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1AZ4
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ECORV ENDONUCLEASE, UNLIGANDED, FORM B, T93A MUTANT
分子名称: ECORV ENDONUCLEASE
著者Perona, J, Martin, A.
登録日1997-11-24
公開日1998-05-27
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Conformational transitions and structural deformability of EcoRV endonuclease revealed by crystallographic analysis.
J.Mol.Biol., 273, 1997
5MKN
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Crystal structure of SmAP (LSm) protein from Methanococcus vannielii
分子名称: Like-Sm ribonucleoprotein core, TETRAETHYLENE GLYCOL, URIDINE-5'-MONOPHOSPHATE
著者Nikulin, A.D, Lekontseva, N.V, Tishchenko, S.V, Kravchenko, O.V.
登録日2016-12-05
公開日2017-12-20
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献Crystal structure of SmAP (LSm) protein from Methanococcus vannielii in complex with URIDINE-5'-MONOPHOSPHATE
To Be Published
1ASL
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BU of 1asl by Molmil
CRYSTAL STRUCTURES OF ESCHERICHIA COLI ASPARTATE AMINOTRANSFERASE IN TWO CONFORMATIONS: COMPARISON OF AN UNLIGANDED OPEN AND TWO LIGANDED CLOSED FORMS
分子名称: 2-[(3-HYDROXY-2-METHYL-5-PHOSPHONOOXYMETHYL-PYRIDIN-4-YLMETHYL)-AMINO]-2-METHYL-SUCCINIC ACID, ASPARTATE AMINOTRANSFERASE
著者Jaeger, J, Jansonius, J.N.
登録日1993-09-16
公開日1994-01-31
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Crystal structures of Escherichia coli aspartate aminotransferase in two conformations. Comparison of an unliganded open and two liganded closed forms.
J.Mol.Biol., 239, 1994
1ASZ
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THE ACTIVE SITE OF YEAST ASPARTYL-TRNA SYNTHETASE: STRUCTURAL AND FUNCTIONAL ASPECTS OF THE AMINOACYLATION REACTION
分子名称: ADENOSINE-5'-TRIPHOSPHATE, ASPARTYL-tRNA SYNTHETASE, T-RNA (75-MER)
著者Cavarelli, J, Rees, B, Thierry, J.C, Moras, D.
登録日1995-01-19
公開日1995-05-08
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献The active site of yeast aspartyl-tRNA synthetase: structural and functional aspects of the aminoacylation reaction.
EMBO J., 13, 1994
1AUO
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CARBOXYLESTERASE FROM PSEUDOMONAS FLUORESCENS
分子名称: CARBOXYLESTERASE
著者Kim, K.K, Song, H.K, Suh, S.W.
登録日1997-09-01
公開日1998-03-04
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Crystal structure of carboxylesterase from Pseudomonas fluorescens, an alpha/beta hydrolase with broad substrate specificity.
Structure, 5, 1997
1BCM
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BACTERIOPHAGE MU TRANSPOSASE CORE DOMAIN WITH 2 MONOMERS PER ASYMMETRIC UNIT
分子名称: BACTERIOPHAGE MU TRANSPOSASE
著者Rice, P.A, Mizuuchi, K.
登録日1995-05-26
公開日1995-10-15
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structure of the bacteriophage Mu transposase core: a common structural motif for DNA transposition and retroviral integration.
Cell(Cambridge,Mass.), 82, 1995
5F2S
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BU of 5f2s by Molmil
Crystal structure of human KDM4A in complex with compound 15
分子名称: 1,2-ETHANEDIOL, 2-(2-azanyl-1,3-thiazol-4-yl)pyridine-4-carboxylic acid, CHLORIDE ION, ...
著者Le Bihan, Y.-V, Dempster, S, Westwood, I.M, van Montfort, R.L.M.
登録日2015-12-02
公開日2016-01-20
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.08 Å)
主引用文献8-Substituted Pyrido[3,4-d]pyrimidin-4(3H)-one Derivatives As Potent, Cell Permeable, KDM4 (JMJD2) and KDM5 (JARID1) Histone Lysine Demethylase Inhibitors.
J.Med.Chem., 59, 2016
1AV5
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PKCI-SUBSTRATE ANALOG
分子名称: PHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER, PROTEIN KINASE C INTERACTING PROTEIN
著者Lima, C.D, Klein, M.G, Hendrickson, W.A.
登録日1997-09-25
公開日1998-03-25
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure-based analysis of catalysis and substrate definition in the HIT protein family.
Science, 278, 1997
6ZYU
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BU of 6zyu by Molmil
Structure of the GluA2 ligand-binding domain (L483Y-N754S) in complex with glutamate and BPAM549
分子名称: (4~{R})-4-cyclopropyl-7-fluoranyl-3,4-dihydro-2~{H}-thiochromene 1,1-dioxide, (4~{S})-4-cyclopropyl-7-fluoranyl-3,4-dihydro-2~{H}-thiochromene 1,1-dioxide, ACETATE ION, ...
