Dps Protein from Microbacterium Arborescens.
J.Biol.Chem., 286, 2011
1E8S
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Alu domain of the mammalian SRP (potential Alu retroposition intermediate)
分子名称: 7SL RNA, 88-MER, EUROPIUM (III) ION, ...
著者Weichenrieder, O, Wild, K, Strub, K, Cusack, S.
登録日2000-09-29
公開日2000-11-08
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (4 Å)
主引用文献Structure and Assembly of the Alu Domain of the Mammalian Signal Recognition Particle
Nature, 408, 2000
1E97
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Crystal structure of ketosteroid isomerase from Pseudomonas putida ; triple mutant y16f/y32f/y57f
分子名称: STEROID DELTA-ISOMERASE
著者Ha, N.-C, Oh, B.-H.
登録日2000-10-10
公開日2001-10-05
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Peudoreversion of the Catalytic Activity of Y14F by the Additional Substitution(S) of Tyrosine with Phenylalanine in the Hydrogen Bond Network of Delta 5-3-Ketosteroid Isomerase from Pseudomonas Putida Biotype B
Biochemistry, 40, 2001
1E8U
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Structure of the multifunctional paramyxovirus hemagglutinin-neuraminidase
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, HEMAGGLUTININ-NEURAMINIDASE, ...
著者Crennell, S, Takimoto, T, Portner, A, Taylor, G.
登録日2000-10-01
公開日2001-04-03
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal Structure of the Multifunctional Paramyxovirus Hemagglutinin-Neuraminidase
Nat.Struct.Biol., 7, 2000
1EAX
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Crystal structure of MTSP1 (matriptase)
分子名称: BENZAMIDINE, SULFATE ION, SUPPRESSOR OF TUMORIGENICITY 14
著者Friedrich, R, Bode, W.
登録日2001-07-17
公開日2002-01-28
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Catalytic Domain Structures of Mt-Sp1/Matriptase, a Matrix-Degrading Transmembrane Serine Proteinase.
J.Biol.Chem., 277, 2002
5H8L
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Crystal structure of Medicago truncatula N-carbamoylputrescine amidohydrolase (MtCPA) C158S mutant in complex with putrescine
分子名称: 1,2-ETHANEDIOL, 1,4-DIAMINOBUTANE, DI(HYDROXYETHYL)ETHER, ...
著者Sekula, B, Ruszkowski, M, Malinska, M, Dauter, Z.
登録日2015-12-23
公開日2016-04-20
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.29 Å)
主引用文献Structural Investigations of N-carbamoylputrescine Amidohydrolase from Medicago truncatula: Insights into the Ultimate Step of Putrescine Biosynthesis in Plants.
Front Plant Sci, 7, 2016
1EA2
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Pseudoreversion of the Catalytic Activity of Y14F by the Additional Tyrosine-to-Phenylalanine Substitution(s) in the Hydrogen Bond Network of Delta-5-3-Ketosteroid Isomerase from Pheudomonas putida Biotype B
分子名称: STEROID DELTA-ISOMERASE
著者Choi, G, Ha, N.-C, Kim, M.-S, Hong, B.-H, Choi, K.Y.
登録日2000-11-03
公開日2001-11-01
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Pseudoreversion of the Catalytic Activity of Y14F by the Additional Substitution(S) of Tyrosine with Phenylalanine in the Hydrogen Bond Network of Delta (5)-3-Ketosteroid Isomerase from Pseudomonas Putida Biotype B
Biochemistry, 40, 2001
2YA5
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Crystal structure of Streptococcus pneumoniae NanA (TIGR4) in complex with sialic acid
分子名称: CHLORIDE ION, FORMIC ACID, N-acetyl-alpha-neuraminic acid, ...
著者Gut, H, Xu, G, Taylor, G.L, Walsh, M.A.
登録日2011-02-18
公開日2011-04-27
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural Basis for Streptococcus Pneumoniae Nana Inhibition by Influenza Antivirals Zanamivir and Oseltamivir Carboxylate.
J.Mol.Biol., 409, 2011
1ECJ
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ESCHERICHIA COLI GLUTAMINE PHOSPHORIBOSYLPYROPHOSPHATE (PRPP) AMIDOTRANSFERASE COMPLEXED WITH 2 AMP PER TETRAMER
分子名称: ADENOSINE MONOPHOSPHATE, GLUTAMINE PHOSPHORIBOSYLPYROPHOSPHATE AMIDOTRANSFERASE
著者Muchmore, C.R, Krahn, J.M, Smith, J.L.
登録日1997-07-16
公開日1998-04-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of glutamine phosphoribosylpyrophosphate amidotransferase from Escherichia coli.
Protein Sci., 7, 1998
1EDM
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EPIDERMAL GROWTH FACTOR-LIKE DOMAIN FROM HUMAN FACTOR IX
分子名称: CALCIUM ION, FACTOR IX
著者Rao, Z, Handford, P, Mayhew, M, Knott, V, Brownlee, G.G, Stuart, D.
登録日1996-03-21
公開日1996-10-14
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献The structure of a Ca(2+)-binding epidermal growth factor-like domain: its role in protein-protein interactions.
Cell(Cambridge,Mass.), 82, 1995
5IB8
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Structure of T. thermophilus 70S ribosome complex with mRNA, tRNAfMet and near-cognate tRNALys with U-G mismatch in the A-site
分子名称: 16S ribosomal RNA, 23S ribosomal RNA, 30S ribosomal protein S10, ...
著者Rozov, A, Demeshkina, N, Yusupov, M, Yusupova, G.
