8S32
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![BU of 8s32 by Molmil](/molmil-images/mine/8s32) | GroEL with bound GroTAC peptide | 分子名称: | Chaperonin GroEL, GroTAC | 著者 | Wroblewski, K, Izert-Nowakowska, M.A, Goral, T.K, Klimecka, M.M, Kmiecik, S, Gorna, M.W. | 登録日 | 2024-02-19 | 公開日 | 2024-02-28 | 実験手法 | ELECTRON MICROSCOPY (2.45 Å) | 主引用文献 | Depletion of essential GroEL protein in Escherichia coli using Clp-Interacting Peptidic Protein Erasers (CLIPPERs) To Be Published
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5AR7
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![BU of 5ar7 by Molmil](/molmil-images/mine/5ar7) | RIP2 Kinase Catalytic Domain (1 - 310) complex with Biaryl Urea | 分子名称: | 1-(5-TERT-BUTYL-1,2-OXAZOL-3-YL)-3-(4-PYRIDIN-4-YLOXYPHENYL)UREA, RECEPTOR-INTERACTING SERINE/THREONINE-PROTEIN KINASE 2 | 著者 | Charnley, A.K, Convery, M.A, Lakdawala Shah, A, Jones, E, Hardwicke, P, Bridges, A, Votta, B.J, Gough, P.J, Marquis, R.W, Bertin, J, Casillas, L. | 登録日 | 2015-09-24 | 公開日 | 2015-10-21 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.71 Å) | 主引用文献 | Crystal Structures of Human Rip2 Kinase Catalytic Domain Complexed with ATP-Competitive Inhibitors: Foundations for Understanding Inhibitor Selectivity. Bioorg.Med.Chem., 23, 2015
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5AR2
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![BU of 5ar2 by Molmil](/molmil-images/mine/5ar2) | RIP2 Kinase Catalytic Domain (1 - 310) | 分子名称: | CALCIUM ION, RECEPTOR-INTERACTING SERINE/THREONINE-PROTEIN KINASE 2 | 著者 | Charnley, A.K, Convery, M.A, Lakdawala Shah, A, Jones, E, Hardwicke, P, Bridges, A, Votta, B.J, Gough, P.J, Marquis, R.W, Bertin, J, Casillas, L. | 登録日 | 2015-09-23 | 公開日 | 2015-10-21 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.44 Å) | 主引用文献 | Crystal Structures of Human Rip2 Kinase Catalytic Domain Complexed with ATP-Competitive Inhibitors: Foundations for Understanding Inhibitor Selectivity. Bioorg.Med.Chem., 23, 2015
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5AR3
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![BU of 5ar3 by Molmil](/molmil-images/mine/5ar3) | RIP2 Kinase Catalytic Domain (1 - 310) complex with AMP-PCP | 分子名称: | MAGNESIUM ION, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, RECEPTOR-INTERACTING SERINE/THREONINE-PROTEIN KINASE 2 | 著者 | Charnley, A.K, Convery, M.A, Lakdawala Shah, A, Jones, E, Hardwicke, P, Bridges, A, Votta, B.J, Gough, P.J, Marquis, R.W, Bertin, J, Casillas, L. | 登録日 | 2015-09-23 | 公開日 | 2015-10-21 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (3.23 Å) | 主引用文献 | Crystal Structures of Human Rip2 Kinase Catalytic Domain Complexed with ATP-Competitive Inhibitors: Foundations for Understanding Inhibitor Selectivity. Bioorg.Med.Chem., 23, 2015
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3TLK
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![BU of 3tlk by Molmil](/molmil-images/mine/3tlk) | Crystal structure of holo FepB | 分子名称: | 1,4-DIETHYLENE DIOXIDE, FE (III) ION, Ferrienterobactin-binding periplasmic protein, ... | 著者 | Li, N, Gu, L. | 登録日 | 2011-08-30 | 公開日 | 2013-01-16 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.853 Å) | 主引用文献 | Crystal structure of holo FepB To be Published
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4WBQ
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![BU of 4wbq by Molmil](/molmil-images/mine/4wbq) | Crystal structure of the exonuclease domain of QIP (QDE-2 interacting protein) solved by native-SAD phasing. | 分子名称: | CALCIUM ION, QDE-2-interacting protein | 著者 | Boland, A, Weinert, T, Weichenrieder, O, Wang, M. | 登録日 | 2014-09-03 | 公開日 | 2014-12-10 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.693 Å) | 主引用文献 | Fast native-SAD phasing for routine macromolecular structure determination. Nat.Methods, 12, 2015
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7LTB
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![BU of 7ltb by Molmil](/molmil-images/mine/7ltb) | Crystal Structure of Keratinicyclin B | 分子名称: | (2~{S},4~{S},5~{R},6~{S})-4-azanyl-5-methoxy-6-methyl-oxan-2-ol, 3-ammonio-2,3,6-trideoxy-alpha-L-arabino-hexopyranose-(1-2)-beta-D-glucopyranose, FORMIC ACID, ... | 著者 | Davis, K.M, Jeffrey, P.D, Seyedsayamdost, M.R. | 登録日 | 2021-02-19 | 公開日 | 2022-12-07 | 最終更新日 | 2024-07-24 | 実験手法 | X-RAY DIFFRACTION (0.95 Å) | 主引用文献 | Potent and specific antibiotic combination therapy against Clostridioides difficile. Nat.Chem.Biol., 20, 2024