著者Dorosz, J, Christensen, K.M, Kastrup, J.S.
登録日2020-08-03
公開日2021-08-11
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Development of Thiochroman Dioxide Analogues of Benzothiadiazine Dioxides as New Positive Allosteric Modulators of alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptors.
Acs Chem Neurosci, 12, 2021
1AYR
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BU of 1ayr by Molmil
ARRESTIN FROM BOVINE ROD OUTER SEGMENTS
分子名称: ARRESTIN
著者Granzin, J, Wilden, U, Choe, H.-W, Labahn, J, Krafft, B, Bueldt, G.
登録日1997-11-10
公開日1998-11-25
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献X-ray crystal structure of arrestin from bovine rod outer segments.
Nature, 391, 1998
1BFA
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BU of 1bfa by Molmil
RECOMBINANT BIFUNCTIONAL HAGEMAN FACTOR/AMYLASE INHIBITOR FROM MAIZE
分子名称: BIFUNCTIONAL AMYLASE/SERINE PROTEASE INHIBITOR
著者Behnke, C.A, Yee, V.C, Le Trong, I, Pedersen, L.C, Stenkamp, R.E, Kim, S.S, Reeck, G.R, Teller, D.C.
登録日1998-05-13
公開日1998-08-12
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structural determinants of the bifunctional corn Hageman factor inhibitor: x-ray crystal structure at 1.95 A resolution.
Biochemistry, 37, 1998
1AO6
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BU of 1ao6 by Molmil
CRYSTAL STRUCTURE OF HUMAN SERUM ALBUMIN
分子名称: SERUM ALBUMIN
著者Sugio, S, Mochizuki, S, Noda, M, Kashima, A.
登録日1997-07-18
公開日1998-05-27
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure of human serum albumin at 2.5 A resolution.
Protein Eng., 12, 1999
1ASB
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BU of 1asb by Molmil
THE STRUCTURAL BASIS FOR THE REDUCED ACTIVITY OF THE D223A(D222A) ACTIVE SITE MUTANT OF E. COLI ASPARTATE AMINOTRANSFERASE
分子名称: ASPARTATE AMINOTRANSFERASE, MALEIC ACID, PYRIDOXAL-5'-PHOSPHATE
著者Schumacher, C, Ringe, D.
登録日1993-08-27
公開日1994-04-30
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献The Structural Basis for the Reduced Activity of the D223A(D222A) Active Site Mutant of E. Coli Aspartate Aminotransferase
To be Published
5XCS
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BU of 5xcs by Molmil
Crystal structure of 12CA5 Fv-clasp fragment with its antigen peptide
分子名称: HA peptide, SULFATE ION, VH-SARAH(Y35C) chimera, ...
著者Arimori, T, Takagi, J.
登録日2017-03-23
公開日2017-10-04
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Fv-clasp: An Artificially Designed Small Antibody Fragment with Improved Production Compatibility, Stability, and Crystallizability
Structure, 25, 2017
1AYP
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BU of 1ayp by Molmil
A PROBE MOLECULE COMPOSED OF SEVENTEEN PERCENT OF TOTAL DIFFRACTING MATTER GIVES CORRECT SOLUTIONS IN MOLECULAR REPLACEMENT
分子名称: 1-OCTADECYL-2-ACETAMIDO-2-DEOXY-SN-GLYCEROL-3-PHOSPHOETHYLMETHYL SULFIDE, CALCIUM ION, PHOSPHOLIPASE A2
著者Oh, B.-H.
登録日1994-07-19
公開日1995-07-31
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.57 Å)
主引用文献A probe molecule composed of seventeen percent of total diffracting matter gives correct solutions in molecular replacement.
Acta Crystallogr.,Sect.D, 51, 1995
5XP8
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Crystal structure of T. thermophilus Argonaute protein complexed with a bulge 4A5 on the guide strand
分子名称: DNA (5'-D(*AP*GP*T)-3'), DNA (5'-D(*CP*AP*AP*CP*C*AP*TP*AP*CP*TP*AP*CP*CP*TP*CP*G)-3'), DNA (5'-D(P*TP*GP*AP*GP*AP*GP*TP*AP*GP*TP*AP*GP*GP*TP*TP*GP*T)-3'), ...
著者Sheng, G, Gogakos, T, Wang, J, Zhao, H, Serganov, A, Juranek, S, Tuschl, T, Patel, J.D, Wang, Y.
登録日2017-06-01
公開日2018-04-18
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structure/cleavage-based insights into helical perturbations at bulge sites within T. thermophilus Argonaute silencing complexes.
Nucleic Acids Res., 45, 2017
1AQC
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BU of 1aqc by Molmil
X11 PTB DOMAIN-10MER PEPTIDE COMPLEX
分子名称: PEPTIDE, X11
著者Lee, C.-H, Zhang, Z, Kuriyan, J.
登録日1997-07-28
公開日1997-12-24
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Sequence-specific recognition of the internalization motif of the Alzheimer's amyloid precursor protein by the X11 PTB domain.