登録日2016-02-22
公開日2016-05-25
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (3.13 Å)
主引用文献The ribosome prohibits the GU wobble geometry at the first position of the codon-anticodon helix.
Nucleic Acids Res., 44, 2016
1ERU
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HUMAN THIOREDOXIN (OXIDIZED FORM)
分子名称: THIOREDOXIN
著者Weichsel, A, Gasdaska, J.R, Powis, G, Montfort, W.R.
登録日1996-02-07
公開日1996-08-01
最終更新日2018-04-18
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystal structures of reduced, oxidized, and mutated human thioredoxins: evidence for a regulatory homodimer.
Structure, 4, 1996
1EI4
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B-DNA DODECAMER CGCGAAT(TLC)CGCG WITH INCORPORATED [3.3.0]BICYCLO-ARABINO-THYMINE-5'-PHOSPHATE
分子名称: DNA (5'-D(*CP*GP*CP*GP*AP*AP*(TLC)P*(TLC)P*CP*GP*CP*G)-3'), MAGNESIUM ION, SPERMINE
著者Minasov, G, Teplova, M, Nielsen, P, Wengel, J, Egli, M.
登録日2000-02-24
公開日2000-03-27
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.43 Å)
主引用文献Structural basis of cleavage by RNase H of hybrids of arabinonucleic acids and RNA.
Biochemistry, 39, 2000
1ETJ
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AZURIN MUTANT WITH MET 121 REPLACED BY GLU
分子名称: AZURIN, COPPER (II) ION
著者Karlsson, B.G, Tsai, L.-C, Nar, H, Sanders-Loehr, J, Bonander, N, Langer, V, Sjolin, L.
登録日1997-01-11
公開日1997-04-21
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献X-ray structure determination and characterization of the Pseudomonas aeruginosa azurin mutant Met121Glu.
Biochemistry, 36, 1997
1ENA
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CRYSTAL STRUCTURES OF THE BINARY CA2+ AND PDTP COMPLEXES AND THE TERNARY COMPLEX OF THE ASP 21->GLU MUTANT OF STAPHYLOCOCCAL NUCLEASE. IMPLICATIONS FOR CATALYSIS AND LIGAND BINDING
分子名称: CALCIUM ION, STAPHYLOCOCCAL NUCLEASE
著者Libson, A, Gittis, A, Lattman, E.E.
登録日1994-02-14
公開日1994-05-31
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Crystal structures of the binary Ca2+ and pdTp complexes and the ternary complex of the Asp21-->Glu mutant of staphylococcal nuclease. Implications for catalysis and ligand binding.
Biochemistry, 33, 1994
1EUS
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SIALIDASE COMPLEXED WITH 2-DEOXY-2,3-DEHYDRO-N-ACETYLNEURAMINIC ACID
分子名称: 2-DEOXY-2,3-DEHYDRO-N-ACETYL-NEURAMINIC ACID, SIALIDASE
著者Gaskell, A, Crennell, S.J, Taylor, G.L.
登録日1996-06-21
公開日1997-01-11
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献The three domains of a bacterial sialidase: a beta-propeller, an immunoglobulin module and a galactose-binding jelly-roll.
Structure, 3, 1995
1EXP
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BETA-1,4-GLYCANASE CEX-CD
分子名称: BETA-1,4-D-GLYCANASE CEX-CD, beta-D-glucopyranose-(1-4)-2-deoxy-2-fluoro-alpha-D-glucopyranose
著者White, A, Tull, D, Johns, K.L, Withers, S.G, Rose, D.R.
登録日1996-01-11
公開日1997-01-27
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystallographic observation of a covalent catalytic intermediate in a beta-glycosidase.
Nat.Struct.Biol., 3, 1996
1EAH
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PV2L COMPLEXED WITH ANTIVIRAL AGENT SCH48973
分子名称: 1[2-CHLORO-4-METHOXY-PHENYL-OXYMETHYL]-4-[2,6-DICHLORO-PHENYL-OXYMETHYL]-BENZENE, MYRISTIC ACID, POLIOVIRUS TYPE 2 COAT PROTEINS VP1 TO VP4
著者Lentz, K, Arnold, E.
登録日1997-07-22
公開日1998-09-16
最終更新日2023-04-19
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structure of poliovirus type 2 Lansing complexed with antiviral agent SCH48973: comparison of the structural and biological properties of three poliovirus serotypes.
Structure, 5, 1997
1E6Y
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Methyl-coenzyme M reductase from Methanosarcina barkeri
分子名称: 1-THIOETHANESULFONIC ACID, Coenzyme B, FACTOR 430, ...
著者Grabarse, W, Ermler, U.
登録日2000-08-23
公開日2000-10-18
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Comparison of Three Methyl-Coenzyme M Reductases from Phylogenetically Distant Organisms: Unusual Amino Acid Modification, Conservation and Adaptation
J.Mol.Biol., 303, 2000
1EUH
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APO FORM OF A NADP DEPENDENT ALDEHYDE DEHYDROGENASE FROM STREPTOCOCCUS MUTANS
分子名称: NADP DEPENDENT NON PHOSPHORYLATING GLYCERALDEHYDE-3-PHOSPHATE DEHYDROGENASE, SULFATE ION
著者Cobessi, D, Tete-Favier, F, Marchal, S, Branlant, G, Aubry, A.
登録日1998-11-05
公開日1999-07-22
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.82 Å)
主引用文献Apo and holo crystal structures of an NADP-dependent aldehyde dehydrogenase from Streptococcus mutans.
J.Mol.Biol., 290, 1999

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