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7LKC
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![BU of 7lkc by Molmil](/molmil-images/mine/7lkc) | Crystal Structure of Keratinimicin A | 分子名称: | (2~{S},4~{S},5~{R},6~{S})-4-azanyl-5-methoxy-6-methyl-oxan-2-ol, CHLORIDE ION, FORMIC ACID, ... | 著者 | Davis, K.M, Jeffrey, P.D, Seyedsayamdost, M.R. | 登録日 | 2021-02-02 | 公開日 | 2022-12-07 | 最終更新日 | 2024-07-24 | 実験手法 | X-RAY DIFFRACTION (0.95 Å) | 主引用文献 | Potent and specific antibiotic combination therapy against Clostridioides difficile. Nat.Chem.Biol., 20, 2024
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7M5M
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![BU of 7m5m by Molmil](/molmil-images/mine/7m5m) | PCNA bound to peptide mimetic | 分子名称: | N-BUTANE, Peptide mimetic (ACE)RQCSMTCFYHSK(NH2) with linker, Proliferating cell nuclear antigen | 著者 | Vandborg, B.A, Bruning, J.B. | 登録日 | 2021-03-24 | 公開日 | 2021-08-11 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | A cell permeable bimane-constrained PCNA-interacting peptide. Rsc Chem Biol, 2, 2021
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7M5L
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4NEU
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![BU of 4neu by Molmil](/molmil-images/mine/4neu) | X-ray structure of Receptor Interacting Protein 1 (RIP1)kinase domain with a 1-aminoisoquinoline inhibitor | 分子名称: | 1-[4-(1-aminoisoquinolin-5-yl)phenyl]-3-(5-tert-butyl-1,2-oxazol-3-yl)urea, MAGNESIUM ION, Receptor-interacting serine/threonine-protein kinase 1 | 著者 | Nolte, R.T, Ward, P, kahler, K.M, Campobasso, N. | 登録日 | 2013-10-30 | 公開日 | 2013-11-20 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.57 Å) | 主引用文献 | Discovery of Small Molecule RIP1 Kinase Inhibitors for the Treatment of Pathologies Associated with Necroptosis. ACS Med Chem Lett, 4, 2013
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7M5N
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![BU of 7m5n by Molmil](/molmil-images/mine/7m5n) | PCNA bound to peptide mimetic with linker | 分子名称: | 1,3-dimethylbenzene, Peptide mimetic (ACE)RQCSMTCFYHSK(NH2) with linker, Proliferating cell nuclear antigen | 著者 | Vandborg, B.A, Bruning, J.B. | 登録日 | 2021-03-24 | 公開日 | 2021-08-11 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (3.11 Å) | 主引用文献 | A cell permeable bimane-constrained PCNA-interacting peptide. Rsc Chem Biol, 2, 2021
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5AR5
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![BU of 5ar5 by Molmil](/molmil-images/mine/5ar5) | RIP2 Kinase Catalytic Domain (1 - 310) complex with Benzimidazole | 分子名称: | 2-(2-(4-CHLOROPHENYL)-1H-IMIDAZOL-5-YL)-N,1-BIS(2-METHOXYETHYL)-1H-BENZO[D]IMIDAZOLE-5-CARBOXAMIDE, CALCIUM ION, RECEPTOR-INTERACTING SERINE/THREONINE-PROTEIN KINASE 2 | 著者 | Charnley, A.K, Convery, M.A, Lakdawala Shah, A, Jones, E, Hardwicke, P, Bridges, A, Votta, B.J, Gough, P.J, Marquis, R.W, Bertin, J, Casillas, L. | 登録日 | 2015-09-24 | 公開日 | 2015-10-21 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.66 Å) | 主引用文献 | Crystal Structures of Human Rip2 Kinase Catalytic Domain Complexed with ATP-Competitive Inhibitors: Foundations for Understanding Inhibitor Selectivity. Bioorg.Med.Chem., 23, 2015
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5AR4
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![BU of 5ar4 by Molmil](/molmil-images/mine/5ar4) | RIP2 Kinase Catalytic Domain (1 - 310) complex with SB-203580 | 分子名称: | 4-[5-(4-FLUORO-PHENYL)-2-(4-METHANESULFINYL-PHENYL)-3H-IMIDAZOL-4-YL]-PYRIDINE, RECEPTOR-INTERACTING SERINE/THREONINE-PROTEIN KINASE 2 | 著者 | Charnley, A.K, Convery, M.A, Lakdawala Shah, A, Jones, E, Hardwicke, P, Bridges, A, Votta, B.J, Gough, P.J, Marquis, R.W, Bertin, J, Casillas, L. | 登録日 | 2015-09-24 | 公開日 | 2015-10-21 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Crystal Structures of Human Rip2 Kinase Catalytic Domain Complexed with ATP-Competitive Inhibitors: Foundations for Understanding Inhibitor Selectivity. Bioorg.Med.Chem., 23, 2015
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3STB
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![BU of 3stb by Molmil](/molmil-images/mine/3stb) | A complex of two editosome proteins and two nanobodies | 分子名称: | MP18 RNA editing complex protein, RNA-editing complex protein MP42, single domain antibody VHH | 著者 | Park, Y.-J, Hol, W. | 登録日 | 2011-07-09 | 公開日 | 2011-11-02 | 最終更新日 | 2019-07-17 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structure of a heterodimer of editosome interaction proteins in complex with two copies of a cross-reacting nanobody. Nucleic Acids Res., 40, 2012