EMBO J., 16, 1997
5XE5
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BU of 5xe5 by Molmil
Discovery and structural analysis of a phloretin hydrolase from the opportunistic pathogen Mycobacterium abscessus
分子名称: 1,2-ETHANEDIOL, MAGNESIUM ION, phloretin hydrolase
著者He, Y.X, Han, J.T, Jia, W.J, Zhang, Z.
登録日2017-04-01
公開日2018-05-02
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.17 Å)
主引用文献Discovery and structural analysis of a phloretin hydrolase from the opportunistic human pathogen Mycobacterium abscessus.
FEBS J., 2019
1ASD
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BU of 1asd by Molmil
THE STRUCTURE OF WILD TYPE E. COLI ASPARTATE AMINOTRANSFERASE RECONSTITUTED WITH N-MEPLP
分子名称: ASPARTATE AMINOTRANSFERASE, MALEIC ACID, N-METHYL-PYRIDOXAL-5'-PHOSPHATE
著者Schumacher, C, Ringe, D.
登録日1993-08-27
公開日1994-04-30
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The Structure of Wild Type E. Coli Aspartate Aminotransferase Reconstituted with N-Meplp
To be Published
1B5L
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OVINE INTERFERON TAU
分子名称: INTERFERON TAU, SULFATE ION
著者Radhakrishnan, R, Walter, L.J, Subramaniam, P.S, Johnson, H.J, Walter, M.R.
登録日1999-01-07
公開日1999-05-18
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystal structure of ovine interferon-tau at 2.1 A resolution.
J.Mol.Biol., 286, 1999
5XPR
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BU of 5xpr by Molmil
Human endothelin receptor type-B in complex with antagonist bosentan
分子名称: 4-tert-butyl-N-[6-(2-hydroxyethyloxy)-5-(2-methoxyphenoxy)-2-pyrimidin-2-yl-pyrimidin-4-yl]benzenesulfonamide, Endothelin B receptor,Endolysin,Endothelin B receptor, SULFATE ION
著者Shihoya, W, Nishizawa, T, Yamashita, K, Hirata, K, Okuta, A, Tani, K, Fujiyoshi, Y, Doi, T, Nureki, O.
登録日2017-06-04
公開日2017-08-16
最終更新日2017-11-15
実験手法X-RAY DIFFRACTION (3.6 Å)
主引用文献X-ray structures of endothelin ETB receptor bound to clinical antagonist bosentan and its analog
Nat. Struct. Mol. Biol., 24, 2017
5EY6
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BU of 5ey6 by Molmil
CRYSTAL STRUCTURE OF GLUTATHIONE TRANSFERASE F2 FROM POPULUS TRICHOCARPA
分子名称: Phi class glutathione transferase GSTF2
著者Didierjean, C, Rouhier, N, Pegeot, H, Gense, F.
登録日2015-11-24
公開日2016-12-07
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural plasticity among glutathione transferase Phi members: natural combination of catalytic residues confers dual biochemical activities.
FEBS J., 284, 2017
1ASE
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BU of 1ase by Molmil
THE STRUCTURE OF WILD TYPE E. COLI ASPARTATE AMINOTRANSFERASE RECONSTITUTED WITH PLP-N-OXIDE
分子名称: ASPARTATE AMINOTRANSFERASE, MALEIC ACID, PYRIDOXAL-5'-PHOSPHATE-N-OXIDE
著者Schumacher, C, Ringe, D.
登録日1993-08-27
公開日1994-04-30
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The Structure of Wild Type E. Coli Aspartate Aminotransferase Reconstituted with Plp-N-Oxide
To be Published
5IVC
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Linked KDM5A Jmj Domain Bound to the Inhibitor N3 (4'-[(2-phenylethyl)carbamoyl][2,2'-bipyridine]-4-carboxylic acid)
分子名称: 1,2-ETHANEDIOL, 4'-[(2-phenylethyl)carbamoyl][2,2'-bipyridine]-4-carboxylic acid, GLYCEROL, ...
著者Horton, J.R, Cheng, X.
登録日2016-03-20
公開日2016-07-27
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.573 Å)
主引用文献Structural Basis for KDM5A Histone Lysine Demethylase Inhibition by Diverse Compounds.
Cell Chem Biol, 23, 2016
1ASF
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THE STRUCTURAL BASIS FOR THE REDUCED ACTIVITY OF THE Y226F(Y225F) ACTIVE SITE MUTANT OF E. COLI ASPARTATE AMINOTRANSFERASE
分子名称: ASPARTATE AMINOTRANSFERASE, PYRIDOXAL-5'-PHOSPHATE, SULFATE ION
著者Schumacher, C, Ringe, D.
登録日1993-08-27
公開日1994-04-30
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献The Structural Basis for the Reduced Activity of the Y226F(Y225F) Active Site Mutant of E. Coli Aspartate Aminotransferase
To be Published

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