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5A1N
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2EHB
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![BU of 2ehb by Molmil](/molmil-images/mine/2ehb) | |
3F9K
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![BU of 3f9k by Molmil](/molmil-images/mine/3f9k) | |
2POM
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![BU of 2pom by Molmil](/molmil-images/mine/2pom) | TAB1 with manganese ion | 分子名称: | MANGANESE (II) ION, Mitogen-activated protein kinase kinase kinase 7-interacting protein 1 | 著者 | Lin, S.C. | 登録日 | 2007-04-26 | 公開日 | 2007-07-03 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.27 Å) | 主引用文献 | XIAP Induces NF-kappaB Activation via the BIR1/TAB1 Interaction and BIR1 Dimerization. Mol.Cell, 26, 2007
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7MU2
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![BU of 7mu2 by Molmil](/molmil-images/mine/7mu2) | Crystal Structure of WIPI2 in complex with W2IR of ATG16L1 | 分子名称: | Autophagy-related protein 16-1, WD repeat domain phosphoinositide-interacting protein 2 | 著者 | Strong, L.M, Flower, T.G, Buffalo, C.Z, Hurley, J.H. | 登録日 | 2021-05-14 | 公開日 | 2021-05-26 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Structural basis for membrane recruitment of ATG16L1 by WIPI2 in autophagy. Elife, 10, 2021
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2POP
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![BU of 2pop by Molmil](/molmil-images/mine/2pop) | The Crystal Structure of TAB1 and BIR1 complex | 分子名称: | Baculoviral IAP repeat-containing protein 4, Mitogen-activated protein kinase kinase kinase 7-interacting protein 1, ZINC ION | 著者 | Lin, S.C. | 登録日 | 2007-04-27 | 公開日 | 2007-07-03 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | XIAP Induces NF-kappaB Activation via the BIR1/TAB1 Interaction and BIR1 Dimerization. Mol.Cell, 26, 2007
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5ZAP
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![BU of 5zap by Molmil](/molmil-images/mine/5zap) | Atomic structure of the herpes simplex virus type 2 B-capsid | 分子名称: | Major capsid protein, Small capsomere-interacting protein, Triplex capsid protein 1, ... | 著者 | Yuan, S, Wang, J.L, Zhu, D.J, Wang, N, Gao, Q, Chen, W.Y, Tang, H, Wang, J.Z, Zhang, X.Z, Liu, H.R, Rao, Z.H, Wang, X.X. | 登録日 | 2018-02-08 | 公開日 | 2018-04-18 | 最終更新日 | 2018-09-05 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Cryo-EM structure of a herpesvirus capsid at 3.1 angstrom. Science, 360, 2018
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6DKQ
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![BU of 6dkq by Molmil](/molmil-images/mine/6dkq) | Crystal structure of the Shr Hemoglobin Interacting Domain 2 | 分子名称: | Heme-binding protein Shr, SULFATE ION | 著者 | Macdonald, R, Cascio, D, Collazo, M.J, Clubb, R.T. | 登録日 | 2018-05-30 | 公開日 | 2018-10-24 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | The Streptococcus pyogenes Shr protein captures human hemoglobin using two structurally unique binding domains. J.Biol.Chem., 293, 2018
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6ZSD
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![BU of 6zsd by Molmil](/molmil-images/mine/6zsd) | Human mitochondrial ribosome in complex with mRNA, P-site tRNA and E-site tRNA | 分子名称: | 12S mitochondrial rRNA, 16S mitochondrial rRNA, 28S ribosomal protein S10, ... | 著者 | Aibara, S, Singh, V, Modelska, A, Amunts, A. | 登録日 | 2020-07-15 | 公開日 | 2020-09-16 | 最終更新日 | 2024-07-10 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | Structural basis of mitochondrial translation. Elife, 9, 2020
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6ZSE
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![BU of 6zse by Molmil](/molmil-images/mine/6zse) | Human mitochondrial ribosome in complex with mRNA, A/P-tRNA and P/E-tRNA | 分子名称: | 12S mitochondrial rRNA, 16S mitochondrial rRNA, 28S ribosomal protein S10, ... | 著者 | Aibara, S, Singh, V, Modelska, A, Amunts, A. | 登録日 | 2020-07-15 | 公開日 | 2020-09-16 | 最終更新日 | 2024-07-10 | 実験手法 | ELECTRON MICROSCOPY (5 Å) | 主引用文献 | Structural basis of mitochondrial translation. Elife, 9, 2020
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